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AR089887A1 - PIRIMIDINE FUNGICIDE COMPOUNDS - Google Patents

PIRIMIDINE FUNGICIDE COMPOUNDS

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Publication number
AR089887A1
AR089887A1 ARP130100331A AR089887A1 AR 089887 A1 AR089887 A1 AR 089887A1 AR P130100331 A ARP130100331 A AR P130100331A AR 089887 A1 AR089887 A1 AR 089887A1
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Argentina
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alkyl
alkoxy
haloalkoxy
haloalkyl
alkynyl
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Spanish (es)
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Basf Se
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Publication of AR089887A1 publication Critical patent/AR089887A1/en

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

Uso y métodos para combatir los hongos fitopatogénicos. Las semillas tratadas al menos con un compuesto de este tipo. Procedimientos para preparar los compuestos de fórmula (1) y composiciones agroquímicas. Reivindicación 1: Compuestos de fórmula (1) en donde: Rᵃ² es halógeno, CN, NO₂, OH, SH, alquilo C₁₋₄, haloalquilo C₁₋₄, alcoxi C₁₋₄, haloalcoxi C₁₋₄, alquiltio C₁₋₄, haloalquiltio C₁₋₄, alquilsulfinilo C₁₋₄, haloalquilsulfinilo C₁₋₄, alquilsulfonilo C₁₋₄, haloalquilsulfonilo C₁₋₄, alcoxi C₁₋₄-alquilo C₁₋₄, alcoxi C₁₋₄-alcoxi C₁₋₄, alquenilo C₂₋₄-, alquinilo C₂₋₄, haloalquenilo C₂₋₄-, haloalquinilo C₂₋₄-, cicloalquilo C₃₋₈, cicloalquiloxi C₃₋₈, cicloalquil C₃₋₈-alquilo C₁₋₄, NRARB, C(=O)R, C(=NOR)R o -C(=NH)-O-R; RA, RB independientemente uno de otro son hidrógeno, alquilo C₁₋₄, alquenilo C₂₋₄, alquinilo C₂₋₄, fenilo, bencilo, cicloalquilo C₃₋₈, cicloalquenilo C₃₋₈ o C(=O)-R; R es hidrógeno, OH, NH₂, alquilo C₁₋₄-, haloalquilo C₁₋₄-, alquenilo C₂₋₄-, alquinilo C₂₋₄-, alcoxi C₁₋₄-, haloalcoxi C₁₋₄-, alquilamino C₁₋₄- o di(alquil C₁₋₄-)amino; R es hidrógeno, alquilo C₁₋₄-, haloalquilo C₁₋₄-, alquenilo C₂₋₄-, alquinilo C₂₋₄- o alcoxi C₁₋₄-alquilo C₁₋₄; R es hidrógeno o alquilo C₁₋₄; Rᵃ⁵, Rᵃ⁶ independientemente uno de otro, son hidrógeno, CN, NH₂, OH, SH, alquilo C₁₋₄, haloalquilo C₁₋₄, alcoxi C₁₋₄, haloalcoxi C₁₋₄, alquiltio C₁₋₄-, haloalquiltio C₁₋₄, alquilsulfinilo C₁₋₄, haloalquilsulfinilo C₁₋₄, alquilsulfonilo C₁₋₄-, haloalquilsulfonilo C₁₋₄, alcoxi C₁₋₄-alquilo C₁₋₄, alcoxi C₁₋₄-alcoxi C₁₋₄-, alquenilo C₁₋₄, alquinilo C₁₋₄, haloalquenilo C₂₋₄-, haloalquinilo C₂₋₄, cicloalquilo C₂₋₄, cicloalquiloxi C₃₋₈, cicloalquil C₃₋₈-alquilo C₁₋₄, NRARB, C(=O)R, C(=NOR)R o C(=NH)-O-R; R es hidrógeno, alquilo C₁₋₄, haloalquilo C₁₋₄, alcoxi C₁₋₄, haloalcoxi C₁₋₄, alcoxi C₁₋₄-alquilo C₁₋₄, haloalcoxi C₁₋₄-alquilo C₁₋₄, alquenilo C₂₋₄, haloalquenilo C₂₋₄, alquinilo C₂₋₄, haloalquinilo C₂₋₄, CN, CH₂CN, NRARB o CH₂-O-C(=O)R; R¹, R² independientemente uno de otro son hidrógeno, halógeno, CN, OH, alquilo C₁₋₄, haloalquilo C₁₋₄, alcoxi C₁₋₄, haloalcoxi C₁₋₄, alcoxi C₁₋₄-alquilo C₁₋₄, haloalcoxi C₁₋₄-alquilo C₁₋₄, alquenilo C₂₋₄, haloalquenilo C₂₋₄, alquinilo C₂₋₄, haloalquinilo C₂₋₄, cicloalquilo C₃₋₈-, cicloalquil C₃₋₈-alquilo C₁₋₄, cicloalquiloxi C₃₋₈, NRARB, C(=O)R, C(=NOR)R, -C(=NH)-O-R o bencilo en donde el resto fenilo de bencilo está no sustituido o transporta 1, 2, 3, 4, ó 5 sustituyentes seleccionados del grupo que consiste en CN, halógeno, alquilo C₁₋₄, haloalquilo C₁₋₄, alcoxi C₁₋₄, haloalcoxi C₁₋₄, (alcoxi C₁₋₄)carbonilo y di(alquilo C₁₋₄)aminocarbonilo, o dos radicales R¹ y R² que están unidos al mismo átomos de carbono forman juntos con dicho átomo de carbono un carbociclo saturado o parcialmente insaturado de 3, 4, 5, 6 ó 7-miembros o un heterociclo saturado o parcialmente insaturado de 3, 4, 5, 6 ó 7-miembros, en donde los átomos del miembro del anillo del heterociclo antes mencionado incluyen además de los átomos de carbono 1, 2, 3 ó 4 heteroátomos seleccionados del grupo de N, O y S, y en donde el ciclo antes mencionado está no sustituido o transporta 1, 2, 3 ó 4 sustituyentes seleccionados de halógeno, CN, OH, SH, alquilo C₁₋₄-, alcoxi C₁₋₄ o alquiltio C₁₋₄; y uno o dos grupos CH₂ de los ciclos antes mencionados pueden ser reemplazados por uno o dos grupos C(=O) o C(=S) respectivamente; X es un grupo divalente seleccionado de -CR³R⁴-, -C(=O)-, -C(=S)-, -C(=NRD)- y -C(=NORD)-, en donde RD es hidrógeno o alquilo C₁₋₄-, y en donde R³ y R⁴ independientemente uno de otro son hidrógeno, hidrógeno, CN, hidroxialquilo C₁₋₄, haloalquilo C₁₋₄, alcoxi C₁₋₄, haloalcoxi C₁₋₄, alcoxi C₁₋₄-alquilo C₁₋₄, haloalcoxi C₁₋₄-alquilo C₁₋₄, alquenilo C₂₋₄, haloalquenilo C₂₋₄, alquinilo C₂₋₄, haloalquinilo C₂₋₄, cicloalquilo C₃₋₈-, cicloalcoxi C₃₋₈, cicloalquil C₁₋₄-alquilo-C₃₋₈, NRARB, C(=O)R, C(=NOR)R, C(=NH)-O-R o bencilo, en donde el resto fenilo de bencilo está no sustituido o transporta 1, 2, 3, 4, ó 5 sustituyentes seleccionados del grupo que consiste en CN, halógeno, alquilo C₁₋₄, haloalquilo C₁₋₄, alcoxi C₁₋₄, haloalcoxi C₁₋₄, (alcoxi C₁₋₄-)carbonilo y di(alquil C₁₋₄)aminocarbonilo, o dos radicales R³ y R⁴ que están unidos al mismo átomos de carbono forman juntos con dicho átomo de carbono un carbociclo saturado o parcialmente insaturado de 3, 4, 5, 6 ó 7-miembros o un heterociclo saturado o parcialmente insaturado de 3, 4, 5, 6 ó 7-miembros, en donde los átomos del miembro del anillo del heterociclo antes mencionado incluyen además de los átomos de carbono 1, 2, 3 ó 4 heteroátomos seleccionados del grupo de N, O y S, y en donde el ciclo antes mencionado está no sustituido o transporta 1, 2, 3 ó 4 sustituyentes seleccionados de halógeno, CN, OH, SH, alquilo C₁₋₄-, alcoxi C₁₋₄ o alquiltio C₁₋₄; y uno o dos grupos CH₂ de los ciclos antes mencionados pueden ser reemplazados por uno o dos grupos C(=O) o C(=S) respectivamente; n indica el número de sustituyentes Rᵇ en el anillo fenilo y n es 0, 1, 2, 3 ó 4; Rᵇ es halógeno, CN, NO₂, alquilo C₁₋₄-, haloalquilo C₁₋₄-, alcoxi C₁₋₄-, haloalcoxi C₁₋₄-, alquenilo C₂₋₄-, haloalquenilo C₂₋₄-, alquinilo C₂₋₄-, haloalquinilo C₂₋₄-, NRARB, C(=NOR)R o C(=NH)-O-R, siendo posible para n = 2, 3, ó 4 que Rᵇ sean