AU2001281806A1 - Method for preparing substituted 5-amino-n-phenyl-1,2,4-triazole-3-sulfonamides - Google Patents
Method for preparing substituted 5-amino-n-phenyl-1,2,4-triazole-3-sulfonamidesInfo
- Publication number
- AU2001281806A1 AU2001281806A1 AU2001281806A AU8180601A AU2001281806A1 AU 2001281806 A1 AU2001281806 A1 AU 2001281806A1 AU 2001281806 A AU2001281806 A AU 2001281806A AU 8180601 A AU8180601 A AU 8180601A AU 2001281806 A1 AU2001281806 A1 AU 2001281806A1
- Authority
- AU
- Australia
- Prior art keywords
- triazole
- amino
- sulfonamides
- phenyl
- formula
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
- 229940124530 sulfonamide Drugs 0.000 title 1
- 125000004178 (C1-C4) alkyl group Chemical class 0.000 abstract 1
- DEJGAOOTMIMNDX-UHFFFAOYSA-N 3-amino-1h-1,2,4-triazole-5-sulfonyl chloride Chemical compound NC1=NC(S(Cl)(=O)=O)=NN1 DEJGAOOTMIMNDX-UHFFFAOYSA-N 0.000 abstract 1
- OAJFLKUHZAKFPE-UHFFFAOYSA-N 3-amino-n-phenyl-1h-1,2,4-triazole-5-sulfonamide Chemical class NC1=NNC(S(=O)(=O)NC=2C=CC=CC=2)=N1 OAJFLKUHZAKFPE-UHFFFAOYSA-N 0.000 abstract 1
- 150000001448 anilines Chemical class 0.000 abstract 1
- 125000004093 cyano group Chemical group *C#N 0.000 abstract 1
- 229910052736 halogen Inorganic materials 0.000 abstract 1
- 125000005843 halogen group Chemical group 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 1
- 239000002904 solvent Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
- C07D249/10—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D249/14—Nitrogen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Abstract
The present invention relates to a process for preparing 5-amino-N-phenyl-1,2,4-triazole-3-sulfonamides of the formula (I)whereX is halogen, cyano or nitro,R is hydrogen or optionally halogen-substituted C1-C4-alkyl, andn is 1 or 2,by reacting 5-amino-3-chlorosulfonyl-1,2,4-triazole of the formula (II)with substituted anilines of the formula (III)where X, n and R are as defined for formula (I), in the absence of a solvent.
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10029878 | 2000-06-16 | ||
| DE10029878 | 2000-06-16 | ||
| DE10038020 | 2000-08-04 | ||
| DE10038020A DE10038020A1 (en) | 2000-06-16 | 2000-08-04 | Pure 5-amino-N-phenyl-1,2,4-triazole-3-sulfonamide preparation in high yield for use as agrochemical intermediate, by reacting corresponding sulfonyl chloride and aniline compounds in the absence of solvents |
| PCT/EP2001/006386 WO2001096316A1 (en) | 2000-06-16 | 2001-06-05 | Method for preparing substituted 5-amino-n-phenyl-1,2,4-triazole-3-sulfonamides |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AU2001281806A1 true AU2001281806A1 (en) | 2001-12-24 |
Family
ID=26006116
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2001281806A Abandoned AU2001281806A1 (en) | 2000-06-16 | 2001-06-05 | Method for preparing substituted 5-amino-n-phenyl-1,2,4-triazole-3-sulfonamides |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US6680388B2 (en) |
| EP (1) | EP1296962B1 (en) |
| JP (1) | JP2004503544A (en) |
| CN (1) | CN1436177A (en) |
| AT (1) | ATE372326T1 (en) |
| AU (1) | AU2001281806A1 (en) |
| BR (1) | BR0111697A (en) |
| DE (1) | DE50112967D1 (en) |
| HU (1) | HUP0302821A2 (en) |
| IL (1) | IL153144A0 (en) |
| WO (1) | WO2001096316A1 (en) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MX2007004155A (en) * | 2004-10-08 | 2007-09-11 | Johnson & Johnson | 1,2,4-triazolylaminoaryl (heteroaryl) sulfonamide derivatives. |
| US7297810B2 (en) * | 2004-12-30 | 2007-11-20 | 3M Innovative Properties Company | High refractive index monomers for optical applications |
| US7919629B2 (en) * | 2005-12-12 | 2011-04-05 | Phostech Lithium Inc. | Sulphonyl-1,2,4-triazole salts |
| CN104059027B (en) * | 2014-07-01 | 2015-10-28 | 河北大学 | One class contains (E)-methoxyimino methyl phenylacetate compounds of 1,2,4-triazole and its production and use |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB951652A (en) | 1960-06-28 | 1964-03-11 | Wallace Broadbent | Sulphamyl triazolopyrimidines and their preparation |
| EP0330137B1 (en) | 1983-11-14 | 1994-03-02 | DowElanco | Intermediate compounds for the preparation of 1,2,4-triazolo [1,5-a]pyrimidine-2-sulfonamides |
| US4818273A (en) | 1983-11-14 | 1989-04-04 | The Dow Chemical Company | Substituted 1,2,4-triazolo[1,5-a]pyrimidine-2-sulfonamides, compositions containing them, and their utility as herbicides |
| US4886883A (en) | 1983-11-14 | 1989-12-12 | The Dow Chemical Company | Substituted 1,2,4-triazolo[1,5-a]pyrimidine-2-sulfonyl chlorides |
