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AU2001268589A1 - Cross linked solid supports for solid phase synthesis - Google Patents

Cross linked solid supports for solid phase synthesis

Info

Publication number
AU2001268589A1
AU2001268589A1 AU2001268589A AU6858901A AU2001268589A1 AU 2001268589 A1 AU2001268589 A1 AU 2001268589A1 AU 2001268589 A AU2001268589 A AU 2001268589A AU 6858901 A AU6858901 A AU 6858901A AU 2001268589 A1 AU2001268589 A1 AU 2001268589A1
Authority
AU
Australia
Prior art keywords
phase synthesis
cross linked
solid
solid phase
supports
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2001268589A
Inventor
H. Mario Geysen
Patrick F. Kiser
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Glaxo Group Ltd
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of AU2001268589A1 publication Critical patent/AU2001268589A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C40—COMBINATORIAL TECHNOLOGY
    • C40B—COMBINATORIAL CHEMISTRY; LIBRARIES, e.g. CHEMICAL LIBRARIES
    • C40B50/00—Methods of creating libraries, e.g. combinatorial synthesis
    • C40B50/14—Solid phase synthesis, i.e. wherein one or more library building blocks are bound to a solid support during library creation; Particular methods of cleavage from the solid support
    • B—PERFORMING OPERATIONS; TRANSPORTING
    • B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
    • B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
    • B01J2219/00—Chemical, physical or physico-chemical processes in general; Their relevant apparatus
    • B01J2219/00274—Sequential or parallel reactions; Apparatus and devices for combinatorial chemistry or for making arrays; Chemical library technology
    • B01J2219/00277—Apparatus
    • B01J2219/00452—Means for the recovery of reactants or products
    • B01J2219/00454—Means for the recovery of reactants or products by chemical cleavage from the solid support
    • B—PERFORMING OPERATIONS; TRANSPORTING
    • B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
    • B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
    • B01J2219/00—Chemical, physical or physico-chemical processes in general; Their relevant apparatus
    • B01J2219/00274—Sequential or parallel reactions; Apparatus and devices for combinatorial chemistry or for making arrays; Chemical library technology
    • B01J2219/00277—Apparatus
    • B01J2219/00497—Features relating to the solid phase supports
    • B—PERFORMING OPERATIONS; TRANSPORTING
    • B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
    • B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
    • B01J2219/00—Chemical, physical or physico-chemical processes in general; Their relevant apparatus
    • B01J2219/00274—Sequential or parallel reactions; Apparatus and devices for combinatorial chemistry or for making arrays; Chemical library technology
    • B01J2219/00583—Features relative to the processes being carried out
    • B01J2219/00596—Solid-phase processes
    • B—PERFORMING OPERATIONS; TRANSPORTING
    • B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
    • B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
    • B01J2219/00—Chemical, physical or physico-chemical processes in general; Their relevant apparatus
    • B01J2219/00274—Sequential or parallel reactions; Apparatus and devices for combinatorial chemistry or for making arrays; Chemical library technology
    • B01J2219/00718—Type of compounds synthesised
    • B01J2219/0072—Organic compounds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/11—Compounds covalently bound to a solid support

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Structural Engineering (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Physical Or Chemical Processes And Apparatus (AREA)
AU2001268589A 2000-06-21 2001-06-19 Cross linked solid supports for solid phase synthesis Abandoned AU2001268589A1 (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US09/598,217 US6582726B1 (en) 2000-06-21 2000-06-21 Cross linked solid supports for solid phase synthesis
US09598217 2000-06-21
US09/598,217 2000-06-21
PCT/US2001/019633 WO2001097964A2 (en) 2000-06-21 2001-06-19 Cross linked solid supports for solid phase synthesis

Publications (1)

Publication Number Publication Date
AU2001268589A1 true AU2001268589A1 (en) 2002-01-02

Family

ID=24394691

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2001268589A Abandoned AU2001268589A1 (en) 2000-06-21 2001-06-19 Cross linked solid supports for solid phase synthesis

Country Status (5)

Country Link
US (1) US6582726B1 (en)
EP (1) EP1292553A2 (en)
JP (1) JP2003535685A (en)
AU (1) AU2001268589A1 (en)
WO (1) WO2001097964A2 (en)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6584411B1 (en) 2000-07-26 2003-06-24 Smithkline Beecham Corporation Methods to facilitate the calculation of yields of reaction products
US20040235053A1 (en) * 2003-03-28 2004-11-25 The Regents Of The University Of California Preparation and application of encoded bead aggregates in combinatorial chemistry
US20050095648A1 (en) * 2003-10-30 2005-05-05 Mario Geysen Method for designing linear epitopes and algorithm therefor and polypeptide epitopes
ES2986867T3 (en) 2005-03-03 2024-11-12 Mirus Llc Enhanced metal alloys for medical devices
US9107899B2 (en) 2005-03-03 2015-08-18 Icon Medical Corporation Metal alloys for medical devices
US8131339B2 (en) * 2007-11-27 2012-03-06 Vivant Medical, Inc. System and method for field ablation prediction
US8398916B2 (en) 2010-03-04 2013-03-19 Icon Medical Corp. Method for forming a tubular medical device
EP3160397A4 (en) 2014-06-24 2018-03-21 Icon Medical Corp. Improved metal alloys for medical devices
EP4512394A3 (en) 2015-06-03 2025-10-22 Triastek, Inc. Dosage forms and use thereof
US11766506B2 (en) 2016-03-04 2023-09-26 Mirus Llc Stent device for spinal fusion
CN121129781A (en) 2017-01-26 2025-12-16 南京三迭纪医药科技有限公司 Dosage form for controlled release at specific gastrointestinal sites
CN116270513A (en) 2018-01-09 2023-06-23 南京三迭纪医药科技有限公司 A combination oral pharmaceutical dosage form comprising a fixed-dose ADHD non-stimulant and an ADHD stimulant

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1989005305A1 (en) 1987-12-09 1989-06-15 3I Research Exploitation Limited Polymers and polymer-peptide conjugates
WO1997026002A1 (en) * 1996-01-17 1997-07-24 California Institute Of Technology Synthesis of conformationally restricted amino acids, peptides and peptidomimetics by catalytic ring closing metathesis
EP0863858B1 (en) 1996-04-08 2004-02-04 Glaxo Group Limited Mass-based encoding and qualitative analysis of combinatorial libraries
US5916585A (en) 1996-06-03 1999-06-29 Gore Enterprise Holdings, Inc. Materials and method for the immobilization of bioactive species onto biodegradable polymers
DE19626762A1 (en) 1996-07-03 1998-01-08 Basf Ag Enzymatically cleavable linker for solid phase synthesis

Also Published As

Publication number Publication date
WO2001097964A2 (en) 2001-12-27
EP1292553A2 (en) 2003-03-19
WO2001097964A3 (en) 2002-07-18
US6582726B1 (en) 2003-06-24
JP2003535685A (en) 2003-12-02

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