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AR226527A1 - Procedimiento para preparar derivados de acido dibenzo(b,f)tiepin-3-carboxilico - Google Patents

Procedimiento para preparar derivados de acido dibenzo(b,f)tiepin-3-carboxilico

Info

Publication number
AR226527A1
AR226527A1 AR273031A AR27303178A AR226527A1 AR 226527 A1 AR226527 A1 AR 226527A1 AR 273031 A AR273031 A AR 273031A AR 27303178 A AR27303178 A AR 27303178A AR 226527 A1 AR226527 A1 AR 226527A1
Authority
AR
Argentina
Prior art keywords
tiepin
carboxylic
procedure
acid derivatives
preparing
Prior art date
Application number
AR273031A
Other languages
English (en)
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Application granted granted Critical
Publication of AR226527A1 publication Critical patent/AR226527A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D337/00Heterocyclic compounds containing rings of more than six members having one sulfur atom as the only ring hetero atom
    • C07D337/02Seven-membered rings
    • C07D337/06Seven-membered rings condensed with carbocyclic rings or ring systems
    • C07D337/10Seven-membered rings condensed with carbocyclic rings or ring systems condensed with two six-membered rings
    • C07D337/14[b,f]-condensed
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/14Antitussive agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C321/00Thiols, sulfides, hydropolysulfides or polysulfides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
AR273031A 1977-07-26 1978-07-21 Procedimiento para preparar derivados de acido dibenzo(b,f)tiepin-3-carboxilico AR226527A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US81919977A 1977-07-26 1977-07-26
US91721278A 1978-06-23 1978-06-23

Publications (1)

Publication Number Publication Date
AR226527A1 true AR226527A1 (es) 1982-07-30

Family

ID=27124337

Family Applications (2)

Application Number Title Priority Date Filing Date
AR273031A AR226527A1 (es) 1977-07-26 1978-07-21 Procedimiento para preparar derivados de acido dibenzo(b,f)tiepin-3-carboxilico
AR278140A AR222666A1 (es) 1977-07-26 1979-09-20 Procedimiento para preparar derivados de 5-tetrazolil dibenzo-(b,f)tiepinas

Family Applications After (1)

Application Number Title Priority Date Filing Date
AR278140A AR222666A1 (es) 1977-07-26 1979-09-20 Procedimiento para preparar derivados de 5-tetrazolil dibenzo-(b,f)tiepinas

Country Status (16)

Country Link
EP (1) EP0011067B1 (es)
JP (1) JPS5444691A (es)
AR (2) AR226527A1 (es)
AU (1) AU517813B2 (es)
CA (1) CA1128048A (es)
DD (1) DD140746A5 (es)
DE (1) DE2861754D1 (es)
DK (1) DK330578A (es)
ES (5) ES471871A1 (es)
FI (1) FI782323A7 (es)
GR (1) GR67276B (es)
IE (1) IE47553B1 (es)
IT (1) IT1107485B (es)
NO (1) NO782539L (es)
PL (3) PL117756B1 (es)
PT (1) PT68303A (es)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4536507A (en) * 1977-07-26 1985-08-20 Merck & Co., Inc. Prostaglandin antagonists
PT71280B (en) * 1979-06-01 1981-09-17 Merck & Co Inc Process for preparing prostaglandin antagonists
DE3068250D1 (en) * 1979-11-27 1984-07-19 Merck Sharp & Dohme 3-hydroxymethyldibenzo(b,f)thiepins and dibenzo(b,f)thiepin-3-carboxaldehydes as prostaglandin antagonists, process for their preparation and pharmaceutical compositions
US4237160A (en) * 1979-11-27 1980-12-02 Merck Sharp & Dohme (I.A.) Corp. 3-Hydroxymethyldibenzo[b,f]thiepins as prostaglandin antagonists
NO811187L (no) * 1980-11-24 1982-05-25 Merck & Co Inc Fremgangsmaate ved fremstilling av 7-fluor-dibenzo-(b,f)-thiepinderivater
US4535171A (en) * 1982-11-18 1985-08-13 Merck Frosst Canada, Inc. Dibenzo[b,f]thiepin-3-carboxaldehydes as prostaglandin antagonists
US4622403A (en) * 1983-10-11 1986-11-11 Merck Frosst Canada, Inc. 6-H dibenz[b,f]thiepin compounds
US4663347A (en) 1983-10-31 1987-05-05 Merck Frosst Canada, Inc. Benzofuran 2-carboxylic acid esters useful as inhibitors of leukotriene biosynthesis
CA1309557C (en) 1985-06-18 1992-10-27 Robert N. Young Leukotriene antagonists
EP0239306B1 (en) 1986-03-27 1993-06-02 Merck Frosst Canada Inc. Tetrahydrocarbazole esters
CA2053216C (en) 1990-10-12 2003-04-08 Michel L. Belley Saturated hydroxyalkylquinoline acids as leukotriene antagonists
US5410054A (en) * 1993-07-20 1995-04-25 Merck Frosst Canada, Inc. Heteroaryl quinolines as inhibitors of leukotriene biosynthesis
US6180659B1 (en) * 1996-01-19 2001-01-30 Nippon Suisan Kaisha, Ltd. Tracheal smooth muscle relaxant
JP3471778B2 (ja) 1999-06-03 2003-12-02 日本水産株式会社 三環性縮合複素環化合物、その製造方法および用途
TWI275495B (en) * 2004-09-21 2007-03-11 Sony Corp Printer and printing method

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4101667A (en) * 1975-05-30 1978-07-18 Nippon Chemiphar Co., Ltd. Benzo[b,f]thiepin derivatives
JPS5346989A (en) * 1976-10-06 1978-04-27 Nippon Chemiphar Co Ltd Novel dibenzo(b,f)thiepin derivatives and their preparation
JPS6021156B2 (ja) * 1976-12-03 1985-05-25 日本ケミフア株式会社 ベンゾチエピン誘導体およびその製法

Also Published As

Publication number Publication date
PL117756B1 (en) 1981-08-31
AU3817778A (en) 1980-01-24
FI782323A7 (fi) 1979-01-27
JPS5444691A (en) 1979-04-09
ES479218A1 (es) 1979-11-01
PL208653A1 (pl) 1979-06-04
EP0011067B1 (en) 1982-04-21
ES479217A1 (es) 1979-07-01
CA1128048A (en) 1982-07-20
JPS6250470B2 (es) 1987-10-24
PT68303A (en) 1978-08-01
PL116355B1 (en) 1981-06-30
DE2861754D1 (en) 1982-06-03
ES471871A1 (es) 1979-10-01
IE47553B1 (en) 1984-04-18
DK330578A (da) 1979-01-27
DD140746A5 (de) 1980-03-26
PL120813B1 (en) 1982-03-31
EP0011067A1 (en) 1980-05-28
AU517813B2 (en) 1981-08-27
ES479215A1 (es) 1979-07-01
IT1107485B (it) 1985-11-25
ES479216A1 (es) 1979-07-01
GR67276B (es) 1981-06-26
IE781488L (en) 1979-01-26
IT7850375A0 (it) 1978-07-19
AR222666A1 (es) 1981-06-15
NO782539L (no) 1979-01-29

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