AR086744A1 - HETEROCICLIC COMPOUND CONTAINING NITROGEN AND FUNGICIDE FOR USE IN AGRICULTURE AND GARDENING - Google Patents
HETEROCICLIC COMPOUND CONTAINING NITROGEN AND FUNGICIDE FOR USE IN AGRICULTURE AND GARDENINGInfo
- Publication number
- AR086744A1 AR086744A1 ARP120102265A AR086744A1 AR 086744 A1 AR086744 A1 AR 086744A1 AR P120102265 A ARP120102265 A AR P120102265A AR 086744 A1 AR086744 A1 AR 086744A1
- Authority
- AR
- Argentina
- Prior art keywords
- substituted
- unsubstituted
- alkyl
- heterocyclyl
- alkynyl
- Prior art date
Links
- 229910052757 nitrogen Inorganic materials 0.000 title abstract 5
- IJGRMHOSHXDMSA-UHFFFAOYSA-N Atomic nitrogen Chemical compound N#N IJGRMHOSHXDMSA-UHFFFAOYSA-N 0.000 title abstract 4
- 230000000855 fungicidal effect Effects 0.000 title abstract 3
- 239000000417 fungicide Substances 0.000 title abstract 3
- 238000010413 gardening Methods 0.000 title abstract 3
- 150000001875 compounds Chemical class 0.000 title 1
- 125000004209 (C1-C8) alkyl group Chemical group 0.000 abstract 11
- 125000000623 heterocyclic group Chemical group 0.000 abstract 9
- 125000003342 alkenyl group Chemical group 0.000 abstract 7
- 125000000392 cycloalkenyl group Chemical group 0.000 abstract 7
- 125000006552 (C3-C8) cycloalkyl group Chemical group 0.000 abstract 6
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 6
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 abstract 6
- 125000002252 acyl group Chemical group 0.000 abstract 5
- 125000000304 alkynyl group Chemical group 0.000 abstract 5
- 125000003917 carbamoyl group Chemical group [H]N([H])C(*)=O 0.000 abstract 5
- 125000003178 carboxy group Chemical group [H]OC(*)=O 0.000 abstract 5
- 125000000472 sulfonyl group Chemical group *S(*)(=O)=O 0.000 abstract 5
- 125000003396 thiol group Chemical class [H]S* 0.000 abstract 4
- 125000000041 C6-C10 aryl group Chemical group 0.000 abstract 3
- 125000004122 cyclic group Chemical group 0.000 abstract 3
- 125000000753 cycloalkyl group Chemical group 0.000 abstract 3
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 3
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 3
- 125000004649 C2-C8 alkynyl group Chemical group 0.000 abstract 2
- 125000003118 aryl group Chemical group 0.000 abstract 2
- 125000004093 cyano group Chemical group *C#N 0.000 abstract 2
- 229910052736 halogen Inorganic materials 0.000 abstract 2
- 150000002367 halogens Chemical class 0.000 abstract 2
- 125000004433 nitrogen atom Chemical group N* 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
- MYMOFIZGZYHOMD-UHFFFAOYSA-N Dioxygen Chemical group O=O MYMOFIZGZYHOMD-UHFFFAOYSA-N 0.000 abstract 1
- 125000004429 atom Chemical group 0.000 abstract 1
- 229910052799 carbon Inorganic materials 0.000 abstract 1
- 125000004432 carbon atom Chemical group C* 0.000 abstract 1
- 150000002391 heterocyclic compounds Chemical class 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 150000002829 nitrogen Chemical group 0.000 abstract 1
- -1 nitrogen-containing heterocyclic compound Chemical class 0.000 abstract 1
- 229910052760 oxygen Inorganic materials 0.000 abstract 1
- 239000001301 oxygen Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/20—Oxygen atoms
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
- A01N43/40—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
- A01N43/42—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings condensed with carbocyclic rings
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/60—1,4-Diazines; Hydrogenated 1,4-diazines
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
Landscapes
- Life Sciences & Earth Sciences (AREA)
- Wood Science & Technology (AREA)