idénticos o diferentes; m indica el número de sustituyentes Rᶜ en el anillo fenilo y n es 0, 1, ó 2; Rᶜ es halógeno, CN, NO₂, NH₂, alquilo C₁₋₆-, haloalquilo C₁₋₆-, alcoxi C₁₋₆-, haloalcoxi C₁₋₆-, alquilamino C₁₋₆-, di(alquil C₁₋₆-)amino, alquiltio C₁₋₆-, haloalquiltio C₁₋₆-, alquilsulfinilo C₁₋₆-, haloalquilsulfinilo C₁₋₆-, alquilsulfonilo C₁₋₆-, haloalquilsulfonilo C₁₋₆-, alcoxi C₁₋₆-alquilo-C₁₋₄-, haloalcoxi C₁₋₆-alquilo-C₁₋₄-, alquenilo C₂₋₆-, alquinilo C₂₋₆-, C(=O)R, C(=NOR)R, cicloalquilo C₃₋₈-, cicloalquil C₃₋₈-alquilo C₁₋₄, fenilo, fenoxi, fenoxi-alquilo C₁₋₄ o un heteroarilo de 5 ó 6 miembros, en donde los átomos del miembro del anillo del heteroarilo incluyen además de átomos de carbono 1, 2, 3 ó 4 heteroátomos seleccionados del grupo de N, O y S, y en donde los radicales cíclicos antes mencionados están no sustituidos o transportan 1, 2, 3 ó 4 sustituyentes Rᵈ idénticos o diferentes: Rᵈ es halógeno, CN, alquilo C₁₋₄-, haloalquilo C₁₋₄-, alcoxi C₁₋₄- o haloalcoxi C₁₋₄-; o dos radicales Rᶜ que están unidos a los átomos del miembro del anillo adyacente del grupo piridinilo forman junto con dichos átomos del miembro del anillo un carbociclo o heterociclo fusionado de 5, 6, ó 7 miembros sUse and methods to combat phytopathogenic fungi. Seeds treated with at least one such compound. Procedures for preparing the compounds of formula (1) and agrochemical compositions. Claim 1: Compounds of formula (1) wherein: Rᵃ² is halogen, CN, NO₂, OH, SH, C alquilo alkyl, C₁₋₄ haloalkyl, C₁₋₄ alkoxy, C₁₋₄ haloalkoxy, C₁₋₄ alkylthio, haloalkylthio C₁₋₄, C₁₋₄ alkylsulfinyl, C₁₋₄ haloalkylsulfinyl, C₁₋₄ alkylsulfonyl, C₁₋₄ haloalkylsulfonyl, C₁₋₄ alkoxyC₁₋₄ alkyl, C₁₋₄ alkoxyC₁₋₄ alkoxy, C₂₋₄ alkenyl, C₂₋₄ alkynyl, C₂₋₄- haloalkenyl, C₂₋₄- haloalkynyl, C₃₋₈ cycloalkyl, C₃₋₈ cycloalkyloxy, C₃₋₈ cycloalkyl-C alquilo alkyl, NRARB, C (= O) R, C (= NOR ) R or -C (= NH) -OR; RA, RB independently of each other are hydrogen, C₁₋₄ alkyl, C₂₋₄ alkenyl, C₂₋₄ alkynyl, phenyl, benzyl, C₃₋₈ cycloalkyl, C₃₋₈ or C (= O) -R cycloalkenyl; R is hydrogen, OH, NH₂, C₁₋₄- alkyl, C₁₋₄- haloalkyl, C₂₋₄- alkenyl, C₂₋₄- alkynyl, C₁₋₄- alkoxy, C₁₋₄- haloalkoxy, C₁₋₄- alkylamino di (C₁₋₄-) alkyl; R is hydrogen, C₁₋₄- alkyl, C₁₋₄- haloalkyl, C₂₋₄- alkenyl, C₂₋₄- alkynyl or C₁₋₄ alkoxy-C₁₋₄ alkyl; R is hydrogen or C₁₋₄ alkyl; Rᵃ⁵, Rᵃ⁶ independently of each other, are hydrogen, CN, NH₂, OH, SH, C₁₋₄ alkyl, C₁₋₄ haloalkyl, C₁₋₄ alkoxy, C₁₋₄ haloalkoxy, C₁₋₄- alkylthio, C₁₋₄ haloalkylthio, C₁₋₄ alkylsulfinyl, C₁₋₄ haloalkylsulfinyl, C₁₋₄- alkylsulfonyl, C₁₋₄ haloalkylsulfonyl, C₁₋₄ alkoxyC₁₋₄ alkyl, C₁₋₄ alkoxyC₁₋₄- alkoxy, C₁₋₄ alkenyl, C₁₋ alkynyl ₄, C₂₋₄- haloalkenyl, C₂₋₄ haloalkynyl, C₂₋₄ cycloalkyl, C₃₋₈ cycloalkyloxy, C₁₋₄ cycloalkyl, NRARB, C (= O) R, C (= NOR) R or C (= NH) -OR; R is hydrogen, C₁₋₄ alkyl, C₁₋₄ haloalkyl, C₁₋₄ alkoxy, C₁₋₄ haloalkoxy, C₁₋₄ alkoxy-C₁₋₄ alkyl, C₁₋₄ haloalkoxy-C₁₋₄ alkyl, C₂₋₄ alkenyl, haloalkenyl C₂₋₄, C₂₋₄ alkynyl, C₂₋₄ haloalkynyl, CN, CH₂CN, NRARB or CH₂-OC (= O) R; R¹, R² independently