ATE481384T1 - Isoindolderivate als ep4-rezeptoragonisten - Google Patents
Isoindolderivate als ep4-rezeptoragonistenInfo
- Publication number
- ATE481384T1 ATE481384T1 AT07821299T AT07821299T ATE481384T1 AT E481384 T1 ATE481384 T1 AT E481384T1 AT 07821299 T AT07821299 T AT 07821299T AT 07821299 T AT07821299 T AT 07821299T AT E481384 T1 ATE481384 T1 AT E481384T1
- Authority
- AT
- Austria
- Prior art keywords
- receptor agonists
- isoindole derivatives
- derivatives
- isoindole
- medicine
- Prior art date
Links
- 150000002518 isoindoles Chemical class 0.000 title 1
- 239000000018 receptor agonist Substances 0.000 title 1
- 229940044601 receptor agonist Drugs 0.000 title 1
- 229940054051 antipsychotic indole derivative Drugs 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 150000002475 indoles Chemical class 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/56—Ring systems containing three or more rings
- C07D209/58—[b]- or [c]-condensed
- C07D209/62—Naphtho [c] pyrroles; Hydrogenated naphtho [c] pyrroles
- C07D209/66—Naphtho [c] pyrroles; Hydrogenated naphtho [c] pyrroles with oxygen atoms in positions 1 and 3
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Pain & Pain Management (AREA)
- Immunology (AREA)
- Rheumatology (AREA)
- Physical Education & Sports Medicine (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Urology & Nephrology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Indole Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0620619.7A GB0620619D0 (en) | 2006-10-17 | 2006-10-17 | Novel compounds |
| PCT/EP2007/060932 WO2008046798A1 (en) | 2006-10-17 | 2007-10-15 | Isoindol derivatives as ep4 receptor agonists |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE481384T1 true ATE481384T1 (de) | 2010-10-15 |
Family
ID=37507899
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT07821299T ATE481384T1 (de) | 2006-10-17 | 2007-10-15 | Isoindolderivate als ep4-rezeptoragonisten |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US20100076048A1 (de) |
| EP (1) | EP2081897B1 (de) |
| JP (1) | JP2010506878A (de) |
| AT (1) | ATE481384T1 (de) |
| DE (1) | DE602007009286D1 (de) |
| ES (1) | ES2352305T3 (de) |
| GB (1) | GB0620619D0 (de) |
| WO (1) | WO2008046798A1 (de) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2488168A1 (de) | 2009-10-14 | 2012-08-22 | Gemmus Pharma Inc. | Kombinationstherapie zur behandlung von virusinfektionen |
| AU2014305843B2 (en) | 2013-08-09 | 2019-08-29 | Ardelyx, Inc. | Compounds and methods for inhibiting phosphate transport |
| CN114340631A (zh) | 2019-05-21 | 2022-04-12 | 阿德利克斯股份有限公司 | 用于降低患者的血清磷酸盐的组合 |
Family Cites Families (24)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3300889A (en) * | 1965-04-22 | 1967-01-31 | Su Ev Inc | Recoil snubber for guns |
| US3707797A (en) * | 1970-11-18 | 1973-01-02 | K Ruth | Recoil absorber |
| US3714726A (en) * | 1970-11-25 | 1973-02-06 | P Braun | Recoil stock |
| US3754344A (en) * | 1972-04-28 | 1973-08-28 | J Spiliotis | Gun recoil absorber |
| US4439943A (en) * | 1982-03-09 | 1984-04-03 | Brakhage Rodney D | Recoil reducer |
| US4910904A (en) * | 1989-03-27 | 1990-03-27 | Browning | Recoil reducer for firearms |
| US5031348A (en) * | 1990-10-01 | 1991-07-16 | Carey Donald C | Gun stock assembly with coordinated comb and recoil |
| US5173564A (en) * | 1992-01-07 | 1992-12-22 | Hammond Jr Claude R | Quick detachable stock system and method |
| US5726377A (en) * | 1996-06-19 | 1998-03-10 | Colt's Manufacturing Company, Inc. | Gas operated firearm |
| EP1442744B1 (de) * | 1999-08-10 | 2006-12-20 | Glaxo Group Limited | EP4 Rezeptor Ligand und Verwendung gegen neuropatischen Schmerzen, Colon Krebs, HIV und Migräne |
| US6481143B2 (en) * | 2000-11-03 | 2002-11-19 | Mccarthy Patrick M. | Gun stock with recoil reduction device |
| GB0103269D0 (en) * | 2001-02-09 | 2001-03-28 | Glaxo Group Ltd | Napthalene derivatives |
| US6651371B2 (en) * | 2001-06-25 | 2003-11-25 | Richard Mark Fitzpatrick | Modular gunstock |
| US6688031B2 (en) * | 2002-05-30 | 2004-02-10 | Gerald Dale Steele | Replacement adjustable competition buttstock |
| US6732466B2 (en) * | 2002-08-19 | 2004-05-11 | James K. Bentley | Recoil system for the receiver of a firearm |
| US7398616B1 (en) * | 2004-05-21 | 2008-07-15 | Robert Weir | Adjustable length heavy duty butt stock assembly for a firearm |
| US7124529B1 (en) * | 2004-12-16 | 2006-10-24 | Havelka Jr Alfred J | Axially displaced gun stock recoil system |
| US7162822B1 (en) * | 2005-01-03 | 2007-01-16 | The United States Of America As Represented By The Secretary Of The Army | Collapsible buttstock for firearm |
| KR20080098597A (ko) * | 2006-02-03 | 2008-11-11 | 글락소 그룹 리미티드 | 통증의 치료를 위한 벤조이소인돌 유도체 |
| UY30121A1 (es) * | 2006-02-03 | 2007-08-31 | Glaxo Group Ltd | Nuevos compuestos |
| US7992337B2 (en) * | 2006-03-16 | 2011-08-09 | Ochoa Adam A | Method and apparatus to mount recoil dampening apparatus on rifle |
| GB0615111D0 (en) * | 2006-07-28 | 2006-09-06 | Glaxo Group Ltd | Novel compounds |
| GB0615105D0 (en) * | 2006-07-28 | 2006-09-06 | Glaxo Group Ltd | Novel compounds |
| US7681351B2 (en) * | 2006-11-15 | 2010-03-23 | Enidine, Inc. | Hydraulic recoil buffer assembly |
-
2006
- 2006-10-17 GB GBGB0620619.7A patent/GB0620619D0/en active Pending
-
2007
- 2007-10-15 AT AT07821299T patent/ATE481384T1/de not_active IP Right Cessation
- 2007-10-15 US US12/445,125 patent/US20100076048A1/en not_active Abandoned
- 2007-10-15 EP EP07821299A patent/EP2081897B1/de active Active
- 2007-10-15 WO PCT/EP2007/060932 patent/WO2008046798A1/en not_active Ceased
- 2007-10-15 DE DE602007009286T patent/DE602007009286D1/de active Active
- 2007-10-15 JP JP2009532780A patent/JP2010506878A/ja active Pending
- 2007-10-15 ES ES07821299T patent/ES2352305T3/es active Active
Also Published As
| Publication number | Publication date |
|---|---|
| EP2081897B1 (de) | 2010-09-15 |
| DE602007009286D1 (de) | 2010-10-28 |
| ES2352305T3 (es) | 2011-02-17 |
| US20100076048A1 (en) | 2010-03-25 |
| GB0620619D0 (en) | 2006-11-29 |
| JP2010506878A (ja) | 2010-03-04 |
| EP2081897A1 (de) | 2009-07-29 |
| WO2008046798A1 (en) | 2008-04-24 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |