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AR087609A1 - Microbiocidas - Google Patents

Microbiocidas

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Publication number
AR087609A1
AR087609A1 ARP120103063A AR087609A1 AR 087609 A1 AR087609 A1 AR 087609A1 AR P120103063 A ARP120103063 A AR P120103063A AR 087609 A1 AR087609 A1 AR 087609A1
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AR
Argentina
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alkyl
independently selected
heterocycle
adjacent
halogen
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Syngenta Participations Ag
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    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
    • A01N43/40—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
    • A01N43/40—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
    • A01N43/42—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings condensed with carbocyclic rings
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/713—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with four or more nitrogen atoms as the only ring hetero atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/44—Radicals substituted by doubly-bound oxygen, sulfur, or nitrogen atoms, or by two such atoms singly-bound to the same carbon atom
    • C07D213/53—Nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/54—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/55—Acids; Esters
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/61—Halogen atoms or nitro radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/84—Nitriles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/89—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members with hetero atoms directly attached to the ring nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/20—Oxygen atoms
    • C07D215/24—Oxygen atoms attached in position 8
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/38—Nitrogen atoms
    • C07D215/40—Nitrogen atoms attached in position 8
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Dentistry (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Reivindicación 1: Un método para aplicar a plantas útiles, al emplazamiento de estas o a su material de propagación un compuesto de fórmula (1) donde L¹ es N o C-D¹; L² es N o C-D²; L³ es N o C-D³; L⁴ es N o C-D⁴; L⁵ es N o C-D⁵; L⁶ es N o C-D⁶; D¹, D², D³, D⁴, D⁵ y D⁶ independientemente de los demás, representan hidrógeno, halógeno, CN, NO₂, alquilo C₁₋₈, cicloalquilo C₃₋₈, alquenilo C₂₋₈, alquinilo C₂₋₈, fenilo, un heterociclo de 5 ó 6 miembros que contiene de uno a cuatro heteroátomos seleccionados independientemente entre O, S y N, siempre que el heterociclo no contenga átomos de oxígeno adyacentes, átomos de azufre adyacentes ni átomos de azufre y oxígeno adyacentes, COR¹, OR², SH, alquiltio C₁₋₈, alquilsulfinilo C₁₋₈, alquilsulfonilo C₁₋₈, feniltio, fenilsulfinilo, fenilsulfonilo, N(R³)₂, CO₂R², O(CO)R¹, CON(R³)₂, NR³COR¹, CR¹N-OR², donde el alquilo, cicloalquilo, alquenilo, alquinilo, fenilo y heterociclo están opcionalmente sustituidos con uno o más grupos seleccionados independientemente entre halógeno, CN, NH₂, NO₂, OR², alquilo C₁₋₄ y haloalquilo C₁₋₄; o D¹ y D⁵, D² y D⁵, D³ y D⁶ o D⁴ y D6, independientemente del otro, junto con el fragmento al que están enlazados, pueden formar un anillo carbocíclico de 5 a 7 miembros parcial o completamente insaturado o un anillo heterocíclico de 5 a 7 miembros