of each other are hydrogen, halogen, CN, OH, C₁₋₄ alkyl, C₁₋₄ haloalkyl, C₁₋₄ alkoxy, C₁₋₄ haloalkoxy, C₁₋₄ alkoxy-C₁₋₄ alkyl, C₁₋₄ haloalkoxy -C₁₋₄ alkyl, C₂₋₄ alkenyl, C₂₋₄ haloalkenyl, C₂₋₄ alkynyl, C₂₋₄ haloalkynyl, C₃₋₈ cycloalkyl, C₃₋₈ cycloalkyl-C₁₋₄ alkyl, C₃₋₈ cycloalkyloxy, NRARB, C (= O) R, C (= NOR) R, -C (= NH) -OR or benzyl where the phenyl benzyl moiety is unsubstituted or carries 1, 2, 3, 4, or 5 substituents selected from the group that It consists of CN, halogen, C₁₋₄ alkyl, C₁₋₄ haloalkyl, C₁₋₄ alkoxy, C₁₋₄ haloalkoxy, (C₁₋₄ alkoxy) carbonyl and di (C₁₋₄ alkyl) aminocarbonyl, or two radicals R¹ and R² which are attached to the same carbon atoms together with said carbon atom a saturated or partially unsaturated carbocycle of 3, 4, 5, 6 or 7-members or a heterocycle sa cured or partially unsaturated of 3, 4, 5, 6 or 7-members, wherein the atoms of the ring member of the above-mentioned heterocycle include in addition to the carbon atoms 1, 2, 3 or 4 heteroatoms selected from the group of N, O and S, and wherein the above-mentioned cycle is unsubstituted or transports 1, 2, 3 or 4 substituents selected from halogen, CN, OH, SH, C₁₋₄- alkyl, C₁₋₄ alkoxy or C₁₋₄ alkylthio; and one or two CH₂ groups of the aforementioned cycles may be replaced by one or two groups C (= O) or C (= S) respectively; X is a divalent group selected from -CR³R⁴-, -C (= O) -, -C (= S) -, -C (= NRD) - and -C (= NORD) -, where RD is hydrogen or alkyl C₁₋₄-, and where R³ and R⁴ independently of each other are hydrogen, hydrogen, CN, C₁₋₄ hydroxyalkyl, C₁₋₄ haloalkyl, C₁₋₄ alkoxy, C₁₋₄ haloalkoxy, C₁₋₄ alkoxy-C₁₋ alkyl ₄, C₁₋₄ haloalkoxy-C₁₋₄ alkyl, C₂₋₄ alkenyl, C₂₋₄ haloalkenyl, C₂₋₄ alkynyl, C₂₋₄ haloalkynyl, C₃₋₈- cycloalkyl, C₃₋₈ cycloalkoxy, C₁₋₄-alkylcycloalkyl- C₃₋₈, NRARB, C (= O) R, C (= NOR) R, C (= NH) -OR or benzyl, wherein the benzyl phenyl moiety is unsubstituted or transports 1, 2, 3, 4, or 5 substituents selected from the group consisting of CN, halogen, C₁₋₄ alkyl, C₁₋₄ haloalkyl, C₁₋₄ alkoxy, C₁₋₄ haloalkoxy, (C₁₋₄-) alkoxycarbonyl and di (C₁₋₄ alkyl) aminocarbonyl , or two radicals R³ and R⁴ that are attached to it together with said carbon atom together with a carbon atom a saturated or partially unsaturated carbocycle of 3, 4, 5, 6 or 7-members or a saturated or partially unsaturated heterocycle of 3, 4, 5, 6 or 7-members, wherein the atoms of the heterocycle ring member mentioned above include in addition to carbon atoms 1, 2, 3 or 4 heteroatoms selected from the group of N, O and S, and wherein the above-mentioned cycle is unsubstituted or transports 1, 2 , 3 or 4 substituents selected from halogen, CN, OH, SH, C₁₋₄- alkyl, C₁₋₄ alkoxy or C₁₋₄ alkylthio; and one or two CH₂ groups of the aforementioned cycles may be replaced by one or two groups C (= O) or C (= S) respectively; n indicates the number of substituents Rᵇ in the phenyl ring and n is 0, 1, 2, 3 or 4; Rᵇ is halogen, CN, NO₂, C₁₋₄- alkyl, C₁₋₄- haloalkyl, C₁₋₄- alkoxy, C₁₋₄- haloalkoxy, C₂₋₄- alkenyl, C₂₋₄- haloalkenyl, C₂₋₄- alkynyl, haloalkynyl C₂₋₄-, NRARB, C (= NOR) R or C (= NH) -OR, it being possible for n = 2, 3, or 4 that Rᵇ be identical or different; m indicates the number of substituents Rᶜ in the phenyl ring and n is 0, 1, or 2; Rᶜ is halogen, CN, NO₂, NH₂, C₁₋₆- alkyl, C₁₋₆- haloalkyl, C₁₋₆- alkoxy, C₁₋₆- haloalkoxy, C₁₋₆- alkylamino, di (C₁₋₆-) alkyl, C₁₋₆- alkylthio, C₁₋₆- haloalkylthio, C₁₋₆- alkylsulfinyl, C₁₋₆- haloalkylsulfinyl, C₁₋₆- alkylsulfonyl, C₁₋₆- haloalkylsulfonyl, C₁₋₆-C - alkoxy, C₁ haloalkoxy ₋₆-C₁₋₄-alkyl, C₂₋₆- alkenyl, C₂₋₆- alkynyl, C (= O) R, C (= NOR) R, C₃₋₈- cycloalkyl, C₃₋₈-cycloalkyl-C₁₋ alkyl ₄, phenyl, phenoxy, phenoxy-C₁₋₄ alkyl or a 5- or 6-membered heteroaryl, wherein the atoms of the heteroaryl ring member include in addition to carbon atoms 1, 2, 3 or 4 heteroatoms selected from the group of N , O and S, and wherein the aforementioned cyclic radicals are unsubstituted or carry 1, 2, 3 or 4 identical or different Rᵈ substituents: Rᵈ is halogen, CN, C₁₋₄- alkyl , C₁₋₄- haloalkyl, C₁₋₄- alkoxy or C₁₋₄- haloalkoxy; or two radicals Rᶜ which are attached to the atoms of the adjacent ring member of the pyridinyl group together with said atoms of the ring member a fused carbocycle or heterocycle of 5, 6, or 7 members s

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* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2913325B1 (en) * 2012-10-25 2021-04-21 Shenyang Sinochem Agrochemicals R & D Co., Ltd. Substituted pyrimidine compound and uses thereof
JP2016179944A (en) * 2013-08-09 2016-10-13 石原産業株式会社 Difluoromethylene compound
JP2017001954A (en) * 2013-11-08 2017-01-05 石原産業株式会社 Nitrogen-containing saturated heterocyclic compound
CN105753791B (en) * 2014-12-19 2019-09-13 沈阳中化农药化工研发有限公司 Substituted uracil compound and application thereof
EP3593637B1 (en) * 2018-07-11 2023-09-06 Fine Agrochemicals Limited Plant growth regulator concentrate and use thereof

Family Cites Families (100)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3325503A (en) 1965-02-18 1967-06-13 Diamond Alkali Co Polychloro derivatives of mono- and dicyano pyridines and a method for their preparation
US3296272A (en) 1965-04-01 1967-01-03 Dow Chemical Co Sulfinyl- and sulfonylpyridines
JPS54115388A (en) 1978-03-01 1979-09-07 Nippon Chemiphar Co Ltd Acetic acid derivative and its preparation
GB2059955A (en) 1979-09-13 1981-04-29 Merck & Co Inc Process for preparing methylvanillyl ketone
DE3338292A1 (en) 1983-10-21 1985-05-02 Basf Ag, 6700 Ludwigshafen 7-AMINO-AZOLO (1,5-A) -PYRIMIDINE AND FUNGICIDES CONTAINING THEM
CA1249832A (en) 1984-02-03 1989-02-07 Shionogi & Co., Ltd. Azolyl cycloalkanol derivatives and agricultural fungicides
DE3545319A1 (en) 1985-12-20 1987-06-25 Basf Ag ACRYLIC ACID ESTERS AND FUNGICIDES THAT CONTAIN THESE COMPOUNDS
CN1015981B (en) 1986-05-02 1992-03-25 施托福化学公司 The preparation method of pyridyl imidate
DE256503T1 (en) 1986-08-12 1990-02-08 Mitsubishi Kasei Corp., Tokio/Tokyo PYRIDINE CARBOXAMIDE DERIVATIVES AND THEIR USE AS A FUNGICIDAL AGENT.
