[go: up one dir, main page]

AU2001272719A1 - Macrolide antibiotics - Google Patents

Macrolide antibiotics

Info

Publication number
AU2001272719A1
AU2001272719A1 AU2001272719A AU7271901A AU2001272719A1 AU 2001272719 A1 AU2001272719 A1 AU 2001272719A1 AU 2001272719 A AU2001272719 A AU 2001272719A AU 7271901 A AU7271901 A AU 7271901A AU 2001272719 A1 AU2001272719 A1 AU 2001272719A1
Authority
AU
Australia
Prior art keywords
macrolide antibiotics
macrolide
antibiotics
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2001272719A
Inventor
Yan Chen
Wei-Guo Su
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Products Inc
Original Assignee
Pfizer Products Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc filed Critical Pfizer Products Inc
Publication of AU2001272719A1 publication Critical patent/AU2001272719A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Genetics & Genomics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Molecular Biology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
AU2001272719A 2000-08-07 2001-08-06 Macrolide antibiotics Abandoned AU2001272719A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US22359100P 2000-08-07 2000-08-07
US60223591 2000-08-07
PCT/IB2001/001403 WO2002012260A1 (en) 2000-08-07 2001-08-06 Macrolide antibiotics

Publications (1)

Publication Number Publication Date
AU2001272719A1 true AU2001272719A1 (en) 2002-02-18

Family

ID=22837162

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2001272719A Abandoned AU2001272719A1 (en) 2000-08-07 2001-08-06 Macrolide antibiotics

Country Status (17)

Country Link
US (2) US20020115621A1 (en)
EP (1) EP1307468A1 (en)
JP (1) JP2004505987A (en)
AP (1) AP2001002236A0 (en)
AR (1) AR034695A1 (en)
AU (1) AU2001272719A1 (en)
BR (1) BR0112863A (en)
CA (1) CA2419044A1 (en)
DO (1) DOP2001000228A (en)
GT (1) GT200100159A (en)
HN (1) HN2001000176A (en)
MX (1) MXPA03001148A (en)
PA (1) PA8524501A1 (en)
PE (1) PE20020468A1 (en)
TN (1) TNSN01121A1 (en)
UY (1) UY26870A1 (en)
WO (1) WO2002012260A1 (en)

