AU2616199A - Novel bicyclene-substituted oxazolidinones - Google Patents

Novel bicyclene-substituted oxazolidinones

Info

Publication number: AU2616199A
Authority: AU; Australia
Prior art keywords: bicyclene; novel; substituted oxazolidinones; oxazolidinones; substituted
Prior art date: 1998-01-22
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Abandoned

Application number

AU26161/99A

Inventor

Stephan Bartel

Rainer Endermann

Walter Guarnieri

Dieter Habich

Hein-Peter Kroll

Siegfried Raddatz

Bernd dr. Riedl

Ulrich Rosentreter

Martin Dr. Ruppelt

Andreas Stolle

Hanno dr. Wild

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Bayer AG

Original Assignee

Bayer AG

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1998-01-22

Filing date

1999-01-09

Publication date

1999-08-09

1999-01-09 Application filed by Bayer AG filed Critical Bayer AG

1999-08-09 Publication of AU2616199A publication Critical patent/AU2616199A/en

Status Abandoned legal-status Critical Current

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

AU26161/99A 1998-01-22 1999-01-09 Novel bicyclene-substituted oxazolidinones Abandoned AU2616199A (en)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
DE19802239A DE19802239A1 (en)	1998-01-22	1998-01-22	New oxazolidinone derivatives useful as antimicrobial agents against Gram-positive and some Gram-negative bacteria, mycobacteria, etc.
DE19802239		1998-01-22
PCT/EP1999/000096 WO1999037641A1 (en)	1998-01-22	1999-01-09	Novel bicyclene-substituted oxazolidinones

Publications (1)

Publication Number	Publication Date
AU2616199A true AU2616199A (en)	1999-08-09

Family

ID=7855292

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AU26161/99A Abandoned AU2616199A (en)	1998-01-22	1999-01-09	Novel bicyclene-substituted oxazolidinones

Country Status (5)

Country	Link
EP (1)	EP1049692A1 (en)
JP (1)	JP2002501065A (en)
AU (1)	AU2616199A (en)
DE (1)	DE19802239A1 (en)
WO (1)	WO1999037641A1 (en)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
BR0010982A (en) *	1999-05-27	2002-03-05	Upjohn Co	New bicyclic oxazolidinones as antibacterial agents
US6441005B1 (en) *	1999-07-28	2002-08-27	Pharmacia & Upjohn Company	Oxazolidinone compounds and compositions, and methods of using the same
GB9928568D0 (en)	1999-12-03	2000-02-02	Zeneca Ltd	Chemical compounds
DE19962924A1 (en)	1999-12-24	2001-07-05	Bayer Ag	Substituted oxazolidinones and their use
PE20011124A1 (en) *	2000-03-31	2001-10-28	Upjohn Co	NEW BENZOSULTAM OXAZOLIDINONE ANTIBACTERIAL AGENTS
GB0009803D0 (en)	2000-04-25	2000-06-07	Astrazeneca Ab	Chemical compounds
ATE321024T1 (en)	2000-10-17	2006-04-15	Pharmacia & Upjohn Co Llc	METHOD FOR PRODUCING OXAZOLIDINONE COMPOUNDS
PE20020689A1 (en) *	2000-11-17	2002-08-03	Upjohn Co	OXAZOLIDINONES WITH A HETEROCYCLE OF 6 OR 7 MEMBERS UNITED WITH ANNULAR LINK TO BENZENE
DE10129725A1 (en)	2001-06-20	2003-01-02	Bayer Ag	Combination therapy of substituted oxazolidinones
AR038536A1 (en)	2002-02-25	2005-01-19	Upjohn Co	N-ARIL-2-OXAZOLIDINONA-5- CARBOXAMIDS AND ITS DERIVATIVES
US7141588B2 (en)	2002-02-25	2006-11-28	Pfizer, Inc.	N-aryl-2-oxazolidinone-5-carboxamides and their derivatives
DE60304360T2 (en)	2002-08-12	2006-11-16	Pharmacia & Upjohn Co. Llc, Kalamazoo	N-ARYL-2-OXAZOLIDINONE AND DERIVATIVES
WO2004026848A1 (en) *	2002-09-20	2004-04-01	Lupin Limited	Oxazolidinone derivatives, process for their preperation and their use as antimycobacterial agents
AR042086A1 (en)	2002-11-21	2005-06-08	Upjohn Co	N-ARIL-2- OXAZOLIDINON -5- CARBOXAMIDS AND THEIR DERIVATIVES, USED AS ANTIBACTERIAL AGENTS
DE10300111A1 (en)	2003-01-07	2004-07-15	Bayer Healthcare Ag	Process for the preparation of 5-chloro-N - ({(5S) -2-oxo-3- [4- (3-oxo-4-morpholinyl) phenyl] -1,3-oxazolidin-5-yl} methyl ) -2-thiophenecarboxamide
US7304050B2 (en)	2003-09-16	2007-12-04	Pfizer Inc.	Antibacterial agents
DE10355461A1 (en)	2003-11-27	2005-06-23	Bayer Healthcare Ag	Solid, high bioavailabilty oral formulations of N-substituted 5-chloro-2-thiophene-carboxamide derivative in hydrophilized form, useful for combating thrombo-embolic diseases
DE102005045518A1 (en)	2005-09-23	2007-03-29	Bayer Healthcare Ag	New 5-thienylaminocarbonylmethyl-oxazolidin-2-one derivatives, useful for treating and preventing thromboembolic disease, are selective inhibitors of coagulation factor Xa
US7790745B2 (en)	2005-10-21	2010-09-07	Bristol-Myers Squibb Company	Tetrahydroisoquinoline LXR Modulators
CA2642406A1 (en) *	2006-02-14	2007-08-23	Pfizer Products Inc.	Benzoxazinone and benzoxazepinone oxazolidinones as antibacterial agents
WO2012166586A1 (en) *	2011-05-27	2012-12-06	Temple University - Of The Commonwealth System Of Higher Education	SUBSTITUTED 2-BENZYLIDENE-2H-BENZO[b][1,4]THIAZIN-3(4H)-ONES, DERIVATIVES THEREOF, AND THERAPEUTIC USES THEREOF
SG11201508479RA (en)	2013-04-16	2015-11-27	Actelion Pharmaceuticals Ltd	Antibacterial biaromatic derivatives
AR102256A1 (en)	2014-10-15	2017-02-15	Actelion Pharmaceuticals Ltd	ANTIBACTERIAL BASIC BIAROMATIC DERIVATIVES WITH REPLACEMENT OF AMINOALCOXI

