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AR065280A1 - Agentes antiparasitarios - Google Patents

Agentes antiparasitarios

Info

Publication number
AR065280A1
AR065280A1 ARP080100563A ARP080100563A AR065280A1 AR 065280 A1 AR065280 A1 AR 065280A1 AR P080100563 A ARP080100563 A AR P080100563A AR P080100563 A ARP080100563 A AR P080100563A AR 065280 A1 AR065280 A1 AR 065280A1
Authority
AR
Argentina
Prior art keywords
compounds
agents
tautomer
prodrug
antiparasitary
Prior art date
Application number
ARP080100563A
Other languages
English (en)
Inventor
Stuart Nicholas Comlay
Joanne Clare Hannam
William Howson
Christelle Lauret
Yogesh Anil Sabins
Original Assignee
Pfizer Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Ltd filed Critical Pfizer Ltd
Publication of AR065280A1 publication Critical patent/AR065280A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C381/00—Compounds containing carbon and sulfur and having functional groups not covered by groups C07C301/00 - C07C337/00
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N41/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a sulfur atom bound to a hetero atom
    • A01N41/12—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a sulfur atom bound to a hetero atom not containing sulfur-to-oxygen bonds, e.g. polysulfides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A61K31/166—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the carbon of a carboxamide group directly attached to the aromatic ring, e.g. procainamide, procarbazine, metoclopramide, labetalol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
    • A61K31/343—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide condensed with a carbocyclic ring, e.g. coumaran, bufuralol, befunolol, clobenfurol, amiodarone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Agronomy & Crop Science (AREA)
  • Wood Science & Technology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pyridine Compounds (AREA)

Abstract

La presente se refiere a compuestos de formula (1) o un tautomero o profármaco de los mismos, o una sal farmacéuticamente aceptable de dicho compuesto, tautomero o profármaco, en la que R1, R2. R3, R4 y R5 se selecciona cada uno independientemente de H, halogeno, CN, CF3 y CONH2; composiciones que contienen dichos compuestos y a los usos de dichos compuestos como agentes antiparasitarios.
ARP080100563A 2007-02-09 2008-02-08 Agentes antiparasitarios AR065280A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US88904107P 2007-02-09 2007-02-09
US94682007P 2007-06-28 2007-06-28

Publications (1)

Publication Number Publication Date
AR065280A1 true AR065280A1 (es) 2009-05-27

Family

ID=39402647

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP080100563A AR065280A1 (es) 2007-02-09 2008-02-08 Agentes antiparasitarios

Country Status (21)

Country Link
US (2) US7608604B2 (es)
EP (1) EP2118055B1 (es)
JP (1) JP4592819B2 (es)
KR (2) KR101136251B1 (es)
AR (1) AR065280A1 (es)
AU (1) AU2008212594C1 (es)
BR (1) BRPI0807137A2 (es)
CA (1) CA2676147C (es)
CL (1) CL2008000403A1 (es)
CO (1) CO6220853A2 (es)
CY (1) CY1114932T1 (es)
DK (1) DK2118055T3 (es)
ES (1) ES2435191T3 (es)
MX (1) MX2009007482A (es)
NZ (1) NZ578259A (es)
PL (1) PL2118055T3 (es)
PT (1) PT2118055E (es)
RU (1) RU2425825C2 (es)
TW (1) TWI352695B (es)
UY (1) UY30897A1 (es)
WO (1) WO2008096231A1 (es)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2002087334A1 (en) * 2001-04-17 2002-11-07 Nihon Nohyaku Co., Ltd. Pest control agent composition and method of using the same
JP5413855B2 (ja) 2007-06-07 2014-02-12 バイエル・アニマル・ヘルス・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツング 外寄生生物の制御
EP2173171A2 (en) * 2007-07-30 2010-04-14 E. I. du Pont de Nemours and Company Flea control method
NZ592382A (en) 2008-10-21 2013-03-28 Merial Ltd Thioamide compounds, method of making and method of using thereof
MX2011005011A (es) 2008-11-14 2011-07-29 Merial Ltd Compuestos de arilazol-2-il-cianoetilamino enantiomericamente enriquecidos, metodo de elaboracion y de uso de los mismos.
AU2009324074B2 (en) 2008-12-03 2014-10-23 Elanco Tiergesundheit Ag Amidoacetonitrile compounds and pesticidal composition thereof
GB0905365D0 (en) 2009-03-27 2009-05-13 Norbrook Lab Ltd A topical parasiticide composition
TWI510189B (zh) * 2009-06-19 2015-12-01 Lilly Co Eli 殺外寄生蟲之方法及調配物
EP2314292A1 (en) * 2009-10-20 2011-04-27 Novartis AG Endoparasiticidal compositions
WO2011091122A1 (en) 2010-01-25 2011-07-28 Eli Lilly And Company Methods for internally controlling or treating equine bot larvae
US8962681B2 (en) 2011-10-19 2015-02-24 Zoetis Llc Use of aminoacetonitrile derivatives against endoparasites
TWI580442B (zh) * 2011-10-19 2017-05-01 傑特大學 醫藥毫微懸浮物
EP2789603B1 (en) * 2011-12-06 2016-08-10 Ube Industries, Ltd. Method for producing pentafluorosulfanyl benzoic acid
KR101978620B1 (ko) * 2011-12-21 2019-08-28 바이엘 파마 악티엔게젤샤프트 무정형 에모뎁시드를 함유하는 제제
NZ627473A (en) * 2012-02-14 2015-12-24 Nippon Soda Co Aryloxyacetamide compound and pesticide
ES2898617T3 (es) 2012-11-14 2022-03-08 Elanco Us Inc Procedimientos y formulaciones ectoparasiticidas que comprenden spinetoram
CN111718281A (zh) * 2013-03-22 2020-09-29 默克专利有限公司 用于制备有机电致发光器件用材料的合成结构单元
CN104230743B (zh) * 2013-06-24 2017-02-08 海正药业南通有限公司 一种4-苄基-1-苯乙基哌嗪-2,6-二酮的制备方法
MX2016000055A (es) * 2013-07-01 2016-08-18 Univ Zuerich Derivados de n-(1-ciano-2-hidroxi-1-metil-etil)-4-(trifluorometils ulfanil)benzamida para su uso como farmacos nematicidas.
EP3257852B1 (en) * 2015-02-12 2020-01-01 Zhejiang Hisun Pharmaceutical Co., Ltd. Preparation method for praziquantel and intermediate compounds thereof
CN106018571A (zh) * 2015-11-09 2016-10-12 中华人民共和国淮安出入境检验检疫局 检测水生蔬菜中氯虫苯甲酰胺残留量的方法