| US4954163A (en) | 1983-11-14 | 1990-09-04 | The Dow Chemical Company | Substituted 1,2,4-triazolo[1,5-a]pyrimidine-2-sulfonamides, compositions containing them, and their utility as herbicides |
| US4734123A (en) | 1986-05-06 | 1988-03-29 | The Dow Chemical Company | Novel sulfonamides and method of making |
| EP0246749A3 (en) * | 1986-05-17 | 1988-08-31 | AgrEvo UK Limited | Triazole herbicides |
| DE3640155A1 (en) | 1986-11-25 | 1988-05-26 | Bayer Ag | TRIAZOLO-PYRIMIDINE-2-SULPHONAMIDE |
| US5382674A (en) | 1988-12-19 | 1995-01-17 | Dowelanco | Preparation of 5-amino-1,2,4-triazole-3-sulfonamides |
| US4937350A (en) | 1989-06-05 | 1990-06-26 | The Dow Chemical Company | Preparation of N-(-3(((aryl)amino)suldonyl)-1H-1,2,4-triazol-5-yl)amines |
| US4988812A (en) | 1989-11-06 | 1991-01-29 | Dow Elanco | Aqueous process for the preparation of 5-methyl-n-(aryl)-1,2,4-triazolo(1,5-A)pyrimidine-2-sulfonamides |
-
2001
- 2001-06-05 HU HU0302821A patent/HUP0302821A2/en unknown
- 2001-06-05 WO PCT/EP2001/006386 patent/WO2001096316A1/en not_active Ceased
- 2001-06-05 EP EP01960270A patent/EP1296962B1/en not_active Expired - Lifetime
- 2001-06-05 AU AU2001281806A patent/AU2001281806A1/en not_active Abandoned
- 2001-06-05 CN CN01811145A patent/CN1436177A/en active Pending
- 2001-06-05 IL IL15314401A patent/IL153144A0/en unknown
- 2001-06-05 US US10/311,038 patent/US6680388B2/en not_active Expired - Lifetime
- 2001-06-05 DE DE50112967T patent/DE50112967D1/en not_active Expired - Lifetime
- 2001-06-05 BR BR0111697-5A patent/BR0111697A/en active Search and Examination
- 2001-06-05 JP JP2002510459A patent/JP2004503544A/en active Pending
- 2001-06-05 AT AT01960270T patent/ATE372326T1/en not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| ATE372326T1 (en) | 2007-09-15 |
| EP1296962A1 (en) | 2003-04-02 |
| US6680388B2 (en) | 2004-01-20 |
| WO2001096316A1 (en) | 2001-12-20 |
| DE50112967D1 (en) | 2007-10-18 |
| IL153144A0 (en) | 2003-06-24 |
| CN1436177A (en) | 2003-08-13 |
| JP2004503544A (en) | 2004-02-05 |
| HUP0302821A2 (en) | 2004-05-28 |
| US20030162975A1 (en) | 2003-08-28 |
| EP1296962B1 (en) | 2007-09-05 |
| BR0111697A (en) | 2003-07-08 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| PT900240E (en) | PROCESS FOR THE PRODUCTION OF POLYALCENOAMINES | |
| MY129613A (en) | Cannabinoid receptor binding compounds | |
| HRP990167B1 (en) | Sulphinic acid derivatives, method for producing them, and their use | |
| WO2002032898A3 (en) | Novel anticholinergics, method for the production thereof and use thereof as medicaments | |
| BG103778A (en) | Process for preparing pyrazole derivatives | |
| DK1255747T3 (en) | Synthesis of 3,6-dialkyl-5,6-dihydro-4-hydroxy-pyran-2-one | |
| MY132507A (en) | Process for substituted pyridines | |
| AU2001281806A1 (en) | Method for preparing substituted 5-amino-n-phenyl-1,2,4-triazole-3-sulfonamides | |
| CA2362217A1 (en) | Process for preparing phenylpyrazole pesticidal intermediates | |
| IL144288A0 (en) | Process for the preparation of organosilylalkylpolysulfanes | |
| AU2003269363A1 (en) | Azo compounds | |
| IN187760B (en) | ||
| AU2102400A (en) | Naphthalenehydrazamimides and perylenehydrazamimides | |
| MXPA02001406A (en) | Substituted heterocyclyl-2h-chromenes. | |
| AU2003302301A1 (en) | Process for preparing 4-aminodiphenylamine intermediates | |
| AU3259997A (en) | Ring-fused dihydropyranes, process for the preparation and use thereof | |
| ID27440A (en) | PROCESS FOR PREPARING | |
| IL148161A0 (en) | Process for the preparation of 2-cyanopyridines | |
| ZA983231B (en) | Substituted benzyloxyimino compounds. | |
| AU2002359985A1 (en) | Diaryl 1,2,4-triazole derivatives as a highly selective cyclooxygenase-2 inhibitor | |
| AU7206898A (en) | Method for producing 1,3-di-substituted 2-nitroguanidines | |
| ATE253553T1 (en) | METHOD FOR PRODUCING 2-ALKYLTHIOBENZONITRIL DERIVATIVES | |
| ES557083A0 (en) | A METHOD FOR PREPARING PYROLE (1,2-B) (1,2,5) TRIAZEPINES | |
| ATE192439T1 (en) | PRODUCTION OF N-(3-HALOPROPYL)IMINOSTILBENE AND ITS IMPLEMENTATION IN OPIPRAMOL | |
| PT1296983E (en) | A novel process for the preparation of pyrazolopyridinidones |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MK6 | Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase | ||
| TH | Corrigenda |
Free format text: IN VOL 16, NO 12, PAGE(S) 2688-2711 UNDER THE HEADING APPLICATIONS LAPSED, REFUSED OR WITHDRAWN PLEASE DELETE ALL REFERENCE TO APPLICATION NO. 63955/01, 70675/01, 74564/01, 81806/01 AND 85733/01 |
|
| MK4 | Application lapsed section 142(2)(d) - no continuation fee paid for the application |