- Environmental Sciences (AREA)
- Plant Pathology (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Dentistry (AREA)
- Pest Control & Pesticides (AREA)
- General Health & Medical Sciences (AREA)
- Zoology (AREA)
- Agronomy & Crop Science (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Plural Heterocyclic Compounds (AREA)
- Quinoline Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
Se proporciona un fungicida para el uso en agricultura y jardinería que tiene una buena eficiencia y seguridad, y un compuesto heterocíclico conteniendo nitrógeno o una sal del mismo que es útil como principio activo de un fungicida para el uso en agricultura y jardinería. Reivindicación 1: Un compuesto heterocíclico conteniendo nitrógeno que presenta la fórmula (1) o una sal del mismo. (En la fórmula (1), R representa OR¹, NR¹R², SR¹, S(=O)R³, SO₂R³, S(=O)(=NR⁴)R⁵, N=S(=O)R⁴R⁵ o nitro; R¹ representa un átomo de hidrógeno, alquilo C₁₋₈ sin sustituir o sustituido, alquenilo C₂₋₈ sin sustituir o sustituido, alquinilo C₂₋₈ sin sustituir o sustituido, cicloalquilo C₃₋₈ sin sustituir o sustituido, cicloalquenilo C₄₋₈ sin sustituir o sustituido, arilo C₆₋₁₀ sin sustituir o sustituido, heterociclilo sin sustituir o sustituido, acilo C₁₋₈ sin sustituir o sustituido, carboxilo sin sustituir o sustituido, carbamoilo sin sustituir o sustituido, sulfonilo sustituido, o amino sin sustituir o sustituido. R² representa un átomo de hidrógeno, alquilo C₁₋₈ sin sustituir o sustituido, alquenilo C₂₋₈ sin sustituir o sustituido, alquinilo C₂₋₈ sin sustituir o sustituido, cicloalquilo C₃₋₈ sin sustituir o sustituido, cicloalquenilo C₄₋₈ sin sustituir o sustituido, arilo C₆₋₁₀ sin sustituir o sustituido, heterociclilo sin sustituir o sustituido, acilo C₁₋₈ sin sustituir o sustituido, carboxilo sin sustituir o sustituido, carbamoilo sin sustituir o sustituido, sulfonilo sustituido, hidroxi sin sustituir o sustituido, o amino sin sustituir o sustituido. R³ representa alquilo C₁₋₈ sin sustituir o sustituido, alquenilo C₂₋₈ sin sustituir o sustituido, alquinilo C₂₋₈ sin sustituir o sustituido, cicloalquilo C₃₋₈ sin sustituir o sustituido, cicloalquenilo C₄₋₈ sin sustituir o sustituido, arilo C₆₋₁₀ sin sustituir o sustituido, heterociclilo sin sustituir o sustituido, mercapto sin sustituir o sustituido, hidroxi sin sustituir o sustituido, o amino sin sustituir o sustituido. R⁴ y R⁵ representan, independientemente entre sí, alquilo C₁₋₈ sin sustituir o sustituido, alquenilo C₂₋₈ sin sustituir o sustituido, alquinilo C₂₋₈ sin sustituir o sustituido, cicloalquilo C₃₋₈ sin sustituir o sustituido, cicloalquenilo C₄₋₈ sin sustituir o sustituido, arilo C₆₋₁₀ sin sustituir o sustituido, o heterociclilo sin sustituir o sustituido. En el grupo NR¹R², el conjunto de R¹ y R² puede formar cíclilo de 3 - 8 miembros sin sustituir o sustituido, =CRᵃRᵇ o =NRᶜ. Rᵃ y Rᵇ representan, independientemente entre sí, un átomo de hidrógeno, alquilo C₁₋₈ sin sustituir o sustituido, alquenilo C₂₋₈ sin sustituir o sustituido, alquinilo C₂₋₈ sin sustituir o sustituido, cicloalquilo C₃₋₈ sin sustituir o sustituido, cicloalquenilo C₄₋₈ sin sustituir o sustituido, arilo C₆₋₁₀ sin sustituir o sustituido, heterociclilo sin sustituir o sustituido, acilo C₁₋₈ sin sustituir o sustituido, carboxilo sin sustituir o sustituido, carbamoilo sin sustituir o sustituido, sulfonilo sustituido, mercapto sin sustituir o sustituido, hidroxilo sin sustituir o sustituido, o amino sin sustituir o sustituido. Rᶜ representa hidroxilo sin sustituir o sustituido, o alquilo C₁₋₈ sin sustituir o sustituido. En el grupo N=S(=O)R⁴R⁵, el conjunto de R⁴ y R⁵ puede formar cíclilo de 5 - 8 miembros sin sustituir