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AR103781A1 - Combinación de un retinoide y un diol y éster de ácido graso poliinsaturado - Google Patents

Combinación de un retinoide y un diol y éster de ácido graso poliinsaturado

Info

Publication number
AR103781A1
AR103781A1 ARP160100497A ARP160100497A AR103781A1 AR 103781 A1 AR103781 A1 AR 103781A1 AR P160100497 A ARP160100497 A AR P160100497A AR P160100497 A ARP160100497 A AR P160100497A AR 103781 A1 AR103781 A1 AR 103781A1
Authority
AR
Argentina
Prior art keywords
retinoid
combination
fatty acid
diol
acid ester
Prior art date
Application number
ARP160100497A
Other languages
English (en)
Original Assignee
Pierre Fabre Dermo Cosmetique
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pierre Fabre Dermo Cosmetique filed Critical Pierre Fabre Dermo Cosmetique
Publication of AR103781A1 publication Critical patent/AR103781A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/045Hydroxy compounds, e.g. alcohols; Salts thereof, e.g. alcoholates
    • A61K31/07Retinol compounds, e.g. vitamin A
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/22Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin
    • A61K31/23Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin of acids having a carboxyl group bound to a chain of seven or more carbon atoms
    • A61K31/232Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin of acids having a carboxyl group bound to a chain of seven or more carbon atoms having three or more double bonds, e.g. etretinate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/33Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing oxygen
    • A61K8/37Esters of carboxylic acids
    • A61K8/375Esters of carboxylic acids the alcohol moiety containing more than one hydroxy group
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/67Vitamins
    • A61K8/671Vitamin A; Derivatives thereof, e.g. ester of vitamin A acid, ester of retinol, retinol, retinal
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0014Skin, i.e. galenical aspects of topical compositions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/06Ointments; Bases therefor; Other semi-solid forms, e.g. creams, sticks, gels
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/02Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/10Anti-acne agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61QSPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q19/00Preparations for care of the skin
    • A61Q19/008Preparations for oily skin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Emergency Medicine (AREA)
  • Birds (AREA)
  • Dermatology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Cosmetics (AREA)

Abstract

Reivindicación 1: Una combinación que comprende un retinoide y un compuesto de la fórmula general (1), donde: n es un número entero entre 0 y 15, m es 0, 1, 2 ó 3, y R es la cadena hidrocarbonada de un ácido graso poliinsaturado seleccionado de omega-3s y omega-6s. Reivindicación 5: La combinación de acuerdo con cualquiera de las reivindicaciones 1 a 4, donde el compuesto de fórmula general (1) se selecciona de las moléculas del grupo de fórmulas (2). Reivindicación 6: La combinación de acuerdo con cualquiera de las reivindicaciones 1 a 5, donde el retinoide se selecciona de retinol, retinaldehído, y ácido retinoico en sus diversas formas estereoisoméricas. Reivindicación 15: Un retinoide para uso tópico en la prevención de la formación de lesiones retencionales.
ARP160100497A 2015-02-27 2016-02-25 Combinación de un retinoide y un diol y éster de ácido graso poliinsaturado AR103781A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR1551714A FR3033135B1 (fr) 2015-02-27 2015-02-27 Association d'un retinoide et d'un ester de diol et d'acide gras polyinsature

Publications (1)

Publication Number Publication Date
AR103781A1 true AR103781A1 (es) 2017-05-31

Family

ID=53200134

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP160100497A AR103781A1 (es) 2015-02-27 2016-02-25 Combinación de un retinoide y un diol y éster de ácido graso poliinsaturado

Country Status (15)

Country Link
US (1) US10188625B2 (es)
EP (1) EP3261719B1 (es)
KR (1) KR20170122764A (es)
AR (1) AR103781A1 (es)
BR (1) BR112017017162A2 (es)
CA (1) CA2976605A1 (es)
ES (1) ES2839877T3 (es)
FR (1) FR3033135B1 (es)
MX (1) MX2017011028A (es)
PT (1) PT3261719T (es)
RU (1) RU2704109C2 (es)
TN (1) TN2017000363A1 (es)
TW (1) TW201639549A (es)
WO (1) WO2016135340A1 (es)
ZA (1) ZA201705670B (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2019068288A1 (de) 2017-10-04 2019-04-11 Berlimed International Research Gmbh Wirkstoff und wirkstoffmatrix enthaltendes produkt zur transdermalen wirkstoffabgabe sowie dessen herstellung und verwendung sowie die wirkstoffmatrix, ihre herstellung und verwendung

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5885595A (en) * 1996-05-13 1999-03-23 Elizabeth Arden Co., Division Of Conopco, Inc. Cosmetic composition with a retinol fatty acid ester
US6521237B2 (en) * 1998-11-12 2003-02-18 Johnson & Johnson Consumer Companies, Inc. Skin care composition
US20080139518A1 (en) * 2006-12-04 2008-06-12 Concert, Llc Topical compositions for treatment of skin conditions
FR2940281B1 (fr) * 2008-12-22 2011-04-01 Fabre Pierre Dermo Cosmetique Ester de diol et d'acide gras polyinsature comme agent anti-acne
FR2940907B1 (fr) * 2009-01-15 2011-03-04 Oreal Composition cosmetique ou dermatologique, comprenant un retinoide, un compose non phosphate a base d'adenosine et un polymere semi-cristallin

Also Published As

Publication number Publication date
ZA201705670B (en) 2019-03-27
BR112017017162A2 (pt) 2018-04-03
RU2017131342A3 (es) 2019-05-17
EP3261719A1 (en) 2018-01-03
KR20170122764A (ko) 2017-11-06
RU2704109C2 (ru) 2019-10-24
TW201639549A (zh) 2016-11-16
TN2017000363A1 (en) 2019-01-16
US20180036275A1 (en) 2018-02-08
PT3261719T (pt) 2021-01-05
RU2017131342A (ru) 2019-03-28
MX2017011028A (es) 2017-11-10
ES2839877T3 (es) 2021-07-06
FR3033135A1 (fr) 2016-09-02
WO2016135340A1 (en) 2016-09-01
US10188625B2 (en) 2019-01-29
FR3033135B1 (fr) 2018-03-16
EP3261719B1 (en) 2020-09-30
CA2976605A1 (en) 2016-09-01

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