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AR248127A1 - Procedimiento para la preparacion de nuevas 2-aminotetralinas sustituidas en la posicion 8. - Google Patents

Procedimiento para la preparacion de nuevas 2-aminotetralinas sustituidas en la posicion 8.

Info

Publication number
AR248127A1
AR248127A1 AR91319245A AR31924591A AR248127A1 AR 248127 A1 AR248127 A1 AR 248127A1 AR 91319245 A AR91319245 A AR 91319245A AR 31924591 A AR31924591 A AR 31924591A AR 248127 A1 AR248127 A1 AR 248127A1
Authority
AR
Argentina
Prior art keywords
aminotetralines
replaced
procedure
new
preparation
Prior art date
Application number
AR91319245A
Other languages
English (en)
Original Assignee
Merrell Dow Pharmaceutcals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merrell Dow Pharmaceutcals Inc filed Critical Merrell Dow Pharmaceutcals Inc
Application granted granted Critical
Publication of AR248127A1 publication Critical patent/AR248127A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/30Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/31Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups having the sulfur atoms of the sulfonamide groups bound to acyclic carbon atoms
    • C07C311/35Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups having the sulfur atoms of the sulfonamide groups bound to acyclic carbon atoms of an unsaturated carbon skeleton containing rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/06Antimigraine agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2602/00Systems containing two condensed rings
    • C07C2602/02Systems containing two condensed rings the rings having only two atoms in common
    • C07C2602/04One of the condensed rings being a six-membered aromatic ring
    • C07C2602/10One of the condensed rings being a six-membered aromatic ring the other ring being six-membered, e.g. tetraline

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pain & Pain Management (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

PROCEDIMIENTO PARA PREPARAR NUEVAS 2-AMINOTETRALINAS SUSTITUIDAS EN LA POSICION 8, DE FORMULA (I) LOS ENANTIOMEROS Y SUS MEZCLAS Y LAS SALES FARMACEUTICAMENTE ACEPTABLES DE LOS MISMOS, DONDE CADA UNO DE R1 Y R2 REPRESENTA HIDROGENO O ALQUILO INFERIOR C1-7, Y R3 ES ALQUILO INFERIOR C1- 7.
AR91319245A 1990-03-21 1991-03-19 Procedimiento para la preparacion de nuevas 2-aminotetralinas sustituidas en la posicion 8. AR248127A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP90400781A EP0447727A1 (en) 1990-03-21 1990-03-21 Novel 8-sulfamylmethylene-2-amino tetralins

Publications (1)

Publication Number Publication Date
AR248127A1 true AR248127A1 (es) 1995-06-30

Family

ID=8205692

Family Applications (1)

Application Number Title Priority Date Filing Date
AR91319245A AR248127A1 (es) 1990-03-21 1991-03-19 Procedimiento para la preparacion de nuevas 2-aminotetralinas sustituidas en la posicion 8.

Country Status (18)

Country Link
EP (2) EP0447727A1 (es)
JP (1) JPH04253954A (es)
KR (1) KR910016692A (es)
CN (1) CN1055179A (es)
AR (1) AR248127A1 (es)
AT (1) ATE124392T1 (es)
AU (1) AU634366B2 (es)
CA (1) CA2038748A1 (es)
DE (1) DE69110728D1 (es)
DK (1) DK0451008T3 (es)
FI (1) FI911351L (es)
HU (1) HUT57185A (es)
IE (1) IE910933A1 (es)
IL (1) IL97579A0 (es)
NO (1) NO911118L (es)
NZ (1) NZ237446A (es)
PT (1) PT97084A (es)
ZA (1) ZA911948B (es)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2686339B1 (fr) * 1992-01-22 1994-03-11 Adir Cie Nouveaux amides et sulfonamides naphtaleniques, leurs procedes de preparation et les compositions pharmaceutiques qui les contiennent.
GB9211277D0 (en) 1992-05-28 1992-07-15 Glaxo Group Inc Pharmaceutical compositions
US6586458B1 (en) 1996-08-16 2003-07-01 Pozen Inc. Methods of treating headaches using 5-HT agonists in combination with long-acting NSAIDs
US8022095B2 (en) 1996-08-16 2011-09-20 Pozen, Inc. Methods of treating headaches using 5-HT agonists in combination with long-acting NSAIDs
US7189753B1 (en) 1997-11-06 2007-03-13 Cady Roger K Preemptive prophylaxis of migraine
MXPA05006954A (es) 2002-12-26 2005-09-22 Pozen Inc Formas de dosificacion de capas multiples que contienen nsaids y triptanos.
AR075442A1 (es) * 2009-02-16 2011-03-30 Abbott Gmbh & Co Kg Derivados de aminotetralina, composiciones farmaceuticas que las contienen y sus usos en terapia

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1170387B (it) * 1982-06-07 1987-06-03 Glaxo Group Ltd Composti eterociclici, procedimento per prepararli e composizioni farmaceutiche che li contengono
US4529723A (en) * 1983-04-29 1985-07-16 William H. Rorer, Inc. Bicyclic benzenoid aminoalkylene ethers and thioethers, pharmaceutical compositions and use
DE3719924A1 (de) * 1986-12-22 1988-06-30 Bayer Ag 8-substituierte 2-aminotetraline

Also Published As

Publication number Publication date
ZA911948B (en) 1991-12-24
CA2038748A1 (en) 1991-09-22
PT97084A (pt) 1991-11-29
FI911351A7 (fi) 1991-09-22
AU7295091A (en) 1991-10-03
NZ237446A (en) 1993-11-25
KR910016692A (ko) 1991-11-05
JPH04253954A (ja) 1992-09-09
NO911118L (no) 1991-09-23
DK0451008T3 (da) 1995-09-04
ATE124392T1 (de) 1995-07-15
EP0451008B1 (en) 1995-06-28
EP0447727A1 (en) 1991-09-25
FI911351A0 (fi) 1991-03-20
HU910937D0 (en) 1991-10-28
DE69110728D1 (de) 1995-08-03
IE910933A1 (en) 1991-09-25
HUT57185A (en) 1991-11-28
AU634366B2 (en) 1993-02-18
IL97579A0 (en) 1992-06-21
EP0451008A1 (en) 1991-10-09
CN1055179A (zh) 1991-10-09
NO911118D0 (no) 1991-03-20
FI911351L (fi) 1991-09-22

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