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AR192802A1 - Metodo para preparar 2,4-diamino-5-bencil-pirimidinas - Google Patents

Metodo para preparar 2,4-diamino-5-bencil-pirimidinas

Info

Publication number
AR192802A1
AR192802A1 AR242772A AR24277272A AR192802A1 AR 192802 A1 AR192802 A1 AR 192802A1 AR 242772 A AR242772 A AR 242772A AR 24277272 A AR24277272 A AR 24277272A AR 192802 A1 AR192802 A1 AR 192802A1
Authority
AR
Argentina
Prior art keywords
pyrimidines
diamine
benzyl
preparing
Prior art date
Application number
AR242772A
Other languages
English (en)
Original Assignee
Wellcome Found
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wellcome Found filed Critical Wellcome Found
Application granted granted Critical
Publication of AR192802A1 publication Critical patent/AR192802A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32One oxygen, sulfur or nitrogen atom
    • C07D239/42One nitrogen atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00Carboxylic acid nitriles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00Sulfones; Sulfoxides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/67Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
    • C07C45/68Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48Two nitrogen atoms
    • C07D239/49Two nitrogen atoms with an aralkyl radical, or substituted aralkyl radical, attached in position 5, e.g. trimethoprim
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
AR242772A 1970-10-22 1972-06-27 Metodo para preparar 2,4-diamino-5-bencil-pirimidinas AR192802A1 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB963871*[A GB1375162A (es) 1970-10-22 1970-10-22
GB963871 1971-04-16
GB4749171 1971-10-12

Publications (1)

Publication Number Publication Date
AR192802A1 true AR192802A1 (es) 1973-03-14

Family

ID=27255400

Family Applications (3)

Application Number Title Priority Date Filing Date
AR238596A AR192588A1 (es) 1970-10-22 1971-10-21 Un metodo para preparar derivados de pirimidina
AR242773A AR192803A1 (es) 1970-10-22 1972-06-27 Metodo para preparar 2,4-diamino-5-bencilpirimidinas
AR242772A AR192802A1 (es) 1970-10-22 1972-06-27 Metodo para preparar 2,4-diamino-5-bencil-pirimidinas

Family Applications Before (2)

Application Number Title Priority Date Filing Date
AR238596A AR192588A1 (es) 1970-10-22 1971-10-21 Un metodo para preparar derivados de pirimidina
AR242773A AR192803A1 (es) 1970-10-22 1972-06-27 Metodo para preparar 2,4-diamino-5-bencilpirimidinas

Country Status (20)

Country Link
JP (2) JPS5536662B1 (es)
AR (3) AR192588A1 (es)
AT (1) AT319948B (es)
BE (1) BE774281A (es)
BG (4) BG20365A3 (es)
CA (1) CA967158A (es)
CH (3) CH582681A5 (es)
DD (1) DD100877A5 (es)
DK (1) DK132174C (es)
ES (1) ES396219A1 (es)
FI (1) FI56175C (es)
FR (1) FR2111769B1 (es)
GB (1) GB1375162A (es)
IE (1) IE37452B1 (es)
IL (2) IL45422A (es)
LU (1) LU64129A1 (es)
MC (1) MC894A1 (es)
NL (1) NL175178C (es)
SE (2) SE384505B (es)
ZM (1) ZM14971A1 (es)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE792096A (fr) * 1971-12-01 1973-05-30 Hoffmann La Roche Nouvelles benzylpyrimidines
FR2397407A2 (fr) * 1977-07-11 1979-02-09 Dick Pierre Derives de 2,4-diamino pyrimidines et leur mise en solution en association avec des sulfamides
JPS54154775A (en) * 1978-05-24 1979-12-06 Wellcome Found Benzylpyrimidine derivative
JPS61156909A (ja) * 1984-12-27 1986-07-16 Matsushita Electric Ind Co Ltd カレント・ミラ−回路
JPS62145907A (ja) * 1985-12-20 1987-06-30 Hitachi Ltd トランジスタ回路
MXPA06011080A (es) 2004-03-26 2007-04-16 Astrazeneca Ab Compuesto de 8-oxoadenina 9-sustituido.
WO2008004948A1 (en) 2006-07-05 2008-01-10 Astrazeneca Ab 8-oxoadenine derivatives acting as modulators of tlr7
TW200831105A (en) 2006-12-14 2008-08-01 Astrazeneca Ab Novel compounds
US8067413B2 (en) 2007-03-19 2011-11-29 Astrazeneca Ab 9-substituted-8-oxo-adenine compounds as toll-like receptor (TLR7 ) modulators
WO2008114006A1 (en) 2007-03-19 2008-09-25 Astrazeneca Ab 9-substituted-8-oxo-adenine compounds as toll-like receptor (tlr7) modulators
WO2008114819A1 (ja) 2007-03-20 2008-09-25 Dainippon Sumitomo Pharma Co., Ltd. 新規アデニン化合物
PE20091236A1 (es) * 2007-11-22 2009-09-16 Astrazeneca Ab Derivados de pirimidina como immunomoduladores de tlr7
PE20091156A1 (es) 2007-12-17 2009-09-03 Astrazeneca Ab Sales de (3-{[[3-(6-amino-2-butoxi-8-oxo-7,8-dihidro-9h-purin-9-il)propil](3-morfolin-4-ilpropil)amino]metil}fenil)acetato de metilo
JP5913093B2 (ja) 2009-05-21 2016-04-27 アストラゼネカ アクチボラグ 新規ピリミジン誘導体と、癌とさらなる疾患の治療におけるそれらの使用
GB0908772D0 (en) 2009-05-21 2009-07-01 Astrazeneca Ab New salts 756
CN103370317B (zh) 2010-12-16 2015-10-07 阿斯利康(瑞典)有限公司 可用于治疗的咪唑并[4,5-c]喹啉-1-基衍生物
EP2651943B1 (en) 2010-12-17 2017-03-22 Sumitomo Dainippon Pharma Co., Ltd. Purine derivatives
JP6184423B2 (ja) 2012-05-18 2017-08-23 大日本住友製薬株式会社 カルボン酸化合物

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE710100A (es) * 1967-02-02 1968-07-30
JPS511716A (ja) * 1974-06-25 1976-01-08 Toray Industries Horiesuterumaruchifuiramentono seiho

Also Published As

Publication number Publication date
BG20365A3 (bg) 1975-11-05
MC894A1 (fr) 1972-06-22
BG20364A3 (bg) 1975-11-05
FI56175B (fi) 1979-08-31
NL175178C (nl) 1984-10-01
FR2111769B1 (es) 1974-10-18
IE37452L (en) 1972-04-22
JPS5536662B1 (es) 1980-09-22
BG20797A3 (bg) 1975-12-20
AR192588A1 (es) 1973-02-28
AT319948B (de) 1975-01-10
BG21406A3 (bg) 1976-05-20
NL175178B (nl) 1984-05-01
FR2111769A1 (es) 1972-06-09
DK132174C (da) 1976-03-29
FI56175C (fi) 1979-12-10
AR192803A1 (es) 1973-03-14
DD100877A5 (es) 1973-10-12
ZM14971A1 (en) 1972-07-21
IL37984A0 (en) 1971-12-29
CH568302A5 (es) 1975-10-31
LU64129A1 (es) 1972-06-28
BE774281A (fr) 1972-04-21
IL37984A (en) 1976-03-31
GB1375162A (es) 1974-11-27
IL45422A (en) 1976-03-31
NL7114494A (es) 1972-04-25
JPS53135991A (en) 1978-11-28
IE37452B1 (en) 1977-08-03
CA967158A (en) 1975-05-06
SE384505B (sv) 1976-05-10
DK132174B (da) 1975-11-03
ES396219A1 (es) 1975-09-16
CH568301A5 (es) 1975-10-31
CH582681A5 (es) 1976-12-15
SE409705B (sv) 1979-09-03

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