US4895849A (en) 1986-10-08 1990-01-23 Ube Industries, Ltd. Aralkylaminopyrimidine compounds which are useful as for producing thereof and insecticides
AU628229B2 (en) 1989-11-10 1992-09-10 Agro-Kanesho Co. Ltd. Hexahydrotriazine compounds and insecticides
JP2828186B2 (en) 1991-09-13 1998-11-25 宇部興産株式会社 Acrylate-based compounds, their preparation and fungicides
US5439911A (en) 1992-12-28 1995-08-08 Shionogi & Co., Ltd. Aminopyrimidine derivatives and their production and use
WO1995018795A1 (en) 1994-01-07 1995-07-13 Dowelanco N-(4-pyrimidinyl)amide pesticides
EP0665225B1 (en) 1994-02-01 1996-11-27 Ube Industries, Ltd. 4-Phenethylamino pyrimidine derivative, process for preparing the same and agricultural and horticultural chemical for controlling noxious organisms containing the same
DE19518073A1 (en) 1995-05-17 1996-11-21 Hoechst Ag Substituted benzyloxycarbonylguanidines, process for their preparation, their use as a medicament or diagnostic agent and medicament containing them
DE19603576A1 (en) 1996-02-01 1997-08-07 Bayer Ag Acylated 4-amino and 4-hydrazinopyrimidines
JPH1036355A (en) 1996-07-19 1998-02-10 Ube Ind Ltd Method for producing 4-amino-5-chloro-6- (1-fluoroethyl) pyrimidine derivative
DE19650197A1 (en) 1996-12-04 1998-06-10 Bayer Ag 3-thiocarbamoylpyrazole derivatives
TW460476B (en) 1997-04-14 2001-10-21 American Cyanamid Co Fungicidal trifluoromethylalkylamino-triazolopyrimidines
NZ503594A (en) 1997-09-18 2001-08-31 Basf Ag (Phenyl, thienyl or pyrazolyl)-substituted and alkyl-substituted benzamidoxime derivatives, and benzonitrile intermediates, useful as fungicides
DE19750012A1 (en) 1997-11-12 1999-05-20 Bayer Ag Isothiazole carboxamides
AU1621799A (en) 1997-12-04 1999-06-16 Dow Agrosciences Llc Fungicidal compositions and methods, and compounds and methods for the preparation thereof
AU2006201959B2 (en) 1997-12-22 2008-09-04 Bayer Healthcare Llc Inhibition of Raf Kinase using Substituted Heterocyclic Ureas
AU755538B2 (en) 1998-11-17 2002-12-12 Ihara Chemical Industry Co. Ltd. Pyrimidinylbenzimidazole and triazinylbenzimidazole derivatives and agricultural/horticultural fungicides
IT1303800B1 (en) 1998-11-30 2001-02-23 Isagro Ricerca Srl DIPEPTID COMPOUNDS HAVING HIGH FUNGICIDE AND AGRICULTURAL USE.
JP3417862B2 (en) 1999-02-02 2003-06-16 新東工業株式会社 Silica gel highly loaded with titanium oxide photocatalyst and method for producing the same
AU770077B2 (en) 1999-03-11 2004-02-12 Dow Agrosciences Llc Heterocyclic substituted isoxazolidines and their use as fungicides
US6586617B1 (en) 1999-04-28 2003-07-01 Sumitomo Chemical Takeda Agro Company, Limited Sulfonamide derivatives
UA73307C2 (en) 1999-08-05 2005-07-15 Куміаі Кемікал Індастрі Ко., Лтд. Carbamate derivative and fungicide of agricultural/horticultural destination
DE10021412A1 (en) 1999-12-13 2001-06-21 Bayer Ag Fungicidal active ingredient combinations
DK1250047T3 (en) 2000-01-25 2005-05-30 Syngenta Participations Ag Herbicide agent
US6376548B1 (en) 2000-01-28 2002-04-23 Rohm And Haas Company Enhanced propertied pesticides
IL167957A (en) 2000-02-04 2009-07-20 Sumitomo Chemical Co Hydroxypyridine compound
MXPA03002338A (en) 2000-09-18 2003-09-10 Du Pont Pyridinyl amides and imides for use as fungicides.
NZ525744A (en) 2000-11-17 2004-10-29 Dow Agrosciences Llc Compounds having fungicidal activity and processes to make and use same
JP5034142B2 (en) 2001-04-20 2012-09-26 住友化学株式会社 Plant disease control composition
DE10136065A1 (en) 2001-07-25 2003-02-13 Bayer Cropscience Ag pyrazolylcarboxanilides
AR037228A1 (en) 2001-07-30 2004-11-03 Dow Agrosciences Llc ACID COMPOUNDS 6- (ARIL OR HETEROARIL) -4-AMYNOPYCOLINIC, HERBICIDE COMPOSITION THAT UNDERSTANDS AND METHOD TO CONTROL UNWANTED VEGETATION
FR2828196A1 (en) 2001-08-03 2003-02-07 Aventis Cropscience Sa New iodochromone derivatives, useful for the prevention or cure of plant fungal disorders, especially in cereals, vines, fruits, legumes or ornamental plants
JPWO2003016286A1 (en) 2001-08-17 2004-12-02 三共アグロ株式会社 3-phenoxy-4-pyridazinol derivative and herbicidal composition containing the same
WO2003053145A1 (en) 2001-12-21 2003-07-03 Nissan Chemical Industries, Ltd. Bactericidal composition
TWI327462B (en) 2002-01-18 2010-07-21 Sumitomo Chemical Co Condensed heterocyclic sulfonyl urea compound, a herbicide containing the same, and a method for weed control using the same
US20030166476A1 (en) 2002-01-31 2003-09-04 Winemiller Mark D. Lubricating oil compositions with improved friction properties
DE10204390A1 (en) 2002-02-04 2003-08-14 Bayer Cropscience Ag Disubstituted thiazolylcarboxanilides
HK1079785B (en) 2002-03-05 2007-08-10 辛根塔参与股份公司 O-cyclopropyl-carboxanilides and their use as fungicides
GB0227966D0 (en) 2002-11-29 2003-01-08 Syngenta Participations Ag Organic Compounds
WO2004083193A1 (en) 2003-03-17 2004-09-30 Sumitomo Chemical Company, Limited Amide compound and bactericide composition containing the same
JP2007524626A (en) 2003-06-25 2007-08-30 エラン ファーマシューティカルズ，インコーポレイテッド Methods and compositions for treating rheumatoid arthritis
MXPA06001320A (en) 2003-08-01 2006-05-04 Pfizer Prod Inc 6-menbered heteroaryl compounds for the treatment of neurodegenerative disorders.
