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AR089962A1 - Composiciones farmaceuticas oftalmicas y metodos para su elaboracion y uso - Google Patents

Composiciones farmaceuticas oftalmicas y metodos para su elaboracion y uso

Info

Publication number
AR089962A1
AR089962A1 ARP130100420A ARP130100420A AR089962A1 AR 089962 A1 AR089962 A1 AR 089962A1 AR P130100420 A ARP130100420 A AR P130100420A AR P130100420 A ARP130100420 A AR P130100420A AR 089962 A1 AR089962 A1 AR 089962A1
Authority
AR
Argentina
Prior art keywords
polymer
composition
oil
emulsion
ophthalmic pharmaceutical
Prior art date
Application number
ARP130100420A
Other languages
English (en)
Original Assignee
Bausch & Lomb
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bausch & Lomb filed Critical Bausch & Lomb
Publication of AR089962A1 publication Critical patent/AR089962A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/107Emulsions ; Emulsion preconcentrates; Micelles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/557Eicosanoids, e.g. leukotrienes or prostaglandins
    • A61K31/5575Eicosanoids, e.g. leukotrienes or prostaglandins having a cyclopentane, e.g. prostaglandin E2, prostaglandin F2-alpha
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/715Polysaccharides, i.e. having more than five saccharide radicals attached to each other by glycosidic linkages; Derivatives thereof, e.g. ethers, esters
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/74Synthetic polymeric materials
    • A61K31/765Polymers containing oxygen
    • A61K31/78Polymers containing oxygen of acrylic acid or derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/14Esters of carboxylic acids, e.g. fatty acid monoglycerides, medium-chain triglycerides, parabens or PEG fatty acid esters
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/32Macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. carbomers, poly(meth)acrylates, or polyvinyl pyrrolidone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A61K47/38Cellulose; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0048Eye, e.g. artificial tears
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/04Artificial tears; Irrigation solutions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Inorganic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Ophthalmology & Optometry (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Dispersion Chemistry (AREA)
  • Molecular Biology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Una composición farmacéutica oftálmica estable para el alivio, el tratamiento, el control, la mejoría o la prevención de una afección ocular patológica comprende: (a) un primer polímero, cuya viscosidad cambia con un cambio en una concentración de un electrólito, tal como una sal, cuando se agrega a dicho primer polímero; (b) un segundo polímero que es diferente del primer polímero y que puede modificar la viscosidad del primer polímero; y (c) un aceite. En algunas formas de realización, la composición además comprende un surfactante no iónico. La composición puede formar una emulsión estable de aceite en agua con el almacenamiento, si bien se separa en una fase de aceite y una fase de agua cuando se aplica al ojo. La emulsión puede comprender un ingrediente activo farmacéutico oftálmico disuelto en fase de aceite o de agua. La emulsión puede proporcionar mejorada estabilidad a dicho ingrediente farmacéutico activo. Reivindicación 5: La composición de la reivindicación 4, donde dicho primer polímero comprende un polímero o copolímero de monómeros de carboxivinilo, y dicho segundo polímero comprende un polisacárido polianiónico. Reivindicación 8: La composición de la reivindicación 7, donde dicho polisacárido polianiónico es seleccionado del grupo que consiste en alginato, ácido hialurónico, glucuronoxilomanano, carboximetjlcelulosa, carboxietilcelulosa, glucosaminoglicano, pectina y goma de xantano. Reivindicación 14: La composición de la reivindicación 13, donde dicho ingrediente activo farmacéutico es latanoprost.
ARP130100420A 2012-02-13 2013-02-08 Composiciones farmaceuticas oftalmicas y metodos para su elaboracion y uso AR089962A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261597879P 2012-02-13 2012-02-13
US13/739,018 US9278132B2 (en) 2012-02-13 2013-01-11 Ophthalmic pharmaceutical compositions and methods of making and using same

Publications (1)

Publication Number Publication Date
AR089962A1 true AR089962A1 (es) 2014-10-01

Family

ID=48946121

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP130100420A AR089962A1 (es) 2012-02-13 2013-02-08 Composiciones farmaceuticas oftalmicas y metodos para su elaboracion y uso

Country Status (14)

