[go: up one dir, main page]

AR106405A1 - MICROBIOCIDES PHENYLAMIDINE DERIVATIVES - Google Patents

MICROBIOCIDES PHENYLAMIDINE DERIVATIVES

Info

Publication number
AR106405A1
AR106405A1 ARP160103187A ARP160103187A AR106405A1 AR 106405 A1 AR106405 A1 AR 106405A1 AR P160103187 A ARP160103187 A AR P160103187A AR P160103187 A ARP160103187 A AR P160103187A AR 106405 A1 AR106405 A1 AR 106405A1
Authority
AR
Argentina
Prior art keywords
alkyl
groups
cycloalkyl
alkoxy
hydrogen
Prior art date
Application number
ARP160103187A
Other languages
Spanish (es)
Inventor
Zambach Werner
James Hoffman Thomas
Daniel Henri Gagnepain Julien
Sulzer Mosse Sarah
Weiss Matthias
Original Assignee
Syngenta Participations Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syngenta Participations Ag filed Critical Syngenta Participations Ag
Publication of AR106405A1 publication Critical patent/AR106405A1/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N37/00Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids
    • A01N37/52Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids containing groups, e.g. carboxylic acid amidines
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N51/00Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds having the sequences of atoms O—N—S, X—O—S, N—N—S, O—N—N or O-halogen, regardless of the number of bonds each atom has and with no atom of these sequences forming part of a heterocyclic ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C257/00Compounds containing carboxyl groups, the doubly-bound oxygen atom of a carboxyl group being replaced by a doubly-bound nitrogen atom, this nitrogen atom not being further bound to an oxygen atom, e.g. imino-ethers, amidines
    • C07C257/10Compounds containing carboxyl groups, the doubly-bound oxygen atom of a carboxyl group being replaced by a doubly-bound nitrogen atom, this nitrogen atom not being further bound to an oxygen atom, e.g. imino-ethers, amidines with replacement of the other oxygen atom of the carboxyl group by nitrogen atoms, e.g. amidines
    • C07C257/12Compounds containing carboxyl groups, the doubly-bound oxygen atom of a carboxyl group being replaced by a doubly-bound nitrogen atom, this nitrogen atom not being further bound to an oxygen atom, e.g. imino-ethers, amidines with replacement of the other oxygen atom of the carboxyl group by nitrogen atoms, e.g. amidines having carbon atoms of amidino groups bound to hydrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C259/00Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups
    • C07C259/04Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups without replacement of the other oxygen atom of the carboxyl group, e.g. hydroxamic acids
    • C07C259/10Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups without replacement of the other oxygen atom of the carboxyl group, e.g. hydroxamic acids having carbon atoms of hydroxamic groups bound to carbon atoms of six-membered aromatic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/48Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups having nitrogen atoms of sulfonamide groups further bound to another hetero atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Agronomy & Crop Science (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Además, se proveen composiciones agroquímicas que comprenden éstos compuestos, a la preparación de estas composiciones y al uso de los compuestos o composiciones en agricultura u horticultura para combatir, prevenir o controlar la infestación de plantas, cultivos alimentarios recolectados, semillas o materiales inertes debida a microorganismos fitopatógenos, en particular, hongos. Reivindicación 1: Un compuesto de fórmula (1), donde R¹ y R² son cada uno independientemente alquilo C₁₋₄ o cicloalquilo