parcial o completamente insaturado que contiene de uno a tres heteroátomos seleccionados independientemente entre O, S, N y N(R³), siempre que el heterociclo no contenga átomos de oxígeno adyacentes, átomos de azufre adyacentes ni átomos de oxígeno y azufre adyacentes, y donde el anillo formado por D¹ y D⁵, D² y D⁵, D³ y D⁶ o D⁴ y D⁶ está opcionalmente sustituido con uno o más grupos seleccionados independientemente entre halógeno, CN, NH₂, NO₂, OH, alquilo C₁₋₄, haloalquilo C₁₋₄, alcoxi C₁₋₄ y haloalcoxi C₁₋₄; X representa los restos de fórmula X-2, X-3, X-4 ó X-5; Z¹, Z², Z³, Z⁵, Z⁶, Z⁷, Z⁸, Z⁹, Z¹⁰, Z¹¹, Z¹³ y Z¹⁴, independientemente de los demás, representan CR⁴R⁵, C=O o C=CR⁶R⁷; Z⁴ y Z¹² representan CR⁸R⁹, SiR¹⁰R¹¹, C=O o C=CR⁶R⁷; donde las agrupaciones de fórmula X-2, X-3, X-4 y X-5 contienen como máximo un anillo que contiene solamente uno de los radicales Z¹ - Z¹⁴, dos de los radicales Z¹ - Z¹⁴, tres de los radicales Z¹ - Z¹⁴ o cuatro de los radicales de Z¹ - Z¹⁴ como miembros del anillo; y donde ninguno de Z¹, Z², Z³, Z⁴, Z⁵, Z⁶, Z⁷, Z⁸, Z⁹, Z¹⁰, Z¹¹, Z¹², Z¹³ y Z¹⁴ representa un átomo de carbono sustituido con dos OH; Q se selecciona del grupo compuesto por los compuestos de fórmula Q-1, Q-2, Q-3, Q-4, Q-5, Q-6, Q-7, Q-8 y Q-9; cada Y¹, Y², Y³ e Y⁴, independientemente de los demás, representan hidrógeno, halógeno, CN, NO₂, alquilo C₁₋₈, cicloalquilo C₃₋₈, alquenilo C₂₋₈, alquinilo C₂₋₈, bencilo, fenilo, un heterociclo de 5 ó 6 miembros que contiene de uno a tres heteroátomos seleccionados independientemente entre O, S y N, siempre que el heterociclo no contenga átomos de oxígeno adyacentes, átomos de azufre adyacentes ni átomos de azufre y oxígeno adyacentes, COR¹, OR², SH, alquiltio C₁₋₈, alquilsulfinilo C₁₋₈, alquilsulfonilo C₁₋₈, feniltio, fenilsulfinilo, fenilsulfonilo, N(R³)₂, CO₂R², O(CO)R¹, CON(R³)₂, NR³COR¹, CR¹N-OR², donde el alquilo, cicloalquilo, alquenilo, alquinilo, bencilo, fenilo y heterociclo están opcionalmente sustituidos con uno o más grupos seleccionados independientemente entre halógeno, CN, NH₂, NO₂, OR², alquilo C₁₋₄ y haloalquilo C₁₋₄; cuando Q sea el resto de fórmula Q-1, Q-2, Q-3, Q-4, Q-6 ó Q-7, entonces Y¹ e Y², Y² e Y³, o Y³ e Y⁴, independientemente del otro, junto con el fragmento al que están enlazados, podrán formar un anillo carbocíclico de 5 a 7 miembros parcial o completamente insaturado o un anillo heterocíclico de 5 a 7 miembros parcial o completamente insaturado que contiene de uno a tres heteroátomos seleccionados independientemente entre O, S, N y N(R³), siempre que el heterociclo no contenga átomos de oxígeno adyacentes, átomos de azufre adyacentes ni átomos de oxígeno y azufre adyacentes, y donde el anillo formado por Y¹ e Y², Y² e Y³, o Y³ e Y⁴ está opcionalmente sustituido con uno o más grupos seleccionados independientemente entre halógeno, CN, NH₂, NO₂, OH, alquilo C₁₋₄, haloalquilo C₁₋₄, alcoxi C₁₋₄, haloalcoxi C₁₋₄ y alquiltio C₁₋₄; cuando Q sea un resto de fórmula Q-1, Q-3, Q-4, Q-7 ó Q-8 y L¹ sea C-D¹, entonces Y¹ y D¹, junto con el fragmento al que están enlazados, podrán formar un anillo carbocíclico de 5 a 7 miembros parcial o completamente insaturado o un anillo heterocíclico de 5 a 7 miembros parcial o completamente insaturado que contiene uno o dos heteroátomos seleccionados independientemente entre O, S, N y N(R³), siempre que el heterociclo no contenga átomos de oxígeno adyacentes, átomos de azufre adyacentes ni átomos de oxígeno y azufre adyacentes, y