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AR060926A1 - Solucion anestesica transparente de propofol, con baja irritacion venosa. - Google Patents

Solucion anestesica transparente de propofol, con baja irritacion venosa.

Info

Publication number
AR060926A1
AR060926A1 ARP070102080A ARP070102080A AR060926A1 AR 060926 A1 AR060926 A1 AR 060926A1 AR P070102080 A ARP070102080 A AR P070102080A AR P070102080 A ARP070102080 A AR P070102080A AR 060926 A1 AR060926 A1 AR 060926A1
Authority
AR
Argentina
Prior art keywords
propofol
anesthetic solution
venous irritation
low venous
transparent
Prior art date
Application number
ARP070102080A
Other languages
English (en)
Inventor
Ciriaco Quiroga
Original Assignee
Ciriaco Quiroga
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciriaco Quiroga filed Critical Ciriaco Quiroga
Priority to ARP070102080A priority Critical patent/AR060926A1/es
Priority to AT08750919T priority patent/ATE489938T1/de
Priority to EP08750919A priority patent/EP2186509B1/en
Priority to DE602008003845T priority patent/DE602008003845D1/de
Priority to ES08750919T priority patent/ES2358864T3/es
Priority to CA2706264A priority patent/CA2706264C/en
Priority to PCT/IB2008/001178 priority patent/WO2008139313A2/es
Priority to US12/600,384 priority patent/US20100160456A1/en
Priority to MX2009012439A priority patent/MX2009012439A/es
Publication of AR060926A1 publication Critical patent/AR060926A1/es
Priority to CO09142710A priority patent/CO6140039A2/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/045Hydroxy compounds, e.g. alcohols; Salts thereof, e.g. alcoholates
    • A61K31/05Phenols
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/14Esters of carboxylic acids, e.g. fatty acid monoglycerides, medium-chain triglycerides, parabens or PEG fatty acid esters
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/08Solutions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/107Emulsions ; Emulsion preconcentrates; Micelles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P23/00Anaesthetics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dermatology (AREA)
  • Dispersion Chemistry (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Anesthesiology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cosmetics (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)

Abstract

Solucion anestésica transparente de propofol, con baja irritacion venosa, compuesta por lo menos por un 90% al 55% de Propofol, disuelto en un 10% al 45% de un Macrogol 15 hidroestearato (Solutol), teniendo preferiblemente cada 10,815 mg/ml de Propofol, 25% de un Macrogol 15 hidroestearato (Solutol), y eventualmente 0,0515 mg/ml de EDTA.
ARP070102080A 2007-05-14 2007-05-14 Solucion anestesica transparente de propofol, con baja irritacion venosa. AR060926A1 (es)

Priority Applications (10)

Application Number Priority Date Filing Date Title
ARP070102080A AR060926A1 (es) 2007-05-14 2007-05-14 Solucion anestesica transparente de propofol, con baja irritacion venosa.
AT08750919T ATE489938T1 (de) 2007-05-14 2008-05-13 Transparente propofol-narkoselösung mit geringer venenreizung
EP08750919A EP2186509B1 (en) 2007-05-14 2008-05-13 Propofol transparent anaesthetic solution with low venous irritation
DE602008003845T DE602008003845D1 (de) 2007-05-14 2008-05-13 Transparente propofol-narkoselösung mit geringer venenreizung
ES08750919T ES2358864T3 (es) 2007-05-14 2008-05-13 Solución anestésica transparente de profol, con baja irritación venosa.
CA2706264A CA2706264C (en) 2007-05-14 2008-05-13 Propofol transparent anesthetic solution, with low venous irritation threshold
PCT/IB2008/001178 WO2008139313A2 (es) 2007-05-14 2008-05-13 Propofol transparent anesthehic solution with a low i.v. irration threshold
US12/600,384 US20100160456A1 (en) 2007-05-14 2008-05-13 Propofol Solution for Anesthetic Use
MX2009012439A MX2009012439A (es) 2007-05-14 2008-05-13 Solucion anestesica transparente de profol, con baja irritacion venosa.
CO09142710A CO6140039A2 (es) 2007-05-14 2009-12-14 Solucion anestesica transparente de propofol con baja irrigacion venosa

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ARP070102080A AR060926A1 (es) 2007-05-14 2007-05-14 Solucion anestesica transparente de propofol, con baja irritacion venosa.

Publications (1)

Publication Number Publication Date
AR060926A1 true AR060926A1 (es) 2008-07-23

Family

ID=39681073

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP070102080A AR060926A1 (es) 2007-05-14 2007-05-14 Solucion anestesica transparente de propofol, con baja irritacion venosa.

Country Status (10)

Country Link
US (1) US20100160456A1 (es)
EP (1) EP2186509B1 (es)
AR (1) AR060926A1 (es)
AT (1) ATE489938T1 (es)
CA (1) CA2706264C (es)
CO (1) CO6140039A2 (es)
DE (1) DE602008003845D1 (es)
ES (1) ES2358864T3 (es)
MX (1) MX2009012439A (es)
WO (1) WO2008139313A2 (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2416004B1 (es) * 2012-01-24 2014-01-28 Investigaciones Farmaceuticas Y Veterinarias, S.L. Composición farmacéutica que comprende cloruro de isometamidium en solución para el tratamiento de la tripanosomiasis en animales.
CN103768055B (zh) * 2012-10-26 2015-11-25 上海医药工业研究院 注射用依托咪酯组合物及其制备方法
PL3316860T3 (pl) 2015-07-01 2024-10-14 Yissum Research Development Company Of The Hebrew University Of Jerusalem Ltd Układy dostarczania propofolu

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1202719B1 (en) * 1999-06-21 2006-05-31 Kuhnil Pharmaceutical Co., Ltd. Anesthetic composition for intravenous injection comprising propofol
KR100482269B1 (ko) * 2002-10-08 2005-04-14 센츄론(주) 2,6-디이소프로필페놀을 활성성분으로 하는 수용액상의마취용 주사제 및 그 제조방법
US7326735B2 (en) * 2003-04-30 2008-02-05 Parnell Laboratories (Aust) Pty Limited Formulations for anaesthetic use
US20040225022A1 (en) * 2003-05-09 2004-11-11 Desai Neil P. Propofol formulation containing reduced oil and surfactants
EP1713444A4 (en) * 2004-02-13 2012-06-20 Bioavailability Inc MICROEMULSION PREPARATION OF HIGHLY CONCENTRATED PROPOFOL FOR APPLICATIONS IN ANESTHESIA
JP5068750B2 (ja) * 2005-07-08 2012-11-07 フィジカ ファルマ プロポフオールを含む透明な薬学的水性マイクロエマルジョン及び製造方法

Also Published As

Publication number Publication date
EP2186509A2 (en) 2010-05-19
MX2009012439A (es) 2010-03-11
CO6140039A2 (es) 2010-03-19
EP2186509B1 (en) 2010-12-01
ES2358864T3 (es) 2011-05-16
WO2008139313A8 (es) 2010-03-18
ATE489938T1 (de) 2010-12-15
CA2706264C (en) 2012-07-17
WO2008139313A3 (es) 2009-04-02
CA2706264A1 (en) 2008-11-20
US20100160456A1 (en) 2010-06-24
WO2008139313A2 (es) 2008-11-20
DE602008003845D1 (de) 2011-01-13

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