C₃₋₈; o R¹ y R² junto con el átomo de nitrógeno al que están unidos forman un grupo cíclico saturado de 3, 4 ó 5 miembros; R³ es hidrógeno, halógeno o alquilo C₁₋₄; R⁴ es hidrógeno, ciano, halógeno, alquilo C₁₋₄, alcoxi C₁₋₄, haloalquilo C₁₋₄ o haloalcoxi C₁₋₄; R⁵ es alquilo C₁₋₄, alquenilo C₂₋₆ o alquinilo C₂₋₆; R⁶ es arilo (opcionalmente sustituido con de uno a tres grupos R⁹), heteroarilo (opcionalmente sustituido con de uno a tres grupos R⁹) o alquilo C₁₋₄; X e Y son cada uno independientemente un enlace directo, -C(R⁷)₂-, -C(R⁷)₂A-, -C(R⁷)₂C(R⁷)₂-, -C(R⁷)₂C(R⁷)₂A-, -SO₂- o -SO₂CH₂-; cada R⁷ se selecciona independientemente entre hidrógeno, alquilo C₁₋₄, haloalquilo C₁₋₄, alcoxi C₁₋₄ o haloalcoxi C₁₋₄; o dos grupos R⁷ junto con el átomo de carbono al que están unidos forman C=O o C=S; cada A se selecciona independientemente entre O, S y NR⁸; cada R⁸ se selecciona independientemente entre hidrógeno, alquilo C₁₋₄, alcoxi C₁₋₄ y cicloalquilo C₃₋₈; y cada R⁹ se selecciona independientemente entre halógeno, ciano, hidroxilo, amino, nitro, alquilo C₁₋₄, haloalquilo C₁₋₄, cicloalquilo C₃₋₆, halocicloalquilo C₃₋₆, alcoxi C₁₋₄, haloalcoxi C₁₋₄, cicloalcoxi C₃₋₆, alquiltio C₁₋₄, haloalquiltio C₁₋₄, cicloalquiltio C₃₋₆, alquilsulfinilo C₁₋₄, haloalquilsulfinilo C₁₋₄, alquilsulfonilo C₁₋₄, haloalquilsulfonilo C₁₋₄, (alquil C₁₋₄)carbonilo, alquenilo C₂₋₆, haloalquenilo C₂₋₆, alqueniloxi C₂₋₆, haloalqueniloxi C₂₋₆, alquinilo C₂₋₆, (cicloalquil C₃₋₆)(alquinilo C₂₋₆), alquiniloxi C₂₋₆, arilo, arilalquilo, ariloxi, heteroarilo, heteroarilalquilo y heteroariloxi, donde los grupos arilo y heteroarilo están opcionalmente sustituidos con de uno a tres grupos R⁴; o una de sus sales o N-óxidos.In addition, agrochemical compositions comprising these compounds are provided for the preparation of these compositions and the use of the compounds or compositions in agriculture or horticulture to combat, prevent or control infestation of plants, harvested food crops, seeds or inert materials due to phytopathogenic microorganisms, in particular, fungi. Claim 1: A compound of formula (1), wherein R¹ and R² are each independently C₁₋₄ alkyl or C₃₋₈ cycloalkyl; or R¹ and R² together with the nitrogen atom to which they are attached form a saturated cyclic group of 3, 4 or 5 members; R³ is hydrogen, halogen or C₁₋₄ alkyl; R⁴ is hydrogen, cyano, halogen, C₁₋₄ alkyl, C₁₋₄ alkoxy, C₁₋₄ haloalkyl or C₁₋₄ haloalkoxy; R⁵ is C₁₋₄ alkyl, C₂₋₆ alkenyl or C₂₋₆ alkynyl; R⁶ is aryl (optionally substituted with one to three R⁹ groups), heteroaryl (optionally substituted with one to three R⁹ groups) or C₁₋₄ alkyl; X and Y are each independently a direct link, -C (R⁷) ₂-, -C (R⁷) ₂A-, -C (R⁷) ₂C (R⁷) ₂-, -C (R⁷) ₂C (R⁷) ₂A- , -SO₂- or -SO₂CH₂-; each R⁷ is independently selected from hydrogen, C₁₋₄ alkyl, C₁₋₄ haloalkyl, C₁₋₄ alkoxy or C₁₋₄ haloalkoxy; or two groups R⁷ together with the carbon atom to which they are attached form C = O or C = S; each A is independently selected from O, S and NR⁸; each R⁸ is independently selected from hydrogen, C₁₋₄ alkyl, C₁₋₄ alkoxy and C₃₋₈ cycloalkyl; and each R⁹ is independently selected from halogen, cyano, hydroxyl, amino, nitro, C₁₋₄ alkyl, C₁₋₄ haloalkyl, C₃₋₆ cycloalkyl, C₃₋₆ halocycloalkyl, C₁₋₄ alkoxy, C₁₋₄ haloalkoxy, C₃₋ cycloalkoxy ₆, Cilt alkylthio, C₁₋₄ haloalkylthio, C₃₋₆ cycloalkylthio, C₁₋₄ alkylsulfinyl, C₁₋₄ haloalkylsulfinyl, C₁₋₄ alkylsulfonyl, C₁₋₄ haloalkylsulfonyl, (C₁₋₄ alkyl) carbonyl, C₂₋₆ alkenyl, C₂₋₆ haloalkenyl, C₂₋₆ alkenyloxy, C₂₋₆ haloalkenyloxy, C₂₋₆ alkynyl, (C₂₋₆ cycloalkyl), C₂₋₆ alkynyloxy, aryl, arylalkyl, aryloxy, heteroaryl, heteroarylalkyl and heteroaryloxy, wherein the aryl and heteroaryl groups are optionally substituted with one to three R⁴ groups; or one of its salts or N-oxides.