Families Citing this family (29)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1351608A (en) 1999-05-24 2002-05-29 辉瑞产品公司 13-Methylerythromycin Derivatives
DE60138876D1 (en) * 2000-03-28 2009-07-16 Sandoz Ag TASTE-MASKED GRANULATED PARTICLES
AU2003234650A1 (en) * 2002-05-31 2003-12-19 Janssen Pharmaceutica N.V. 3-descladinosyl-6-o-carbamoyl and 6-o-carbonoyl macrolide antibacterial agents
HRP20020885B1 (en) 2002-11-11 2007-05-31 GlaxoSmithKline istra�iva�ki centar Zagreb d.o.o. SUBSTITUTED 9a-N-{N'-[4-(SULFONYL)PHENYLCARBAMOYL]}DERIVATIVES 9-DEOXO-9-DIHYDRO-9a-AZA-9a-HOMOERITHROMYCIN A AND 5-O-DESOZAMINYL-9-DEOXO-9-DIHYDRO-9a-AZA-9a-HOMOERITHRONOLIDE A
WO2004080391A2 (en) 2003-03-10 2004-09-23 Optimer Pharmaceuticals, Inc. Novel antibacterial agents
GB0310981D0 (en) * 2003-05-13 2003-06-18 Glaxo Group Ltd Novel compounds
HRP20030381B1 (en) * 2003-05-14 2007-05-31 GlaxoSmithKline istra�iva�ki centar Zagreb d.o.o. 3-DECLADINOZYL 9a-N-CARBAMOYL AND 9a-N-THIOCARBAMOYL DERIVATIVES 9-DEOXO-9-DIHYDRO-9a-AZA-9a-HOMOERYTHROMICYNE A
WO2005030227A1 (en) 2003-09-23 2005-04-07 Enanta Pharmaceuticals, Inc. 9a, 11-3C-BICYCLIC 9a-AZALIDE DERIVATIVES
US7468428B2 (en) * 2004-03-17 2008-12-23 App Pharmaceuticals, Llc Lyophilized azithromycin formulation
US20060116336A1 (en) * 2004-03-17 2006-06-01 American Pharmaceutical Partners, Inc. Lyophilized azithromycin formulation
US20080287376A1 (en) * 2004-07-28 2008-11-20 Mohammad Salman Ketolide Derivatives as Antibacterial Agents
US7402568B2 (en) 2004-09-29 2008-07-22 Enanta Pharmaceuticals, Inc. Bicyclic 9a-azalide derivatives
EP1807439A2 (en) * 2004-10-25 2007-07-18 Ranbaxy Laboratories Limited Ketolide derivatives as antibacterial agents
HRP20100253T1 (en) 2004-12-21 2010-06-30 Pfizer Products Inc. macrolides
US7271155B2 (en) 2005-01-07 2007-09-18 Enanta Pharmaceuticals, Inc. 9A, 11-2C-bicyclic 9a-azalide derivatives
ATE419261T1 (en) * 2005-01-13 2009-01-15 Glaxosmithkline Zagreb DECLADINOSYL MACROLIDE WITH ANTI-INFLAMMATORY EFFECT
EP1957508A2 (en) * 2005-11-23 2008-08-20 Ranbaxy Laboratories Limited Ketolide derivatives as antibacterial agents
WO2007060618A2 (en) * 2005-11-23 2007-05-31 Ranbaxy Laboratories Limited Macrolides derivatives as antibacterial agents
EP2023721A2 (en) * 2006-06-05 2009-02-18 Auspex Pharmaceuticals Inc. Preparation and utility of substituted erythromycin analogs
US9453042B2 (en) * 2007-10-25 2016-09-27 Cempra Pharmaceuticals, Inc. Process for the preparation of macrolide antibacterial agents
CN102245195B (en) * 2008-10-24 2016-01-13 森普拉制药公司 Biodefense using triazole-containing macrolides
US9937194B1 (en) 2009-06-12 2018-04-10 Cempra Pharmaceuticals, Inc. Compounds and methods for treating inflammatory diseases
CN102724874B (en) 2009-09-10 2018-06-01 森普拉制药公司 Methods of treating malaria, tuberculosis and MAC disease
PL2550286T3 (en) 2010-03-22 2016-07-29 Cempra Pharmaceuticals Inc Crystalline forms of a macrolide, and uses therefor
CA2799937A1 (en) 2010-05-20 2011-11-24 Cempra Pharmaceuticals, Inc. Processes for preparing macrolides and ketolides and intermediates therefor
JP6042334B2 (en) 2010-09-10 2016-12-14 センプラ ファーマシューティカルズ，インコーポレイテッド Hydrogen bond forming fluoroketolides for disease treatment
SG11201405895UA (en) 2012-03-27 2014-10-30 Cempra Pharmaceuticals Inc Parenteral formulations for administering macrolide antibiotics
RU2015138796A (en) 2013-03-14 2017-04-19 Семпра Фармасьютикалс, Инк. METHODS AND COMPOSITIONS FOR TREATMENT OF RESPIRATORY DISEASES
HK1218864A1 (en) 2013-03-15 2017-03-17 森普拉制药公司 Convergent processes for preparing macrolide antibacterial agents

