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AR066544A1 - Metodos de utilizacion de antagonistas de la vasopresina con agentes para quimioterapia con antracina para reducir la cardiotoxicidad y/o aumentar la supervivencia. composicion farmaceutica. - Google Patents

Metodos de utilizacion de antagonistas de la vasopresina con agentes para quimioterapia con antracina para reducir la cardiotoxicidad y/o aumentar la supervivencia. composicion farmaceutica.

Info

Publication number
AR066544A1
AR066544A1 ARP080102015A ARP080102015A AR066544A1 AR 066544 A1 AR066544 A1 AR 066544A1 AR P080102015 A ARP080102015 A AR P080102015A AR P080102015 A ARP080102015 A AR P080102015A AR 066544 A1 AR066544 A1 AR 066544A1
Authority
AR
Argentina
Prior art keywords
group
methods
vasopresine
antracine
antagonists
Prior art date
Application number
ARP080102015A
Other languages
English (en)
Inventor
Huaquing Liu
Junichi Kambayashi
Original Assignee
Otsuka Pharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Otsuka Pharma Co Ltd filed Critical Otsuka Pharma Co Ltd
Publication of AR066544A1 publication Critical patent/AR066544A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/337Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/04Antineoplastic agents specific for metastasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P39/00General protective or antinoxious agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Cardiology (AREA)
  • Oncology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Toxicology (AREA)
  • Communicable Diseases (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Métodos para reducir la cardiotoxicidad y/o aumentar la supervivencia del tratamiento con agentes de antraciclina que comprende administrar una cantidad efectiva para uso terapéutico de una composicion que comprende un compuesto antagonista de lavasopresina o una sal aceptable para uso farmacéutico del mismo como un componente activo, administrada en forma simultánea o anterior a la administracion de antraciclinas. Reivindicacion 4: El método de la reivindicacion 1, caracterizado porque elantagonista de la vasopresina es un compuesto representado por la formula (1) donde R1 es un átomo de hidrogeno o un átomo de halogeno, R2 es un grupo hidroxi, o un grupo de la formula: --NR5R6 donde R5 y R6 son iguales o diferentes y son cada unoun átomo de hidrogeno o un grupo alquilo inferior, R3 es un átomo de hidrogeno, un átomo de halogeno, un grupo alquilo inferior, o un grupo alcoxi inferior, R4 es un átomo de halogeno, un grupo alquilo inferior, o un grupo alcoxi inferior, o una salaceptable para uso farmacéutico del mismo. Reivindicacion 7: El método de la reivindicacion 1, caracterizado porque la antraciclina se selecciona del grupo que consiste en daunorubicina, doxorubicina, epirubicina e idarubicina. Reivindicacion 8:El método de la reivindicacion 1, caracterizado porque el antagonista de la vasopresina es tolvaptan.
ARP080102015A 2007-05-15 2008-05-13 Metodos de utilizacion de antagonistas de la vasopresina con agentes para quimioterapia con antracina para reducir la cardiotoxicidad y/o aumentar la supervivencia. composicion farmaceutica. AR066544A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US93808907P 2007-05-15 2007-05-15

Publications (1)

Publication Number Publication Date
AR066544A1 true AR066544A1 (es) 2009-08-26

Family

ID=40122254

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP080102015A AR066544A1 (es) 2007-05-15 2008-05-13 Metodos de utilizacion de antagonistas de la vasopresina con agentes para quimioterapia con antracina para reducir la cardiotoxicidad y/o aumentar la supervivencia. composicion farmaceutica.

Country Status (24)