o sustituido. X¹ representa, independientemente entre sí, alquilo C₁₋₈ sin sustituir o sustituido, alquenilo C₂₋₈ sin sustituir o sustituido, alquinilo C₂₋₈ sin sustituir o sustituido, cicloalquilo C₃₋₈ sin sustituir o sustituido, cicloalquenilo C₄₋₈ sin sustituir o sustituido, arilo C₆₋₁₀ sin sustituir o sustituido, heterociclilo sin sustituir o sustituido, acilo C₁₋₈ sin sustituir o sustituido, (1-imino) alquilo C₁₋₈ sin sustituir o sustituido, carboxilo sin sustituir o sustituido, carbamoilo sin sustituir o sustituido, hidroxilo sin sustituir o sustituido, amino sin sustituir o sustituido, mercapto sin sustituir o sustituido, sulfonilo sustituido, halógeno, ciano o nitro. m representa el número de X¹ y un número entero de 0 a 5. B representa un átomo de carbono o de nitrógeno. D representa hidrocarburo cíclico de 5 - 7 miembros sin sustituir o sustituido con X¹ o heterociclilo de 5 - 7 miembros sin sustituir o sustituido con X¹. X² representa, independientemente entre sí, alquilo C₁₋₈ sin sustituir o sustituido, alquenilo C₂₋₈ sin sustituir o sustituido, alquinilo C₂₋₈ sin sustituir o sustituido, cicloalquilo C₃₋₈ sin sustituir o sustituido, cicloalquenilo C₄₋₈ sin sustituir o sustituido, arilo C₆₋₁₀ sin sustituir o sustituido, heterociclilo sin sustituir o sustituido, acilo C₁₋₈ sin sustituir o sustituido, (1-imino) alquilo C₁₋₈ sin sustituir o sustituido, carboxilo sin sustituir o sustituido, carbamoilo sin sustituir o sustituido, hidroxilo sin sustituir o sustituido, amino sin sustituir o sustituido, mercapto sin sustituir o sustituido, sulfonilo sustituido, halógeno, ciano o nitro. n representa el número de X² y un número entero de 0 a 3. El conjunto de uno de X² y R puede formar cíclilo de 5 - 8 miembros sin sustituir o sustituido. E representa hidrocarburo cíclico de 5 - 7 miembros sin sustituir o sustituido con X² o heterociclilo de 5 - 7 miembros sin sustituir o sustituido con X². X representa un átomo de oxígeno o de nitrógeno, o un átomo de nitrógeno sustituido con alquilo C₁₋₈).A fungicide is provided for use in agriculture and gardening that has good efficiency and safety, and a heterocyclic compound containing nitrogen or a salt thereof that is useful as an active principle of a fungicide for use in agriculture and gardening. Claim 1: A nitrogen-containing heterocyclic compound having the formula (1) or a salt thereof. (In formula (1), R represents OR¹, NR¹R², SR¹, S (= O) R³, SO₂R³, S (= O) (= NR⁴) R⁵, N = S (= O) R⁴R⁵ or nitro; R¹ represents a hydrogen atom, unsubstituted or substituted C₁₋₈ alkyl, unsubstituted or substituted Cque alkenyl, unsubstituted or substituted C₂₋₈ alkynyl, unsubstituted or substituted C₃₋₈ cycloalkyl, unsubstituted or substituted C₄₋₈ cycloalkenyl, aryl Unsubstituted or substituted C₆₋₁₀, unsubstituted or substituted heterocyclyl, unsubstituted or substituted C₁₋₈ acyl, unsubstituted or substituted carboxyl, unsubstituted or substituted carbamoyl, substituted sulfonyl, or unsubstituted or substituted amino.R² represents an atom of hydrogen, unsubstituted or substituted C₁₋₈ alkyl, unsubstituted or substituted C alkenyl, unsubstituted or substituted Cin alkynyl, unsubstituted or substituted C₃₋₈ cycloalkyl, unsubstituted or substituted C ciclo cycloalkenyl, C₆₋ aryl ₁₀ no substitute tuir or substituted, unsubstituted or substituted heterocyclyl, unsubstituted or substituted C₁₋₈ acyl, unsubstituted or substituted carboxyl, unsubstituted or substituted carbamoyl, substituted sulfonyl, unsubstituted or substituted hydroxy, or unsubstituted or substituted amino. R³ represents unsubstituted or substituted C₁₋₈ alkyl, unsubstituted or substituted C alkenyl, unsubstituted or substituted C sustitu alkynyl, unsubstituted or substituted C₃₋₈ cycloalkyl, unsubstituted or substituted C₄₋₈ cycloalkenyl, C₆₋ aryl ₁₀ unsubstituted or substituted, unsubstituted or substituted heterocyclyl, unsubstituted or substituted mercapto, unsubstituted or substituted hydroxy, or unsubstituted or substituted amino. R⁴ and R⁵ represent, independently of each other, unsubstituted or substituted C₁₋₈ alkyl, unsubstituted or substituted Cque alkenyl, unsubstituted or substituted Cin alkynyl, unsubstituted or substituted C₃₋₈ cycloalkyl, C₄₋₈ cycloalkenyl without substituted or substituted, unsubstituted or substituted C₆₋₁₀ aryl, or unsubstituted or substituted heterocyclyl. In the NR¹R² group, the set of R¹ and R² can form 3-8 unsubstituted or substituted cyclyl, = CRᵃRᵇ or = NRᶜ. Rᵃ and Rᵇ represent, independently of each other, a hydrogen atom, unsubstituted or substituted C₁₋₈ alkyl, unsubstituted or substituted Cque alkenyl, unsubstituted or substituted Cin alkynyl, unsubstituted or substituted C ciclo cycloalkyl, C sustituir unsubstituted or substituted cycloalkenyl, unsubstituted or substituted Cilo aryl, unsubstituted or substituted heterocyclyl, unsubstituted or substituted C₁₋₈ acyl, unsubstituted or substituted carboxyl, unsubstituted or substituted carbamoyl, substituted sulfonyl, mercapto without substituted or substituted, unsubstituted or substituted hydroxyl, or unsubstituted or substituted amino. Rᶜ represents unsubstituted or substituted hydroxyl, or unsubstituted or substituted C₁₋₈ alkyl. In the group N = S (= O) R⁴R⁵, the set of R⁴ and R⁵ can form 5-8 membered cyclyl unsubstituted or substituted. X¹ represents, independently of each other, unsubstituted or substituted C₁₋₈ alkyl, unsubstituted or substituted Cque alkenyl, unsubstituted or substituted Cin alkynyl, unsubstituted or substituted C₃₋₈ cycloalkyl, unsubstituted or substituted Cal cycloalkenyl substituted, unsubstituted or substituted C₆₋₁₀ aryl, unsubstituted or substituted heterocyclyl, unsubstituted or substituted C₁₋₈ acyl, (1-imino) unsubstituted or substituted C₁₋₈ alkyl, unsubstituted or substituted carboxyl, unsubstituted carbamoyl or substituted, unsubstituted or substituted hydroxyl, unsubstituted or substituted amino, unsubstituted or substituted mercapto, substituted sulfonyl, halogen, cyano or nitro. m represents the number of X¹ and an integer from 0 to 5. B represents a carbon or nitrogen atom. D represents 5-7 membered cyclic hydrocarbon unsubstituted or substituted with X¹ or 5-7 membered heterocyclyl unsubstituted or substituted with X¹. X² represents, independently of each other, unsubstituted or substituted C₁₋₈ alkyl, unsubstituted or substituted Cque alkenyl, unsubstituted or substituted C₂₋₈ alkynyl, unsubstituted or substituted C₃₋₈ cycloalkyl, unsubstituted or substituted C₄₋₈ cycloalkenyl substituted, unsubstituted or substituted C₆₋₁₀ aryl, unsubstituted or substituted heterocyclyl, unsubstituted or substituted C₁₋₈ acyl, (1-imino) unsubstituted or substituted C₁₋₈ alkyl, unsubstituted or substituted carboxyl, unsubstituted carbamoyl or substituted, unsubstituted or substituted hydroxyl, unsubstituted or substituted amino, unsubstituted or substituted mercapto, substituted sulfonyl, halogen, cyano or nitro. n represents the number of X² and an integer from 0 to 3. The set of one of X² and R can form 5-8 membered cyclyl unsubstituted or substituted. E represents 5-7 membered cyclic hydrocarbon unsubstituted or substituted with X² or 5-7 membered heterocyclyl unsubstituted or substituted with X². X represents an oxygen or nitrogen atom, or a nitrogen atom substituted with C₁₋₈ alkyl).