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1643766A1 (de) * 1967-01-06 1971-07-01 Allied Chem Perhalogenierte Jodide sowie Verfahren zu ihrer Herstellung
GB9801851D0 (en) * 1998-01-29 1998-03-25 Pfizer Ltd Parasiticidal agents
US6239077B1 (en) 1998-05-01 2001-05-29 Nihon Nohyaku Co., Ltd. Aminoacetonitrile derivative agricultural and horticultural insecticide containing the same and use thereof
ES2281453T3 (es) * 2000-12-20 2007-10-01 Novartis Ag Amidoacetonitrilos antiendoparasitarios.
WO2002050052A1 (en) 2000-12-20 2002-06-27 Syngenta Participations Ag N-acyl aminoacetonitriles having pesticidal properties
AR035531A1 (es) 2001-01-22 2004-06-02 Novartis Ag Composicion para el control de plagas endoparasiticas en ganados y animales domesticos, un metodo para su control y el uso de dicha composicion para la preparacion de medicamentos
DE10222192A1 (de) * 2002-05-18 2003-11-27 Aventis Pharma Gmbh Pentafluorsulfuranyl-benzoylguanidine, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament
GB0402677D0 (en) * 2003-11-06 2004-03-10 Novartis Ag Organic compounds
DE10353205A1 (de) * 2003-11-13 2005-06-16 Aventis Pharma Deutschland Gmbh Ortho-substituierte Pentafluorsulfuranyl-Benzole, Verfahren zu ihrer Herstellung sowie ihre Verwendung als wertvolle Synthese-Zwischenstufen
US7514464B2 (en) * 2003-12-18 2009-04-07 Pfizer Limited Substituted arylpyrazoles
US7425580B2 (en) 2004-05-19 2008-09-16 Wyeth (Diaryl-methyl)-malononitriles and their use as estrogen receptor ligands
AR049391A1 (es) 2004-06-10 2006-07-26 Novartis Ag Derivados de aminoacetonitrilo y su uso para controlar parasitos en animales de sangre caliente
WO2006043654A1 (ja) 2004-10-22 2006-04-27 Nihon Nohyaku Co., Ltd. アセトニトリル誘導体及び有害生物防除剤並びにその使用方法
EP1878249B1 (en) 2005-04-01 2020-03-04 LG Electronics, Inc. Method for scalably decoding a video signal

Also Published As

Publication number Publication date
BRPI0807137A2 (pt) 2014-04-15
TW200843728A (en) 2008-11-16
HK1133871A1 (en) 2010-04-09
KR20110098012A (ko) 2011-08-31
CO6220853A2 (es) 2010-11-19
US20100010093A1 (en) 2010-01-14
US7608604B2 (en) 2009-10-27
EP2118055A1 (en) 2009-11-18
DK2118055T3 (da) 2013-11-04
RU2425825C2 (ru) 2011-08-10
TWI352695B (en) 2011-11-21
CA2676147A1 (en) 2008-08-14
EP2118055B1 (en) 2013-08-21
KR101136251B1 (ko) 2012-04-25
AU2008212594C1 (en) 2013-04-11
WO2008096231A8 (en) 2009-08-20
NZ578259A (en) 2011-12-22
PL2118055T3 (pl) 2014-01-31
MX2009007482A (es) 2009-08-13
JP4592819B2 (ja) 2010-12-08
UY30897A1 (es) 2008-09-30
CA2676147C (en) 2012-03-13
WO2008096231A1 (en) 2008-08-14
AU2008212594A1 (en) 2008-08-14
AU2008212594B2 (en) 2012-10-04
JP2010518067A (ja) 2010-05-27
RU2009127356A (ru) 2011-03-20
KR20090104856A (ko) 2009-10-06
US20080194694A1 (en) 2008-08-14
ES2435191T3 (es) 2013-12-16
CL2008000403A1 (es) 2008-08-18
PT2118055E (pt) 2013-11-19
CY1114932T1 (el) 2016-12-14

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Legal Events

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