[go: up one dir, main page]

AR227400A1 - PROCEDURE TO OBTAIN N-OXACICLIL-ALKYL-PIPERIDINES AND THEIR SALTS - Google Patents

PROCEDURE TO OBTAIN N-OXACICLIL-ALKYL-PIPERIDINES AND THEIR SALTS

Info

Publication number
AR227400A1
AR227400A1 AR282945A AR28294580A AR227400A1 AR 227400 A1 AR227400 A1 AR 227400A1 AR 282945 A AR282945 A AR 282945A AR 28294580 A AR28294580 A AR 28294580A AR 227400 A1 AR227400 A1 AR 227400A1
Authority
AR
Argentina
Prior art keywords
oxaciclil
piperidines
salts
alkyl
procedure
Prior art date
Application number
AR282945A
Other languages
Spanish (es)
Original Assignee
Ciba Geigy Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy Ag filed Critical Ciba Geigy Ag
Application granted granted Critical
Publication of AR227400A1 publication Critical patent/AR227400A1/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Psychiatry (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
AR282945A 1978-03-20 1980-10-20 PROCEDURE TO OBTAIN N-OXACICLIL-ALKYL-PIPERIDINES AND THEIR SALTS AR227400A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US88808978A 1978-03-20 1978-03-20

Publications (1)

Publication Number Publication Date
AR227400A1 true AR227400A1 (en) 1982-10-29

Family

ID=25392505

Family Applications (4)

Application Number Title Priority Date Filing Date
AR275879A AR227272A1 (en) 1978-03-20 1979-03-20 PROCEDURE FOR OBTAINING COMPOUNDS OF N-OXACICLIL-ALQUIL-PIPERIDIL-DIAZA AND ITS SALTS
AR282945A AR227400A1 (en) 1978-03-20 1980-10-20 PROCEDURE TO OBTAIN N-OXACICLIL-ALKYL-PIPERIDINES AND THEIR SALTS
AR282944A AR231638A1 (en) 1978-03-20 1980-10-20 PROCEDURE FOR OBTAINING COMPOUNDS OF 1-1-2- (1,4-BENZOXATIO OR 1,4-BENZOXATIAN OR 1,4-BENZODIOXAN-2-IL) -ALKYLENE-4-PIPERIDIL-2-IMIDAZOLINONE, 2-HEXAHYDRO-PIRIMIDINONE OR 2-IMINO-IMIDAZOLIDINE
AR282946A AR227527A1 (en) 1978-03-20 1980-10-20 PROCEDURE FOR THE ELABORATION OF NEW COMPOUNDS N-OXACICLILALQUIL-PIPERIDIL-DIAZOICOS

Family Applications Before (1)

Application Number Title Priority Date Filing Date
AR275879A AR227272A1 (en) 1978-03-20 1979-03-20 PROCEDURE FOR OBTAINING COMPOUNDS OF N-OXACICLIL-ALQUIL-PIPERIDIL-DIAZA AND ITS SALTS

Family Applications After (2)

Application Number Title Priority Date Filing Date
AR282944A AR231638A1 (en) 1978-03-20 1980-10-20 PROCEDURE FOR OBTAINING COMPOUNDS OF 1-1-2- (1,4-BENZOXATIO OR 1,4-BENZOXATIAN OR 1,4-BENZODIOXAN-2-IL) -ALKYLENE-4-PIPERIDIL-2-IMIDAZOLINONE, 2-HEXAHYDRO-PIRIMIDINONE OR 2-IMINO-IMIDAZOLIDINE
AR282946A AR227527A1 (en) 1978-03-20 1980-10-20 PROCEDURE FOR THE ELABORATION OF NEW COMPOUNDS N-OXACICLILALQUIL-PIPERIDIL-DIAZOICOS

Country Status (20)

Country Link
EP (1) EP0004358B1 (en)
JP (1) JPS54157570A (en)
AR (4) AR227272A1 (en)
AT (1) AT372088B (en)
AU (1) AU529838B2 (en)
DD (1) DD142341A5 (en)
DE (1) DE2961738D1 (en)
DK (1) DK113079A (en)
ES (4) ES478662A1 (en)
FI (1) FI66373C (en)
GB (1) GB2019837B (en)
GR (1) GR71865B (en)
HU (1) HU182941B (en)
IL (1) IL56908A (en)
MY (1) MY8700122A (en)
NO (1) NO150202C (en)
NZ (1) NZ189939A (en)
PL (1) PL116514B1 (en)
PT (1) PT69369A (en)
ZA (2) ZA79417B (en)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4329348A (en) * 1979-02-26 1982-05-11 Ciba-Geigy Corporation N-Oxacyclic-alkylpiperidines as psychostimulants
DE3124366A1 (en) * 1981-06-20 1982-12-30 Hoechst Ag, 6000 Frankfurt N-OXACYCLYL-ALKYLPIPERIDIN DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF, PHARMACEUTICAL PREPARATIONS CONTAINING IT AND THE USE THEREOF
FR2524887A1 (en) * 1982-04-08 1983-10-14 Bouchara Emile NOVEL CYANOGUANIDINES, PROCESS FOR OBTAINING THEM AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME
FR2525600A1 (en) * 1982-04-21 1983-10-28 Bouchara Emile NOVEL CARBOXAMIDOGUANIDINES, PROCESS FOR OBTAINING SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME
US4556660A (en) * 1982-07-12 1985-12-03 Janssen Pharmaceutica N.V. N-(Bicyclic heterocyclyl)-4-piperidinamines
JP2807577B2 (en) * 1990-06-15 1998-10-08 エーザイ株式会社 Cyclic amide derivative
SI9300097B (en) * 1992-02-27 2001-12-31 Janssen Pharmaceutica Nv (benzodioxan, benzofuran or benzopyran) alkylamino) alkyl substituted guanidines
US5703115A (en) * 1993-02-19 1997-12-30 Janssen Pharmaceutica, N.V. (benzodioxan, benzofuran or benzopyran) alkylamino! alkyl substituted guanidines
US6133277A (en) 1997-12-05 2000-10-17 Janssen Pharmaceutica N.V. (Benzodioxan, benzofuran or benzopyran) derivatives having fundic relaxation properties
PL198552B1 (en) * 1999-06-02 2008-06-30 Janssen Pharmaceutica Nv Derivatives (of benzodioxane, benzophurane or benzopyrane) substituted by aminoalkil
HUP0201344A3 (en) 1999-06-02 2005-09-28 Janssen Pharmaceutica Nv Pyrrolidinyl, piperidinyl or homopiperidinyl substituted (benzodioxan, benzofuran or benzopyran) derivatives, process for their preparation and pharmaceutical compositions containing the compounds
JO2352B1 (en) * 2000-06-22 2006-12-12 جانسين فارماسيوتيكا ان. في Compounds for treating fundic disaccomodation
EP1856126A2 (en) 2005-02-17 2007-11-21 Wyeth a Corporation of the State of Delaware Cycloalkylfused indole, benzothiophene, benzofuran and indene derivatives
CN114920686B (en) * 2022-05-20 2023-11-24 山东农业大学 Synthesis method of 5-(phenylsulfonyl)-N-piperidin-4-yl-2-(trifluoromethyl)benzenesulfonamide hydrochloride

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3910930A (en) * 1973-01-04 1975-10-07 Janssen Pharmaceutica Nv 1-{55 1-{8 2-(1,4-Benzodioxan-2-yl)-2-hydroxyethyl{9 -4-piperidyl{56 -2-benzimidazolinones

Also Published As

Publication number Publication date
MY8700122A (en) 1987-12-31
ZA791276B (en) 1980-03-26
FI790894A7 (en) 1979-09-21
IL56908A0 (en) 1979-05-31
AR227272A1 (en) 1982-10-15
PT69369A (en) 1979-04-01
ES484570A1 (en) 1980-05-16
DK113079A (en) 1979-09-21
AT372088B (en) 1983-08-25
IL56908A (en) 1983-09-30
NO150202C (en) 1984-09-05
EP0004358B1 (en) 1982-01-06
ATA204479A (en) 1983-01-15
AU4524379A (en) 1979-09-27
ZA79417B (en) 1980-01-30
EP0004358A1 (en) 1979-10-03
FI66373C (en) 1984-10-10
NZ189939A (en) 1981-12-15
DE2961738D1 (en) 1982-02-25
PL214206A1 (en) 1980-02-25
ES478662A1 (en) 1980-01-16
AU529838B2 (en) 1983-06-23
ES484571A1 (en) 1980-05-16
DD142341A5 (en) 1980-06-18
PL116514B1 (en) 1981-06-30
NO150202B (en) 1984-05-28
AR227527A1 (en) 1982-11-15
ES484572A1 (en) 1980-05-16
HU182941B (en) 1984-03-28
FI66373B (en) 1984-06-29
GR71865B (en) 1983-07-07
GB2019837B (en) 1982-08-25
NO790917L (en) 1979-09-21
JPS54157570A (en) 1979-12-12
GB2019837A (en) 1979-11-07
AR231638A1 (en) 1985-01-31

Similar Documents

Publication Publication Date Title
AR220539A1 (en) PROCEDURE TO OBTAIN 7 BETA-ARIL-MALONAMIDO-7 ALPHA-METOXI-3- (TIADIAZOLILTIO) 1-OXADETIACEFALOSPORINAS AND ITS SALTS
MX5995E (en) PROCEDURE TO PREPARE 6-N-PROPIL-8-METHYLMARKET-METHYLERGOLINS
AR229081A1 (en) PROCEDURE TO PREPARE NEW MERCAPTOACILPROLINAS
MX5926E (en) PROCEDURE TO PREPARE 4-PYRIMIDONES
AR221699A1 (en) A PROCEDURE TO PREPARE THE D-VAL-GLI-L-CIS-L-LIS-L-ASN-L-FE-L-FE-L-TRP-L-LIS-L-TTR-L-FE-L- SER-L-CIS-OH AND ITS SALTS
AR222828A1 (en) PROCEDURE FOR THE PREPARATION OF 2,3,4,5-TETRAHIDRO-6-FENILTIO-1H-3-BENZAZEPINAS AND ITS SALTS
AR225922A1 (en) PROCEDURE TO PREPARE NEW DERIVATIVES OF 3-CARBAMOIL-SULFONAMIDO-4-AMINO-PIRIDINA AND ITS SALTS
AR227731A1 (en) PROCEDURE TO OBTAIN NEW DERIVATIVES OF ((PIPERIDIL-2) -2-ETIL) -4-QUINOLEIN AND ITS SALTS
ES496713A0 (en) PROCEDURE TO PREPARE ALPHA-ARIL-IN-IMIDAZOLE-1-ETHANOLS
AR227400A1 (en) PROCEDURE TO OBTAIN N-OXACICLIL-ALKYL-PIPERIDINES AND THEIR SALTS
AR230280A1 (en) PROCEDURE FOR OBTAINING CARBOESTIRILE DERIVATIVES AND THEIR SALTS
AR223069A1 (en) POLYETERPOLIAMINS AND THEIR SALTS, PROCEDURE FOR THEIR PREPARATION AND EMPLOYMENT
AR228851A1 (en) PROCEDURE FOR PREPARING 9-HYDROXY-9-AMINO ALKYLFLOURENES AND THEIR SALTS
AR241905A1 (en) PROCEDURE TO OBTAIN NEW CARBOESTIRILE DERIVATIVES AND THEIR SALTS.
AR228019A1 (en) PROCEDURE FOR PREPARING ACID DERIVATIVES- (3-PENOXI-2-AMINO) -PHENYLALCANOIC AND ITS SALTS
AR219948A1 (en) PROCEDURE TO OBTAIN NEW 7-AZABENZIMIDAZOLES WITH BASIC SIDE CHAINS AND THEIR SALTS
AR219792A1 (en) PROCEDURE TO PREPARE S-HALOALQUENIL DIISOALQUILTIOCARBAMATOS
AR227621A1 (en) PROCEDURE FOR THE ELABORATION OF BENZ-ACILBENZIMIDAZOLCARBENIC ACIDS AND THEIR SALTS
AR226288A1 (en) PROCEDURE FOR THE PRODUCTION OF NEW 4-ALQUILTIOFENOXI ALQUILAMINAS AND ITS SALTS
AR228036A1 (en) PROCEDURE FOR OBTAINING DERIVATIVES OF 1-TIO-ALCANOYLPROLIN AND ITS SALTS
AR225318A1 (en) PROCEDURE TO PREPARE SUBSTITUTED PHENYL-PROPIL-MORPHOLINS
AR230453A1 (en) PROCEDURE TO PREPARE NOVELTY DERIVATIVES OF VINCALEUCOBLASTINA AND ITS SALTS
MX3845E (en) PROCEDURE FOR THE PREPARATION OF SUBSTITUTED SULFOXIMIDES AND THEIR SALTS
AR226825A1 (en) PROCEDURE FOR PREPARING 2-HYDROXY-PROPYLAMINOALKYL GUANIDINES DERIVATIVES AND THEIR ADDITIONAL SALTS
MX6013E (en) PROCEDURE FOR PREPARING ARILALQUIL AND ARILOXI-ALQUIL-FOSFONATOS