AU2001291739A1 - 1h-pyrazol derivatives, method for producing them and their use as nitrificationinhibitors - Google Patents
1h-pyrazol derivatives, method for producing them and their use as nitrificationinhibitorsInfo
- Publication number
- AU2001291739A1 AU2001291739A1 AU2001291739A AU9173901A AU2001291739A1 AU 2001291739 A1 AU2001291739 A1 AU 2001291739A1 AU 2001291739 A AU2001291739 A AU 2001291739A AU 9173901 A AU9173901 A AU 9173901A AU 2001291739 A1 AU2001291739 A1 AU 2001291739A1
- Authority
- AU
- Australia
- Prior art keywords
- alkyl
- represent
- aryl
- nitrificationinhibitors
- producing
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
- WTKZEGDFNFYCGP-UHFFFAOYSA-N Pyrazole Chemical class C=1C=NNC=1 WTKZEGDFNFYCGP-UHFFFAOYSA-N 0.000 title abstract 2
- 238000004519 manufacturing process Methods 0.000 title 1
- 125000000041 C6-C10 aryl group Chemical group 0.000 abstract 3
- 125000004178 (C1-C4) alkyl group Chemical group 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 230000002401 inhibitory effect Effects 0.000 abstract 2
- 125000004209 (C1-C8) alkyl group Chemical group 0.000 abstract 1
- 125000002877 alkyl aryl group Chemical group 0.000 abstract 1
- 239000003337 fertilizer Substances 0.000 abstract 1
- 229910052736 halogen Inorganic materials 0.000 abstract 1
- 150000002367 halogens Chemical class 0.000 abstract 1
- 230000007062 hydrolysis Effects 0.000 abstract 1
- 238000006460 hydrolysis reaction Methods 0.000 abstract 1
- 230000002209 hydrophobic effect Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C05—FERTILISERS; MANUFACTURE THEREOF
- C05G—MIXTURES OF FERTILISERS COVERED INDIVIDUALLY BY DIFFERENT SUBCLASSES OF CLASS C05; MIXTURES OF ONE OR MORE FERTILISERS WITH MATERIALS NOT HAVING A SPECIFIC FERTILISING ACTIVITY, e.g. PESTICIDES, SOIL-CONDITIONERS, WETTING AGENTS; FERTILISERS CHARACTERISED BY THEIR FORM
- C05G3/00—Mixtures of one or more fertilisers with additives not having a specially fertilising activity
- C05G3/90—Mixtures of one or more fertilisers with additives not having a specially fertilising activity for affecting the nitrification of ammonium compounds or urea in the soil
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/16—Halogen atoms or nitro radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P60/00—Technologies relating to agriculture, livestock or agroalimentary industries
- Y02P60/20—Reduction of greenhouse gas [GHG] emissions in agriculture, e.g. CO2
- Y02P60/21—Dinitrogen oxide [N2O], e.g. using aquaponics, hydroponics or efficiency measures
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Soil Sciences (AREA)
- Pest Control & Pesticides (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Fertilizers (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Abstract
The invention relates to 1H-pyrazol derivatives corresponding to general formula (I), wherein R<1> and R<3>, independently of each other, represent H or a C1-C4-alkyl radical, R<2> represents H, halogen or a C1-C4-alkyl radical, R<1> and R<2>, together, represent a five or six-membered cycloalkyl radical, R<4> and R<5>, independently of each other, represent H or Cl, and X represents OR<6> or NHR<7>, R<6> representing C1-C4-alkyl, C6-C10-aryl or alkylaryl with C1-C4-alkyl- and C6-C10-aryl groups and R<7> representing C1-C8-alkyl or C6-C10-aryl. The inventive compounds are suitable for inhibiting or controlling nitrification. In addition to their good nitrification-inhibiting effect, the compounds have a low hydrolysis tendency and can be applied particularly well to the surface of the fertiliser due to their hydrophobic properties.
