AU1638095A - Boronic peptide derivatives, preparation and therapeutic application thereof - Google Patents

Boronic peptide derivatives, preparation and therapeutic application thereof

Info

Publication number: AU1638095A
Authority: AU; Australia
Prior art keywords: boronic; preparation; therapeutic application; peptide derivatives; peptide
Prior art date: 1994-04-12
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Abandoned

Application number

AU16380/95A

Inventor

Gilbert Lassalle

Sergio Mallart

Jean Claude Muller

Thomas Andrew Purcell

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Synthelabo SA

Original Assignee

Synthelabo SA

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1994-04-12

Filing date

1995-04-11

Publication date

1995-10-19

1995-04-11 Application filed by Synthelabo SA filed Critical Synthelabo SA

1995-10-19 Publication of AU1638095A publication Critical patent/AU1638095A/en

Status Abandoned legal-status Critical Current

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06191—Dipeptides containing heteroatoms different from O, S, or N
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Organic Chemistry (AREA)
Medicinal Chemistry (AREA)
General Health & Medical Sciences (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Biochemistry (AREA)
Engineering & Computer Science (AREA)
Molecular Biology (AREA)
Genetics & Genomics (AREA)
Pharmacology & Pharmacy (AREA)
Biophysics (AREA)
Animal Behavior & Ethology (AREA)
Bioinformatics & Cheminformatics (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Diabetes (AREA)
General Chemical & Material Sciences (AREA)
Hematology (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Immunology (AREA)
Epidemiology (AREA)
Peptides Or Proteins (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

AU16380/95A 1994-04-12 1995-04-11 Boronic peptide derivatives, preparation and therapeutic application thereof Abandoned AU1638095A (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
FR9404288A FR2718451B1 (en)	1994-04-12	1994-04-12	Boronic peptide derivatives, their preparation and their therapeutic use.
FR9404288		1994-04-12

Publications (1)

Publication Number	Publication Date
AU1638095A true AU1638095A (en)	1995-10-19

Family

ID=9461981

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AU16380/95A Abandoned AU1638095A (en)	1994-04-12	1995-04-11	Boronic peptide derivatives, preparation and therapeutic application thereof

Country Status (17)

Country	Link
EP (1)	EP0677531A1 (en)
JP (1)	JPH07285990A (en)
KR (1)	KR950032225A (en)
CN (1)	CN1113493A (en)
AU (1)	AU1638095A (en)
CA (1)	CA2146833A1 (en)
CZ (1)	CZ92295A3 (en)
FI (1)	FI951726L (en)
FR (1)	FR2718451B1 (en)
HU (1)	HUT71617A (en)
IL (1)	IL113332A0 (en)
NO (1)	NO951418L (en)
NZ (1)	NZ270913A (en)
PL (1)	PL308074A1 (en)
RU (1)	RU95105419A (en)
SK (1)	SK47695A3 (en)
ZA (1)	ZA952983B (en)

Cited By (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5578574A (en) *	1994-03-04	1996-11-26	Eli Lilly And Company	Antithrombotic agents
US5599793A (en) *	1994-03-04	1997-02-04	Eli Lilly And Company	Antithromobotic agents
US5602101A (en) *	1994-03-04	1997-02-11	Eli Lilly And Company	Antithrombotic agents
US5705487A (en) *	1994-03-04	1998-01-06	Eli Lilly And Company	Antithrombotic agents
US5707966A (en) *	1994-03-04	1998-01-13	Eli Lilly And Company	Antithrombotic agents
US5710130A (en) *	1995-02-27	1998-01-20	Eli Lilly And Company	Antithrombotic agents
US5726159A (en) *	1994-03-04	1998-03-10	Eli Lilly And Company	Antithrombotic agents
US5811402A (en) *	1996-03-22	1998-09-22	Eli Lilly And Company	Antithrombotic diamides
US5885967A (en) *	1994-03-04	1999-03-23	Eli Lilly And Company	Antithrombotic agents
US5914319A (en) *	1995-02-27	1999-06-22	Eli Lilly And Company	Antithrombotic agents

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5639739A (en) *	1995-03-24	1997-06-17	The Dupont Merck Pharmaceutical Company	Imidazole containing aminoboronic acids
FR2739858B1 (en) *	1995-10-11	1997-11-14	Synthelabo	N-SULFONYL- AND N-SULFAMOYLPEPTIDYLPROLINAMIDE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION
FR2758329B1 (en) *	1997-01-16	1999-02-12	Synthelabo	BORONIC IMIDAZOLE-4-BUTANE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC USE

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4499082A (en) *	1983-12-05	1985-02-12	E. I. Du Pont De Nemours And Company	α-Aminoboronic acid peptides
US5187157A (en) *	1987-06-05	1993-02-16	Du Pont Merck Pharmaceutical Company	Peptide boronic acid inhibitors of trypsin-like proteases
EP0315574A3 (en) *	1987-11-05	1990-08-22	Hoechst Aktiengesellschaft	Renin inhibitors

1994
- 1994-04-12 FR FR9404288A patent/FR2718451B1/en not_active Expired - Lifetime
1995
- 1995-04-07 EP EP95400776A patent/EP0677531A1/en not_active Withdrawn
- 1995-04-11 NO NO951418A patent/NO951418L/en unknown
- 1995-04-11 CA CA002146833A patent/CA2146833A1/en not_active Abandoned
- 1995-04-11 NZ NZ270913A patent/NZ270913A/en unknown
- 1995-04-11 HU HU9501041A patent/HUT71617A/en unknown
- 1995-04-11 FI FI951726A patent/FI951726L/en unknown
- 1995-04-11 IL IL11333295A patent/IL113332A0/en unknown
- 1995-04-11 CN CN95103889A patent/CN1113493A/en active Pending
- 1995-04-11 PL PL95308074A patent/PL308074A1/en unknown
- 1995-04-11 CZ CZ95922A patent/CZ92295A3/en unknown
- 1995-04-11 RU RU95105419/04A patent/RU95105419A/en unknown
- 1995-04-11 SK SK476-95A patent/SK47695A3/en unknown
- 1995-04-11 ZA ZA952983A patent/ZA952983B/en unknown
- 1995-04-11 AU AU16380/95A patent/AU1638095A/en not_active Abandoned
- 1995-04-11 JP JP7085270A patent/JPH07285990A/en active Pending
- 1995-04-11 KR KR1019950008356A patent/KR950032225A/en not_active Withdrawn

Cited By (12)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5578574A (en) *	1994-03-04	1996-11-26	Eli Lilly And Company	Antithrombotic agents
US5599793A (en) *	1994-03-04	1997-02-04	Eli Lilly And Company	Antithromobotic agents
US5602101A (en) *	1994-03-04	1997-02-11	Eli Lilly And Company	Antithrombotic agents
US5705487A (en) *	1994-03-04	1998-01-06	Eli Lilly And Company	Antithrombotic agents
US5707966A (en) *	1994-03-04	1998-01-13	Eli Lilly And Company	Antithrombotic agents
US5726159A (en) *	1994-03-04	1998-03-10	Eli Lilly And Company	Antithrombotic agents
US5885967A (en) *	1994-03-04	1999-03-23	Eli Lilly And Company	Antithrombotic agents
US6090787A (en) *	1994-03-04	2000-07-18	Eli Lilly And Company	Antithrombotic agents
US6124277A (en) *	1994-03-04	2000-09-26	Eli Lilly And Company	Antithrombotic agents
US5710130A (en) *	1995-02-27	1998-01-20	Eli Lilly And Company	Antithrombotic agents
US5914319A (en) *	1995-02-27	1999-06-22	Eli Lilly And Company	Antithrombotic agents
US5811402A (en) *	1996-03-22	1998-09-22	Eli Lilly And Company	Antithrombotic diamides

Also Published As

Publication number	Publication date
JPH07285990A (en)	1995-10-31
NO951418D0 (en)	1995-04-11
HUT71617A (en)	1996-01-29
FR2718451A1 (en)	1995-10-13
HU9501041D0 (en)	1995-06-28
NO951418L (en)	1995-10-13
EP0677531A1 (en)	1995-10-18
RU95105419A (en)	1997-01-10
KR950032225A (en)	1995-12-20
FR2718451B1 (en)	1996-05-10
IL113332A0 (en)	1995-07-31
CZ92295A3 (en)	1995-11-15
ZA952983B (en)	1996-01-11
FI951726A7 (en)	1995-10-13
SK47695A3 (en)	1995-12-06
CN1113493A (en)	1995-12-20
PL308074A1 (en)	1995-10-16
FI951726A0 (en)	1995-04-11
NZ270913A (en)	1996-05-28
FI951726L (en)	1995-10-13
CA2146833A1 (en)	1995-10-13

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