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AU1027188A - Sweetening agents derived from guanidinoacetic and ethanamidinoacetic acids, process for sweetening various products, and compositions containing such sweetening agents - Google Patents

Sweetening agents derived from guanidinoacetic and ethanamidinoacetic acids, process for sweetening various products, and compositions containing such sweetening agents

Info

Publication number
AU1027188A
AU1027188A AU10271/88A AU1027188A AU1027188A AU 1027188 A AU1027188 A AU 1027188A AU 10271/88 A AU10271/88 A AU 10271/88A AU 1027188 A AU1027188 A AU 1027188A AU 1027188 A AU1027188 A AU 1027188A
Authority
AU
Australia
Prior art keywords
sweetening
sweetening agents
ethanamidinoacetic
guanidinoacetic
acids
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
AU10271/88A
Other versions
AU605228B2 (en
Inventor
Claude Nofre
Farroudja Ouar
Jean-Marie Tinti
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Universite Claude Bernard Lyon 1
Original Assignee
Universite Claude Bernard Lyon 1
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Universite Claude Bernard Lyon 1 filed Critical Universite Claude Bernard Lyon 1
Publication of AU1027188A publication Critical patent/AU1027188A/en
Application granted granted Critical
Publication of AU605228B2 publication Critical patent/AU605228B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A23—FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23G—COCOA; COCOA PRODUCTS, e.g. CHOCOLATE; SUBSTITUTES FOR COCOA OR COCOA PRODUCTS; CONFECTIONERY; CHEWING GUM; ICE-CREAM; PREPARATION THEREOF
    • A23G3/00—Sweetmeats; Confectionery; Marzipan; Coated or filled products
    • A23G3/34—Sweetmeats, confectionery or marzipan; Processes for the preparation thereof
    • A23G3/36—Sweetmeats, confectionery or marzipan; Processes for the preparation thereof characterised by the composition containing organic or inorganic compounds
    • A23G3/42—Sweetmeats, confectionery or marzipan; Processes for the preparation thereof characterised by the composition containing organic or inorganic compounds characterised by the carbohydrates used, e.g. polysaccharides
    • A—HUMAN NECESSITIES
    • A23—FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23L—FOODS, FOODSTUFFS OR NON-ALCOHOLIC BEVERAGES, NOT OTHERWISE PROVIDED FOR; PREPARATION OR TREATMENT THEREOF
    • A23L27/00—Spices; Flavouring agents or condiments; Artificial sweetening agents; Table salts; Dietetic salt substitutes; Preparation or treatment thereof
    • A23L27/30—Artificial sweetening agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/40—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing nitrogen
    • A61K8/44—Aminocarboxylic acids or derivatives thereof, e.g. aminocarboxylic acids containing sulfur; Salts; Esters or N-acylated derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q11/00—Preparations for care of the teeth, of the oral cavity or of dentures; Dentifrices, e.g. toothpastes; Mouth rinses
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C279/00—Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups
    • C07C279/18—Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of guanidine groups bound to carbon atoms of six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/75—Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56—Benzopyrazoles; Hydrogenated benzopyrazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
    • C07D317/44—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D317/46—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D317/48—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring
    • C07D317/62—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to atoms of the carbocyclic ring
    • C07D317/66—Nitrogen atoms not forming part of a nitro radical
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D319/00—Heterocyclic compounds containing six-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D319/10—1,4-Dioxanes; Hydrogenated 1,4-dioxanes
    • C07D319/14—1,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems
    • C07D319/16—1,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D319/18—Ethylenedioxybenzenes, not substituted on the hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/06—Systems containing only non-condensed rings with a five-membered ring
    • C07C2601/08—Systems containing only non-condensed rings with a five-membered ring the ring being saturated

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Polymers & Plastics (AREA)
  • Food Science & Technology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Nutrition Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Inorganic Chemistry (AREA)
  • Epidemiology (AREA)
  • Birds (AREA)
  • Molecular Biology (AREA)
  • Oral & Maxillofacial Surgery (AREA)
  • Seasonings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Circuits Of Receivers In General (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Pyridine Compounds (AREA)
  • Fats And Perfumes (AREA)
  • Medicinal Preparation (AREA)
  • Pyrrole Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
  • Cosmetics (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Sweetening agents of the formula: <IMAGE> in which, in a preferred embodiment, R0 is: either a heterocyclic ring constructed on a cyclopentadienyl or phenyl group by replacement of 1 to 3 cyclic C with N, O or S, or an indanyl, indenyl, naphthyl or tetrahydronaphthyl group or a heterocyclic derivative constructed on these groups by replacement of 1 to 4 cyclic C with N, O or S; R1 is H or CH3; R2 is a 2-13 C hydrocarbon group in which up to 4 C may be replaced by N, O, S, Cl, Br and I and up to 5 H by F; R3 and R4 are H.
AU10271/88A 1987-01-15 1988-01-14 Sweetening agents derived from guanidinoacetic and ethanamidinoacetic acids, process for sweetening various products, and compositions containing such sweetening agents Ceased AU605228B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR8700539 1987-01-15
FR8700539A FR2609603B1 (en) 1987-01-15 1987-01-15 SWEETENING AGENTS DERIVED FROM GUANIDINOACETIC AND ETHANAMIDINOACETIC ACIDS, METHOD FOR SWEETENING VARIOUS PRODUCTS, AND COMPOSITIONS CONTAINING SUCH SWEETENING AGENTS

Publications (2)

Publication Number Publication Date
AU1027188A true AU1027188A (en) 1988-08-11
AU605228B2 AU605228B2 (en) 1991-01-10

Family

ID=9347035

Family Applications (1)

Application Number Title Priority Date Filing Date
AU10271/88A Ceased AU605228B2 (en) 1987-01-15 1988-01-14 Sweetening agents derived from guanidinoacetic and ethanamidinoacetic acids, process for sweetening various products, and compositions containing such sweetening agents

Country Status (16)

Country Link
EP (1) EP0289430B1 (en)
JP (1) JPS63188360A (en)
KR (1) KR880008760A (en)
CN (1) CN88100129A (en)
AT (1) ATE74496T1 (en)
AU (1) AU605228B2 (en)
BR (1) BR8800116A (en)
DE (1) DE3869823D1 (en)
DK (1) DK16188A (en)
FI (1) FI880160L (en)
FR (1) FR2609603B1 (en)
IL (1) IL84983A0 (en)
NO (1) NO880143L (en)
NZ (1) NZ223180A (en)
PT (1) PT86547B (en)
ZA (1) ZA88208B (en)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU595598B2 (en) * 1986-04-10 1990-04-05 Universite Claude Bernard - Lyon 1 High potency sweetening agents
AU612739B2 (en) * 1987-12-18 1991-07-18 Universite Claude Bernard - Lyon 1 Heterocyclic derivatives of n-carbamoyl-, n-thiocarbamoyl- or n-amidino-glycine or beta-alanine useful as sweetening agents

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4900740A (en) * 1987-10-02 1990-02-13 The Nutrasweet Company N,N'-disubstituted guanidines containing a carboxyl or a tetrazolyl moiety
IL95548A0 (en) * 1989-09-15 1991-06-30 Fujisawa Pharmaceutical Co Thiazole derivatives,processes for the preparation thereof and pharmaceutical composition containing the same
US9296697B2 (en) 2005-08-24 2016-03-29 Abbott Laboratories Hetaryl-substituted guanidine compounds and use thereof as binding partners for 5-HT5-receptors
DE102007034102A1 (en) * 2007-07-21 2009-01-22 Alzchem Trostberg Gmbh Abrasion-resistant and free-flowing glycocyamine-containing moldings and process for their preparation
DE102018112496A1 (en) 2018-05-24 2019-11-28 Rockwell Collins Deutschland Gmbh FLYWHEEL WITH TILGERMASSES

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2533210A1 (en) * 1982-09-17 1984-03-23 Lyon I Universite Claude SWEETENERS OF SYNTHESIS
FR2579202B1 (en) * 1985-03-19 1988-04-29 Univ Claude Bernard Lyon NOVEL CHEMICAL COMPOUNDS, USE AS SWEETENERS AND COMPOSITIONS CONTAINING SUCH AGENTS
FR2579201B1 (en) * 1985-03-19 1987-05-07 Bernard Lyon I Universite Clau IMPROVED CHEMICAL COMPOUNDS, USE AS SWEETENING AGENTS AND COMPOSITIONS CONTAINING SUCH AGENTS

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU595598B2 (en) * 1986-04-10 1990-04-05 Universite Claude Bernard - Lyon 1 High potency sweetening agents
AU612739B2 (en) * 1987-12-18 1991-07-18 Universite Claude Bernard - Lyon 1 Heterocyclic derivatives of n-carbamoyl-, n-thiocarbamoyl- or n-amidino-glycine or beta-alanine useful as sweetening agents

Also Published As

Publication number Publication date
BR8800116A (en) 1988-08-23
FR2609603A1 (en) 1988-07-22
DK16188A (en) 1988-07-16
DE3869823D1 (en) 1992-05-14
PT86547A (en) 1988-02-01
ATE74496T1 (en) 1992-04-15
FR2609603B1 (en) 1989-03-24
ZA88208B (en) 1988-06-30
DK16188D0 (en) 1988-01-14
NO880143L (en) 1988-07-18
IL84983A0 (en) 1988-06-30
PT86547B (en) 1991-12-31
AU605228B2 (en) 1991-01-10
EP0289430B1 (en) 1992-04-08
KR880008760A (en) 1988-09-13
NO880143D0 (en) 1988-01-14
FI880160A7 (en) 1988-07-16
JPS63188360A (en) 1988-08-03
FI880160A0 (en) 1988-01-14
NZ223180A (en) 1989-11-28
CN88100129A (en) 1988-07-27
FI880160L (en) 1988-07-16
EP0289430A1 (en) 1988-11-02

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