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10038608 | 2000-08-08 | ||
| DE10038608 | 2000-08-08 | ||
| PCT/EP2001/009074 WO2002012197A1 (en) | 2000-08-08 | 2001-08-06 | 1h-pyrazol derivatives, method for producing them and their use as nitrification inhibitors |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AU2001291739A1 true AU2001291739A1 (en) | 2002-02-18 |
Family
ID=7651681
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2001291739A Abandoned AU2001291739A1 (en) | 2000-08-08 | 2001-08-06 | 1h-pyrazol derivatives, method for producing them and their use as nitrificationinhibitors |
Country Status (5)
| Country | Link |
|---|---|
| EP (1) | EP1309561B1 (en) |
| AT (1) | ATE342255T1 (en) |
| AU (1) | AU2001291739A1 (en) |
| DE (2) | DE10135423A1 (en) |
| WO (1) | WO2002012197A1 (en) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE10224823A1 (en) * | 2002-06-05 | 2003-12-24 | Piesteritz Stickstoff | 1H-pyrazole derivatives, process for their preparation and their use as nitrification inhibitors |
| DE10343277A1 (en) | 2003-09-18 | 2005-04-21 | Piesteritz Stickstoff | N- (1H-Azolyl-methyl) amides, process for their preparation and their use as nitrification inhibitors |
| DE102008020785B4 (en) | 2008-04-25 | 2021-11-04 | Skw Stickstoffwerke Piesteritz Gmbh | Use of simple derivatives of 5-amino-1,2,4-thiadiazole to inhibit or control nitrification |
| DE102011120098B4 (en) | 2011-12-02 | 2021-02-11 | Skw Stickstoffwerke Piesteritz Gmbh | N- (1H-pyrazolyl-methyl) formamides, process for their preparation and their use as nitrification inhibitors |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE19503827A1 (en) * | 1995-02-06 | 1996-08-08 | Basf Ag | Use of low volatility pyrazole derivatives with hydrophilic groups as nitrification inhibitors |
| DE19849496B4 (en) * | 1997-10-28 | 2007-06-14 | Skw Stickstoffwerke Piesteritz Gmbh | Non-volatile alkylpyrazole derivatives, processes for their preparation and their use as nitrification inhibitors |
| DE19913475A1 (en) * | 1999-03-25 | 2000-09-28 | Piesteritz Stickstoff | Use of non-volatile new and known 2-chloro-1-azolyl-ethanol compounds, as nitrification inhibitors in fertilizers |
-
2001
- 2001-07-20 DE DE10135423A patent/DE10135423A1/en not_active Withdrawn
- 2001-08-06 WO PCT/EP2001/009074 patent/WO2002012197A1/en not_active Ceased
- 2001-08-06 AT AT01971875T patent/ATE342255T1/en not_active IP Right Cessation
- 2001-08-06 EP EP01971875A patent/EP1309561B1/en not_active Expired - Lifetime
- 2001-08-06 AU AU2001291739A patent/AU2001291739A1/en not_active Abandoned
- 2001-08-06 DE DE50111217T patent/DE50111217D1/en not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| ATE342255T1 (en) | 2006-11-15 |
| EP1309561B1 (en) | 2006-10-11 |
| EP1309561A1 (en) | 2003-05-14 |
| DE50111217D1 (en) | 2006-11-23 |
| WO2002012197A1 (en) | 2002-02-14 |
| DE10135423A1 (en) | 2002-02-21 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| AU2003284352A1 (en) | Pentafluoropropene-based compositions | |
| WO2002032898A3 (en) | Novel anticholinergics, method for the production thereof and use thereof as medicaments | |
| CA2349227A1 (en) | Substituted 2-phenylbenzimidazoles, the production thereof and their use | |
| MXPA04000622A (en) | Pyrazolylcarboxanilides as fungicides. | |
| MXPA03008755A (en) | 2-amino-propanol derivatives. | |
| MXPA04005802A (en) | Substituted phenyl derivatives. | |
| BG105177A (en) | Novel substituted pyrazole derivatives | |
| AU2795000A (en) | Epothilone derivatives and their use as antitumor agents | |
| WO2004011453A3 (en) | Method for preparing 3-halo-4,5-dihydro-1h-pyrazoles | |
| GB9929552D0 (en) | Compounds | |
| GB0114185D0 (en) | Compounds | |
| SE0004245D0 (en) | Novel compounds and their use | |
| WO2002014439A3 (en) | Process for producing coatings using surface-active photoinitiators | |
| PL335839A1 (en) | Cycloalkylalkane carboxamides as well as their production and application | |
| CA2309474A1 (en) | New 4-arylpiperidine derivatives for the treatment of pruritus | |
| AU2001291739A1 (en) | 1h-pyrazol derivatives, method for producing them and their use as nitrificationinhibitors | |
| AU2003235806A1 (en) | Dibenzodiazepine derivates, their preparation and use | |
| GB0019124D0 (en) | Novel process | |
| WO2002059089A3 (en) | Process for the preparation of heterocyclic indene analogs | |
| AU2001246537A1 (en) | 1h-pyrazole derivatives, method for the production thereof and their use for inhibiting and controlling nitrification | |
| MXPA02001406A (en) | Substituted heterocyclyl-2h-chromenes. | |
| ID27440A (en) | PROCESS FOR PREPARING | |
| WO2002046152A3 (en) | Coniosetin and derivatives thereof, method for producing the same and use thereof | |
| CA2309485A1 (en) | New 4-arylpiperidine derivatives for the treatment of pruritus | |
| AU2002359985A1 (en) | Diaryl 1,2,4-triazole derivatives as a highly selective cyclooxygenase-2 inhibitor |