ARP160103187A 2015-10-23 2016-10-19 MICROBIOCIDES PHENYLAMIDINE DERIVATIVES AR106405A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP15191177 2015-10-23

Publications (1)

Publication Number Publication Date
AR106405A1 true AR106405A1 (en) 2018-01-10

Family

ID=54360120

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP160103187A AR106405A1 (en) 2015-10-23 2016-10-19 MICROBIOCIDES PHENYLAMIDINE DERIVATIVES

Country Status (3)

Country Link
AR (1) AR106405A1 (en)
UY (1) UY36962A (en)
WO (1) WO2017067837A1 (en)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2018193385A1 (en) 2017-04-20 2018-10-25 Pi Industries Ltd. Novel phenylamine compounds
US20200148635A1 (en) 2017-05-18 2020-05-14 Pi Industries Ltd. Formimidamidine compounds useful against phytopathogenic microorganisms
WO2019202459A1 (en) 2018-04-16 2019-10-24 Pi Industries Ltd. Use of 4-substituted phenylamidine compounds for controlling disease rust diseases in plants
AR115966A1 (en) 2018-08-17 2021-03-17 Pi Industries Ltd PHENYLAMIDINE COMPOUNDS AND THEIR USES
EP3643175A1 (en) 2018-10-24 2020-04-29 Basf Se Ternary pesticidal mixtures containing metyltetraprole and fenpropimorph
TW202045008A (en) 2019-02-01 2020-12-16 印度商皮埃企業有限公司 4-substituted isoxazole/isoxazoline (hetero) arylamidine compounds, preparation and use thereof

Family Cites Families (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR8600161A (en) 1985-01-18 1986-09-23 Plant Genetic Systems Nv CHEMICAL GENE, HYBRID, INTERMEDIATE PLASMIDIO VECTORS, PROCESS TO CONTROL INSECTS IN AGRICULTURE OR HORTICULTURE, INSECTICIDE COMPOSITION, PROCESS TO TRANSFORM PLANT CELLS TO EXPRESS A PLANTINIDE TOXIN, PRODUCED BY CULTURES, UNITED BY BACILLA
CA1340685C (en) 1988-07-29 1999-07-27 Frederick Meins Dna sequences encoding polypeptides having beta-1,3-glucanase activity
US5169629A (en) 1988-11-01 1992-12-08 Mycogen Corporation Process of controlling lepidopteran pests, using bacillus thuringiensis isolate denoted b.t ps81gg
NZ231804A (en) 1988-12-19 1993-03-26 Ciba Geigy Ag Insecticidal toxin from leiurus quinquestriatus hebraeus
EP0392225B1 (en) 1989-03-24 2003-05-28 Syngenta Participations AG Disease-resistant transgenic plants
GB8910624D0 (en) 1989-05-09 1989-06-21 Ici Plc Bacterial strains
CA2015951A1 (en) 1989-05-18 1990-11-18 Mycogen Corporation Novel bacillus thuringiensis isolates active against lepidopteran pests, and genes encoding novel lepidopteran-active toxins
DE69018772T2 (en) 1989-11-07 1996-03-14 Pioneer Hi Bred Int Larvae kill lectins and plant resistance to insects based on them.
US5639949A (en) 1990-08-20 1997-06-17 Ciba-Geigy Corporation Genes for the synthesis of antipathogenic substances
UA48104C2 (en) 1991-10-04 2002-08-15 Новартіс Аг Dna fragment including sequence that codes an insecticide protein with optimization for corn, dna fragment providing directed preferable for the stem core expression of the structural gene of the plant related to it, dna fragment providing specific for the pollen expression of related to it structural gene in the plant, recombinant dna molecule, method for obtaining a coding sequence of the insecticide protein optimized for corn, method of corn plants protection at least against one pest insect
US5530195A (en) 1994-06-10 1996-06-25 Ciba-Geigy Corporation Bacillus thuringiensis gene encoding a toxin active against insects
EA001148B1 (en) 1996-03-11 2000-10-30 Новартис Аг Pyrimidin-4-one derivatives
GB9902592D0 (en) 1999-02-06 1999-03-24 Hoechst Schering Agrevo Gmbh Fungicides
WO2002015701A2 (en) 2000-08-25 2002-02-28 Syngenta Participations Ag Bacillus thuringiensis crystal protein hybrids
US7230167B2 (en) 2001-08-31 2007-06-12 Syngenta Participations Ag Modified Cry3A toxins and nucleic acid sequences coding therefor
WO2003052073A2 (en) 2001-12-17 2003-06-26 Syngenta Participations Ag Novel corn event
DE102005007160A1 (en) 2005-02-16 2006-08-24 Basf Ag Pyrazolecarboxylic acid anilides, process for their preparation and compositions containing them for controlling harmful fungi
EP1928818B1 (en) * 2005-09-13 2012-03-21 Bayer CropScience AG Pesticide benzyloxy- and phenetyl-substituted phenyl-amidine derivatives
EP1969929A1 (en) * 2007-03-12 2008-09-17 Bayer CropScience AG Substituted phenylamidines and their use as fungicides
TWI528899B (en) 2010-12-29 2016-04-11 杜邦股份有限公司 Mesoionic pesticides
US9770023B2 (en) * 2014-02-13 2017-09-26 Bayer Cropscience Aktiengesellschaft Active compound combinations comprising phenylamidine compounds and further fungicides
EP2865265A1 (en) * 2014-02-13 2015-04-29 Bayer CropScience AG Active compound combinations comprising phenylamidine compounds and biological control agents

