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AR240834A1 - Procedimiento para preparar derivados de 3beta-colestaniloxifosforilalquilamina - Google Patents

Procedimiento para preparar derivados de 3beta-colestaniloxifosforilalquilamina

Info

Publication number
AR240834A1
AR240834A1 AR297667A AR29766784A AR240834A1 AR 240834 A1 AR240834 A1 AR 240834A1 AR 297667 A AR297667 A AR 297667A AR 29766784 A AR29766784 A AR 29766784A AR 240834 A1 AR240834 A1 AR 240834A1
Authority
AR
Argentina
Prior art keywords
oxyphosphoryl
cholestanyl
3beta
preparing
procedure
Prior art date
Application number
AR297667A
Other languages
English (en)
Other versions
AR240834A2 (es
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Application granted granted Critical
Publication of AR240834A1 publication Critical patent/AR240834A1/es
Publication of AR240834A2 publication Critical patent/AR240834A2/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J1/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J51/00Normal steroids with unmodified cyclopenta(a)hydrophenanthrene skeleton not provided for in groups C07J1/00 - C07J43/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Cardiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Vascular Medicine (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Urology & Nephrology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AR297667A 1983-08-25 1984-08-22 Procedimiento para preparar derivados de 3beta-colestaniloxifosforilalquilamina AR240834A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH464483 1983-08-25

Publications (2)

Publication Number Publication Date
AR240834A1 true AR240834A1 (es) 1991-02-28
AR240834A2 AR240834A2 (es) 1991-02-28

Family

ID=4279973

Family Applications (1)

Application Number Title Priority Date Filing Date
AR297667A AR240834A1 (es) 1983-08-25 1984-08-22 Procedimiento para preparar derivados de 3beta-colestaniloxifosforilalquilamina

Country Status (21)

Country Link
US (1) US4680290A (es)
EP (1) EP0135762B1 (es)
JP (1) JPS6061595A (es)
KR (1) KR850001767A (es)
AR (1) AR240834A1 (es)
AT (1) ATE37883T1 (es)
AU (1) AU574706B2 (es)
CA (1) CA1252778A (es)
DE (1) DE3474552D1 (es)
DK (1) DK347584A (es)
ES (2) ES8602844A1 (es)
FI (1) FI842830A7 (es)
GR (1) GR80196B (es)
HU (1) HU189929B (es)
IL (1) IL72725A (es)
MC (1) MC1618A1 (es)
NO (1) NO161679C (es)
NZ (1) NZ209275A (es)
PH (1) PH19849A (es)
PT (1) PT79130B (es)
ZA (1) ZA846430B (es)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1241947A (en) * 1985-05-31 1988-09-13 Pierre R. Proulx Conjugated polyene sterol derivatives as membrane probes
US5026882A (en) * 1988-12-23 1991-06-25 Smithkline Beecham Corporation Phosphinic acid substituted steroids as inhibitors of steroid 5α-reductase
US4946834A (en) * 1988-12-23 1990-08-07 Smithkline Beecham Corporation Phosphonic acid substituted steroids as steroid 5α-reductase inhibitors
CA2028759A1 (en) * 1989-11-22 1991-05-23 Jean-Marie Cassal Steroids
US5215972A (en) * 1989-11-22 1993-06-01 Hoffmann-La Roche Inc. Steroids
US5244887A (en) * 1992-02-14 1993-09-14 Straub Carl D Stanols to reduce cholesterol absorption from foods and methods of preparation and use thereof
HUT77514A (hu) * 1994-11-30 1998-05-28 Amur Research Corp. Gyógyszerhatóanyagok foszfokolinszármazékai
JPH11507352A (ja) * 1995-06-07 1999-06-29 ジンタ・インコーポレイテッド 新規カルバメート基本カチオン性脂質
CA2223179A1 (en) * 1995-06-07 1996-12-19 Bob Dale Brown Phosphonic acid-based cationic lipids
JP2002514183A (ja) * 1996-09-17 2002-05-14 スーパージェン・インコーポレーテッド リン脂質薬剤誘導体
US5830432A (en) * 1997-03-31 1998-11-03 Amur Pharmacuticals, Inc. Phospholipid drug derivatives
EP1079859B1 (en) 1998-05-22 2010-07-14 The Board Of Trustees Of The Leland Stanford Junior University Bifunctional molecules and therapies based thereon
EP1252137A1 (en) 2000-01-28 2002-10-30 The Procter & Gamble Company Palatable arginine compounds and uses thereof for cardiovascular health
US20030045473A1 (en) * 2002-07-19 2003-03-06 Sarama Robert Joseph Compositions, kits, and methods for cardiovascular health
EP3827747A1 (en) 2005-04-28 2021-06-02 Otsuka Pharmaceutical Co., Ltd. Pharma-informatics system
EP1945240B1 (en) 2005-09-16 2016-12-28 Raptor Pharmaceutical Inc Compositions comprising receptor-associated protein (rap) variants specific for cr-containing proteins and uses thereof
JP2010511648A (ja) * 2006-12-08 2010-04-15 ジャド テクノロジーズ ゲーエムベーハー 感染性疾患の治療及び予防のためのコレステリルアミン
ES2728225T3 (es) 2009-02-20 2019-10-23 2 Bbb Medicines B V Sistema de administración de fármacos a base de glutatión
KR20190116576A (ko) 2009-05-06 2019-10-14 라보라토리 스킨 케어, 인크. 활성제-칼슘 포스페이트 입자 복합체를 포함하는 피부 전달 조성물 및 이들을 이용하는 방법
US20250135007A1 (en) * 2021-12-20 2025-05-01 Ron Weiss Compositions comprising sterol-amino-phosphate compounds and methods of making and use thereof

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3248408A (en) * 1963-07-22 1966-04-26 Merck & Co Inc Purification of steroid phosphates

Also Published As

Publication number Publication date
HUT34997A (en) 1985-05-28
DK347584A (da) 1985-02-26
PT79130A (en) 1984-09-01
ES8606879A1 (es) 1986-05-01
KR850001767A (ko) 1985-04-01
EP0135762A2 (de) 1985-04-03
NO161679C (no) 1989-09-13
PT79130B (en) 1986-11-14
PH19849A (en) 1986-07-22
EP0135762B1 (de) 1988-10-12
JPS6061595A (ja) 1985-04-09
FI842830A0 (fi) 1984-07-13
EP0135762A3 (en) 1986-01-22
CA1252778A (en) 1989-04-18
NO161679B (no) 1989-06-05
US4680290A (en) 1987-07-14
IL72725A (en) 1988-07-31
IL72725A0 (en) 1984-11-30
ES535391A0 (es) 1985-12-01
ES543646A0 (es) 1986-05-01
HU189929B (en) 1986-08-28
MC1618A1 (fr) 1985-07-18
DE3474552D1 (en) 1988-11-17
AR240834A2 (es) 1991-02-28
FI842830A7 (fi) 1985-02-26
DK347584D0 (da) 1984-07-13
ZA846430B (en) 1985-04-24
GR80196B (en) 1985-01-02
ATE37883T1 (de) 1988-10-15
NZ209275A (en) 1987-06-30
AU574706B2 (en) 1988-07-14
NO843406L (no) 1985-02-26
ES8602844A1 (es) 1985-12-01
AU3222584A (en) 1985-02-28

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