AU2003279915A1 - Process for making azetidine-3-carboxylic acid - Google Patents
Process for making azetidine-3-carboxylic acidInfo
- Publication number
- AU2003279915A1 AU2003279915A1 AU2003279915A AU2003279915A AU2003279915A1 AU 2003279915 A1 AU2003279915 A1 AU 2003279915A1 AU 2003279915 A AU2003279915 A AU 2003279915A AU 2003279915 A AU2003279915 A AU 2003279915A AU 2003279915 A1 AU2003279915 A1 AU 2003279915A1
- Authority
- AU
- Australia
- Prior art keywords
- azetidine
- making
- carboxylic acid
- carboxylic
- acid
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
- C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D205/04—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US41856502P | 2002-10-15 | 2002-10-15 | |
| US60/418,565 | 2002-10-15 | ||
| PCT/US2003/032074 WO2004035538A1 (en) | 2002-10-15 | 2003-10-10 | Process for making azetidine-3-carboxylic acid |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AU2003279915A1 true AU2003279915A1 (en) | 2004-05-04 |
Family
ID=32107946
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2003279915A Abandoned AU2003279915A1 (en) | 2002-10-15 | 2003-10-10 | Process for making azetidine-3-carboxylic acid |
Country Status (2)
| Country | Link |
|---|---|
| AU (1) | AU2003279915A1 (en) |
| WO (1) | WO2004035538A1 (en) |
Families Citing this family (34)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2006010379A1 (en) | 2004-07-29 | 2006-02-02 | Actelion Pharmaceuticals Ltd. | Novel thiophene derivatives as immunosuppressive agents |
| PT1650186E (en) * | 2004-10-22 | 2008-09-16 | Bioprojet Soc Civ | Novel dicarboxylic acid derivatives |
| CA2583681A1 (en) * | 2004-10-22 | 2006-05-04 | Merck & Co., Inc. | 2-(aryl)azacyclylmethyl carboxylates, sulfonates, phosphonates, phosphinates and heterocycles as s1p receptor agonists |
| SI1863474T1 (en) | 2005-03-23 | 2009-04-30 | Actelion Pharmaceuticals Ltd | Novel thiophene derivatives as sphingosine-1-phosphate-1 receptor agonists |
| MX2007011670A (en) | 2005-03-23 | 2007-11-15 | Actelion Pharmaceuticals Ltd | Hydrogenated benzo (c) thiophene derivatives as immunomodulators. |
| AU2006256968A1 (en) * | 2005-06-08 | 2006-12-14 | Novartis Ag | Polycyclic oxadiazoles or I soxazoles and their use as SIP receptor ligands |
| TWI404706B (en) * | 2006-01-11 | 2013-08-11 | Actelion Pharmaceuticals Ltd | Novel thiophene derivatives |
| CA2635124C (en) | 2006-01-24 | 2014-04-29 | Actelion Pharmaceuticals Ltd | Novel pyridine derivatives |
| EP2021338A1 (en) | 2006-05-09 | 2009-02-11 | Pfizer Products Inc. | Cycloalkylamino acid derivatives and pharmaceutical compositions thereof |
| AR061841A1 (en) | 2006-09-07 | 2008-09-24 | Actelion Pharmaceuticals Ltd | DERIVATIVES OF THIOFEN-OXADIAZOLS, AGONISTS OF THE S1P1 / EDG1 RECEPTOR, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND USES AS IMMUNOMODULATING AGENTS. |
| AU2007292993B2 (en) | 2006-09-07 | 2013-01-24 | Idorsia Pharmaceuticals Ltd | Pyridin-4-yl derivatives as immunomodulating agents |
| BRPI0716633A2 (en) | 2006-09-08 | 2013-09-24 | Actelion Pharmaceuticals Ltd | pyridin-3-yl derivatives, pharmaceutical composition and use of a compound as an immunomodulatory agent |
| KR20090051774A (en) * | 2006-09-21 | 2009-05-22 | 액테리온 파마슈티칼 리미티드 | Phenyl derivatives and their use as immunomodulators |
| BRPI0720043A2 (en) | 2006-12-15 | 2014-01-07 | Abbott Lab | OXADIAZOL COMPOUND |