Also Published As

Publication number Publication date
WO2017067837A1 (en) 2017-04-27
UY36962A (en) 2017-05-31

Similar Documents

Publication Publication Date Title
AR104046A1 (en) MICROBICIDE HETEROBICYCLIC DERIVATIVES
AR113865A1 (en) MICROBICIDE DERIVATIVES OF PHENYLAMIDINE
AR106405A1 (en) MICROBIOCIDES PHENYLAMIDINE DERIVATIVES
AR093828A1 (en) ACTIVE MIXTURES AS PESTICIDES, WHICH INCLUDE ANTRANILAMIDE COMPOUNDS
CR20180434A (en) MICROBIOCIDE DERIVATIVES OF TYPE (UNCLE) CARBOXAMIDE OF QUINOLINE
MX391739B (en) CONDENSED HETEROCYCLIC COMPOUND HAVING A CYCLOALKYLPYRIDIL GROUP OR A SALT THEREOF, AGRICULTURAL AND HORTICULTURAL INSECTICIDE COMPRISING THE COMPOUND, AND METHOD FOR USING THE INSECTICIDE
AR106947A1 (en) OXADIAZOLS REPLACED TO FIGHT FITOPATHOGEN FUNGI
AR106762A1 (en) OXADIAZOLS REPLACED TO FIGHT FITOPATHOGEN FUNGI
CO2018005946A2 (en) Phenylamine derivatives microbicides
AR105322A1 (en) HITEROCICLES NITROGENATED AS PESTICIDES
AR094139A1 (en) ACTIVE MIXTURES AS PESTICIDES, WHICH INCLUDE ANTRANILAMIDE COMPOUNDS
AR101201A1 (en) DERIVATIVES OF FENIL-PIRIDAZINA-DIONAS BENCILOXI SUBSTITUTED AND FENIL-PIRIDAZINONA BENCILOXI SUBSTITUTED AS HERBICIDES
AR109152A1 (en) HERBICIDE PIRIMIDINE COMPOUNDS
AR110367A1 (en) ACTIVE COMPOUND COMBINATIONS
MX2019012813A (en) Substituted succinimide derivatives as pesticides.
AR104433A1 (en) HERBICIDE COMPOUNDS
AR087528A1 (en) REPLACED CETOENOLS WITH 1,2,4-TRIAZOLIL
AR105425A1 (en) IMIDAZOL DERIVATIVES AS A PESTICIDE WITH SUBSTITUTES CONTAINING SULFUR
AR118054A1 (en) HERBICIDE COMPOUNDS
AR103088A1 (en) HERBICIDE COMPOUNDS
AR093782A1 (en) USE OF ANTRANILAMIDE COMPOUNDS TO REDUCE VIRAL INFECTIONS WHOSE VECTOR IS AN INSECT
AR101489A1 (en) REGULATING COMPOUNDS OF VEGETABLE GROWTH
AR091577A1 (en) HERBICIDE AGENTS CONTAINING FLUFENACET
AR098272A1 (en) HERBICIDE COMPOUNDS
AR096517A1 (en) DERIVATIVES OF 5-HIDROXI-2,3-DIFENYLPENTANONITRILE REPLACED, PROCEDURES FOR THEIR PREPARATION AND ITS USE AS HERBICIDES AND / OR REGULATORS OF GROWTH OF PLANTS

Legal Events

Date Code Title Description
FB Suspension of granting procedure