Country Link
US (1) US8372830B2 (es)
EP (1) EP2146721B1 (es)
KR (1) KR101508797B1 (es)
CN (2) CN101808517A (es)
AR (1) AR066544A1 (es)
AU (1) AU2008254273B2 (es)
BR (1) BRPI0811134A2 (es)
CA (1) CA2685186A1 (es)
CO (1) CO6280574A2 (es)
CY (1) CY1114163T1 (es)
DK (1) DK2146721T3 (es)
ES (1) ES2421639T3 (es)
HR (1) HRP20130920T1 (es)
IL (1) IL202094A (es)
MX (1) MX2009012164A (es)
MY (1) MY150682A (es)
NZ (1) NZ581126A (es)
PL (1) PL2146721T3 (es)
PT (1) PT2146721E (es)
RU (1) RU2470643C2 (es)
SI (1) SI2146721T1 (es)
TW (1) TWI428131B (es)
UA (1) UA99914C2 (es)
WO (1) WO2008144269A2 (es)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2011503085A (ja) * 2007-11-07 2011-01-27 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ アンギオテンシン変換酵素阻害剤及びバソプレッシン受容体拮抗薬を含む複合治療
WO2013176955A1 (en) * 2012-05-21 2013-11-28 The General Hospital Corporation Cardioprotective compounds, their use with chemotherapy, and methods for identifying them
WO2014062888A1 (en) * 2012-10-18 2014-04-24 University Of South Florida Compositions and methods for treating stroke
US9682983B2 (en) 2013-03-14 2017-06-20 The Brigham And Women's Hospital, Inc. BMP inhibitors and methods of use thereof
EP2983674A4 (en) 2013-04-08 2017-05-10 Dennis M. Brown Therapeutic benefit of suboptimally administered chemical compounds
WO2015050983A1 (en) * 2013-10-01 2015-04-09 The United States Of America, As Represented By The Secretary, Department Of Health And Human Services Methods of modulating erythropoiesis with arginine vasopressin receptor 1b molecules
WO2016011019A1 (en) 2014-07-15 2016-01-21 The Brigham And Women's Hospital, Inc. Compositions and methods for inhibiting bmp
WO2017120220A1 (en) 2016-01-04 2017-07-13 Adepthera Llc Peptide analogs
US11701409B2 (en) 2016-02-09 2023-07-18 Adepthera Llc Dosing and use of long-acting CLR/ramp agonists
WO2018226875A2 (en) * 2017-06-07 2018-12-13 University Of Kansas Methods and medicaments for the treatment of renal cell carcinoma
WO2019005623A1 (en) 2017-06-30 2019-01-03 Adepthera Llc PEPTIDE ANALOGS
TWI737974B (zh) 2018-04-09 2021-09-01 美商標徑製藥公司 用於治療增生性失調的劑量方案

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US574455A (en) * 1897-01-05 Switch-lock
US5744455A (en) * 1988-01-27 1998-04-28 New York University Reduction of anthracycline-induced cardiotoxicity
TWI322689B (en) * 2003-02-24 2010-04-01 Otsuka Pharma Co Ltd Method for treating severe heart failure and medicament therefor

Also Published As

Publication number Publication date
DK2146721T3 (da) 2013-07-22
HK1176318A1 (en) 2013-07-26
AU2008254273A1 (en) 2008-11-27
CY1114163T1 (el) 2016-08-31
RU2470643C2 (ru) 2012-12-27
IL202094A (en) 2015-06-30
US8372830B2 (en) 2013-02-12
KR101508797B1 (ko) 2015-04-06
MY150682A (en) 2014-02-28
EP2146721A4 (en) 2010-08-25
ES2421639T3 (es) 2013-09-04
HK1138772A1 (en) 2010-09-03
SI2146721T1 (sl) 2013-10-30
CO6280574A2 (es) 2011-05-20
MX2009012164A (es) 2009-12-09
KR20100019439A (ko) 2010-02-18
CA2685186A1 (en) 2008-11-27
UA99914C2 (ru) 2012-10-25
TW200916104A (en) 2009-04-16
BRPI0811134A2 (pt) 2014-09-30
PL2146721T3 (pl) 2013-12-31
PT2146721E (pt) 2013-07-18
CN101808517A (zh) 2010-08-18
RU2009146376A (ru) 2011-06-20
EP2146721B1 (en) 2013-07-10
AU2008254273B2 (en) 2013-03-28
NZ581126A (en) 2012-04-27
CN103550233A (zh) 2014-02-05
US20100249104A1 (en) 2010-09-30
WO2008144269A3 (en) 2010-01-21
WO2008144269A2 (en) 2008-11-27
TWI428131B (zh) 2014-03-01
HRP20130920T1 (hr) 2013-11-08
IL202094A0 (en) 2010-06-16
EP2146721A2 (en) 2010-01-27

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