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AR192803A1 - METHOD FOR PREPARING 2,4-DIAMINE-5-BENZYLPYRIMIDINES - Google Patents

METHOD FOR PREPARING 2,4-DIAMINE-5-BENZYLPYRIMIDINES

Info

Publication number
AR192803A1
AR192803A1 AR242773A AR24277372A AR192803A1 AR 192803 A1 AR192803 A1 AR 192803A1 AR 242773 A AR242773 A AR 242773A AR 24277372 A AR24277372 A AR 24277372A AR 192803 A1 AR192803 A1 AR 192803A1
Authority
AR
Argentina
Prior art keywords
benzylpyrimidines
diamine
preparing
Prior art date
Application number
AR242773A
Other languages
Spanish (es)
Original Assignee
Wellcome Found
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wellcome Found filed Critical Wellcome Found
Application granted granted Critical
Publication of AR192803A1 publication Critical patent/AR192803A1/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32One oxygen, sulfur or nitrogen atom
    • C07D239/42One nitrogen atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00Carboxylic acid nitriles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00Sulfones; Sulfoxides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/67Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
    • C07C45/68Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48Two nitrogen atoms
    • C07D239/49Two nitrogen atoms with an aralkyl radical, or substituted aralkyl radical, attached in position 5, e.g. trimethoprim
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
AR242773A 1970-10-22 1972-06-27 METHOD FOR PREPARING 2,4-DIAMINE-5-BENZYLPYRIMIDINES AR192803A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB963871*[A GB1375162A (en) 1970-10-22 1970-10-22
GB963871 1971-04-16
GB4749171 1971-10-12

Publications (1)

Publication Number Publication Date
AR192803A1 true AR192803A1 (en) 1973-03-14

Family

ID=27255400

Family Applications (3)

Application Number Title Priority Date Filing Date
AR238596A AR192588A1 (en) 1970-10-22 1971-10-21 A METHOD FOR PREPARING PYRIMIDINE DERIVATIVES
AR242773A AR192803A1 (en) 1970-10-22 1972-06-27 METHOD FOR PREPARING 2,4-DIAMINE-5-BENZYLPYRIMIDINES
AR242772A AR192802A1 (en) 1970-10-22 1972-06-27 METHOD FOR PREPARING 2,4-DIAMINE-5-BENZYL-PYRIMIDINES

Family Applications Before (1)

Application Number Title Priority Date Filing Date
AR238596A AR192588A1 (en) 1970-10-22 1971-10-21 A METHOD FOR PREPARING PYRIMIDINE DERIVATIVES

Family Applications After (1)

Application Number Title Priority Date Filing Date
AR242772A AR192802A1 (en) 1970-10-22 1972-06-27 METHOD FOR PREPARING 2,4-DIAMINE-5-BENZYL-PYRIMIDINES

Country Status (20)

Country Link
JP (2) JPS5536662B1 (en)
AR (3) AR192588A1 (en)
AT (1) AT319948B (en)
BE (1) BE774281A (en)
BG (4) BG20365A3 (en)
CA (1) CA967158A (en)
CH (3) CH568302A5 (en)
DD (1) DD100877A5 (en)
DK (1) DK132174C (en)
ES (1) ES396219A1 (en)
FI (1) FI56175C (en)
FR (1) FR2111769B1 (en)
GB (1) GB1375162A (en)
IE (1) IE37452B1 (en)
IL (2) IL45422A (en)
LU (1) LU64129A1 (en)
MC (1) MC894A1 (en)
NL (1) NL175178C (en)
SE (2) SE384505B (en)
ZM (1) ZM14971A1 (en)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE792096A (en) * 1971-12-01 1973-05-30 Hoffmann La Roche NEW BENZYLPYRIMIDINES
FR2397407A2 (en) * 1977-07-11 1979-02-09 Dick Pierre 2,4-DIAMINO PYRIMIDINE DERIVATIVES AND THEIR SOLUTION IN ASSOCIATION WITH SULFAMIDS
IT1117752B (en) * 1978-05-24 1986-02-24 Wellcome Found PHARMACEUTICAL COMPOSITION BASED ON BENZYLPYRIMIDINE AND PROCEDURE FOR ITS PREPARATION
JPS61156909A (en) * 1984-12-27 1986-07-16 Matsushita Electric Ind Co Ltd Current mirror circuit
JPS62145907A (en) * 1985-12-20 1987-06-30 Hitachi Ltd transistor circuit
EP1728793B1 (en) 2004-03-26 2016-02-03 Sumitomo Dainippon Pharma Co., Ltd. 9-substituted 8-oxoadenine compound
WO2008004948A1 (en) 2006-07-05 2008-01-10 Astrazeneca Ab 8-oxoadenine derivatives acting as modulators of tlr7
TW200831105A (en) 2006-12-14 2008-08-01 Astrazeneca Ab Novel compounds
PT2132209E (en) 2007-03-19 2014-04-15 Astrazeneca Ab 9-substituted-8-oxo-adenine compounds as toll-like receptor (tlr7 ) modulators
US8063051B2 (en) 2007-03-19 2011-11-22 Astrazeneca Ab 9-substituted-8-oxo-adenine compounds as toll-like receptor (TLR7) modulators
US8044056B2 (en) 2007-03-20 2011-10-25 Dainippon Sumitomo Pharma Co., Ltd. Adenine compound
PE20091236A1 (en) 2007-11-22 2009-09-16 Astrazeneca Ab PYRIMIDINE DERIVATIVES AS IMMUNOMODULATORS OF TLR7
UY31531A1 (en) 2007-12-17 2009-08-03 SALTS DERIVED FROM 8-OXOADENINE PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM AND THEIR USE IN THERAPY AS TOLL TYPE RECEIVER MODULATORS (TLR)
GB0908772D0 (en) 2009-05-21 2009-07-01 Astrazeneca Ab New salts 756
CN102482233A (en) 2009-05-21 2012-05-30 阿斯利康(瑞典)有限公司 Novel pyrimidine derivatives and their use in the treatment of cancer and other diseases
ES2575688T3 (en) 2010-12-16 2016-06-30 Sumitomo Dainippon Pharma Co., Ltd. Imidazo [4,5-c] quinolin-1-yl derivative useful in therapy
JP5978226B2 (en) 2010-12-17 2016-08-24 大日本住友製薬株式会社 Purine derivatives
KR102194585B1 (en) 2012-05-18 2020-12-23 다이닛본 스미토모 세이야꾸 가부시끼가이샤 Carboxylic acid compounds

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE710100A (en) * 1967-02-02 1968-07-30
JPS511716A (en) * 1974-06-25 1976-01-08 Toray Industries HORIESUTERUMARUCHIFUIRAMENTONO SEIHO

Also Published As

Publication number Publication date
ZM14971A1 (en) 1972-07-21
AR192588A1 (en) 1973-02-28
SE384505B (en) 1976-05-10
CH568302A5 (en) 1975-10-31
AR192802A1 (en) 1973-03-14
SE409705B (en) 1979-09-03
ES396219A1 (en) 1975-09-16
AT319948B (en) 1975-01-10
JPS5536662B1 (en) 1980-09-22
IL37984A (en) 1976-03-31
DK132174C (en) 1976-03-29
MC894A1 (en) 1972-06-22
BG20797A3 (en) 1975-12-20
BG20364A3 (en) 1975-11-05
NL175178C (en) 1984-10-01
LU64129A1 (en) 1972-06-28
NL7114494A (en) 1972-04-25
IE37452L (en) 1972-04-22
BG20365A3 (en) 1975-11-05
BE774281A (en) 1972-04-21
IL37984A0 (en) 1971-12-29
FI56175C (en) 1979-12-10
GB1375162A (en) 1974-11-27
FR2111769A1 (en) 1972-06-09
FR2111769B1 (en) 1974-10-18
BG21406A3 (en) 1976-05-20
DD100877A5 (en) 1973-10-12
IL45422A (en) 1976-03-31
CA967158A (en) 1975-05-06
CH568301A5 (en) 1975-10-31
FI56175B (en) 1979-08-31
DK132174B (en) 1975-11-03
JPS53135991A (en) 1978-11-28
NL175178B (en) 1984-05-01
CH582681A5 (en) 1976-12-15
IE37452B1 (en) 1977-08-03

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