AR215591A1 - PROCEDURE FOR THE PREPARATION OF 4,5-DIPHENYL-2- (THIO-SUBSTITUTED) IMIDAZOLES AND THEIR CORRESPONDING SULFOXIDES AND SULFONES - Google Patents
PROCEDURE FOR THE PREPARATION OF 4,5-DIPHENYL-2- (THIO-SUBSTITUTED) IMIDAZOLES AND THEIR CORRESPONDING SULFOXIDES AND SULFONESInfo
- Publication number
- AR215591A1 AR215591A1 AR264308A AR26430876A AR215591A1 AR 215591 A1 AR215591 A1 AR 215591A1 AR 264308 A AR264308 A AR 264308A AR 26430876 A AR26430876 A AR 26430876A AR 215591 A1 AR215591 A1 AR 215591A1
- Authority
- AR
- Argentina
- Prior art keywords
- sulfones
- imidazoles
- thio
- diphenyl
- substituted
- Prior art date
Links
- 150000002460 imidazoles Chemical class 0.000 title 1
- 150000003457 sulfones Chemical class 0.000 title 1
- 150000003462 sulfoxides Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/84—Sulfur atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pain & Pain Management (AREA)
- Pharmacology & Pharmacy (AREA)
- Rheumatology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US60365075A | 1975-08-11 | 1975-08-11 | |
| US69128276A | 1976-06-09 | 1976-06-09 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR215591A1 true AR215591A1 (en) | 1979-10-31 |
Family
ID=27084480
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AR264308A AR215591A1 (en) | 1975-08-11 | 1976-08-11 | PROCEDURE FOR THE PREPARATION OF 4,5-DIPHENYL-2- (THIO-SUBSTITUTED) IMIDAZOLES AND THEIR CORRESPONDING SULFOXIDES AND SULFONES |
| AR270672A AR218054A1 (en) | 1975-08-11 | 1978-01-10 | PROCEDURE FOR THE PREPARATION OF 4,5-DIPHENYL-2- (THIO-SUBSTITUTED) IMIDAZOLES AND ITS CORRESPONDING SULFOXIDES AND SULPHONES |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AR270672A AR218054A1 (en) | 1975-08-11 | 1978-01-10 | PROCEDURE FOR THE PREPARATION OF 4,5-DIPHENYL-2- (THIO-SUBSTITUTED) IMIDAZOLES AND ITS CORRESPONDING SULFOXIDES AND SULPHONES |
Country Status (26)
| Country | Link |
|---|---|
| JP (1) | JPS6011702B2 (en) |
| AR (2) | AR215591A1 (en) |
| AU (1) | AU508605B2 (en) |
| CA (1) | CA1074327A (en) |
| CH (1) | CH638791A5 (en) |
| DD (1) | DD126244A5 (en) |
| DE (1) | DE2635876A1 (en) |
| DK (1) | DK361376A (en) |
| ES (2) | ES450601A1 (en) |
| FI (1) | FI66177C (en) |
| FR (1) | FR2320745A1 (en) |
| GB (1) | GB1516908A (en) |
| GR (1) | GR61145B (en) |
| HU (1) | HU174707B (en) |
| IE (1) | IE44019B1 (en) |
| IL (1) | IL50230A (en) |
| LU (1) | LU75578A1 (en) |
| MX (1) | MX3932E (en) |
| NL (1) | NL7608915A (en) |
| NO (1) | NO146571C (en) |
| NZ (1) | NZ181731A (en) |
| PH (1) | PH11857A (en) |
| PT (1) | PT65464B (en) |
| SE (1) | SE428686B (en) |
| SU (1) | SU640662A3 (en) |
| YU (1) | YU198176A (en) |
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DK16778A (en) * | 1977-02-09 | 1978-08-10 | Du Pont | IMIDAZOLE DERIVATIVES THEIR USES AND MANUFACTURE |
| LU77703A1 (en) * | 1977-07-07 | 1979-03-26 | Ciba Geigy Ag | METHOD FOR PRODUCING BICYCLIC THIA-DIAZA COMPOUNDS |
| EP0004648B1 (en) * | 1978-04-11 | 1982-08-25 | Ciba-Geigy Ag | Mercapto-imidazole derivatives, their preparation, mercapto-imidazole derivatives for the treatment of inflammatory diseases and their pharmaceutical compositions |
| DE2823197A1 (en) * | 1978-05-24 | 1979-11-29 | Schering Ag | NEW IMIDAZOLE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND PHARMACEUTICAL PREPARATIONS CONTAINING THEM |
| US4308277A (en) * | 1978-08-10 | 1981-12-29 | Ciba-Geigy Corporation | 2,4,5-Trisubstituted imidazolines and pharmaceutical compositions containing same |
| US4188397A (en) * | 1978-09-22 | 1980-02-12 | Smithkline Corporation | 2,2-Alkyldiylbis(thio)bis(imidazoles) |
| US4215135A (en) * | 1979-06-08 | 1980-07-29 | E. I. Du Pont De Nemours And Company | Antiinflammatory 2-substituted-1H-phenanthro[9,10-d]imidazoles |
| DE2856909A1 (en) * | 1978-12-28 | 1980-07-17 | Schering Ag | NEW IMIDAZOLE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND PHARMACEUTICAL PREPARATIONS CONTAINING THEM |
| GB8907656D0 (en) * | 1989-04-05 | 1989-05-17 | May & Baker Ltd | New compositions of matter |
| PL183931B1 (en) * | 1994-09-26 | 2002-08-30 | Shionogi & Co | Imidazole derivative |
| JP2002515915A (en) * | 1997-06-30 | 2002-05-28 | オーソ−マクニール・フアーマシユーチカル・インコーポレーテツド | 2-Substituted imidazoles useful in treating inflammatory diseases |
| DE10222103A1 (en) * | 2002-05-17 | 2003-11-27 | Merckle Gmbh Chem Pharm Fabrik | New 2-(substituted thio)-imidazole derivatives are immunomodulators and cytokine release inhibitors, useful for treating diseases associated with immune system disorders, e.g. cancer or rheumatoid arthritis |
| CN101415687B (en) * | 2006-02-06 | 2012-02-08 | 大正制药株式会社 | Binding inhibitor of sphingosine-1-phosphate |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SE345453B (en) * | 1965-10-21 | 1972-05-29 | Ciba Geigy Ag | |
| US3651080A (en) * | 1969-11-07 | 1972-03-21 | Ciba Geigy Corp | Certain substituted 2-alkylmercaptoimidazole derivatives |
| US3636003A (en) * | 1969-11-17 | 1972-01-18 | Geigy Chem Corp | Substituted 2-mercaptoimidazole derivatives |
| US3714179A (en) * | 1970-09-08 | 1973-01-30 | Searle & Co | 1-alkyl-2-furfurylthioimidazoles and congeners |
| US3707475A (en) * | 1970-11-16 | 1972-12-26 | Pfizer | Antiinflammatory imidazoles |
-
1976
- 1976-07-02 SE SE7607615A patent/SE428686B/en not_active IP Right Cessation
- 1976-08-05 MX MX762132U patent/MX3932E/en unknown
- 1976-08-09 NO NO762754A patent/NO146571C/en unknown
- 1976-08-09 DD DD194248A patent/DD126244A5/xx unknown
- 1976-08-09 CA CA258,690A patent/CA1074327A/en not_active Expired
- 1976-08-10 DK DK361376A patent/DK361376A/en not_active Application Discontinuation
- 1976-08-10 PT PT65464A patent/PT65464B/en unknown
- 1976-08-10 FR FR7624400A patent/FR2320745A1/en active Granted
- 1976-08-10 SU SU762388413A patent/SU640662A3/en active
- 1976-08-10 AU AU16711/76A patent/AU508605B2/en not_active Expired
- 1976-08-10 DE DE19762635876 patent/DE2635876A1/en not_active Withdrawn
- 1976-08-10 PH PH18773A patent/PH11857A/en unknown
- 1976-08-10 CH CH1019276A patent/CH638791A5/en not_active IP Right Cessation
- 1976-08-10 ES ES450601A patent/ES450601A1/en not_active Expired
- 1976-08-10 FI FI762290A patent/FI66177C/en not_active IP Right Cessation
- 1976-08-10 IL IL50230A patent/IL50230A/en unknown
- 1976-08-10 GB GB33286/76A patent/GB1516908A/en not_active Expired
- 1976-08-10 HU HU76DU252A patent/HU174707B/en unknown
- 1976-08-10 GR GR51440A patent/GR61145B/en unknown
- 1976-08-10 NZ NZ181737A patent/NZ181731A/en unknown
- 1976-08-11 YU YU01981/76A patent/YU198176A/en unknown
- 1976-08-11 JP JP51094991A patent/JPS6011702B2/en not_active Expired
- 1976-08-11 IE IE1775/76A patent/IE44019B1/en unknown
- 1976-08-11 AR AR264308A patent/AR215591A1/en active
- 1976-08-11 NL NL7608915A patent/NL7608915A/en not_active Application Discontinuation
- 1976-08-11 LU LU75578A patent/LU75578A1/xx unknown
-
1977
- 1977-07-28 ES ES461193A patent/ES461193A1/en not_active Expired
-
1978
- 1978-01-10 AR AR270672A patent/AR218054A1/en active
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