AR064564A1 - Derivados de n-alquinilcarboxamida, un procedimiento para su preparacion, una composicion fungicida que los comprende y un metodo para combatir hongos fitopatogenos que los emplea. - Google Patents
Derivados de n-alquinilcarboxamida, un procedimiento para su preparacion, una composicion fungicida que los comprende y un metodo para combatir hongos fitopatogenos que los emplea.Info
- Publication number
- AR064564A1 AR064564A1 ARP070105933A AR064564A1 AR 064564 A1 AR064564 A1 AR 064564A1 AR P070105933 A ARP070105933 A AR P070105933A AR 064564 A1 AR064564 A1 AR 064564A1
- Authority
- AR
- Argentina
- Prior art keywords
- alkyl
- sulfanyl
- halogen atoms
- alkenyl
- halogen
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 5
- 241000233866 Fungi Species 0.000 title 1
- 150000003857 carboxamides Chemical class 0.000 title 1
- 125000005843 halogen group Chemical group 0.000 abstract 15
- 125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 5
- 150000001875 compounds Chemical class 0.000 abstract 5
- 125000004209 (C1-C8) alkyl group Chemical group 0.000 abstract 4
- 125000001188 haloalkyl group Chemical group 0.000 abstract 4
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 4
- 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 abstract 3
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 abstract 3
- 125000003601 C2-C6 alkynyl group Chemical group 0.000 abstract 3
- 125000003545 alkoxy group Chemical group 0.000 abstract 3
- -1 nitro, cyano, sulfanyl Chemical group 0.000 abstract 3
- 125000001181 organosilyl group Chemical group [SiH3]* 0.000 abstract 3
- 125000006272 (C3-C7) cycloalkyl group Chemical group 0.000 abstract 2
- 125000004648 C2-C8 alkenyl group Chemical group 0.000 abstract 2
- 125000004649 C2-C8 alkynyl group Chemical group 0.000 abstract 2
- 125000004438 haloalkoxy group Chemical group 0.000 abstract 2
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
- 125000001424 substituent group Chemical group 0.000 abstract 2
- 125000000171 (C1-C6) haloalkyl group Chemical group 0.000 abstract 1
- 125000004217 4-methoxybenzyl group Chemical group [H]C1=C([H])C(=C([H])C([H])=C1OC([H])([H])[H])C([H])([H])* 0.000 abstract 1
- 150000001204 N-oxides Chemical class 0.000 abstract 1
- 125000003342 alkenyl group Chemical group 0.000 abstract 1
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 125000004414 alkyl thio group Chemical group 0.000 abstract 1
- 125000001797 benzyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])* 0.000 abstract 1
- 125000004432 carbon atom Chemical group C* 0.000 abstract 1
- 150000001732 carboxylic acid derivatives Chemical class 0.000 abstract 1
- 239000003054 catalyst Substances 0.000 abstract 1
- 239000003795 chemical substances by application Substances 0.000 abstract 1
- 125000002485 formyl group Chemical group [H]C(*)=O 0.000 abstract 1
- 230000000855 fungicidal effect Effects 0.000 abstract 1
- 125000005842 heteroatom Chemical group 0.000 abstract 1
- 125000000623 heterocyclic group Chemical group 0.000 abstract 1
- 239000002184 metal Chemical class 0.000 abstract 1
- 229910052752 metalloid Inorganic materials 0.000 abstract 1
- 150000002738 metalloids Chemical class 0.000 abstract 1
- 125000000538 pentafluorophenyl group Chemical group FC1=C(F)C(F)=C(*)C(F)=C1F 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/38—Nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/72—Nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D339/00—Heterocyclic compounds containing rings having two sulfur atoms as the only ring hetero atoms
- C07D339/08—Six-membered rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
Un procedimiento para preparar este compuesto. Una composicion fungicida que comprende un compuesto de formula general (1). Un método para tratar plantas mediante la aplicacion de un compuesto de formula general (1) o una composicion que lo comprende. Reivindicacion 1: Un compuesto de formula general (1), en la que, R1 es un átomo de hidrogeno, un átomo de halogeno, un alquilo C1-6, un alquenilo C2-6, un alquinilo C2-6, un tri(alquilo C1-8)sililo, un cicloalquilo C3-6, un halogenocicloalquilo C3-6 que tiene 1 a 5 átomos de halogeno; R2 y R3 se seleccionan independientemente uno de otro para que sean un átomo de hidrogeno, un átomo de halogeno, un alquilo C1-6 , un alquenilo C2-6, un alquinilo C2-6, un tri(alquilo C1- 8)sililo, un cicloalquilo C3-6, un halogenocicloalquilo C3-6 que tiene 1 a 5 átomos de halogeno; R4 y R5 se seleccionan independientemente uno de otro para que sean un átomo de hidrogeno, un átomo de halogeno, un alquilo C1-6, un alquenilo C2-6, un alquinilo C2-6, un tri(alquilo C1-8)sililo, un cicloalquilo C3-6 un halogenocicloalquilo C3-6 que tiene 1 a 5 átomos de halogeno; o R2 o R3 pueden formar junto con R4 o R5 un cicloalquilo C3-7; R6 es un átomo de hidrogeno, un alquilo C1-6, o un cicloalquilo C3-7, y Het representa un heterociclo no condensado de 5, 6 o 7 elementos, opcionalmente sustituido con uno, dos o tres heteroátomos que pueden ser iguales o diferentes, estando Het unido por un átomo de C; estando sustituido Het en la porcion orto por un sustituyente seleccionado para que sea un átomo de halogeno, un grupo nitro, ciano, sulfanilo, pentafluoro-gamma6-sulfanilo, alquilo C1-8- halogenoalquilo C1-8 que tiene 1 a 5 átomos de halogeno, alquenilo C2-8, alquinilo C2-8, alcoxi C1-8, halogenoalcoxi C1-8 que tiene 1 a 5 átomos de halogeno, alcoxi C1-8-alquenilo C2-8, un alquil C1-8-sulfanilo, o un halogenoalquil C1-8-sulfanilo que tiene 1 a 5 átomos de halogeno, y opcionalmente sustituidos en cualquier otra posicion por uno o más sustituyentes seleccionados independientemente uno de otro de un átomo de halogeno, un grupo nitro, ciano, sulfanilo, pentafluoro-gamma6-sulfanilo, formilo, formiloxi, formilamino, carboxi, alquilo C1-8, halogenoalquilo C1-8 que tiene 1 a 5 átomos de halogeno, alquenilo C2-8, alquinilo C2-8, alcoxi C1-8, halogenoalcoxi C1-8 que tiene 1 a 5 átomos de halogeno, alcoxi C1-8alquenilo C2-8, alquil C1-8-sulfanilo o un halogenoalquil C1-8-sulfanilo con 1 a 5 átomos de halogeno; así como sus sales, N-oxidos, complejos metálicos, complejos metaloides e isomeros opticamente activos. Reivindicacion 10: Un procedimiento para la preparacion de un compuesto de formula general (1) como se define en la reivindicacion 1, que comprende hacer reaccionar un derivado de la N-alquinilcarboxamida de formula general (2) o una de sus sales: en la que R1, R2, R3, R4, R5 y R6 son como se definio en la reivindicacion 1; con un derivado de ácido carboxílico de formula general (3), en la que: Het es como se definio en la reivindicacion 1; y - L1 es un grupo saliente seleccionado para que sea un átomo de halogeno, un grupo hidroxilo, -ORa, -OCORa, siendo Ra un alquilo C1-6, un haloalquilo C1-6, un bencilo, 4-metoxibencilo, pentafluorofenilo o un grupo de formula (4) en presencia de un catalizador y, si L1 es un grupo hidroxilo, en presencia de un agente de condensacion.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP07100063 | 2007-01-03 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR064564A1 true AR064564A1 (es) | 2009-04-08 |
Family
ID=37969863
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP070105933 AR064564A1 (es) | 2007-01-03 | 2007-12-27 | Derivados de n-alquinilcarboxamida, un procedimiento para su preparacion, una composicion fungicida que los comprende y un metodo para combatir hongos fitopatogenos que los emplea. |
Country Status (3)
| Country | Link |
|---|---|
| AR (1) | AR064564A1 (es) |
| CL (1) | CL2008000005A1 (es) |
| WO (1) | WO2008081017A1 (es) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PL2576517T3 (pl) | 2010-06-03 | 2015-06-30 | Bayer Ip Gmbh | N-[(het)aryloalkilo)]pirazolo(tio)karboksyamidy i ich analogi heteropodstawione |
| BR112013017060A2 (pt) * | 2011-01-05 | 2016-09-20 | Syngenta Participations Ag | derivados de pirasol-4-il carboxamida como microbiocidas |
| WO2020244970A1 (en) * | 2019-06-06 | 2020-12-10 | Basf Se | New carbocyclic pyridine carboxamides |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4064135A (en) * | 1976-07-19 | 1977-12-20 | Syntex (U.S.A.) Inc. | Certain thiazole-5-carboxamide compounds |
| DE4029654A1 (de) * | 1990-09-19 | 1992-04-02 | Hoechst Ag | 2-phenyl-pyrimidine, verfahren zu ihrer herstellung, sie enthaltende mittel und ihre verwendung als fungizide |
| DE10136065A1 (de) * | 2001-07-25 | 2003-02-13 | Bayer Cropscience Ag | Pyrazolylcarboxanilide |
| US7355053B2 (en) * | 2002-10-18 | 2008-04-08 | Basf Aktiengesellschaft | 1-phenylpyrrolidine-2-one-3-carboxamides |
| DE102004059725A1 (de) * | 2004-12-11 | 2006-06-22 | Bayer Cropscience Ag | 2-Alkyl-cycloalk(en)yl-carboxamide |
| PT1885712E (pt) * | 2005-05-18 | 2011-04-29 | Bayer Cropscience Ag | Novos derivados de 2-piridinilcicloalquilcrboxamida como fungicidas |
-
2007
- 2007-12-27 AR ARP070105933 patent/AR064564A1/es unknown
-
2008
- 2008-01-02 WO PCT/EP2008/050014 patent/WO2008081017A1/en not_active Ceased
- 2008-01-02 CL CL2008000005A patent/CL2008000005A1/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CL2008000005A1 (es) | 2008-07-11 |
| WO2008081017A1 (en) | 2008-07-10 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FB | Suspension of granting procedure |