|
AU749214C
(en)
*
|
1997-11-21 |
2006-03-30 |
Purdue Neuroscience Company |
Substituted 2-aminoacetamides and the use thereof
|
|
DE60112272T2
(en)
*
|
2000-04-27 |
2006-05-24 |
Astellas Pharma Inc. |
Imidazopyridine DERIVATIVES
|
|
DE10117184A1
(en)
*
|
2001-04-05 |
2002-10-17 |
Gruenenthal Gmbh |
Substituted imidazole [1,2-a] pyridin-3-yl amide and amine compounds
|
|
PL366827A1
(en)
|
2001-06-21 |
2005-02-07 |
Smithkline Beecham Corporation |
Imidazo[1,2-a]pyridine derivatives for the prophylaxis and treatment of herpes viral infections
|
|
IL159811A0
(en)
*
|
2001-07-13 |
2004-06-20 |
Neurogen Corp |
Heteroaryl substituted fused bicyclic heteroaryl compounds as gabaa receptor ligands
|
|
DE60211539T2
(en)
|
2001-10-05 |
2006-09-21 |
Smithkline Beecham Corp. |
IMIDAZOPYRIDINE DERIVATIVES FOR USE IN THE TREATMENT OF HERPES VIRUS INFECTION
|
|
AU2002357740A1
(en)
|
2001-12-11 |
2003-06-23 |
Smithkline Beecham Corporation |
Pyrazolo-pyridine derivatives as antiherpes agents
|
|
WO2003076441A1
(en)
|
2002-03-07 |
2003-09-18 |
Smithkline Beecham Corporation |
Pyrazolopyrimidine and pyrazolotriazine derivatives and pharmaceutical compositions containing them
|
|
CN100537571C
(en)
|
2002-04-19 |
2009-09-09 |
细胞基因组公司 |
Imidazo[1,2-a]pyrazin-8-ylamines, method of making and method of use thereof
|
|
JP2005529919A
(en)
|
2002-05-10 |
2005-10-06 |
スミスクライン ビーチャム コーポレーション |
Therapeutic compounds
|
|
US7312341B2
(en)
|
2002-09-09 |
2007-12-25 |
Cgi Pharmaceuticals, Inc. |
6-aryl-imidazo[1,2-a] pyrazin-8-ylamines, method of making, and method of use thereof
|
|
MXPA05003058A
(en)
*
|
2002-09-19 |
2005-05-27 |
Schering Corp |
Imidazopyridines as cyclin dependent kinase inhibitors.
|
|
DE10246890A1
(en)
*
|
2002-10-08 |
2004-04-22 |
Grünenthal GmbH |
New C-(imidazo-(1,2-a)-pyridin-3-yl)-methylamines, are nitrogen monoxide synthase inhibitors useful e.g. for treating migraine, septic shock, neurodegenerative diseases, inflammatory pain or cancer
|
|
WO2004072080A1
(en)
|
2003-02-10 |
2004-08-26 |
Cellular Genomics, Inc. |
Certain 8-heteroaryl-6-phenyl-imidazo[1,2-a]pyrazines as modulators of hsp90 complex activity
|
|
US7405295B2
(en)
|
2003-06-04 |
2008-07-29 |
Cgi Pharmaceuticals, Inc. |
Certain imidazo[1,2-a]pyrazin-8-ylamines and method of inhibition of Bruton's tyrosine kinase by such compounds
|
|
US7393848B2
(en)
|
2003-06-30 |
2008-07-01 |
Cgi Pharmaceuticals, Inc. |
Certain heterocyclic substituted imidazo[1,2-A]pyrazin-8-ylamines and methods of inhibition of Bruton's tyrosine kinase by such compounds
|
|
WO2005019220A2
(en)
|
2003-08-11 |
2005-03-03 |
Cellular Genomics Inc. |
Substituted imidazo[1,2-a]pyrazines as modulators of kinase activity
|
|
JP5206405B2
(en)
*
|
2005-03-21 |
2013-06-12 |
エムイーアイ・ファーマ・インコーポレイテッド |
Imidazo [1,2-a] pyridine derivatives: production and pharmaceutical use
|
|
US7777040B2
(en)
|
2005-05-03 |
2010-08-17 |
Cgi Pharmaceuticals, Inc. |
Certain substituted ureas, as modulators of kinase activity
|
|
TW200800213A
(en)
|
2005-09-02 |
2008-01-01 |
Abbott Lab |
Novel imidazo based heterocycles
|
|
MX2008015747A
(en)
|
2006-06-06 |
2008-12-19 |
Schering Corp |
Imidazopyrazines as protein kinase inhibitors.
|
|
PL2121687T3
(en)
|
2006-12-22 |
2016-03-31 |
Astex Therapeutics Ltd |
Tricyclic amine derivatives as protein tyrosine kinase inhibitors
|
|
JP5442448B2
(en)
|
2006-12-22 |
2014-03-12 |
アステックス、セラピューティックス、リミテッド |
Bicyclic heterocyclic compounds as FGFR inhibitors
|
|
GB0720038D0
(en)
|
2007-10-12 |
2007-11-21 |
Astex Therapeutics Ltd |
New compounds
|
|
GB0720041D0
(en)
|
2007-10-12 |
2007-11-21 |
Astex Therapeutics Ltd |
New Compounds
|
|
EP2252617A1
(en)
|
2008-02-13 |
2010-11-24 |
CGI Pharmaceuticals, Inc. |
6-aryl-imidaz0[l, 2-a]pyrazine derivatives, method of making, and method of use thereof
|
|
EP2291187B1
(en)
|
2008-04-24 |
2018-08-15 |
Newlink Genetics Corporation |
Ido inhibitors
|
|
KR20110019385A
(en)
*
|
2008-05-29 |
2011-02-25 |
서트리스 파마슈티컬즈, 인코포레이티드 |
Imidazopyridine and related analogs as sirtuin modulators
|
|
GB0810902D0
(en)
|
2008-06-13 |
2008-07-23 |
Astex Therapeutics Ltd |
New compounds
|
|
US8450321B2
(en)
|
2008-12-08 |
2013-05-28 |
Gilead Connecticut, Inc. |
6-(1H-indazol-6-yl)-N-[4-(morpholin-4-yl)phenyl]imidazo-[1,2-A]pyrazin-8-amine, or a pharmaceutically acceptable salt thereof, as a SYK inhibitor
|
|
ES2590804T3
(en)
|
2008-12-08 |
2016-11-23 |
Gilead Connecticut, Inc. |
Imidazopyrazine Syk inhibitors
|
|
WO2010068258A1
(en)
|
2008-12-08 |
2010-06-17 |
Cgi Pharmaceuticals, Inc. |
Imidazopyrazine syk inhibitors
|
|
GB0906470D0
(en)
|
2009-04-15 |
2009-05-20 |
Astex Therapeutics Ltd |
New compounds
|
|
GB0906472D0
(en)
|
2009-04-15 |
2009-05-20 |
Astex Therapeutics Ltd |
New compounds
|
|
WO2011051342A1
(en)
|
2009-10-30 |
2011-05-05 |
Janssen Pharmaceutica Nv |
IMIDAZO[1,2-b]PYRIDAZINE DERIVATIVES AND THEIR USE AS PDE10 INHIBITORS
|
|
AR080754A1
(en)
|
2010-03-09 |
2012-05-09 |
Janssen Pharmaceutica Nv |
IMIDAZO DERIVATIVES (1,2-A) PIRAZINA AND ITS USE AS PDE10 INHIBITORS
|
|
KR101717809B1
(en)
|
2010-03-11 |
2017-03-17 |
질레드 코네티컷 인코포레이티드 |
Imidazopyridines syk inhibitors
|
|
US9173887B2
(en)
|
2010-12-22 |
2015-11-03 |
Abbvie Inc. |
Hepatitis C inhibitors and uses thereof
|
|
CA2838645C
(en)
|
2011-06-27 |
2020-03-10 |
Janssen Pharmaceutica Nv |
1-aryl-4-methyl-[1,2,4]triazolo[4,3-a]quinoxaline derivatives
|
|
DE102012200349A1
(en)
|
2012-01-11 |
2013-07-11 |
Bayer Intellectual Property Gmbh |
Substituted fused pyrimidines and triazines and their use
|
|
US9669035B2
(en)
|
2012-06-26 |
2017-06-06 |
Janssen Pharmaceutica Nv |
Combinations comprising PDE 2 inhibitors such as 1-aryl-4-methyl-[1,2,4]triazolo-[4,3-A]]quinoxaline compounds and PDE 10 inhibitors for use in the treatment of neurological of metabolic disorders
|
|
WO2014009305A1
(en)
|
2012-07-09 |
2014-01-16 |
Janssen Pharmaceutica Nv |
Inhibitors of phosphodiesterase 10 enzyme
|
|
US8778964B2
(en)
|
2012-11-05 |
2014-07-15 |
Bayer Pharma Aktiengesellschaft |
Hydroxy-substituted imidazo[1,2-a]-pyridinecarboxamides and their use
|
|
US8796305B2
(en)
|
2012-11-05 |
2014-08-05 |
Bayer Pharma Aktiengesellschaft |
Carboxy-substituted imidazo[1,2-a]pyridinecarboxamides and their use
|
|
US9126998B2
(en)
|
2012-11-05 |
2015-09-08 |
Bayer Pharma AG |
Amino-substituted imidazo[1,2-a]pyridinecarboxamides and their use
|
|
US9624214B2
(en)
|
2012-11-05 |
2017-04-18 |
Bayer Pharma Aktiengesellschaft |
Amino-substituted imidazo[1,2-a]pyridinecarboxamides and their use
|
|
DK2925757T3
(en)
|
2012-11-19 |
2018-01-15 |
Novartis Ag |
Compounds and compositions for the treatment of parasitic diseases
|
|
US9243001B2
(en)
*
|
2013-03-15 |
2016-01-26 |
Epizyme, Inc. |
Substituted benzene compounds
|
|
US20160031907A1
(en)
*
|
2013-03-15 |
2016-02-04 |
Epizyme, Inc. |
Substituted Benzene Compounds
|
|
CN105339368B
(en)
|
2013-06-04 |
2017-08-15 |
拜耳制药股份公司 |
Imidazo [1,2 a] pyridine of 3 aryl substitution and application thereof
|
|
CN105745215A
(en)
|
2013-07-10 |
2016-07-06 |
拜耳制药股份公司 |
Benzyl-1h-pyrazolo[3,4-b]pyridines and use thereof
|
|
US9918939B2
(en)
|
2013-07-30 |
2018-03-20 |
Gilead Connecticut, Inc. |
Formulation of Syk inhibitors
|
|
EP3027618B1
(en)
|
2013-07-30 |
2020-07-08 |
Gilead Connecticut, Inc. |
Polymorph of syk inhibitors
|
|
AU2014360537B2
(en)
|
2013-12-04 |
2017-09-07 |
Gilead Sciences, Inc. |
Methods for treating cancers
|
|
US9290505B2
(en)
|
2013-12-23 |
2016-03-22 |
Gilead Sciences, Inc. |
Substituted imidazo[1,2-a]pyrazines as Syk inhibitors
|
|
TWI735853B
(en)
|
2013-12-23 |
2021-08-11 |
美商克洛諾斯生技有限公司 |
Syk inhibitors
|
|
WO2015124544A1
(en)
|
2014-02-19 |
2015-08-27 |
Bayer Pharma Aktiengesellschaft |
3-(pyrimidine-2-yl)imidazo[1,2-a]pyridines
|
|
WO2015140199A1
(en)
|
2014-03-21 |
2015-09-24 |
Bayer Pharma Aktiengesellschaft |
Cyano-substituted imidazo[1,2-a]pyridinecarboxamides and their use
|
|
US20170057958A1
(en)
|
2014-05-02 |
2017-03-02 |
Bayer Pharma Aktiengesellschaft |
Enantiomers of the n-(2-amino-5-fluoro-2-methylpentyl)-8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]pyridine-3-carboxamide, as well as of the di- and trifluoro derivatives for the treatment of cardiovascular diseases
|
|
JP6310144B2
(en)
|
2014-07-14 |
2018-04-18 |
ギリアード サイエンシーズ, インコーポレイテッド |
Combinations for treating cancer
|
|
US10174021B2
(en)
|
2014-12-02 |
2019-01-08 |
Bayer Pharma Aktiengesellschaft |
Substituted pyrazolo[1,5-A]pyridines and their use
|
|
EP3227287B1
(en)
|
2014-12-02 |
2019-08-07 |
Bayer Pharma Aktiengesellschaft |
Heteroaryl-substituted imidazo[1,2-a]pyridines and their use
|
|
WO2016124564A1
(en)
|
2015-02-05 |
2016-08-11 |
Bayer Pharma Aktiengesellschaft |
N-substituted 8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyrazin-3-carboxamide derivatives as stimulators of soluble guanylate cylase (sgc) for the treatment of cardiovascular diseases
|
|
WO2016124565A1
(en)
|
2015-02-05 |
2016-08-11 |
Bayer Pharma Aktiengesellschaft |
Substituted pyrazolo[1,5-a]-pyridine-3-carboxamides and use thereof
|
|
WO2016161572A1
(en)
*
|
2015-04-08 |
2016-10-13 |
Merck Sharp & Dohme Corp. |
TrkA KINASE INHIBITORS, COMPOSITIONS AND METHODS THEREOF
|
|
WO2018184976A1
(en)
|
2017-04-05 |
2018-10-11 |
Bayer Pharma Aktiengesellschaft |
Substituted imidazo[1,2-a]pyridinecarboxamides and use of same
|
|
CN115028640A
(en)
|
2017-08-25 |
2022-09-09 |
吉利德科学公司 |
Polymorphic forms of a SYK inhibitor
|
|
CN113950479A
(en)
|
2019-02-22 |
2022-01-18 |
克洛诺斯生物股份有限公司 |
Solid forms of condensed pyrazines as SYK inhibitors
|
|
US11718622B2
(en)
|
2020-03-16 |
2023-08-08 |
Exelixis Inc. |
Heterocyclic adenosine receptor antagonists
|