Country Link
US (1) US9278132B2 (es)
EP (1) EP2814463B1 (es)
JP (1) JP5898789B2 (es)
KR (1) KR101760990B1 (es)
CN (1) CN104203215B (es)
AR (1) AR089962A1 (es)
AU (1) AU2013219822B2 (es)
CA (1) CA2864417C (es)
ES (1) ES2576113T3 (es)
HU (1) HUE029276T2 (es)
MX (1) MX349169B (es)
PL (1) PL2814463T3 (es)
TW (1) TWI535462B (es)
WO (1) WO2013122801A1 (es)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11596599B2 (en) 2012-05-03 2023-03-07 The Johns Hopkins University Compositions and methods for ophthalmic and/or other applications
EP4008355A1 (en) 2012-05-03 2022-06-08 Kala Pharmaceuticals, Inc. Pharmaceutical nanoparticles showing improved mucosal transport
US9827191B2 (en) 2012-05-03 2017-11-28 The Johns Hopkins University Compositions and methods for ophthalmic and/or other applications
EP2844227B1 (en) 2012-05-03 2020-11-18 Kala Pharmaceuticals, Inc. Pharmaceutical nanoparticles showing improved mucosal transport
JP6537775B2 (ja) * 2014-03-10 2019-07-03 小林製薬株式会社 乳化組成物
US10245324B2 (en) 2014-10-31 2019-04-02 Johnson & Johnson Consumer Inc. Ophthalmic composition
PT3373976T (pt) 2015-11-10 2024-04-02 Sun Pharmaceutical Ind Ltd Formulações tópicas e suas utilizações
DK3423076T3 (da) 2016-02-29 2024-07-08 Sun Pharmaceutical Ind Ltd Topisk cyclosporinholdige formuleringer og anvendelser deraf
EP3231417B1 (de) * 2016-04-15 2018-12-05 Dr. Gerhard Mann Chem.-Pharm. Fabrik GmbH Lagerungsstabile, ophthalmische zusammensetzung
RU2019130955A (ru) * 2017-03-05 2021-04-07 Ресдевко Рисёрч Энд Дивелопмент Ко. Лтд. Глазные капли для лечения раздражения, не вызванного инфекцией
US10933111B2 (en) * 2019-01-08 2021-03-02 Boston Biotechnology US CORP Treating dry eye disorders
DE102021212692A1 (de) 2021-11-11 2023-05-11 Ursapharm Arzneimittel Gmbh Selbstemulgierende öl-in wasser-mikro- oder nanoemulsion so-wie emulgierende zusammensetzung

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4409205A (en) 1979-03-05 1983-10-11 Cooper Laboratories, Inc. Ophthalmic solution
US5209927A (en) 1985-01-23 1993-05-11 Alcon Laboratories, Inc. Ophthalmic solution
EP0459148B1 (en) 1990-05-29 1996-01-03 Ocular Research Of Boston Inc. Dry eye treatment composition
US5474979A (en) * 1994-05-17 1995-12-12 Allergan, Inc. Nonirritating emulsions for sensitive tissue
ES2094688B1 (es) * 1994-08-08 1997-08-01 Cusi Lab Manoemulsion del tipo de aceite en agua, util como vehiculo oftalmico y procedimiento para su preparacion.
DE69807281T2 (de) * 1997-05-14 2003-04-17 Mitsubishi Chemical Corp., Tokio/Tokyo Difluprednat enthaltende Zusammensetzungen
CN1456157A (zh) 2002-05-10 2003-11-19 刘继东 左旋氧氟沙星眼用凝胶
CN1180776C (zh) 2002-12-02 2004-12-22 刘继东 凝胶型氧氟沙星眼膏
WO2005044276A1 (ja) * 2003-11-07 2005-05-19 Senju Pharmaceutical Co., Ltd. プロスタグランジン含有医薬組成物
US9161905B2 (en) * 2005-01-12 2015-10-20 Ocular Research Of Boston, Inc. Dry eye treatment
US7288520B2 (en) * 2005-07-13 2007-10-30 Allergan, Inc. Cyclosporin compositions
EP1985298A1 (en) * 2007-04-24 2008-10-29 Azad Pharma AG Ophtalmic oil-in-water emulsions containing prostaglandins
PT2437762T (pt) 2009-06-05 2017-11-14 Allergan Inc Lágrimas artificiais e usos terapêuticos
FR2962044B1 (fr) * 2010-04-21 2013-02-22 Horus Pharma Emulsion lacrymimetique
FR2961694B1 (fr) 2010-06-29 2013-01-25 Thea Lab Systeme de delivrance polymerique d'une solution non visqueuse a base de prostaglandine sans conservateur
US8957048B2 (en) 2011-10-06 2015-02-17 Allergan, Inc. Compositions for the treatment of dry eye

Also Published As

Publication number Publication date
US20130210912A1 (en) 2013-08-15
CN104203215A (zh) 2014-12-10
JP2015507010A (ja) 2015-03-05
JP5898789B2 (ja) 2016-04-06
CA2864417A1 (en) 2013-08-22
PL2814463T3 (pl) 2016-11-30
TW201345564A (zh) 2013-11-16
US9278132B2 (en) 2016-03-08
KR20140121479A (ko) 2014-10-15
MX349169B (es) 2017-07-17
EP2814463A1 (en) 2014-12-24
AU2013219822B2 (en) 2016-01-14
CN104203215B (zh) 2017-04-12
MX2014009620A (es) 2014-11-10
HUE029276T2 (en) 2017-02-28
CA2864417C (en) 2018-10-16
KR101760990B1 (ko) 2017-07-24
AU2013219822A1 (en) 2014-08-28
TWI535462B (zh) 2016-06-01
EP2814463B1 (en) 2016-05-18
ES2576113T3 (es) 2016-07-05
WO2013122801A1 (en) 2013-08-22

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