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2011143479 | 2011-06-28 | ||
| JP2012006279 | 2012-01-16 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR086744A1 true AR086744A1 (en) | 2014-01-22 |
Family
ID=47424097
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP120102265 AR086744A1 (en) | 2011-06-28 | 2012-06-25 | HETEROCICLIC COMPOUND CONTAINING NITROGEN AND FUNGICIDE FOR USE IN AGRICULTURE AND GARDENING |
Country Status (4)
| Country | Link |
|---|---|
| JP (1) | JP5753583B2 (en) |
| AR (1) | AR086744A1 (en) |
| TW (1) | TW201304681A (en) |
| WO (1) | WO2013002205A1 (en) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR106515A1 (en) | 2015-10-29 | 2018-01-24 | Bayer Cropscience Ag | SILISPHENOXYHETEROCICLES, TRISUSTITUTED AND ANALOG |
| TWI782983B (en) * | 2017-04-27 | 2022-11-11 | 德商拜耳廠股份有限公司 | Heteroarylphenylaminoquinolines and analogues |
| CN110582484A (en) | 2017-05-03 | 2019-12-17 | 拜耳公司 | Trisubstituted silylmethylphenoxyquinolines and their analogues |
| JP2020518592A (en) | 2017-05-03 | 2020-06-25 | バイエル・アクチエンゲゼルシヤフト | Trisubstituted silylheteroaryloxyquinolines and analogs |
| TW201927768A (en) | 2017-12-21 | 2019-07-16 | 德商拜耳廠股份有限公司 | Trisubstitutedsilylmethylheteroaryloxyquinolines and analogues |
| WO2021209490A1 (en) | 2020-04-16 | 2021-10-21 | Bayer Aktiengesellschaft | Cyclaminephenylaminoquinolines as fungicides |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3666814A (en) * | 1970-03-03 | 1972-05-30 | Delta W Gier | Chloronitrophenyl ethers as herbicides |
| JPS6097964A (en) * | 1983-11-02 | 1985-05-31 | Nissan Chem Ind Ltd | N-quinoxalinylaniline compound, its production and fungicidal, insecticidal and miticidal agent for agricultural and horticultural use |
| ZA864580B (en) * | 1985-06-20 | 1988-02-24 | Du Pont | Herbicidal aryloxybenzeneacetic acid derivatives |
| PT86297B (en) * | 1986-12-05 | 1990-11-07 | Du Pont | PROCESS FOR THE PREPARATION OF DERIVATIVES OF ARYLOXIBENZENOACETIC ACID AND HERBICIDAL COMPOSITIONS CONTAINING THEM |
| BR9609001A (en) * | 1995-06-20 | 1999-06-29 | Du Pont | Method for controlling arthropods composed of fungicidal composition and method for controlling plant diseases |
| WO1998023155A1 (en) * | 1996-11-26 | 1998-06-04 | E.I. Du Pont De Nemours And Company | Arthropodicidal and fungicidal cyclic amides |
| BR9917036A (en) * | 1999-02-09 | 2002-07-30 | Dimensional Pharm Inc | Heteroaryl amidines, methylamidines and guanidines as protease inhibitors |
| DE10013318A1 (en) * | 2000-03-17 | 2001-09-20 | Merck Patent Gmbh | Quinoxaline derivatives are used as photo-stable UV filters in cosmetic or pharmaceutical sunscreens for the hair or skin |
| US7470712B2 (en) * | 2004-01-21 | 2008-12-30 | Bristol-Myers Squibb Company | Amino-benzazoles as P2Y1 receptor inhibitors |
| BRPI0615613A2 (en) * | 2005-09-01 | 2009-05-19 | Hoffmann La Roche | diaminopyrimidines as p2x3 and p3x2 / 3 modulators |
| GB0707704D0 (en) * | 2007-04-20 | 2007-05-30 | Glaxo Group Ltd | Compounds |
| EP1990342A1 (en) * | 2007-05-10 | 2008-11-12 | AEterna Zentaris GmbH | Pyridopyrazine Derivatives, Process of Manufacturing and Uses thereof |
| WO2009017838A2 (en) * | 2007-08-01 | 2009-02-05 | Exelixis, Inc. | Combinations of jak-2 inhibitors and other agents |
-
2012
- 2012-06-25 AR ARP120102265 patent/AR086744A1/en not_active Application Discontinuation
- 2012-06-26 WO PCT/JP2012/066240 patent/WO2013002205A1/en not_active Ceased
- 2012-06-26 TW TW101122765A patent/TW201304681A/en unknown
- 2012-06-26 JP JP2013522864A patent/JP5753583B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| WO2013002205A1 (en) | 2013-01-03 |
| JPWO2013002205A1 (en) | 2015-02-23 |
| JP5753583B2 (en) | 2015-07-22 |
| TW201304681A (en) | 2013-02-01 |
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