US7501538B2 (en) 2003-08-08 2009-03-10 Transtech Pharma, Inc. Aryl and heteroaryl compounds, compositions and methods of use
TWI355894B (en) 2003-12-19 2012-01-11 Du Pont Herbicidal pyrimidines
HRP20100538T1 (en) 2004-03-10 2010-12-31 Basf Se 5,6-dialkyl-7-amino-triazolopyrimidines, method for their production, their use for controlling pathogenic fungi and agents containing said compounds
JP2007527886A (en) 2004-03-10 2007-10-04 ビーエーエスエフ　アクチェンゲゼルシャフト 5,6-Dialkyl-7-aminotriazolopyrimidines, their preparation, and their use for controlling harmful fungi, and compositions containing these compounds
AU2005227997A1 (en) 2004-03-30 2005-10-13 Arena Pharmaceuticals, Inc. Pyrimidine derivatives and methods of treatment related to the use thereof
US7459562B2 (en) 2004-04-23 2008-12-02 Bristol-Myers Squibb Company Monocyclic heterocycles as kinase inhibitors
WO2005120234A2 (en) 2004-06-03 2005-12-22 E.I. Dupont De Nemours And Company Fungicidal mixtures of amidinylphenyl compounds
EP1761498A1 (en) 2004-06-18 2007-03-14 Basf Aktiengesellschaft 1-methyl-3-difluoromethyl-pyrazol-4-carbonic acid-(ortho-phenyl)-anilides, and use thereof as a fungicide
ATE458722T1 (en) 2004-06-18 2010-03-15 Basf Se 1-METHYL-3-TRIFLUORMETHYL-PYRAZOLE-4-CARBONIC ACID (ORTHO-PHENYL) ANILIDES AND THEIR USE AS A FUNGICIDE
GB0418048D0 (en) 2004-08-12 2004-09-15 Syngenta Participations Ag Method for protecting useful plants or plant propagation material
AP2007004061A0 (en) 2005-01-10 2007-08-31 Galloway & Company Pyrrolopyrazoles, potent kinase inhibitors
CA2593439C (en) 2005-01-14 2014-02-25 F. Hoffmann-La Roche Ag Thiazole-4-carboxamide derivatives as mglur5 antagonists
DE102005007160A1 (en) 2005-02-16 2006-08-24 Basf Ag Pyrazolecarboxylic acid anilides, process for their preparation and compositions containing them for controlling harmful fungi
WO2006087325A1 (en) 2005-02-16 2006-08-24 Basf Aktiengesellschaft 5-alkoxyalkyl-6-alkyl-7-amino-azolopyrimidines, method for their production, their use for controlling pathogenic fungi and agents containing said substances
DE102005009458A1 (en) 2005-03-02 2006-09-07 Bayer Cropscience Ag pyrazolylcarboxanilides
KR20070113267A (en) 2005-03-09 2007-11-28 쉐링 코포레이션 Compound for inhibiting PSP kinesin activity
US20070021435A1 (en) 2005-06-10 2007-01-25 Gaul Michael D Aminopyrimidines as kinase modulators
GB0513841D0 (en) 2005-07-07 2005-08-10 Medivir Ab Cysteine protease inhibitors
GB0516705D0 (en) 2005-08-15 2005-09-21 Syngenta Participations Ag Process
DK1917253T3 (en) 2005-08-15 2015-03-30 Boehringer Ingelheim Int Method of Preparation of Beta Mimetics
EP1937691A1 (en) 2005-10-21 2008-07-02 Dow Agrosciences LLC Thieno-pyrimidine compounds having fungicidal activity
TWI382974B (en) 2005-12-20 2013-01-21 英塞特公司 N-hydroxymethyl hydrazine heterocyclic compound as a guanamine 2,3-dioxygenase modulator
PL1973881T3 (en) 2006-01-13 2010-04-30 Dow Agrosciences Llc 6-(poly-substituted aryl)-4-aminopicolinates and their use as herbicides
EP1983832A2 (en) 2006-02-09 2008-10-29 Syngeta Participations AG A method of protecting a plant propagation material, a plant, and/or plant organs
CA2643670A1 (en) 2006-02-27 2007-08-30 Sterix Limited Diaryl compounds as non-steroidal inhibitors of 17-beta hydroxysteroid dehydrogenase and/or steroid sulphatase for the treatment of oestrogen-related diseases such as hormone dependent breast cancer
MX2009002781A (en) 2006-09-15 2009-03-30 Reviva Pharmaceuticals Inc Synthesis, methods of using, and compositions of cycloalkylmethylamines.
US8779154B2 (en) 2006-09-26 2014-07-15 Qinglin Che Fused ring compounds for inflammation and immune-related uses
WO2008039882A1 (en) 2006-09-30 2008-04-03 Sanofi-Aventis U.S. Llc A combination of niacin and a prostaglandin d2 receptor antagonist
ES2302447B1 (en) 2006-10-20 2009-06-12 Laboratorios Almirall S.A. DERIVATIVES OF 4- (2-AMINO-1-HYDROXYETHYL) Phenol as agonists of the BETA2 ADRENERGIC RECEIVER.
TW200831488A (en) 2006-11-29 2008-08-01 Astrazeneca Ab Novel compounds
PE20081559A1 (en) 2007-01-12 2008-11-20 Merck & Co Inc SPIROCHROMANONE DERIVATIVES SUBSTITUTED AS ACETYL COA CARBOXYLASE INHIBITORS
CN101679406B (en) 2007-04-10 2013-07-10 百时美施贵宝公司 Thiazolyl compounds useful as kinase inhibitors
JP5478488B2 (en) 2007-06-20 2014-04-23 メルク・シャープ・アンド・ドーム・コーポレーション JANUS kinase inhibitors
HUE026195T2 (en) 2008-01-22 2016-05-30 Dow Agrosciences Llc 4-amino-5-fluoro-pyrimidine derivatives as fungicides
KR101638326B1 (en) 2008-06-24 2016-07-12 사노피 Substituted isoquinolines and isoquinolinones as Rho kinase inhibitors
DE102008040168A1 (en) 2008-07-04 2010-01-07 Robert Bosch Gmbh Solenoid valve for a fuel injector and fuel injector
US20100068197A1 (en) 2008-07-11 2010-03-18 Myriad Pharmaceuticals, Inc. Pharmaceutical compounds as inhibitors of cell proliferation and the use thereof
WO2010025451A2 (en) 2008-08-29 2010-03-04 Dow Agrosciences Llc 5,8-difluoro-4-(2-(4-(heteroaryloxy)-phenyl)ethylamino)quinazolines and their use as agrochemicals
AP2011005613A0 (en) 2008-09-11 2011-04-30 Pfizer Heteroaryls amide derivatives and their use as glucokinase activators.
TW201024281A (en) 2008-11-24 2010-07-01 Boehringer Ingelheim Int New compounds
EP2210890A1 (en) 2009-01-19 2010-07-28 Almirall, S.A. Oxadiazole derivatives as S1P1 receptor agonists
JP5420761B2 (en) 2009-05-28 2014-02-19 ノバルティス アーゲー Substituted aminopropionic acid derivatives as neprilysin inhibitors
US8461164B2 (en) 2009-08-31 2013-06-11 Dow Agrosciences, Llc. Pteridines and their use as agrochemicals
BR112012008044A2 (en) 2009-08-31 2019-09-24 Dow Agrosciences Llc pteridines and their use as agrochemicals
MX2012002579A (en) 2009-09-01 2012-07-23 Dow Agrosciences Llc Synergistic fungicidal compositions containing a 5-fluoropyrimidine derivative for fungal control in cereals.
US20110230465A1 (en) 2009-09-18 2011-09-22 Boehringer Ingleheim International Gmbh Viral polymerase inhibitors
WO2011053835A1 (en) 2009-10-30 2011-05-05 Aton Pharma, Inc. Stereoselective synthesis of metyrosine
EP2533783B8 (en) 2010-01-13 2015-12-16 Tempero Pharmaceuticals, Inc. COMPOUNDS AND METHODS for the inhibition of HDAC
WO2011100285A1 (en) 2010-02-10 2011-08-18 Lexicon Pharmaceuticals, Inc. Tryptophan hydroxylase inhibitors for the treatment of metastatic bone disease
CN102260263A (en) 2010-05-26 2011-11-30 四川大学 Diphenylamine purine derivatives, and preparation method and medicinal application thereof

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