| CN101627034B (en) | 2007-03-16 | 2013-05-15 | 埃科特莱茵药品有限公司 | Amino-pyridine derivatives as S1P1/EDG1 receptor agonists |
| EP2014653A1 (en) * | 2007-06-15 | 2009-01-14 | Bioprojet | Novel dicarboxylic acid derivatives as S1P1 receptor agonists |
| PL2195311T3 (en) | 2007-08-17 | 2011-08-31 | Actelion Pharmaceuticals Ltd | Pyridine derivatives as s1p1/edg1 receptor modulators |
| CA2700917A1 (en) | 2007-11-01 | 2009-05-07 | Actelion Pharmaceuticals Ltd | Novel pyrimidine derivatives |
| US8148410B2 (en) | 2007-12-10 | 2012-04-03 | Actelion Pharmaceuticals Ltd. | Thiophene derivatives as agonists of S1P1/EDG1 |
| CA2715317A1 (en) * | 2008-03-07 | 2009-09-11 | Actelion Pharmaceuticals Ltd | Novel aminomethyl benzene derivatives |
| PL2252609T3 (en) * | 2008-03-07 | 2013-09-30 | Idorsia Pharmaceuticals Ltd | Pyridin-2-yl derivatives as immunomodulating agents |
| ES2441845T3 (en) | 2009-07-16 | 2014-02-06 | Actelion Pharmaceuticals Ltd. | Pyridin-4-yl derivatives as S1P1 / EDG1 agonists |
| US8399451B2 (en) | 2009-08-07 | 2013-03-19 | Bristol-Myers Squibb Company | Heterocyclic compounds |
| US8791100B2 (en) | 2010-02-02 | 2014-07-29 | Novartis Ag | Aryl benzylamine compounds |
| TWI546300B (en) | 2011-01-19 | 2016-08-21 | 艾克泰聯製藥有限公司 | 2-methoxy-pyridin-4-yl derivative |
| CN105189487B (en) | 2013-03-15 | 2017-12-26 | 爱杜西亚药品有限公司 | Pyridin-4-yl derivatives |
| CN103450171B (en) * | 2013-09-22 | 2015-07-08 | 苏州康乃德生物医药有限公司 | Novel immune adjustment compound, application thereof and medicine combination comprising same |
| CN105315266B (en) * | 2014-08-01 | 2019-10-01 | 苏州康乃德生物医药有限公司 | The crystal form of 1- { the fluoro- 4- of 2- [5- (4- isobutyl phenenyl) -1,2,4- oxadiazoles -3- base]-benzyl } -3- azetidinecarboxylic acid |
| BR112017024785B1 (en) | 2015-05-20 | 2022-05-17 | Idorsia Pharmaceuticals Ltd | CRYSTALLINE FORM OF COMPOUND (S)-3-{4-[5-(2-CYCLOPENTYL-6-METOXY-PYRIDIN-4-YL)-[1,2,4]OXADIAZOLE-3-YL]-2-ETHYL- 6-METHYLPHENOXY}-PROPANE-1,2-DIOL, PHARMACEUTICAL COMPOSITION, AND USE |
| CN107857760A (en) * | 2017-11-21 | 2018-03-30 | 南京天翔医药科技有限公司 | The phosphate receptor modulators of sphingol 1 and its application |
| CN109956912B (en) * | 2017-12-26 | 2021-10-22 | 中国医学科学院药物研究所 | Carboxylic acid compound containing diphenyloxadiazole, its preparation method and medical use |
| ES2978392T3 (en) | 2018-05-04 | 2024-09-11 | Suzhou Connect Biopharmaceuticals Ltd | Addition salt of S1P1 receptor agonist and crystalline form thereof, and pharmaceutical composition |
| JP7692032B2 (en) * | 2020-06-30 | 2025-06-12 | 上海 インスティテュート オブ マテリア メディカ、チャイニーズ アカデミー オブ サイエンシーズ | Oxadiazole compounds, their preparation, pharmaceutical compositions and uses |
| WO2025151705A1 (en) * | 2024-01-10 | 2025-07-17 | Vrise Therapeutics, Inc. | Novel inhibitors of dna damage repair pathway |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2005533058A (en) * | 2002-06-17 | 2005-11-04 | メルク エンド カムパニー インコーポレーテッド | 1-((5-Aryl-1,2,4-oxadiazol-3-yl) benzyl) azetidine-3-carboxylate and 1-((5-aryl-1,2,4) as EDG receptor agonists -Oxadiazol-3-yl) benzyl) pyrrolidine-3-carboxylate |
-
2003
- 2003-10-10 AU AU2003279915A patent/AU2003279915A1/en not_active Abandoned
- 2003-10-10 WO PCT/US2003/032074 patent/WO2004035538A1/en not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| WO2004035538A1 (en) | 2004-04-29 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MK6 | Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase |