AR065109A1 - PROCESO PARA LA PREPARACIoN DE (R)-5-(2-AMINOETIL)-1-(6,8-DIFLUOROCROMAN-3-IL)-1,3-DIHIDROIMIDAZOL-2-TIONA E INTERMEDIARIOS - Google Patents
PROCESO PARA LA PREPARACIoN DE (R)-5-(2-AMINOETIL)-1-(6,8-DIFLUOROCROMAN-3-IL)-1,3-DIHIDROIMIDAZOL-2-TIONA E INTERMEDIARIOSInfo
- Publication number
- AR065109A1 AR065109A1 ARP080100397A ARP080100397A AR065109A1 AR 065109 A1 AR065109 A1 AR 065109A1 AR P080100397 A ARP080100397 A AR P080100397A AR P080100397 A ARP080100397 A AR P080100397A AR 065109 A1 AR065109 A1 AR 065109A1
- Authority
- AR
- Argentina
- Prior art keywords
- preparation
- difluorocroman
- aminoetil
- tiona
- dihydroimidazol
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 4
- ZMZDMBWJUHKJPS-UHFFFAOYSA-M Thiocyanate anion Chemical compound [S-]C#N ZMZDMBWJUHKJPS-UHFFFAOYSA-M 0.000 abstract 1
- ZMZDMBWJUHKJPS-UHFFFAOYSA-N hydrogen thiocyanate Natural products SC#N ZMZDMBWJUHKJPS-UHFFFAOYSA-N 0.000 abstract 1
- 150000007524 organic acids Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Cardiology (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Heart & Thoracic Surgery (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pyrane Compounds (AREA)
Abstract
Reivindicacion 1:un proceso para la preparacion de un compuestote la formula 1:que comprende la reaccion de un compuesto de la formula 2; con un compuesto de la formula 3 y un tiocianato hidrosoluble y un acido organico reivindicacion 15: un compuesto de la formula 4 ;reivindicacion 16 un compuesto de la formula 5
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0701966.4A GB0701966D0 (en) | 2007-02-01 | 2007-02-01 | Process |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR065109A1 true AR065109A1 (es) | 2009-05-13 |
Family
ID=37891143
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP080100397A AR065109A1 (es) | 2007-02-01 | 2008-01-31 | PROCESO PARA LA PREPARACIoN DE (R)-5-(2-AMINOETIL)-1-(6,8-DIFLUOROCROMAN-3-IL)-1,3-DIHIDROIMIDAZOL-2-TIONA E INTERMEDIARIOS |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US8158666B2 (es) |
| EP (1) | EP2114927B1 (es) |
| JP (2) | JP2010518000A (es) |
| KR (1) | KR20090104899A (es) |
| CN (1) | CN101636396A (es) |
| AR (1) | AR065109A1 (es) |
| AU (1) | AU2008211847A1 (es) |
| BR (1) | BRPI0806428A2 (es) |
| CA (1) | CA2677204C (es) |
| ES (1) | ES2648223T3 (es) |
| GB (1) | GB0701966D0 (es) |
| IL (1) | IL200183A0 (es) |
| MX (1) | MX2009008245A (es) |
| PT (1) | PT2114927T (es) |
| RU (1) | RU2009132667A (es) |
| WO (1) | WO2008094056A1 (es) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0701966D0 (en) | 2007-02-01 | 2007-03-14 | Portela & Ca Sa | Process |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5438150A (en) * | 1994-04-26 | 1995-08-01 | Syntex (U.S.A.) Inc. | Process for making 1-benzocycloalkyl-1,3-dihydroimidazole-2-thione derivatives |
| US7125904B2 (en) * | 2002-10-11 | 2006-10-24 | Portela & C.A., S.A. | Peripherally-selective inhibitors of dopamine-β-hydroxylase and method of their preparation |
| GB0701966D0 (en) | 2007-02-01 | 2007-03-14 | Portela & Ca Sa | Process |
-
2007
- 2007-02-01 GB GBGB0701966.4A patent/GB0701966D0/en not_active Ceased
-
2008
- 2008-01-31 CA CA2677204A patent/CA2677204C/en active Active
- 2008-01-31 RU RU2009132667/04A patent/RU2009132667A/ru not_active Application Discontinuation
- 2008-01-31 MX MX2009008245A patent/MX2009008245A/es unknown
- 2008-01-31 US US12/525,043 patent/US8158666B2/en not_active Expired - Fee Related
- 2008-01-31 CN CN200880003954A patent/CN101636396A/zh active Pending
- 2008-01-31 KR KR1020097017871A patent/KR20090104899A/ko not_active Withdrawn
- 2008-01-31 EP EP08712688.4A patent/EP2114927B1/en not_active Not-in-force
- 2008-01-31 JP JP2009548189A patent/JP2010518000A/ja active Pending
- 2008-01-31 AR ARP080100397A patent/AR065109A1/es unknown
- 2008-01-31 AU AU2008211847A patent/AU2008211847A1/en not_active Abandoned
- 2008-01-31 WO PCT/PT2008/000006 patent/WO2008094056A1/en not_active Ceased
- 2008-01-31 PT PT87126884T patent/PT2114927T/pt unknown
- 2008-01-31 ES ES08712688.4T patent/ES2648223T3/es active Active
- 2008-01-31 BR BRPI0806428-8A patent/BRPI0806428A2/pt not_active IP Right Cessation
-
2009
- 2009-07-30 IL IL200183A patent/IL200183A0/en unknown
-
2014
- 2014-03-03 JP JP2014040896A patent/JP5789687B2/ja not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| US20100121073A1 (en) | 2010-05-13 |
| EP2114927A1 (en) | 2009-11-11 |
| JP5789687B2 (ja) | 2015-10-07 |
| KR20090104899A (ko) | 2009-10-06 |
| RU2009132667A (ru) | 2011-03-10 |
| MX2009008245A (es) | 2009-08-12 |
| ES2648223T3 (es) | 2017-12-29 |
| JP2014193858A (ja) | 2014-10-09 |
| GB0701966D0 (en) | 2007-03-14 |
| IL200183A0 (en) | 2010-04-15 |
| US8158666B2 (en) | 2012-04-17 |
| AU2008211847A1 (en) | 2008-08-07 |
| CA2677204A1 (en) | 2008-08-07 |
| JP2010518000A (ja) | 2010-05-27 |
| WO2008094056A1 (en) | 2008-08-07 |
| CN101636396A (zh) | 2010-01-27 |
| EP2114927B1 (en) | 2017-08-23 |
| PT2114927T (pt) | 2017-11-24 |
| BRPI0806428A2 (pt) | 2011-09-13 |
| CA2677204C (en) | 2015-06-23 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FB | Suspension of granting procedure |