AU2001264044A1 - 1,4-diazabicyclo(3.2.2)nonabenzoxazole, -benzothiazole and benzimidazole derivatives, preparation and therapeutic use thereof - Google Patents

1,4-diazabicyclo(3.2.2)nonabenzoxazole, -benzothiazole and benzimidazole derivatives, preparation and therapeutic use thereof

Info

Publication number: AU2001264044A1
Authority: AU; Australia
Prior art keywords: nonabenzoxazole; benzothiazole; diazabicyclo; preparation; therapeutic use
Prior art date: 2000-05-31
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Abandoned

Application number

AU2001264044A

Inventor

Frederic Galli

Alistair Lochead

Axelle Samson

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Sanofi Aventis France

Original Assignee

Sanofi Synthelabo SA

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-05-31

Filing date

2001-05-29

Publication date

2001-12-11

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=8850826&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AU2001264044(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2001-05-29 Application filed by Sanofi Synthelabo SA filed Critical Sanofi Synthelabo SA

2001-12-11 Publication of AU2001264044A1 publication Critical patent/AU2001264044A1/en

Status Abandoned legal-status Critical Current

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/08—Bridged systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/32—Alcohol-abuse
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/34—Tobacco-abuse
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Veterinary Medicine (AREA)
Pharmacology & Pharmacy (AREA)
Public Health (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
Biomedical Technology (AREA)
Neurosurgery (AREA)
Neurology (AREA)
Psychiatry (AREA)
Addiction (AREA)
Pain & Pain Management (AREA)
Cardiology (AREA)
Psychology (AREA)
Heart & Thoracic Surgery (AREA)
Vascular Medicine (AREA)
Urology & Nephrology (AREA)
Hospice & Palliative Care (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

AU2001264044A 2000-05-31 2001-05-29 1,4-diazabicyclo(3.2.2)nonabenzoxazole, -benzothiazole and benzimidazole derivatives, preparation and therapeutic use thereof Abandoned AU2001264044A1 (en)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
FR0006975		2000-05-31
FR0006975A FR2809730B1 (en)	2000-05-31	2000-05-31	1,4-DIAZABICYCLO [3.2.2] NONANEBENZOXAZOLE, -BENZOTHIAZOLE AND -BENZIMIDAZOLE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION
PCT/FR2001/001651 WO2001092261A1 (en)	2000-05-31	2001-05-29	1,4-diazabicyclo[3.2.2]nonabenzoxazole, -benzothiazole and benzimidazole derivatives, preparation and therapeutic use thereof

Publications (1)

Publication Number	Publication Date
AU2001264044A1 true AU2001264044A1 (en)	2001-12-11

Family

ID=8850826

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AU2001264044A Abandoned AU2001264044A1 (en)	2000-05-31	2001-05-29	1,4-diazabicyclo(3.2.2)nonabenzoxazole, -benzothiazole and benzimidazole derivatives, preparation and therapeutic use thereof

Country Status (11)

Country	Link
US (1)	US7220740B2 (en)
EP (1)	EP1289988B1 (en)
JP (1)	JP4939721B2 (en)
AR (1)	AR028647A1 (en)
AT (1)	ATE267202T1 (en)
AU (1)	AU2001264044A1 (en)
DE (1)	DE60103395T2 (en)
FR (1)	FR2809730B1 (en)
HU (1)	HU229102B1 (en)
TW (1)	TW541307B (en)
WO (1)	WO2001092261A1 (en)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
SE0000540D0 (en)	2000-02-18	2000-02-18	Astrazeneca Ab	New compounds
US20020086871A1 (en) *	2000-12-29	2002-07-04	O'neill Brian Thomas	Pharmaceutical composition for the treatment of CNS and other disorders
DE60215172T2 (en) *	2001-07-06	2007-08-30	Neurosearch A/S	NEW COMPOUNDS, THEIR PREPARATION AND USE
FR2832714B1 (en)	2001-11-23	2004-07-16	Sanofi Synthelabo	DERIVATIVES OF 4- (OXAZOLOPYRIDIN-2-YL) -1,4-DIAZABICYCLO [3.2.2] NONANE, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION
SE0202465D0 (en) *	2002-08-14	2002-08-14	Astrazeneca Ab	New compounds
US7456171B2 (en)	2002-10-08	2008-11-25	Sanofi-Aventis	1,4-Diazabicyclo[3.2.2]nonanecarboxamide derivatives, preparation and therapeutic use thereof
FR2845388B1 (en) *	2002-10-08	2004-11-12	Sanofi Synthelabo	1,4-DIAZABICYCLO [3.2.2] NONANECARBOXAMIDES DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION
US7223753B2 (en)	2002-11-11	2007-05-29	Neurosearch A/S	Diazabicyclic biaryl derivatives
AU2003280309A1 (en) *	2002-11-11	2004-06-03	Neurosearch A/S	1,4-diazabicyclo (3,2,2)nonane derivatives, preparation and therapeutical use thereof
NZ540998A (en) *	2003-02-27	2008-06-30	Neurosearch As	Novel diazabicyclic aryl derivatives
FR2865208B1 (en) *	2004-01-16	2009-01-16	Sanofi Synthelabo	1,4-DIAZABICYCLO [3.2.1] OCTANECARBOXMIQUE DERIVATIVES, THEIR PREPARATION AND THERAPEUTIC USE THEREOF
DE602005018020D1 (en)	2004-02-04	2010-01-14	Neurosearch As	DIAZABICYCLIC ARYL DERIVATIVES AS CHOLINERGE RECEPTOR MODULATORS
JP2008519820A (en) *	2004-11-15	2008-06-12	ファイザー・プロダクツ・インク	Azabenzoxazole for the treatment of CNS disorders
WO2006051410A1 (en) *	2004-11-15	2006-05-18	Pfizer Inc.	Azabenzoxazoles for the treatment of cns disorders
WO2006051413A1 (en) *	2004-11-15	2006-05-18	Pfizer Inc.	Azabenoxazoles for the treatment of cns disorders
US7662812B2 (en)	2005-02-16	2010-02-16	Neurosearch A/S	Diazabicyclic aryl derivatives and their use as chinolinergic ligands at nicotinic acetylcholine receptors
EP2029607A1 (en)	2006-05-23	2009-03-04	NeuroSearch A/S	Novel 8,10-diaza-bicycloý4.3.1¨decane derivatives and their medical use
CN104262348B (en) *	2014-08-15	2017-12-15	北京师范大学	A kind of alpha 7 nicotinic acetylcholine receptors part and preparation method thereof
CN107188900B (en) *	2017-05-27	2019-09-06	北京师范大学	Ligand compound of α7 nicotinic acetylcholine receptor and its application

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
IN166416B (en) *	1985-09-18	1990-05-05	Pfizer
NZ226000A (en) *	1987-09-10	1991-06-25	Merck Sharp & Dohme	Oxadiazolyl-azabicycloheptanes and pharmaceutical compositions
US5478939A (en) *	1994-07-20	1995-12-26	American Cyanamid Company	(R,R) and (S,S) 2,5-diazabicyclo [2,2,1]heptane derivatives
FR2786770B1 (en)	1998-12-04	2001-01-19	Synthelabo	NONANE 1,4-DIAZABICYCLO [3.2.2.] DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION
US20020086871A1 (en) *	2000-12-29	2002-07-04	O'neill Brian Thomas	Pharmaceutical composition for the treatment of CNS and other disorders

2000
- 2000-05-31 FR FR0006975A patent/FR2809730B1/en not_active Expired - Fee Related
2001
- 2001-05-29 EP EP01938363A patent/EP1289988B1/en not_active Expired - Lifetime
- 2001-05-29 JP JP2002500874A patent/JP4939721B2/en not_active Expired - Fee Related
- 2001-05-29 HU HU0302193A patent/HU229102B1/en not_active IP Right Cessation
- 2001-05-29 AT AT01938363T patent/ATE267202T1/en not_active IP Right Cessation
- 2001-05-29 WO PCT/FR2001/001651 patent/WO2001092261A1/en not_active Ceased
- 2001-05-29 AU AU2001264044A patent/AU2001264044A1/en not_active Abandoned
- 2001-05-29 DE DE60103395T patent/DE60103395T2/en not_active Expired - Lifetime
- 2001-05-29 US US10/276,646 patent/US7220740B2/en not_active Expired - Lifetime
- 2001-05-30 AR ARP010102574A patent/AR028647A1/en active IP Right Grant
- 2001-05-30 TW TW090113060A patent/TW541307B/en not_active IP Right Cessation

Also Published As

Publication number	Publication date
JP2003535091A (en)	2003-11-25
AR028647A1 (en)	2003-05-21
HUP0302193A2 (en)	2003-11-28
EP1289988B1 (en)	2004-05-19
TW541307B (en)	2003-07-11
ATE267202T1 (en)	2004-06-15
FR2809730A1 (en)	2001-12-07
US7220740B2 (en)	2007-05-22
HU229102B1 (en)	2013-07-29
FR2809730B1 (en)	2002-07-19
EP1289988A1 (en)	2003-03-12
US20030153574A1 (en)	2003-08-14
WO2001092261A1 (en)	2001-12-06
HUP0302193A3 (en)	2012-02-28
DE60103395D1 (en)	2004-06-24
DE60103395T2 (en)	2005-06-16
JP4939721B2 (en)	2012-05-30

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