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AU2002230409A1 - Process for preparing 3-aryl-benzo(b)thiophenes - Google Patents

Process for preparing 3-aryl-benzo(b)thiophenes

Info

Publication number
AU2002230409A1
AU2002230409A1 AU2002230409A AU3040902A AU2002230409A1 AU 2002230409 A1 AU2002230409 A1 AU 2002230409A1 AU 2002230409 A AU2002230409 A AU 2002230409A AU 3040902 A AU3040902 A AU 3040902A AU 2002230409 A1 AU2002230409 A1 AU 2002230409A1
Authority
AU
Australia
Prior art keywords
thiophenes
benzo
aryl
preparing
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2002230409A
Inventor
Wayne Douglas Luke
Heidi Ann Sanderson
Hua Zheng
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eli Lilly and Co
Original Assignee
Eli Lilly and Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eli Lilly and Co filed Critical Eli Lilly and Co
Publication of AU2002230409A1 publication Critical patent/AU2002230409A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/62—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
    • C07D333/64—Oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/54—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • C07D333/56—Radicals substituted by oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
AU2002230409A 2000-11-27 2001-11-14 Process for preparing 3-aryl-benzo(b)thiophenes Abandoned AU2002230409A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US25321200P 2000-11-27 2000-11-27
US60/253,212 2000-11-27
PCT/US2001/042940 WO2002042289A2 (en) 2000-11-27 2001-11-14 Process for preparing 3-aryl-benzo[b]thiophenes

Publications (1)

Publication Number Publication Date
AU2002230409A1 true AU2002230409A1 (en) 2002-06-03

Family

ID=22959343

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2002230409A Abandoned AU2002230409A1 (en) 2000-11-27 2001-11-14 Process for preparing 3-aryl-benzo(b)thiophenes

Country Status (3)

Country Link
US (1) US6921827B2 (en)
AU (1) AU2002230409A1 (en)
WO (1) WO2002042289A2 (en)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2499819A1 (en) 2002-09-30 2004-04-08 A/S Gea Farmaceutisk Fabrik Novel raloxifene acid addition salts and/or solvates thereof, improved method for purification of said raloxifene acid addition salts and/or solvates thereof and pharmaceutical compositions comprising these
AU2002953533A0 (en) 2002-12-24 2003-01-16 Arthron Limited Fc receptor modulating compounds and compositions

Family Cites Families (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4133814A (en) 1975-10-28 1979-01-09 Eli Lilly And Company 2-Phenyl-3-aroylbenzothiophenes useful as antifertility agents
AU509682B2 (en) 1975-10-28 1980-05-22 Eli Lilly And Company 2-Aroyl-3-Phenylbenzothiophene Derivatives
US4418068A (en) 1981-04-03 1983-11-29 Eli Lilly And Company Antiestrogenic and antiandrugenic benzothiophenes
US4358593A (en) 1981-04-03 1982-11-09 Eli Lilly And Company Process for preparing 3-(4-aminoethoxybenzoyl)benzo[b]thiophenes
US4380635A (en) 1981-04-03 1983-04-19 Eli Lilly And Company Synthesis of acylated benzothiophenes
US5523416A (en) 1994-07-22 1996-06-04 Eli Lilly And Company Process for preparing 3-(4-aminoethoxy-benzoyl) benzo (B)-thiophenes
CO4410190A1 (en) 1994-09-19 1997-01-09 Lilly Co Eli 3- [4- (2-AMINOETOXI) -BENZOIL] -2-ARIL-6-HYDROXYBENZO [b] CRYSTALLINE THIOPHEN
US5629425A (en) 1994-09-19 1997-05-13 Eli Lilly And Company Haloalkyl hemisolvates of 6-hydroxy-2-(4-hydroxyphenyl)-3-[4-piperidinoethoxy)-benzoyl]benzo[b]thiophene
US5510357A (en) 1995-02-28 1996-04-23 Eli Lilly And Company Benzothiophene compounds as anti-estrogenic agents
US5552401A (en) 1995-02-28 1996-09-03 Eli Lilly And Company 2-benzyl-3-arylbenzothiophenes
ZA978372B (en) 1996-09-25 1999-03-17 Lilly Co Eli Process for the synthesis of benzothiophenes
ZA9710262B (en) 1996-11-19 1999-05-13 Lilly Co Eli Process for the synthesis of benzothiophenes
RU2186065C1 (en) * 1998-03-31 2002-07-27 Сионоги Энд Ко., Лтд. Method of synthesis of derivatives of 5-hydroxy-benzo[b]thiophene-3- carboxylic acid (variants) and thiophenic acid derivatives
DE19913349A1 (en) * 1999-03-24 2000-09-28 Clariant Gmbh Use of benzothiophene derivatives as components of liquid crystal mixtures, especially for use in ferroelectric switching and display devices
EP1204655B1 (en) 1999-07-29 2003-10-01 Eli Lilly And Company A crystalline form of 6-hydroxy-3-(4-[2-(piperidin-1-yl)ethoxy] phenoxy)-2-(4-methoxyphenyl)benzo[b]thiophene hydrochloride
AU6335600A (en) 1999-07-29 2001-02-19 Eli Lilly And Company A novel crystalline form of 6-hydroxy-3-(4-[2-(piperidin-1-yl)ethoxy]phenoxy)-2-(4-metho yphenyl)benzo[b]thiophene hydrochloride
ATE319702T1 (en) * 1999-08-02 2006-03-15 METHOD FOR PRODUCING BENZOTHIOPHENE DERIVATIVES
EP1222181B1 (en) * 1999-10-21 2003-12-10 Rhodia Chimie Method for preparing a benzofuran or benzothiophene compound
AU2002228593A8 (en) 2000-11-27 2008-06-12 Lilly Co Eli Process for preparing alpha-(3-arylthio)-acetophenones
US6388105B1 (en) * 2001-09-27 2002-05-14 Allergan Sales, Inc. Benzofuran, indole or benzothiophene 2,4-pentadienoic acid derivatives having selective activity for retinoid X (RXR) receptors

Also Published As

Publication number Publication date
WO2002042289A3 (en) 2002-09-06
US20040132775A1 (en) 2004-07-08
US6921827B2 (en) 2005-07-26
WO2002042289A8 (en) 2004-02-12
WO2002042289A2 (en) 2002-05-30

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