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AR050574A1 - Uso de un compuesto para estimulacion del crecimiento de pelo - Google Patents

Uso de un compuesto para estimulacion del crecimiento de pelo

Info

Publication number
AR050574A1
AR050574A1 ARP050100480A ARP050100480A AR050574A1 AR 050574 A1 AR050574 A1 AR 050574A1 AR P050100480 A ARP050100480 A AR P050100480A AR P050100480 A ARP050100480 A AR P050100480A AR 050574 A1 AR050574 A1 AR 050574A1
Authority
AR
Argentina
Prior art keywords
compound
pharmaceutically acceptable
alopecia
hair growth
stimulation
Prior art date
Application number
ARP050100480A
Other languages
English (en)
Original Assignee
Warner Lambert Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Warner Lambert Co filed Critical Warner Lambert Co
Publication of AR050574A1 publication Critical patent/AR050574A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D237/00Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
    • C07D237/02Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings
    • C07D237/06Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D237/10Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D237/14Oxygen atoms
    • C07D237/16Two oxygen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/50Pyridazines; Hydrogenated pyridazines
    • A61K31/501Pyridazines; Hydrogenated pyridazines not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/50Pyridazines; Hydrogenated pyridazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/14Drugs for dermatological disorders for baldness or alopecia
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cosmetics (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Se refiere a compuesto (3S,4R)-3,4-dihidro-4-(2,3-dihidro-2-metil-3-oxopiridazin-6-il)oxi-3-hidroxi-6-(3-hidroxifenil)sulfonil-2,2,3-trimietl-2H-benzo[b]pirano y su uso para promover el crecimiento de pelo y aliviar la alopecia. Reivindicacion 1: Uso de un compuesto de formula (1), una sal farmacéuticamente aceptable del mismo, o un solvato del mismo, en la fabricacion de un medicamento para alopecia. Reivindicacion 7: Una formulacion topica que comprende un compuesto de formula (1); una sal farmacéuticamente aceptable del mismo, o un solvato del mismo, en mezcla con al menos un vehículo topico farmacéuticamente aceptable. Reivindicacion 8: Un artículo de fabricacion que comprende una formulacion farmacéutica segun la reivindicacion 7 envasada para la distribucion al por menor, en asociacion con instrucciones que explican como usar dicha formulacion para tratar alopecia.
ARP050100480A 2004-02-12 2005-02-10 Uso de un compuesto para estimulacion del crecimiento de pelo AR050574A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US54411604P 2004-02-12 2004-02-12

Publications (1)

Publication Number Publication Date
AR050574A1 true AR050574A1 (es) 2006-11-08

Family

ID=34886004

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP050100480A AR050574A1 (es) 2004-02-12 2005-02-10 Uso de un compuesto para estimulacion del crecimiento de pelo

Country Status (15)

Country Link
US (2) US20050182065A1 (es)
EP (1) EP1715869A1 (es)
JP (1) JP2007522201A (es)
KR (1) KR100802848B1 (es)
CN (1) CN1917878A (es)
AR (1) AR050574A1 (es)
AU (1) AU2005215258A1 (es)
BR (1) BRPI0507669A (es)
CA (1) CA2555741C (es)
IL (1) IL177001A0 (es)
NO (1) NO20064057L (es)
RU (1) RU2006129320A (es)
TW (1) TW200526222A (es)
WO (1) WO2005079804A1 (es)
ZA (1) ZA200606428B (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6733714B2 (en) * 2001-08-13 2004-05-11 Edwin J. Oakey Method for forming high-impact, transparent, distortion-free polymeric material
AU2003274569B2 (en) * 2002-11-12 2008-07-31 Warner-Lambert Company Llc Method of stimulating hair growth using benzopyrans
EP1773820A1 (en) * 2004-07-16 2007-04-18 Warner-Lambert Company LLC Hair growth promoting agents
JP2008506767A (ja) * 2004-07-19 2008-03-06 ワーナー−ランバート カンパニー リミテッド ライアビリティー カンパニー 発毛を刺激する製剤
CN102791284A (zh) * 2010-02-24 2012-11-21 艾德宛金国际私人有限公司 治疗或预防毛发脱落或促进毛发生长的方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL108841A0 (en) * 1993-03-10 1994-06-24 Pfizer Res & Dev Benzopyrans
GB9316111D0 (en) * 1993-08-04 1993-09-22 Pfizer Ltd Benzopyrans
US5547957A (en) * 1993-10-15 1996-08-20 Merck & Co., Inc. Method of treating androgenic alopecia with 5-α reductase inhibitors
AU2003274569B2 (en) * 2002-11-12 2008-07-31 Warner-Lambert Company Llc Method of stimulating hair growth using benzopyrans

Also Published As

Publication number Publication date
WO2005079804A8 (en) 2006-05-18
US20050182065A1 (en) 2005-08-18
WO2005079804A1 (en) 2005-09-01
CA2555741C (en) 2010-03-23
KR100802848B1 (ko) 2008-02-12
US20090143393A1 (en) 2009-06-04
NO20064057L (no) 2006-11-08
TW200526222A (en) 2005-08-16
JP2007522201A (ja) 2007-08-09
IL177001A0 (en) 2006-12-10
BRPI0507669A (pt) 2007-07-17
CA2555741A1 (en) 2005-09-01
CN1917878A (zh) 2007-02-21
RU2006129320A (ru) 2008-02-27
KR20060114005A (ko) 2006-11-03
ZA200606428B (en) 2008-01-30
EP1715869A1 (en) 2006-11-02
AU2005215258A1 (en) 2005-09-01

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Legal Events

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