Family Cites Families (30)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US25937A (en) 1859-11-01 ballou
US100518A (en) 1870-03-08 Roland s
US61857A (en) 1867-02-05 Improvement in top-drivers or spinners
US61856A (en) 1867-02-05 Enos s
US156027A (en) 1874-10-20 Improvement in loom-shuttles
US40007A (en) 1863-09-22 Improvement in railroad-car brakes
US3923784A (en) * 1973-09-10 1975-12-02 Hoffmann La Roche Erythromycin a derivatives
SI8110592A8 (en) * 1981-03-06 1996-06-30 Pliva Pharm & Chem Works Process for preparing of n-methyl-11-aza-10-deoxo-10-dihydroerythromycine a and derivatives thereof
US4474768A (en) * 1982-07-19 1984-10-02 Pfizer Inc. N-Methyl 11-aza-10-deoxo-10-dihydro-erytromycin A, intermediates therefor
US5141926A (en) * 1990-04-18 1992-08-25 Abbott Laboratories Erythromycin derivatives
US5523399A (en) 1991-12-27 1996-06-04 Taisho Pharmaceutical Co., Ltd. 5-O-desosaminylerythronolide derivatives
FR2745290B1 (en) * 1996-02-28 1998-04-03 Roussel Uclaf NOVEL ERYTHROMYCIN DERIVATIVES, THEIR PREPARATION PROCESS AND THEIR APPLICATION AS MEDICAMENTS
FR2748746B1 (en) * 1996-05-14 1998-08-14 Hoechst Marion Roussel Inc NEW PROCESS FOR ISOMERIZATION OF RADICAL METHYL IN 10 FROM ERYTHROMYCIN DERIVATIVES
US5804565A (en) * 1996-09-24 1998-09-08 Taisho Pharmaceutical Co., Ltd. Erythromycin A derivatives
WO1998023628A1 (en) * 1996-11-27 1998-06-04 Taisho Pharmaceutical Co., Ltd. Erythromycin a derivatives
US6162794A (en) * 1997-05-09 2000-12-19 Pfizer Inc. Erythromycin derivatives
EP0895999A1 (en) * 1997-08-06 1999-02-10 Pfizer Products Inc. C-4" substituted macrolide antibiotics
ZA987689B (en) * 1997-09-02 1999-02-24 Abbott Lab 3-descladinose 6-O substituted erythromycin derivatives
PA8461401A1 (en) * 1997-10-29 2000-05-24 Pfizer Prod Inc TRICYCLIC ERYTHROMYCINE DERIVATIVES
AU9649698A (en) 1997-10-29 1999-05-17 Taisho Pharmaceutical Co., Ltd. Erythromycin a 11, 12-carbamate derivatives
AU9649598A (en) 1997-10-29 1999-05-17 Taisho Pharmaceutical Co., Ltd. Erythromycin a, 11,12-carbamate derivatives
HN1998000159A (en) * 1997-10-29 1999-02-09 Monsanto Co DERIVATIVES OF 9- AMINO - 3 CETO ERITROMICINA
AU1504899A (en) * 1997-12-11 1999-06-28 Hokuriku Seiyaku Co. Ltd Erythromycin derivatives
AP1060A (en) 1998-01-02 2002-04-23 Pfizer Prod Inc Novel erythromycin derivatives.
US6248719B1 (en) * 1998-06-03 2001-06-19 Pfizer Inc Tricyclic 3-keto derivatives of 6-O-methylerthromycin
ID30233A (en) 1999-01-27 2001-11-15 Pfizer Prod Inc ANTIBIOTICS OF TETOLIDA
WO2001010880A1 (en) 1999-08-06 2001-02-15 Taisho Pharmaceutical Co., Ltd. Erythromycin a derivatives
WO2001010878A1 (en) 1999-08-06 2001-02-15 Taisho Pharmaceutical Co., Ltd. Erythromycin a derivatives
US6498146B1 (en) * 1999-10-28 2002-12-24 Pfizer Inc Erythromycin derivatives
EP1101769A3 (en) * 1999-11-18 2001-10-24 Pfizer Products Inc. Nitrogen containing erythromycin derivatives

Also Published As

Publication number Publication date
GT200100159A (en) 2002-03-22
AP2001002236A0 (en) 2001-09-30
DOP2001000228A (en) 2002-09-30
EP1307468A1 (en) 2003-05-07
TNSN01121A1 (en) 2005-11-10
US20020115621A1 (en) 2002-08-22
US6849608B2 (en) 2005-02-01
HN2001000176A (en) 2001-10-08
UY26870A1 (en) 2002-03-22
BR0112863A (en) 2003-07-01
US20040009930A1 (en) 2004-01-15
WO2002012260A1 (en) 2002-02-14
PE20020468A1 (en) 2002-06-14
AR034695A1 (en) 2004-03-17
JP2004505987A (en) 2004-02-26
CA2419044A1 (en) 2002-02-14
MXPA03001148A (en) 2003-06-09
PA8524501A1 (en) 2002-08-29

Similar Documents

Publication Publication Date Title
EP1363925B8 (en) Macrolide antibiotics
AU2002217277A1 (en) Macrolide antibiotics
AU2001272719A1 (en) Macrolide antibiotics
AU2001284934A1 (en) Steroid derived antibiotics
IL144178A0 (en) Ketolide antibiotics
AU2001228708A1 (en) Coin-validation arrangement
AU2001254546A1 (en) Aminopiperidines
AU2001220246A1 (en) Neckphone
IL142628A0 (en) Novel macrolide antibiotics
AU2001258349A1 (en) Bisacylguanidine
AU4657001A (en) Displacing arrangement
AU2001278694A1 (en) Avermectin derivatives
AU2002221895A1 (en) Macrolide solvates
AU2001257490A1 (en) Improved beta-lactam antibiotics
AU2001253911A1 (en) Bifunctional antibiotics
AU2001258924A1 (en) Microsatellite-aflp
AU2002230386A1 (en) Sixteen-membered macrolide compounds
AU2002359761A1 (en) Antibiotic compounds
AU2001246864A1 (en) Hypotensors
AU2001226668A1 (en) Crankshaft-starter-generator
AU2001238020A1 (en) Glycopeptide derivatives having antibiotic activity
EP1201403A3 (en) Electrofusible units
AU2002246567A1 (en) Aminoglycosides as antibiotics
AU2001260192A1 (en) Glycinamides
HK1062443A (en) Macrolide antibiotics