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AR067997A1 - ORGANIC COMPOUNDS - Google Patents

ORGANIC COMPOUNDS

Info

Publication number
AR067997A1
AR067997A1 ARP080103643A ARP080103643A AR067997A1 AR 067997 A1 AR067997 A1 AR 067997A1 AR P080103643 A ARP080103643 A AR P080103643A AR P080103643 A ARP080103643 A AR P080103643A AR 067997 A1 AR067997 A1 AR 067997A1
Authority
AR
Argentina
Prior art keywords
inhibitor
antagonist
agonist
colipid
composition
Prior art date
Application number
ARP080103643A
Other languages
Spanish (es)
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40149638&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR067997(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of AR067997A1 publication Critical patent/AR067997A1/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0043Nose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/007Pulmonary tract; Aromatherapy
    • A61K9/0073Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
    • A61K9/0075Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy for inhalation via a dry powder inhaler [DPI], e.g. comprising micronized drug mixed with lactose carrier particles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/127Synthetic bilayered vehicles, e.g. liposomes or liposomes with cholesterol as the only non-phosphatidyl surfactant
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/127Synthetic bilayered vehicles, e.g. liposomes or liposomes with cholesterol as the only non-phosphatidyl surfactant
    • A61K9/1271Non-conventional liposomes, e.g. PEGylated liposomes or liposomes coated or grafted with polymers

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Dispersion Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Otolaryngology (AREA)
  • Pulmonology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

La presente se refiere a una composicion farmacéutica que comprende: (A) una o más sustancias medicamentosas; (B) un lípido; (C) un colípido; y (D) un mejorador de flujo; en donde el colípido y el mejorador de flujo juntos forman una dispersion liposomal que contiene vesículas lipídicas que encapsulan la una o más sustancias medicamentosas. La composicion farmacéutica opcionalmente se seca para formar una formulacion en polvo seco que tiene flujo suelto y de preferencia es adecuada para administracion por inhalacion o nasal. También se describe un proceso para preparar la composicion y la formulacion en polvo seco. Reivindicacion 2: La composicion de conformidad con la reivindicacion 1 en donde el diámetro promedio de las vesículas lipídicas está entre 70 y 550 nm. Reivindicacion 3: La composicion de conformidad con la reivindicacion 1 o 2, en donde la o cada sustancia medicamentosa es un agonista del adrenoceptor-beta2, un antagonista muscarínico, un glucocorticosteriode, un agonista del receptor de glucocorticoides no esteroide, un agonista de A2a, un antagonista de A2b, un antihistamínico, un inhibidor de caspasa, un antagonista de LTB4, un antagonista de LTD4, un inhibidor de fosfodiesterasa, un mucolitico, un inhibidor de metaloproteinasa de matriz metálica, un antagonista del receptor de leucotrieno, una hormona del crecimiento, heparina, estradiol, un antagonista de prostaglandina D2, un antagonista del receptor de CRTH2, cromoglicato de sodio, un inhibidor de la síntesis de IgE un antibiotico, un interferon, un inhibidor del canal de potasio, un inmunomodulador, un agente citostático, un inhibidor de elastasa, un antineoplásico, un inhibidor de prostatina, un péptido, un oIigonucleotido ARN (tal como ARNic), ADN, un plásmido, insulina, una interleucina, GLP-1, un agente antineoplásico, o un anticuerpo.This refers to a pharmaceutical composition comprising: (A) one or more medicinal substances; (B) a lipid; (C) a colipid; and (D) a flow improver; wherein the colipid and the flow improver together form a liposomal dispersion containing lipid vesicles that encapsulate the one or more drug substances. The pharmaceutical composition is optionally dried to form a dry powder formulation that has loose flow and is preferably suitable for inhalation or nasal administration. A process for preparing the composition and dry powder formulation is also described. Claim 2: The composition according to claim 1 wherein the average diameter of the lipid vesicles is between 70 and 550 nm. Claim 3: The composition according to claim 1 or 2, wherein the or each drug substance is an adrenoceptor-beta2 agonist, a muscarinic antagonist, a glucocorticosteriode, a non-steroidal glucocorticoid receptor agonist, an A2a agonist, an A2b antagonist, an antihistamine, a caspase inhibitor, an LTB4 antagonist, an LTD4 antagonist, a phosphodiesterase inhibitor, a mucolytic, a metal matrix metalloproteinase inhibitor, a leukotriene receptor antagonist, a growth hormone , heparin, estradiol, a prostaglandin D2 antagonist, a CRTH2 receptor antagonist, sodium cromoglycate, an inhibitor of IgE synthesis an antibiotic, an interferon, a potassium channel inhibitor, an immunomodulator, a cytostatic agent, a elastase inhibitor, an antineoplastic, a prostatin inhibitor, a peptide, an RNA oligonucleotide (such as siRNA), DNA, a plasmid, insu lina, an interleukin, GLP-1, an antineoplastic agent, or an antibody.

ARP080103643A 2007-08-24 2008-08-21 ORGANIC COMPOUNDS AR067997A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP07114981 2007-08-24
EP07123163 2007-12-13

Publications (1)

Publication Number Publication Date
AR067997A1 true AR067997A1 (en) 2009-10-28

Family

ID=40149638

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP080103643A AR067997A1 (en) 2007-08-24 2008-08-21 ORGANIC COMPOUNDS

Country Status (5)

Country Link
AR (1) AR067997A1 (en)
CL (1) CL2008002479A1 (en)
PE (1) PE20090607A1 (en)
TW (1) TW200916126A (en)
WO (1) WO2009027337A1 (en)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP5508003B2 (en) 2006-06-30 2014-05-28 アイスイティカ ピーティーワイ リミテッド Process for the preparation of biologically active compounds in nanoparticulate form
BRPI1014275B8 (en) 2009-04-24 2021-05-25 Iceutica Pty Ltd composition comprising indomethacin particles dispersed in at least two partially ground mill materials
US8808734B2 (en) 2011-07-11 2014-08-19 Full Spectrum Laboratories Limited Cannabinoid formulations
CN104394846B (en) * 2012-05-03 2018-10-19 爱尔兰詹森科学公司 Polyinosinic acid-polycytidylic acid (poly(I:C)) formulations for the treatment of upper respiratory infections
WO2018160295A1 (en) * 2017-01-25 2018-09-07 Yiannios James John Dietary supplement compositions with enhanced delivery matrix, gummies, chocolates, atomizers and powders containing same, and methods of making same
US9526734B2 (en) 2014-06-09 2016-12-27 Iceutica Pty Ltd. Formulation of meloxicam
JP2021512860A (en) 2018-02-01 2021-05-20 コーバス・ファーマシューティカルズ・インコーポレイテッド Pharmaceutical product
US20190231783A1 (en) * 2018-02-01 2019-08-01 Corvus Pharmaceuticals, Inc. Pharmaceutical formulations
MX2021005508A (en) * 2018-11-13 2021-09-08 Civitas Therapeutics Inc Respirable polynucleotide powder formulations for inhalation.
US10729687B1 (en) * 2019-07-09 2020-08-04 Orexo Ab Pharmaceutical composition for nasal delivery
US20220249678A1 (en) * 2019-07-10 2022-08-11 The University Of Hong Kong PEGylated synthetic KL4 peptide, Compositions and Methods Thereof
CN114209651A (en) * 2021-11-18 2022-03-22 上海欣峰制药有限公司 Pharmaceutical preparation of cefotaxime sodium compound and preparation method thereof
CN114053226A (en) * 2021-11-18 2022-02-18 上海欣峰制药有限公司 Pharmaceutical preparation of cefminox sodium compound and preparation method thereof

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2227989A1 (en) * 1995-08-01 1997-02-13 Karen Ophelia Hamilton Liposomal oligonucleotide compositions
EP2660322A3 (en) * 2003-04-17 2013-11-13 Alnylam Pharmaceuticals Inc. Modified iRNA agents
US20070160657A1 (en) * 2003-08-01 2007-07-12 National Institute Of Advanced Industrial Science Targeting and intestinal-absorption controlled liposome having sugar chain and therapeutic drug for cancer and diagnostic drug containing the liposome
DK1771206T3 (en) * 2004-05-05 2018-05-22 Silence Therapeutics Gmbh LIPIDS, LIPID COMPLEXES AND USE THEREOF
GB0418172D0 (en) * 2004-08-13 2004-09-15 Ic Vec Ltd Vector
AU2005326371A1 (en) * 2005-01-28 2006-08-03 Kyowa Hakko Kirin Co., Ltd. Composition for inhibiting expression of target gene
US20070172430A1 (en) * 2006-01-20 2007-07-26 Nastech Pharmaceutical Company Inc. Dry powder compositions for rna influenza therapeutics
WO2007121947A1 (en) * 2006-04-20 2007-11-01 Silence Therapeutics Ag. Lipoplex formulations for specific delivery to vascular endothelium
GB0608838D0 (en) * 2006-05-04 2006-06-14 Novartis Ag Organic compounds

Also Published As

Publication number Publication date
TW200916126A (en) 2009-04-16
PE20090607A1 (en) 2009-06-11
CL2008002479A1 (en) 2009-05-08
WO2009027337A1 (en) 2009-03-05

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