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
EP0609905B1 (en) *	1988-09-15	2001-06-06	PHARMACIA & UPJOHN COMPANY	3-(Nitrogen substituted)phenyl-5beta-amidomethyloxazolidin-2-ones
DE4425612A1 (en) *	1994-07-20	1996-04-04	Bayer Ag	6-membered nitrogen-containing heteroaryl oxazolidinones
ZA968661B (en) *	1995-11-17	1998-04-14	Upjohn Co	Oxazolidinone antibacterial agent with tricyclic substituents.
DE19601265A1 (en) *	1996-01-16	1997-07-17	Bayer Ag	2-oxo and 2-thio-1,2-dihydroquinolinyl oxazolidinones
DE19604223A1 (en) *	1996-02-06	1997-08-07	Bayer Ag	New substituted oxazolidinones
DE19649095A1 (en) *	1996-02-06	1997-08-07	Bayer Ag	New 5-(acyl-aminomethyl)-3-hetero-aryl-oxazolidinone compounds

1998
- 1998-01-22 DE DE19802239A patent/DE19802239A1/en not_active Withdrawn
1999
- 1999-01-09 WO PCT/EP1999/000096 patent/WO1999037641A1/en not_active Ceased
- 1999-01-09 EP EP99906112A patent/EP1049692A1/en not_active Withdrawn
- 1999-01-09 AU AU26161/99A patent/AU2616199A/en not_active Abandoned
- 1999-01-09 JP JP2000528563A patent/JP2002501065A/en active Pending

Also Published As

Publication number	Publication date
JP2002501065A (en)	2002-01-15
DE19802239A1 (en)	1999-07-29
EP1049692A1 (en)	2000-11-08
WO1999037641A1 (en)	1999-07-29

Publication	Publication Date	Title
AU1251697A (en)	1997-08-14	New substituted oxazolidinones
AU3485999A (en)	1999-11-01	Neo-tryptophan
AU8441798A (en)	1999-02-10	Tricyclically substituted oxazolidinones
AU2616199A (en)	1999-08-09	Novel bicyclene-substituted oxazolidinones
AU9392998A (en)	1999-09-20	Pack-a-pillow
AU2623899A (en)	1999-09-06	Novel thiobenzamides
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AU4037699A (en)	1999-11-29	Novel aryl-hydro naphthalenal kanamines
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AU3253699A (en)	1999-09-06	Myxochelines
AU8363398A (en)	2000-01-24	Capotasto
AU2724799A (en)	1999-08-30	Novel endo-xylogalacturonase
AU2609599A (en)	2000-07-12	Sensor-coupling
AU3204999A (en)	1999-10-18	Futureball
AU2069199A (en)	1999-08-09	Codelets
AU1055399A (en)	1999-11-08	Rollerboard
AU5223199A (en)	2000-02-14	Bathtub-bathseat
AU3347599A (en)	1999-12-13	Aeromobile
AU9347498A (en)	2000-03-21	Imidazotriazolopyrimidines
AU2840799A (en)	1999-10-11	1-phosphanorbornadienes
AU9218098A (en)	2000-03-27	Exocyclic-phosphoethanolamines
AU1779099A (en)	1999-08-09	Heterocyclyl-derivatives

Legal Events

Date	Code	Title	Description
2000-10-05	MK6	Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase