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AR243887A1 - Procedimiento para la preparacion de piridilcarbonil-tiazolonas cardiotonicas. - Google Patents

Procedimiento para la preparacion de piridilcarbonil-tiazolonas cardiotonicas.

Info

Publication number
AR243887A1
AR243887A1 AR86304762A AR30476286A AR243887A1 AR 243887 A1 AR243887 A1 AR 243887A1 AR 86304762 A AR86304762 A AR 86304762A AR 30476286 A AR30476286 A AR 30476286A AR 243887 A1 AR243887 A1 AR 243887A1
Authority
AR
Argentina
Prior art keywords
tiazolonas
piridilcarbonil
cardiotonicas
procedure
preparation
Prior art date
Application number
AR86304762A
Other languages
English (en)
Original Assignee
Merrell Dow Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merrell Dow Pharma filed Critical Merrell Dow Pharma
Application granted granted Critical
Publication of AR243887A1 publication Critical patent/AR243887A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D407/00Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
    • C07D407/02Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/06Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Cardiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
AR86304762A 1985-10-15 1986-08-01 Procedimiento para la preparacion de piridilcarbonil-tiazolonas cardiotonicas. AR243887A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/787,225 US4623651A (en) 1985-10-15 1985-10-15 Cardiotonic heterocyclocarbonyl- and acetyl-thiazolones

Publications (1)

Publication Number Publication Date
AR243887A1 true AR243887A1 (es) 1993-09-30

Family

ID=25140796

Family Applications (1)

Application Number Title Priority Date Filing Date
AR86304762A AR243887A1 (es) 1985-10-15 1986-08-01 Procedimiento para la preparacion de piridilcarbonil-tiazolonas cardiotonicas.

Country Status (21)

Country Link
US (1) US4623651A (es)
EP (1) EP0219625B1 (es)
JP (1) JPS6287586A (es)
KR (1) KR890005203B1 (es)
CN (1) CN1020730C (es)
AR (1) AR243887A1 (es)
AT (1) ATE48275T1 (es)
AU (1) AU588900B2 (es)
CA (1) CA1287833C (es)
DE (1) DE3667175D1 (es)
DK (1) DK368986A (es)
ES (1) ES2000594A6 (es)
FI (1) FI863159L (es)
GR (1) GR862045B (es)
HU (1) HU197004B (es)
IL (1) IL79343A0 (es)
NO (1) NO863113L (es)
NZ (1) NZ217068A (es)
PH (1) PH22193A (es)
PT (1) PT83137B (es)
ZA (1) ZA865839B (es)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4734422A (en) * 1985-10-15 1988-03-29 Merrell Dow Pharmaceuticals Inc. Cardiotonic aroylthiazolones and the use thereof
US4762849A (en) * 1985-10-15 1988-08-09 Merrell Dow Pharmaceuticals Inc. Cardiotonic alkanoylthiazolones
US4927939A (en) * 1985-10-15 1990-05-22 Merrell Dow Pharmaceuticals Cardiotonic aroylthiazolones
US4670450A (en) * 1985-11-13 1987-06-02 Merrell Dow Pharmaceuticals Inc. Cardiotonic thiazolones
US4868182A (en) * 1986-11-05 1989-09-19 Merrell Dow Pharmaceuticals Inc. Enhancement of prazosin
US4866182A (en) * 1988-02-18 1989-09-12 Merrell Dow Pharmaceuticals Inc. Cardiotonic alkanoyl and aroyl oxazolones
US5095028A (en) * 1988-01-14 1992-03-10 Kureha Kagaku Kogyo Kabushiki Kaisha 2-(4-chlorobenzyl)-1-(1H-imidazole-1-ylmethyl)-1-cyclohexanol and cycloheptanol

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3514465A (en) * 1966-12-30 1970-05-26 Degussa Certain thiazolyl- and pyridinylaminoketones
FR2209560A1 (en) * 1972-12-07 1974-07-05 Degussa N-(Trialkoxyaroyl)-ethylenediamine derivs - useful as cardioactive medicaments, exhibit anti-ischaemic activity comparable to nitroglycerin
US4405635A (en) 1979-06-18 1983-09-20 Merrell Dow Pharmaceuticals Inc. 4-Aroylimidazol-2-ones and their use as pharmaceuticals
IE52884B1 (en) 1981-05-11 1988-03-30 Sigma Tau Ind Farmaceuti 2-methoxyphenyl esters of n-substituted amino acids, their preparation and pharmaceutical use

Also Published As

Publication number Publication date
KR890005203B1 (ko) 1989-12-18
US4623651A (en) 1986-11-18
AU588900B2 (en) 1989-09-28
EP0219625A1 (en) 1987-04-29
FI863159A7 (fi) 1987-04-16
PT83137B (pt) 1988-07-29
FI863159L (fi) 1987-04-16
NO863113L (no) 1987-04-21
KR870004025A (ko) 1987-05-07
DK368986A (da) 1987-04-16
ES2000594A6 (es) 1988-03-01
ATE48275T1 (de) 1989-12-15
DK368986D0 (da) 1986-08-01
CN86104968A (zh) 1987-04-22
ZA865839B (en) 1987-03-25
IL79343A0 (en) 1986-10-31
CA1287833C (en) 1991-08-20
PH22193A (en) 1988-06-28
DE3667175D1 (de) 1990-01-04
EP0219625B1 (en) 1989-11-29
PT83137A (en) 1986-09-01
NZ217068A (en) 1989-01-27
HU197004B (en) 1989-02-28
GR862045B (en) 1986-12-24
HUT44785A (en) 1988-04-28
JPS6287586A (ja) 1987-04-22
NO863113D0 (no) 1986-08-01
CN1020730C (zh) 1993-05-19
AU6084286A (en) 1987-04-16
FI863159A0 (fi) 1986-08-01

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