AU2002213978A1 - Substituted C-cyclohexylmethylamine derivatives - Google Patents

Substituted C-cyclohexylmethylamine derivatives

Info

Publication number: AU2002213978A1
Authority: AU; Australia
Prior art keywords: substituted; cyclohexylmethylamine derivatives; cyclohexylmethylamine; derivatives
Prior art date: 2000-09-29
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Granted

Application number

AU2002213978A

Other versions

AU2002213978B2 (en

Inventor

Helmut Buschmann

Michael Finkam

Babette-Yvonne Kogel

Corinna Maul

Bernd Sundermann

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Gruenenthal GmbH

Original Assignee

Gruenenthal GmbH

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-09-29

Filing date

2001-09-28

Publication date

2002-06-27

2000-09-29 Priority claimed from DE10049481A external-priority patent/DE10049481A1/en

2001-09-28 Application filed by Gruenenthal GmbH filed Critical Gruenenthal GmbH

2002-06-27 Publication of AU2002213978A1 publication Critical patent/AU2002213978A1/en

2007-10-18 Application granted granted Critical

2007-10-18 Publication of AU2002213978B2 publication Critical patent/AU2002213978B2/en

2021-09-28 Anticipated expiration legal-status Critical

Status Ceased legal-status Critical Current

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
DE10049481A DE10049481A1 (en)	2000-09-29	2000-09-29	Substituted C-cyclohexylmethylamine derivatives
DE10049481.1		2000-09-29
PCT/EP2001/011246 WO2002030870A2 (en)	2000-09-29	2001-09-28	Substituted c-cyclohexylmethylamine derivatives

Publications (2)

Publication Number	Publication Date
AU2002213978A1 true AU2002213978A1 (en)	2002-06-27
AU2002213978B2 AU2002213978B2 (en)	2007-10-18

Family

ID=7658870

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
AU2002213978A Ceased AU2002213978B2 (en)	2000-09-29	2001-09-28	Substituted C-cyclohexylmethylamine derivatives
AU1397802A Pending AU1397802A (en)	2000-09-29	2001-09-28	Substituted c-cyclohexylmethylamine derivatives

Family Applications After (1)

Application Number	Title	Priority Date	Filing Date
AU1397802A Pending AU1397802A (en)	2000-09-29	2001-09-28	Substituted c-cyclohexylmethylamine derivatives

Country Status (29)

Country	Link
US (1)	US7273952B2 (en)
EP (2)	EP1571140B1 (en)
JP (1)	JP2004524274A (en)
KR (1)	KR100893672B1 (en)
CN (1)	CN1547570A (en)
AR (1)	AR035062A1 (en)
AT (2)	ATE414056T1 (en)
AU (2)	AU2002213978B2 (en)
BR (1)	BR0114379A (en)
CA (1)	CA2423935A1 (en)
CY (2)	CY1105247T1 (en)
CZ (1)	CZ2003906A3 (en)
DE (3)	DE10049481A1 (en)
DK (2)	DK1571140T3 (en)
EC (1)	ECSP034531A (en)
ES (2)	ES2267833T3 (en)
HU (1)	HUP0303184A3 (en)
IL (1)	IL155103A0 (en)
MX (1)	MXPA03002348A (en)
NO (1)	NO20031386L (en)
NZ (2)	NZ525170A (en)
PE (1)	PE20030618A1 (en)
PL (1)	PL366057A1 (en)
PT (2)	PT1368299E (en)
RU (1)	RU2295515C2 (en)
SI (2)	SI1571140T1 (en)
SK (1)	SK3412003A3 (en)
WO (1)	WO2002030870A2 (en)
ZA (1)	ZA200303224B (en)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE10153346A1 (en)	2001-10-29	2004-04-22	Grünenthal GmbH	Substituted indoles
DE10153347A1 (en) *	2001-10-29	2003-05-08	Gruenenthal Gmbh	Substituted 1H-quinolin-2-one compounds
DE10161644A1 (en) *	2001-12-14	2003-06-26	Gruenenthal Gmbh	New N,N'-disubstituted piperazine derivatives are noradrenaline reuptake inhibitors, useful e.g. for the treatment of arrhythmia, emesis, diarrhea, inflammation or especially depression or pain
DE10261091A1 (en) *	2002-12-20	2004-07-01	Grünenthal GmbH	Saturated and unsaturated heteroarylcycloalkylmethyl amines
DE102004039382A1 (en) *	2004-08-13	2006-02-23	Grünenthal GmbH	Spirocyclic cyclohexane derivatives
DE102005061428A1 (en) *	2005-12-22	2007-08-16	Grünenthal GmbH	Substituted cyclohexylmethyl derivatives
TWI496762B (en)	2006-07-24	2015-08-21		Method for preparing (1R,2R)-3-(3-dimethylamino-1-ethyl-2-methyl-propyl)-phenol
CN103936605B (en)	2007-05-31	2017-09-01	赛诺维信制药公司	The cycloalkanes amine of phenyl substitution is used as monoamine reuptaking inhibitor
CN101906056B (en) *	2009-06-04	2013-10-30	中国科学院广州生物医药与健康研究院	Cycloalkane amine compound as M2 inhibitor and application thereof
RU2431479C2 (en) *	2010-07-19	2011-10-20	Государственное образовательное учреждение высшего профессионального образования Казанский государственный медицинский университет	2-(1'-hydroxy-4'-isopropylene-1'-methylcyclohexyl-2'-thio)-methyl ethanoate exhibiting fungicidal and anti-inflammatory action
WO2012100423A1 (en) *	2011-01-27	2012-08-02	Eli Lilly And Company	Analgesic compounds, methods, and formulations
CN105837454B (en) *	2016-04-21	2018-06-08	河南师范大学	A kind of synthetic method of 3,3- difiuorocyclohexyls methylamine
CN112759545B (en) *	2019-11-06	2022-12-13	复旦大学	3- (dimethylamino methyl) piperidine-4-alcohol derivative and preparation method and pharmaceutical application thereof
WO2021088758A1 (en) *	2019-11-06	2021-05-14	复旦大学	Opioid receptor agonist, preparation method therefor and pharmaceutical use thereof
CN112759538B (en) *	2019-11-06	2022-01-18	复旦大学	3- (dimethylaminomethyl) cyclohexan-4-ol derivative, preparation method and pharmaceutical application thereof
CN112759546B (en) *	2019-11-06	2022-08-26	复旦大学	3- (dimethylaminomethyl) piperidin-4-ol derivatives, their preparation and their pharmaceutical use
CN112759587B (en) *	2019-11-06	2022-12-30	复旦大学	3- (dimethylamino methyl) piperidine-4-alcohol derivative and preparation method and pharmaceutical application thereof
CN112759544B (en) *	2019-11-06	2022-08-26	复旦大学	Preparation method and pharmaceutical application of 3- (dimethylaminomethyl) piperidine-4-alcohol derivative

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
BE615646A (en)	1961-03-27	1900-01-01
US3165428A (en)	1962-12-27	1965-01-12	Westinghouse Electric Corp	Production of thin goss oriented magnetic materials
US3975436A (en) *	1974-03-27	1976-08-17	American Home Products Corporation	Benzylamine narcotic antagonists
DE2614244A1 (en) *	1976-04-02	1977-10-20	Bayer Ag	CYCLOALIPHATIC TRIAMINES
IL103096A (en) *	1992-09-08	1996-12-05	Chemagis Ltd	Process for the purification of 2-[(dimethyllamino)methyl]-1-(3-methoxyphenyl) cyclohexanol and its salts
DE19525137C2 (en) *	1995-07-11	2003-02-27	Gruenenthal Gmbh	6-Dimethylaminomethyl-1-phenyl-cyclohexane compounds as intermediates for the preparation of pharmaceutical agents
DE19547766A1 (en) *	1995-12-20	1997-06-26	Gruenenthal Gmbh	1-phenyl-2-dimethylaminomethyl-cyclohexan-1-ol compounds as active pharmaceutical ingredients
DE19609847A1 (en) *	1996-03-13	1997-09-18	Gruenenthal Gmbh	Dimethyl- (3-aryl-but-3-enyl) amine compounds as active pharmaceutical ingredients
JP4334766B2 (en)	1998-04-01	2009-09-30	カーディオムファーマコーポレイション	Aminocyclohexyl ether compounds and uses thereof
EP1077923B1 (en)	1998-05-22	2004-01-02	Mallinckrodt Inc.	An improved synthesis and purification of (r,r)-2- (dimethylamino) methyl]-1-( 3-methoxyphenyl) cyclohexanol hydrochloride
DE19915601A1 (en) *	1999-04-07	2000-10-19	Gruenenthal Gmbh	3-Amino-3-arylpropan-1-ol derivatives, their preparation and use
DE19957342A1 (en) *	1999-11-29	2001-05-31	Gruenenthal Gmbh	Treatment of interleukin (IL)-12 mediated illnesses comprises simultaneous administration of thalidomide or analogue and antiinflammatory cytokine
DE10004926A1 (en) *	2000-02-04	2001-08-09	Gruenenthal Gmbh	Process for the enzymatic resolution of aminomethyl aryl cyclohexanol derivatives

2000
- 2000-09-29 DE DE10049481A patent/DE10049481A1/en not_active Withdrawn
2001
- 2001-09-28 RU RU2003111757/04A patent/RU2295515C2/en not_active IP Right Cessation
- 2001-09-28 PT PT01982379T patent/PT1368299E/en unknown
- 2001-09-28 ES ES01982379T patent/ES2267833T3/en not_active Expired - Lifetime
- 2001-09-28 SI SI200130896T patent/SI1571140T1/en unknown
- 2001-09-28 AU AU2002213978A patent/AU2002213978B2/en not_active Ceased
- 2001-09-28 DK DK05011581T patent/DK1571140T3/en active
- 2001-09-28 PE PE2001000972A patent/PE20030618A1/en not_active Application Discontinuation
- 2001-09-28 KR KR1020037004578A patent/KR100893672B1/en not_active Expired - Fee Related
- 2001-09-28 PL PL01366057A patent/PL366057A1/en not_active Application Discontinuation
- 2001-09-28 DE DE50110569T patent/DE50110569D1/en not_active Expired - Lifetime
- 2001-09-28 AT AT05011581T patent/ATE414056T1/en active
- 2001-09-28 DE DE50114491T patent/DE50114491D1/en not_active Expired - Lifetime
- 2001-09-28 WO PCT/EP2001/011246 patent/WO2002030870A2/en not_active Ceased
- 2001-09-28 AU AU1397802A patent/AU1397802A/en active Pending
- 2001-09-28 JP JP2002534259A patent/JP2004524274A/en active Pending
- 2001-09-28 EP EP05011581A patent/EP1571140B1/en not_active Expired - Lifetime
- 2001-09-28 IL IL15510301A patent/IL155103A0/en unknown
- 2001-09-28 DK DK01982379T patent/DK1368299T3/en active
- 2001-09-28 MX MXPA03002348A patent/MXPA03002348A/en active IP Right Grant
- 2001-09-28 BR BR0114379-4A patent/BR0114379A/en not_active IP Right Cessation
- 2001-09-28 CZ CZ2003906A patent/CZ2003906A3/en unknown
- 2001-09-28 EP EP01982379A patent/EP1368299B1/en not_active Expired - Lifetime
- 2001-09-28 ES ES05011581T patent/ES2317103T3/en not_active Expired - Lifetime
- 2001-09-28 SK SK341-2003A patent/SK3412003A3/en not_active Application Discontinuation
- 2001-09-28 SI SI200130633T patent/SI1368299T1/en unknown
- 2001-09-28 CA CA002423935A patent/CA2423935A1/en not_active Abandoned
- 2001-09-28 CN CNA018164951A patent/CN1547570A/en active Pending
- 2001-09-28 NZ NZ525170A patent/NZ525170A/en unknown
- 2001-09-28 AT AT01982379T patent/ATE334114T1/en active
- 2001-09-28 HU HU0303184A patent/HUP0303184A3/en unknown
- 2001-09-28 AR ARP010104582A patent/AR035062A1/en unknown
- 2001-09-28 NZ NZ545879A patent/NZ545879A/en unknown
- 2001-09-28 PT PT05011581T patent/PT1571140E/en unknown
2003
- 2003-03-26 NO NO20031386A patent/NO20031386L/en not_active Application Discontinuation
- 2003-03-28 EC EC2003004531A patent/ECSP034531A/en unknown
- 2003-03-31 US US10/402,260 patent/US7273952B2/en not_active Expired - Fee Related
- 2003-04-24 ZA ZA200303224A patent/ZA200303224B/en unknown
2006
- 2006-09-12 CY CY20061101292T patent/CY1105247T1/en unknown
2009
- 2009-02-03 CY CY20091100123T patent/CY1110258T1/en unknown

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