AU2003272077A1 - Alpha-amino acid benzothiazolylthio ester as intermediates for manufacture of ace inhibitors and process for preparation thereof - Google Patents
Alpha-amino acid benzothiazolylthio ester as intermediates for manufacture of ace inhibitors and process for preparation thereofInfo
- Publication number
- AU2003272077A1 AU2003272077A1 AU2003272077A AU2003272077A AU2003272077A1 AU 2003272077 A1 AU2003272077 A1 AU 2003272077A1 AU 2003272077 A AU2003272077 A AU 2003272077A AU 2003272077 A AU2003272077 A AU 2003272077A AU 2003272077 A1 AU2003272077 A1 AU 2003272077A1
- Authority
- AU
- Australia
- Prior art keywords
- intermediates
- alpha
- manufacture
- preparation
- amino acid
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
- 239000005541 ACE inhibitor Substances 0.000 title 1
- -1 Alpha-amino acid benzothiazolylthio ester Chemical class 0.000 title 1
- 235000008206 alpha-amino acids Nutrition 0.000 title 1
- 229940044094 angiotensin-converting-enzyme inhibitor Drugs 0.000 title 1
- 239000000543 intermediate Substances 0.000 title 1
- 238000004519 manufacturing process Methods 0.000 title 1
- 238000000034 method Methods 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
- C07K5/022—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2
- C07K5/0222—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2 with the first amino acid being heterocyclic, e.g. Pro, Trp
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D277/70—Sulfur atoms
- C07D277/74—Sulfur atoms substituted by carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
- General Health & Medical Sciences (AREA)
- Genetics & Genomics (AREA)
- Medicinal Chemistry (AREA)
- Molecular Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Peptides Or Proteins (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PCT/IN2003/000257 WO2005010028A1 (en) | 2003-07-31 | 2003-07-31 | Alpha-amino acid benzothiazolylthio ester as intermediates for manufacture of ace inhibitors and process for preparation thereof |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AU2003272077A1 true AU2003272077A1 (en) | 2005-02-14 |
Family
ID=34090467
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2003272077A Abandoned AU2003272077A1 (en) | 2003-07-31 | 2003-07-31 | Alpha-amino acid benzothiazolylthio ester as intermediates for manufacture of ace inhibitors and process for preparation thereof |
Country Status (2)
| Country | Link |
|---|---|
| AU (1) | AU2003272077A1 (en) |
| WO (1) | WO2005010028A1 (en) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2006131828A1 (en) * | 2005-06-08 | 2006-12-14 | Aurobindo Pharma Limited | A process for the preparation of perindopril |
| CN106349185B (en) * | 2016-08-26 | 2018-07-06 | 河北科技大学 | 3- hydroxyadamantane glycine benzothiazole -2- thiol actives ester, preparation method and the application of a kind of amido protecting |
| CN106699592B (en) | 2016-11-17 | 2020-12-08 | 浙江华海药业股份有限公司 | Method for preparing lisinopril intermediate |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4847384A (en) * | 1987-03-12 | 1989-07-11 | Sandoz Pharm. Corp. | Process for the preparation of certain nitrogen-containing mono- and bicyclic ace inhibitors, and novel intermediates useful therefor |
| SI8811355A (en) * | 1988-07-13 | 1995-04-30 | Krka Tovarna Zdravil | Process for preparing of L-alanine-L-proline derivatives |
-
2003
- 2003-07-31 AU AU2003272077A patent/AU2003272077A1/en not_active Abandoned
- 2003-07-31 WO PCT/IN2003/000257 patent/WO2005010028A1/en not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| WO2005010028A1 (en) | 2005-02-03 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MK6 | Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase |