AR128896A1 - IKZF2 DEGRADERS AND USES OF THESE - Google Patents
IKZF2 DEGRADERS AND USES OF THESEInfo
- Publication number
- AR128896A1 AR128896A1 ARP230100748A ARP230100748A AR128896A1 AR 128896 A1 AR128896 A1 AR 128896A1 AR P230100748 A ARP230100748 A AR P230100748A AR P230100748 A ARP230100748 A AR P230100748A AR 128896 A1 AR128896 A1 AR 128896A1
- Authority
- AR
- Argentina
- Prior art keywords
- compound
- formula
- pharmaceutically acceptable
- ikzf2
- degraders
- Prior art date
Links
- 101000599037 Homo sapiens Zinc finger protein Helios Proteins 0.000 title 1
- 102100037796 Zinc finger protein Helios Human genes 0.000 title 1
- 239000001064 degrader Substances 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 5
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 239000000546 pharmaceutical excipient Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 239000012453 solvate Substances 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Un compuesto de formula (1). El compuesto de reivindicación 9, en donde el compuesto es un compuesto de fórmula (I-2-ii), (I-2-iii), (I-2-iv), (I-2-v), (I-2-vi), (I-2-vii), (I-2-ix) o (I-2-xii) del grupo de fórmulas (2), o una sal, solvato o estereoisómero farmacéuticamente aceptable de este. Una composición farmacéutica que comprende el compuesto de una cualquiera de las reivindicaciones 1 - 36, y un excipiente farmacéuticamente aceptable.A compound of formula (1). The compound of claim 9, wherein the compound is a compound of formula (I-2-ii), (I-2-iii), (I-2-iv), (I-2-v) , (I-2-vi), (I-2-vii), (I-2-ix) or (I-2-xii) of the group of formulas (2), or a salt, solvate or pharmaceutically acceptable stereoisomer thereof. A pharmaceutical composition comprising the compound of any one of claims 1-36, and a pharmaceutically acceptable excipient.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US202063446105P | 2020-02-16 | 2020-02-16 | |
| US202263323792P | 2022-03-25 | 2022-03-25 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR128896A1 true AR128896A1 (en) | 2024-06-26 |
Family
ID=91665054
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP230100748A AR128896A1 (en) | 2020-02-16 | 2023-03-27 | IKZF2 DEGRADERS AND USES OF THESE |
Country Status (1)
| Country | Link |
|---|---|
| AR (1) | AR128896A1 (en) |
-
2023
- 2023-03-27 AR ARP230100748A patent/AR128896A1/en unknown
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