donde el anillo formado por D¹ e Y¹ está opcionalmente sustituido con uno o más grupos seleccionados independientemente entre halógeno, CN, NH₂, NO₂, OH, alquilo C₁₋₄, haloalquilo C₁₋₄, alcoxi C₁₋₄, haloalcoxi C₁₋₄ y alquiltio C₁₋₄; cuando Q sea el resto de fórmula Q-9 y L¹ sea C-D¹, entonces R¹² y D¹ juntos podrán ser -(G¹)ₚ-G²-G³-; Q se selecciona del grupo compuesto por los restos de fórmulas Q-1, Q-2, Q-3, Q-4, Q-5, Q-6, Q-7, Q-8 y Q-9; cada Y¹, Y², Y³ e Y⁴, independientemente de los demás, representan hidrógeno, halógeno, CN, NO₂, alquilo C₁₋₈, cicloalquilo C₃₋₈, alquenilo C₂₋₈, alquinilo C₂₋₈, bencilo, fenilo, un heterociclo de 5 ó 6 miembros que contiene de uno a tres heteroátomos seleccionados independientemente entre O, S y N, siempre que el heterociclo no contenga átomos de oxígeno adyacentes, átomos de azufre adyacentes ni átomos de azufre y oxígeno adyacentes, COR¹, OR², SH, alquiltio C₁₋₈, alquilsulfinilo C₁₋₈, alquilsulfonilo C₁₋₈, feniltio, fenilsulfinilo, fenilsulfonilo, N(R³)₂, CO₂R², O(CO)R¹, CON(R³)₂, NR³COR¹, CR¹N-OR², donde el alquilo, cicloalquilo, alquenilo, alquinilo, bencilo, fenilo y heterociclo están opcionalmente sustituidos con uno o más grupos seleccionados independientemente entre halógeno, CN, NH₂, NO₂, OR², alquilo C₁₋₄ y haloalquilo C₁₋₄; cuando Q sea un compuesto de fórmula Q-1, Q-2, Q-3, Q-4, Q-6 ó Q-7, entonces Y¹ e Y², Y² e Y³, o Y³ e Y⁴, independientemente del otro, junto con el fragmento al que están enlazados, podrán formar un anillo carbocíclico de 5 a 7 miembros parcial o completamente insaturado o un anillo heterocíclico de 5 a 7 miembros parcial o completamente insaturado que contiene de uno a tres heteroátomos seleccionados independientemente entre O, S, N y N(R³), siempre que el heterociclo no contenga átomos de oxígeno adyacentes, átomos de azufre adyacentes ni átomos de oxígeno y azufre adyacentes, y donde el anillo formado por Y¹ e Y², Y² e Y³, o Y³ e Y⁴ está opcionalmente sustituido con uno o más grupos seleccionados independientemente entre halógeno, CN, NH₂, NO₂, OH, alquilo C₁₋₄, haloalquilo C₁₋₄, alcoxi C₁₋₄, haloalcoxi C₁₋₄ y alquiltio C₁₋₄; cuando Q sea un resto de fórmula Q-1, Q-3, Q-4, Q-7 ó Q-8 y L⁴ sea C-D⁴, entonces Y¹ y D⁴, junto con el fragmento al que están enlazados, podrán formar un anillo carbocíclico de 5 a 7 miembros parcial o completamente insaturado o un anillo heterocíclico de 5 a 7 miembros parcial o completamente insaturado que contiene uno o dos heteroátomos seleccionados independientemente entre O, S, N y N(R³), siempre que el heterociclo no contenga átomos de oxígeno adyacentes, átomos de azufre adyacentes ni átomos de oxígeno y azufre adyacentes, y donde el anillo formado por D⁴ e Y¹ está opcionalmente sustituido con uno o más grupos seleccionados independientemente entre halógeno, CN, NH₂, NO₂, OH, alquilo C₁₋₄, haloalquilo C₁₋₄, alcoxi C₁₋₄, haloalcoxi C₁₋₄ y alquiltio C₁₋₄; cuando Q sea el compuesto de fórmula Q-9 y L⁴ sea C-D⁴, entonces R¹² y D⁴ juntos podrán ser -(G¹)ₚ-G²-G³-; cada G¹ y G², independientemente de los demás, representan -C(R¹⁴R¹⁵)-; cada G³, independientemente de los demás, representa -C(R¹⁴R¹⁵)-, O, N(R¹⁶) o S; o cada combinación de G¹ y G², o G² y G³, o G¹ y G¹, independientemente unas de otras, pueden representar juntos -CR¹⁴=CR¹⁵-; cada p, independientemente de los demás, representa 0, 1 ó 2; cada R¹, independientemente de los demás, representa hidrógeno, alquilo C₁&#
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