AR204660A1 - Procedimiento para preparar compuestos derivados del acido 2(1-piperazinil)-5-oxopirido-(2,3-d)pirimidino-6-carboxilico - Google Patents
Procedimiento para preparar compuestos derivados del acido 2(1-piperazinil)-5-oxopirido-(2,3-d)pirimidino-6-carboxilicoInfo
- Publication number
- AR204660A1 AR204660A1 AR258571A AR25857175A AR204660A1 AR 204660 A1 AR204660 A1 AR 204660A1 AR 258571 A AR258571 A AR 258571A AR 25857175 A AR25857175 A AR 25857175A AR 204660 A1 AR204660 A1 AR 204660A1
- Authority
- AR
- Argentina
- Prior art keywords
- oxopyride
- piperazinil
- pyrimidine
- procedure
- preparing compounds
- Prior art date
Links
- 239000002253 acid Substances 0.000 title 1
- 150000001875 compounds Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/48—Two nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP3845373A JPS5546400B2 (es) | 1973-04-03 | 1973-04-03 | |
| JP5654473A JPS565753B2 (es) | 1973-05-21 | 1973-05-21 | |
| JP6446473A JPS565755B2 (es) | 1973-06-07 | 1973-06-07 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR204660A1 true AR204660A1 (es) | 1976-02-20 |
Family
ID=27289838
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AR253060A AR204003A1 (es) | 1973-04-03 | 1974-01-01 | Procedimiento para preparar compuestos derivados del acido 2-(1-piperazinil)-5-oxopirido-(2,3-d)pirimidino-6-carboxilico y sus sales farmaceuticamente aceptables |
| AR258571A AR204660A1 (es) | 1973-04-03 | 1975-01-01 | Procedimiento para preparar compuestos derivados del acido 2(1-piperazinil)-5-oxopirido-(2,3-d)pirimidino-6-carboxilico |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AR253060A AR204003A1 (es) | 1973-04-03 | 1974-01-01 | Procedimiento para preparar compuestos derivados del acido 2-(1-piperazinil)-5-oxopirido-(2,3-d)pirimidino-6-carboxilico y sus sales farmaceuticamente aceptables |
Country Status (11)
| Country | Link |
|---|---|
| AR (2) | AR204003A1 (es) |
| AT (1) | AT340931B (es) |
| CA (1) | CA1066701A (es) |
| CH (1) | CH593281A5 (es) |
| ES (1) | ES424851A1 (es) |
| FI (1) | FI56011C (es) |
| IE (1) | IE39102B1 (es) |
| NL (1) | NL186087C (es) |
| NO (1) | NO142221C (es) |
| PH (2) | PH10529A (es) |
| SE (1) | SE416051B (es) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IT1209163B (it) * | 1979-12-21 | 1989-07-10 | Unibios S P A Trecate Novara | Procedimento per la fabbricazione di: 6-alcossicarbonil-8-etil-5-oxo-5,8diidro-aperta par. quadrata 2,3-dchiusa par. quadrata-primidine 2-sostituite ed acidi libri corrispondenti. |
| CA2766100C (en) | 2009-06-29 | 2018-05-22 | Incyte Corporation | Pyrimidinones as pi3k inhibitors |
| WO2011075643A1 (en) | 2009-12-18 | 2011-06-23 | Incyte Corporation | Substituted heteroaryl fused derivatives as pi3k inhibitors |
| WO2011075630A1 (en) | 2009-12-18 | 2011-06-23 | Incyte Corporation | Substituted fused aryl and heteroaryl derivatives as pi3k inhibitors |
| ES2764848T3 (es) | 2010-12-20 | 2020-06-04 | Incyte Holdings Corp | N-(1-(fenilo sustituido)etilo)-9H-purina-6-aminas como inhibidores de PI3K |
| KR102131612B1 (ko) | 2011-09-02 | 2020-07-08 | 인사이트 홀딩스 코포레이션 | Pi3k 억제제로서 헤테로시클릴아민 |
| AR090548A1 (es) | 2012-04-02 | 2014-11-19 | Incyte Corp | Azaheterociclobencilaminas biciclicas como inhibidores de pi3k |
| WO2015191677A1 (en) | 2014-06-11 | 2015-12-17 | Incyte Corporation | Bicyclic heteroarylaminoalkyl phenyl derivatives as pi3k inhibitors |
| SI3831833T1 (sl) | 2015-02-27 | 2023-03-31 | Incyte Holdings Corporation | Postopki za pripravo inhibitorja PI3K |
| WO2016183063A1 (en) | 2015-05-11 | 2016-11-17 | Incyte Corporation | Crystalline forms of a pi3k inhibitor |
| WO2016183060A1 (en) | 2015-05-11 | 2016-11-17 | Incyte Corporation | Process for the synthesis of a phosphoinositide 3-kinase inhibitor |
| IL278889B2 (en) | 2018-06-01 | 2025-11-01 | Incyte Corp | Dosing regimen for the treatment of pi3k related disorders |
-
1974
- 1974-01-01 AR AR253060A patent/AR204003A1/es active
- 1974-01-30 CA CA191,286A patent/CA1066701A/en not_active Expired
- 1974-02-01 SE SE7401361A patent/SE416051B/xx not_active IP Right Cessation
- 1974-02-04 NO NO740349A patent/NO142221C/no unknown
- 1974-02-04 FI FI298/74A patent/FI56011C/fi active
- 1974-02-04 NL NLAANVRAGE7401509,A patent/NL186087C/xx not_active IP Right Cessation
- 1974-02-14 CH CH205474A patent/CH593281A5/de not_active IP Right Cessation
- 1974-03-25 IE IE00650/74A patent/IE39102B1/xx unknown
- 1974-04-02 ES ES424851A patent/ES424851A1/es not_active Expired
- 1974-04-03 AT AT277774A patent/AT340931B/de not_active IP Right Cessation
- 1974-04-03 PH PH15698A patent/PH10529A/en unknown
-
1975
- 1975-01-01 AR AR258571A patent/AR204660A1/es active
- 1975-09-05 PH PH17546A patent/PH10984A/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| NO740349L (no) | 1974-10-04 |
| AT340931B (de) | 1978-01-10 |
| CA1066701A (en) | 1979-11-20 |
| NL186087B (nl) | 1990-04-17 |
| FI56011B (fi) | 1979-07-31 |
| IE39102B1 (en) | 1978-08-02 |
| NO142221B (no) | 1980-04-08 |
| AR204003A1 (es) | 1975-11-12 |
| IE39102L (en) | 1974-10-03 |
| CH593281A5 (en) | 1977-11-30 |
| SE416051B (sv) | 1980-11-24 |
| NO142221C (no) | 1980-07-16 |
| PH10984A (en) | 1977-10-18 |
| NL186087C (nl) | 1990-09-17 |
| ES424851A1 (es) | 1976-06-01 |
| FI56011C (fi) | 1979-11-12 |
| PH10529A (en) | 1977-05-30 |
| NL7401509A (es) | 1974-10-07 |
| ATA277774A (de) | 1977-05-15 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| AR213608A1 (es) | Procedimiento para preparar compuestos derivados de 1a-hidroxi vitamina d | |
| AR206409A1 (es) | Un procedimento para preparar compuestos de hexahidro-dibenzo(b,d)piran-ona | |
| AR213169A1 (es) | Procedimiento de obtencion de nuevos compuestos derivados de acido(1-oxo-2,2-disubstituido-6,7-dihaloindaniloxi alcanaicos | |
| SE420720B (sv) | Forfarande for framstellning av 2,6-disubstuerade fenylaminoguanidinforeningar | |
| AR204660A1 (es) | Procedimiento para preparar compuestos derivados del acido 2(1-piperazinil)-5-oxopirido-(2,3-d)pirimidino-6-carboxilico | |
| SE416725B (sv) | Forfarande for framstellning av p-nitrobensoesyra | |
| IT1011276B (it) | Procedimento per produrre acido p nitro toluol 2 solfonic | |
| AR218221A1 (es) | Procedimiento para preparar 5-glutamida del acido 2-aminoetansulfonico | |
| SE422212B (sv) | Forfarande for framstellning av 7beta-amino-3-metyl-cefam-4-karbonsyraforeningar | |
| AR208885A1 (es) | Procedimiento mejorado para preparar compuestos de 2-amino-5-alquil-1,3,4-tiadiazol | |
| IT1010309B (it) | Processo per la preparazione di composti aromatici del fosforo | |
| AR212692A1 (es) | Procedimiento para preparar 5,6-dihidro-s-triazolo(5,1-a)isoquinolinas | |
| AR214173A1 (es) | Un procedimiento para preparar alfa-esteres del acido 6alfa-metoxi,6beta-(2-carboxifenil o tienil-acetamido)-penicilanico | |
| BE810087A (fr) | Procede de preparation de triceto-2,4,5- imidazolidines | |
| MX4655E (es) | Procedimiento para preparar derivados del acido 3,3,'-triarilmetanodicarboxilico | |
| AR204577A1 (es) | Procedimiento para la preparacion de derivados del acido 7-mesilamino-fenilglicinamido-3-substituido-3-cefem-4-carboxilico | |
| AR204250A1 (es) | Procedimiento para preparar compuestos derivados del acido tricloroacetamido-6 penicilanico-5-oxido | |
| AR218217A1 (es) | Proceso para la preparacion de acido 3,6-dicloropicolinico | |
| BE819212A (fr) | Procede de preparation de 2,6-di-tert-butyl-4-cumyl-phenol | |
| AR208712A1 (es) | Procedimiento para preparar compuestos de acido 7-beta-acilamino-7-alfa-metoxi-3-cefemcarboxilico | |
| IT1025936B (it) | Procedimento per preparare acido metacrilico | |
| AR199285A1 (es) | Procedimiento para preparar compuestos del acido 1,4,6,9-tetrahidro-4-6-dioxopirido <3,2-g> quinolin-2,8-dicarboxilico | |
| SE402920B (sv) | Forfarande for framstellning av nya 21-alkylerade 16alfa, 17alfa-alkylidendioxi-pregn-4-en-3,20-dioner | |
| AR208274A1 (es) | Procedimiento para preparar nuevos compuestos derivados acidos xantona-2-carboxilicos-5,7-disustituidos | |
| MX5979E (es) | Procedimiento para la preparacion de bis-(dihidroxipropilamidas)del acido 5-hidroxipropionilamino-2,4,6-triyodo isoftalico |