[go: up one dir, main page]

AU4752785A - 13-halo and 13 hydroxymilbemycins - Google Patents

13-halo and 13 hydroxymilbemycins

Info

Publication number
AU4752785A
AU4752785A AU47527/85A AU4752785A AU4752785A AU 4752785 A AU4752785 A AU 4752785A AU 47527/85 A AU47527/85 A AU 47527/85A AU 4752785 A AU4752785 A AU 4752785A AU 4752785 A AU4752785 A AU 4752785A
Authority
AU
Australia
Prior art keywords
hydroxymilbemycins
halo
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU47527/85A
Inventor
Bruno Frei
Peter Maienfisch
Anthony Cornelius O'sullivan
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Original Assignee
Ciba Geigy AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy AG filed Critical Ciba Geigy AG
Publication of AU4752785A publication Critical patent/AU4752785A/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AU47527/85A 1984-09-18 1985-09-17 13-halo and 13 hydroxymilbemycins Abandoned AU4752785A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH445784 1984-09-18
CH4457/84 1984-09-18

Publications (1)

Publication Number Publication Date
AU4752785A true AU4752785A (en) 1986-03-27

Family

ID=4276475

Family Applications (1)

Application Number Title Priority Date Filing Date
AU47527/85A Abandoned AU4752785A (en) 1984-09-18 1985-09-17 13-halo and 13 hydroxymilbemycins

Country Status (6)

Country Link
EP (1) EP0180539A1 (en)
JP (1) JPS6185390A (en)
AU (1) AU4752785A (en)
DK (1) DK420785A (en)
IL (1) IL76392A0 (en)
ZA (1) ZA857124B (en)

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU576029B2 (en) * 1984-11-26 1988-08-11 Ciba-Geigy Ag 5-azolylacetoxymilbemycins
AU587895B2 (en) * 1986-04-03 1989-08-31 Merck & Co., Inc. Avermectins as growth promotant agents
US5208222A (en) * 1991-03-28 1993-05-04 Merck & Co., Inc. 4"-and 4'-alkylthio avermectin derivatives
CN111217828A (en) * 2018-11-26 2020-06-02 浙江海正药业股份有限公司 Preparation method of lepithromycin and intermediate thereof

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FI860233A7 (en) * 1985-01-22 1986-07-23 Ciba Geigy Ag 13-alkyl-milbemycin derivatives for the control of animal and plant parasites.
US4587247A (en) * 1985-02-25 1986-05-06 Merck & Co., Inc. Substituted and unsubstituted 13-(alkoxy)methoxy derivatives of the avermectin aglycones, compositions and use
EP0235085A1 (en) * 1986-02-20 1987-09-02 Ciba-Geigy Ag 13-Beta-sugar derivatives of milbemycine, their preparation and use as ekto- and endo-parasitic agents for treatment of animals and plants
US4897416A (en) * 1987-02-18 1990-01-30 Ciba-Geigy Corporation Insecticides and parasiticides
US4918097A (en) * 1988-03-11 1990-04-17 Ciba-Geigy Corporation Insecticides and parasiticides
US5428034A (en) * 1988-09-02 1995-06-27 Sankyo Co., Ltd. Milbemycin derivatives, their preparation and their use
DE69100177T2 (en) * 1990-02-08 1994-01-27 Merck & Co Inc Flea control methods.
JP2622197B2 (en) * 1990-03-01 1997-06-18 三共株式会社 13-ether substituted milbemycin derivative
US5229416A (en) * 1992-04-29 1993-07-20 Merck & Co., Inc. Avermectin difluoro derivatives
WO1999055171A1 (en) * 1998-04-24 1999-11-04 Künzle Farma Ag Licking stone
HUP0301040A3 (en) 2000-04-27 2005-11-28 Sankyo Lifetech Company Ltd Bu Paraziticidal 13-substituted milbemycin derivatives, composition and use thereof

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4093629A (en) * 1977-04-11 1978-06-06 Merck & Co., Inc. Derivatives of antibiotic substance milbemycin and processes therefor
NZ186851A (en) * 1977-04-11 1984-12-14 Merck & Co Inc Glycosyloxy derivatives of milbemycin and parasiticidal compositions
PH16612A (en) * 1977-12-19 1983-11-28 Merck & Co Inc 13-halo and 13-deoxy derivatives of c-076 compounds
US4285963A (en) * 1980-08-07 1981-08-25 Merck & Co., Inc. Novel derivatives of C-076 compounds
NZ201681A (en) * 1981-09-03 1985-11-08 Merck & Co Inc Avermectin derivatives and parasiticidal compositions

Cited By (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU576029B2 (en) * 1984-11-26 1988-08-11 Ciba-Geigy Ag 5-azolylacetoxymilbemycins
AU587895B2 (en) * 1986-04-03 1989-08-31 Merck & Co., Inc. Avermectins as growth promotant agents
US5208222A (en) * 1991-03-28 1993-05-04 Merck & Co., Inc. 4"-and 4'-alkylthio avermectin derivatives
CN111217828A (en) * 2018-11-26 2020-06-02 浙江海正药业股份有限公司 Preparation method of lepithromycin and intermediate thereof
WO2020108146A1 (en) * 2018-11-26 2020-06-04 浙江海正药业股份有限公司 Preparation method for lepimectin, and intermediate thereof

Also Published As

Publication number Publication date
DK420785A (en) 1986-03-19
DK420785D0 (en) 1985-09-17
IL76392A0 (en) 1986-01-31
JPS6185390A (en) 1986-04-30
ZA857124B (en) 1987-05-27
EP0180539A1 (en) 1986-05-07

Similar Documents

Publication Publication Date Title
AU584321B2 (en) 17 ```(N-t-butylcarbamoyl)-4-aza-5```-androst-1-en-3-one
AU4177785A (en) Polyaminodithiols and radiopharmaceuticals
AU583361B2 (en) see form 10
AU576466B2 (en) Novel 4h-1-benzopyran-4-ones and benzothiopyran-4-ones
AU4752785A (en) 13-halo and 13 hydroxymilbemycins
GB2224742B (en) Polyanhydride-siloxanes and polymide-siloxanes obtained therefrom
AU583489B2 (en) 8alpha-acylamino-ergolines uses and production thereof
AU581445B2 (en) N-arylsulfonyl-N'-triazinylureas and N-arylsulfonyl-N'- pyrimidinylureas
AU6697086A (en) Immunoamplifiers and related compositions
CS304985A2 (en) Zpusob vyroby derivatu substituovaneho 3 fenyliminothiazolidinu
AU4617185A (en) Ketofin and anti-asthmatically effective xanthine
AU568750B2 (en) Imidazo-pyrrolo-pyridines and their use as herbacides
AU4064785A (en) Kraftspannfutter 300mm - 5000mm 0
AU4001785A (en) Substituted isochromanes and oxepines
AU3828585A (en) Imidazolo-isoindole and imidazolo-pyrrolo-pyridine derivatives
AU4914785A (en) Substituted 1-phenyl-3-benzoyl ureas and thioureas - pesticidal agents
CS733884A1 (en) Zpusob izolace 8 chinolinolu
IE842224L (en) Flavene and thioflavene derivatives
IE842223L (en) Flavene and thioflavene derivatives
CS328984A1 (en) Zpusob stanoveni 5 sulfoisoftalove kyseliny v elektrolytickych vybarvovacich roztocich
CS61384A2 (en) Zpusob vyroby derivatu pyridazinu substituovanych v poloze 3 substituovanou aminoskupinou
PL249544A2 (en) Three-socket 10-16a 250 v branch-joint with earthing and without earthing
CS55586A2 (en) Zpusob vyroby noveho derivatu 3 fenyl 2 propenaminu
CS598584A1 (en) Zpusob pripravy 1
CS392886A2 (en) Zpusob vyroby derivatu substituovaneho 3 fenyliminothiazolidinu