AU5181779A - 5h-2,3-benzodiazepine derivatives - Google Patents

5h-2,3-benzodiazepine derivatives

Info

Publication number: AU5181779A
Authority: AU; Australia
Prior art keywords: benzodiazepine derivatives; benzodiazepine; derivatives
Prior art date: 1978-10-19
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Granted

Application number

AU51817/79A

Other versions

AU532079B2 (en

Inventor

Ferenc Andrasi

Jozef Borsy

Tamas Hamori

Katalin Goldschmidt Nee Horvath

Jeno Korosi

Tibor Land

Erzsebet Miglecz

Jozsef Szekely

Gabor Zolyomi

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Egyt Gyogyszervegyeszeti Gyar

Original Assignee

Egyt Gyogyszervegyeszeti Gyar

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1978-10-19

Filing date

1979-10-16

Publication date

1980-04-24

1978-10-19 Priority claimed from HU78GO1426A external-priority patent/HU179018B/en

1979-10-16 Application filed by Egyt Gyogyszervegyeszeti Gyar filed Critical Egyt Gyogyszervegyeszeti Gyar

1980-04-24 Publication of AU5181779A publication Critical patent/AU5181779A/en

1983-09-15 Application granted granted Critical

1983-09-15 Publication of AU532079B2 publication Critical patent/AU532079B2/en

1999-10-16 Anticipated expiration legal-status Critical

Status Ceased legal-status Critical Current

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
HUGO-1426		1978-10-19
HU78GO1426A HU179018B (en)	1978-10-19	1978-10-19	Process for producing new 5h-2,3-benzodiazepine derivatives

Publications (2)

Publication Number	Publication Date
AU5181779A true AU5181779A (en)	1980-04-24
AU532079B2 AU532079B2 (en)	1983-09-15

Family

ID=10996876

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AU51817/79A Ceased AU532079B2 (en)	1978-10-19	1979-10-16	5h-2,3-benzodiazepine derivatives

Country Status (25)

Country	Link
US (1)	US4322346A (en)
JP (1)	JPS5592377A (en)
AT (1)	AT373589B (en)
AU (1)	AU532079B2 (en)
BE (1)	BE879404A (en)
BG (1)	BG60270B1 (en)
CA (1)	CA1125749A (en)
CH (1)	CH643835A5 (en)
CS (1)	CS236456B2 (en)
DD (1)	DD146596A5 (en)
DE (1)	DE2940483A1 (en)
DK (1)	DK155327C (en)
ES (1)	ES485163A1 (en)
FI (1)	FI66604C (en)
FR (1)	FR2439189A1 (en)
GB (1)	GB2034706B (en)
GR (1)	GR74034B (en)
HU (1)	HU179018B (en)
IT (1)	IT1220947B (en)
NL (1)	NL190552C (en)
NO (1)	NO152048C (en)
PL (1)	PL124063B1 (en)
SE (1)	SE439919B (en)
SU (1)	SU1402258A3 (en)
YU (1)	YU41887B (en)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
AU648111B2 (en) *	1990-10-17	1994-04-14	Egis Gyogyszergyar	A new 5H-benzodiazepine derivative, pharmaceutical compositions containing same and process for preparing them

Families Citing this family (38)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
HU186760B (en) *	1981-03-12	1985-09-30	Gyogyszerkutato Intezet	Process for preparing 3,4-dihydro-5h-2,3-aenzodiazepine derivatives
HU191702B (en) *	1984-06-27	1987-03-30	Gyogyszerkutato Intezet	New process for preparing 1-aryl-5 h-2,3-benzodiazepines
HU191698B (en) *	1984-07-27	1987-03-30	Gyogyszerkutato Intezet	Process for producing new 1-aryl-5h-2beta-benzodiazepines
HU195788B (en) *	1986-05-21	1988-07-28	Gyogyszerkutato Intezet	Process for producing 1-/hydroxy-stiryl/-5h-2,3-benzobiazepines and pharmaceutical compositions containing them
JPH01311400A (en) *	1988-06-09	1989-12-15	Kyocera Corp	Method for lighting light emitting symbol body
JPH0251568U (en) *	1988-10-07	1990-04-11
JPH0324693U (en) *	1989-07-18	1991-03-14
HU208429B (en) *	1991-05-03	1993-10-28	Gyogyszerkutato Intezet	Process for producing 1-/3-chloro-phenyl/-4-methyl-7,8-dimethoxy-5h-2,3-benzodiazepine of high purity
US5939412A (en) *	1992-06-26	1999-08-17	Smithkline Beecham Corporation	Bicyclic fibrinogen antagonists
JP3497164B2 (en) *	1991-06-28	2004-02-16	スミスクライン・ビーチャム・コーポレイション	Bicyclic fibrinogen antagonist
US6458784B1 (en)	1994-06-29	2002-10-01	Smithkline Beecham Corporation	Vitronectin receptor antagonists
SK283859B6 (en) *	1995-02-09	2004-03-02	Egis Gy�Gyszergy�R Rt.	1- [2 '- (Substituted) vinyl] -5H-2,3-benzodiazepine derivatives, process for their preparation and intermediates for their preparation, medicaments containing them and their use
HU224435B1 (en) *	1995-02-09	2005-10-28	EGIS Gyógyszergyár Rt.	Benzodiazepine derivatives, process for producing them, their use and pharmaceutical compositions containing them
DE69612413T2 (en) *	1995-02-09	2001-09-27	Egis Gyogyszergyar Rt., Budapest	1- (hetero) arylvinyl-5H-2,3-benzodiazepine derivatives can be used for the treatment of diseases of the central nervous system, as well as benzopyrylium intermediates for their production
US5977101A (en) *	1995-06-29	1999-11-02	Smithkline Beecham Corporation	Benzimidazoles/Imidazoles Linked to a Fibrinogen Receptor Antagonist Template Having Vitronectin Receptor Antagonist Activity
DE19604920A1 (en) *	1996-02-01	1997-08-07	Schering Ag	New 2,3-benzodiazepine derivatives, their production and use as medicines
DE19604919A1 (en) *	1996-02-01	1997-08-07	Schering Ag	New 2,3-benzodiazepine derivatives, their production and use as medicines
ES2111493B1 (en) *	1996-02-08	1999-08-01	Egyt Gyogyszervegyeszeti Gyar	DERIVATIVES OF 1- (2- (SUBSTITUTED VINYL)) -5H-2,3-BENZO-DIAZEPINE, PROCEDURE FOR ITS PREPARATION, PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM AND CORRESPONDING UTILIZATIONS.
HU9600871D0 (en) *	1996-04-04	1996-05-28	Gyogyszerkutato Intezet	New 2,3-benzodiazepine derivatives
ZA972746B (en) *	1996-04-04	1998-10-09	Egyt Gyogyszervegyeszeti Gyar	Novel 2,3-benzodiazepine derivatives
HUP9701284A3 (en) *	1997-07-24	2005-11-28	Egyt Gyogyszervegyeszeti Gyar	Use of 2,3-benzodiazepine derivatives for producing pharmaceutical compositions for treating and prophylacting illnesses and conditions connected with the endogene opioide system
HU227128B1 (en) *	1999-07-07	2010-07-28	Egyt Gyogyszervegyeszeti Gyar	New 2,3-benzodiazepine derivatives
FR2824065A1 (en) *	2001-04-26	2002-10-31	Neuro3D	COMPOUNDS INHIBITORS OF CYCLIC NUCLEOTIDE PHOSPHODIESTERASES, PREPARATION AND USES
US6649607B2 (en) *	2001-05-18	2003-11-18	Vela Pharmaceuticals, Inc.	Compositions and methods for treating or preventing convulsions or seizures
DK1545546T3 (en) *	2002-09-13	2007-08-06	Motac Neuroscience Ltd	Treatment of dyskinesia with 2,3-benzodiazepines
DE60313474T2 (en) *	2002-09-17	2008-01-03	Motac Neuroscience Ltd.	TREATMENT OF DYSKINESIA
US6638928B1 (en)	2002-12-03	2003-10-28	Vela Pharmaceuticals, Inc.	Treatment of irritable bowel syndrome and nonulcer dyspepsia with substituted 2,3-benzodiazepines
US7022700B2 (en) *	2002-12-03	2006-04-04	Vela Pharmaceuticals, Inc.	Method of increasing neutrophil production using optically-pure (R)-2,3-benzodiazepines
WO2004050040A2 (en) *	2002-12-03	2004-06-17	Vela Pharmaceuticals, Inc.	Pharmaceutical composition of 1-(3,4-dimethoxyphenyl)-4-methyl-5-ethyl-7-methoxy-8-hydroxy-5h-2,3-benzodiazepine and uses thereof
AU2003303312A1 (en) *	2002-12-03	2004-08-30	Vela Pharmaceuticals, Inc.	Pharmaceutical composition of 1-(3-hydroxy-4-methoxyphenyl)-4-methyl-5-ethyl-7,8-dimethoxy-5h-2,3-benzodiazepine and uses therof
US6864251B2 (en) *	2002-12-03	2005-03-08	Vela Pharmaceuticals, Inc.	Treatment of LTB4-mediated inflammatory disorders with optically-pure (R)-2,3-benzodiazepines
US20040224943A1 (en) *	2003-02-19	2004-11-11	Leventer Steven M.	Method of lowering body temperature with (R) - 2,3-benzodiazepines
US20040162284A1 (en) *	2003-02-19	2004-08-19	Harris Herbert W.	Method of lowering body temperature with (S) tofisopam
US20070021412A1 (en) *	2003-05-16	2007-01-25	Vela Pharmaceuticals, Inc.	Treatment of gastrointestinal dysfunction and related stress with an enantiomerically-pure (S) 2,3-benzodiazepine
JP4611308B2 (en) *	2003-05-16	2011-01-12	ヴェラアクイジションコーポレイション	Treatment of gastrointestinal dysfunction and associated stress using enantiomerically pure (R) 2,3-benzodiazepines
US20040254173A1 (en) *	2003-06-13	2004-12-16	Leventer Steven M.	Modulation of dopamine responses with substituted (S)-2,3-benzodiazepines
HUP0302449A3 (en) *	2003-08-04	2005-06-28	Egis Gyogyszergyar Nyilvanosan	8-chloro-2,3-benzodiazepine derivatives, pharmaceutical compositions containing them and process for producing them
US7541355B2 (en) *	2005-05-23	2009-06-02	Vela Acquisition Corporation	Conversion process for 2,3-benzodiazepine enantiomers

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
USRE30014E (en)	1966-12-09	1979-05-29	Egyesult Gyogyazer-es Tapozergyar	1-(3,4-Dimethoxy-phenyl)-4-methyl-5-ethyl-7,8-dimethoxy-5H-2,3-benzodiazepine
GB1202579A (en) *	1966-12-09	1970-08-19	Egyt Gyogyszervegyeszeti Gyar	Pharmacologically active new isoquinoline derivative and process for preparing same
DK118660B (en) *	1966-12-09	1970-09-21	Egyt Gyogyszervegyeszeti Gyar	Analogous process for the preparation of 1- (3 ', 4'-dimethoxyphenyl) -3-methyl-4-ethyl-6,7-dimethoxy-isoquinoline-N-imide.
ZA712798B (en) *	1970-11-06	1972-02-23	Egyt Gyogyszervegyeszeti Gyar	New,pharmaceutically active 2,3-diazabicyclo(5.4.0)undecapentaene derivative and process for preparing same

1978
- 1978-10-19 HU HU78GO1426A patent/HU179018B/en not_active IP Right Cessation
1979
- 1979-10-03 YU YU2410/79A patent/YU41887B/en unknown
- 1979-10-04 AT AT0647279A patent/AT373589B/en not_active IP Right Cessation
- 1979-10-05 DE DE19792940483 patent/DE2940483A1/en active Granted
- 1979-10-12 SE SE7908481A patent/SE439919B/en not_active IP Right Cessation
- 1979-10-15 BE BE1/9569A patent/BE879404A/en not_active IP Right Cessation
- 1979-10-16 CH CH929279A patent/CH643835A5/en not_active IP Right Cessation
- 1979-10-16 AU AU51817/79A patent/AU532079B2/en not_active Ceased
- 1979-10-16 FI FI793209A patent/FI66604C/en not_active IP Right Cessation
- 1979-10-16 FR FR7925698A patent/FR2439189A1/en active Granted
- 1979-10-16 CS CS797020A patent/CS236456B2/en unknown
- 1979-10-17 DD DD79216290A patent/DD146596A5/en not_active IP Right Cessation
- 1979-10-17 GR GR60290A patent/GR74034B/el unknown
- 1979-10-18 NL NLAANVRAGE7907692,A patent/NL190552C/en not_active IP Right Cessation
- 1979-10-18 DK DK440179A patent/DK155327C/en not_active IP Right Cessation
- 1979-10-18 BG BG045206A patent/BG60270B1/en unknown
- 1979-10-18 NO NO793349A patent/NO152048C/en unknown
- 1979-10-18 IT IT7926579A patent/IT1220947B/en active
- 1979-10-18 GB GB7936185A patent/GB2034706B/en not_active Expired
- 1979-10-18 ES ES485163A patent/ES485163A1/en not_active Expired
- 1979-10-18 JP JP13471879A patent/JPS5592377A/en active Granted
- 1979-10-18 SU SU792832177A patent/SU1402258A3/en active
- 1979-10-18 CA CA337,955A patent/CA1125749A/en not_active Expired
- 1979-10-18 PL PL1979219034A patent/PL124063B1/en unknown
1980
- 1980-09-26 US US06/191,811 patent/US4322346A/en not_active Expired - Lifetime

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
AU648111B2 (en) *	1990-10-17	1994-04-14	Egis Gyogyszergyar	A new 5H-benzodiazepine derivative, pharmaceutical compositions containing same and process for preparing them

Publication	Publication Date	Title
AU532079B2 (en)	1983-09-15	5h-2,3-benzodiazepine derivatives
AU5181779A (en)	1980-04-24	5h-2,3-benzodiazepine derivatives
AU550388B2 (en)	1986-03-20	3,4-dihydro-5h-2,3-benzodiazepine derivatives
FI852906L (en)	1986-01-28	PROCEDURE FOR FRAMSTAELLNING AV 5H-2,3-BENZODIAZEPINE DERIVATIVES.
AU541679B2 (en)	1985-01-17	Ergolinyl -n:,n:-diethylurea derivatives
AU550032B2 (en)	1986-02-27	Benzodiazepine derivatives
AU7339781A (en)	1982-02-04	Benzodiazepine derivatives
AU533578B2 (en)	1983-12-01	4-phenyl-1,3-benzodiazepines
AU545491B2 (en)	1985-07-18	Benzodiazepine derivatives
AU530398B2 (en)	1983-07-14	N-substituted-2,6-dimethylmorpholine derivatives
AU509147B2 (en)	1980-04-24	Benzodiazepine derivatives
AU6881081A (en)	1981-10-08	Substituted-2,4,5-triarylthiazole derivatives
AU540897B2 (en)	1984-12-06	Carbamoyloxyamino-1,4-benzodiazepines
AU6048080A (en)	1981-01-15	1-substituted-3-cycloalkyl-sulphonyl-pyrrolidine-2,5-dione derivatives
AU528800B2 (en)	1983-05-12	Benzodiazepines
AU522783B2 (en)	1982-06-24	2phenyl-5,6-dihydro-4-pyrone derivatives
AU529072B2 (en)	1983-05-26	25-hydroxycholecalciferol-26,23-lactone
AU5709380A (en)	1980-10-09	5-aryl-1-hetero-1h-1,4-benzodiazepines
AU539507B2 (en)	1984-10-04	Methyl-quinaxoline-1,4-dioxide derivatives
AU5767980A (en)	1980-10-30	Tdm concentrator-deconcentrator
AU534512B2 (en)	1984-02-02	Spiro(dibenz(b,f)oxepin-piperidine)s
AU6212280A (en)	1981-08-20	Benzodiazepine derivatives
AU519623B2 (en)	1981-12-17	Pyrand [4,3-e]-as-triazines
AU518438B2 (en)	1981-10-01	Substituted 6-aryl-4h-s-triazolo-3,4-c-thieno-2,3-e-1,4-diazepines
AU3337178A (en)	1978-05-25	Mononitro-n-alkyl-3, 4-xylidines

AU5181779A - 5h-2,3-benzodiazepine derivatives - Google Patents

Info

Links

Applications Claiming Priority (2)

Publications (2)

Family

ID=10996876

Family Applications (1)

Country Status (25)

Cited By (1)

Families Citing this family (38)

Family Cites Families (4)

Cited By (1)

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