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AR059696A1 - Medicamentos que contienen fluoroquinolonas - Google Patents

Medicamentos que contienen fluoroquinolonas

Info

Publication number
AR059696A1
AR059696A1 ARP070100842A ARP070100842A AR059696A1 AR 059696 A1 AR059696 A1 AR 059696A1 AR P070100842 A ARP070100842 A AR P070100842A AR P070100842 A ARP070100842 A AR P070100842A AR 059696 A1 AR059696 A1 AR 059696A1
Authority
AR
Argentina
Prior art keywords
fluoroquinolones
medicines containing
quaternary ammonium
containing fluoroquinolones
fluoroquinolone
Prior art date
Application number
ARP070100842A
Other languages
English (en)
Original Assignee
Bayer Healthcare Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38171208&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR059696(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bayer Healthcare Ag filed Critical Bayer Healthcare Ag
Publication of AR059696A1 publication Critical patent/AR059696A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/472Non-condensed isoquinolines, e.g. papaverine
    • A61K31/4725Non-condensed isoquinolines, e.g. papaverine containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/02Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/16Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing nitrogen, e.g. nitro-, nitroso-, azo-compounds, nitriles, cyanates
    • A61K47/18Amines; Amides; Ureas; Quaternary ammonium compounds; Amino acids; Oligopeptides having up to five amino acids
    • A61K47/186Quaternary ammonium compounds, e.g. benzalkonium chloride or cetrimide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/08Solutions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Engineering & Computer Science (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Dermatology (AREA)
  • Inorganic Chemistry (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Uso de compuestos de amonio cuaternario para evitar las precipitaciones de fluoroquinolonas a partir de sus disoluciones, así como a medicamentos estables tolerables, particularmente adecuados para aplicacion parenteral, que contienen en forma disuelta una fluoroquinolona y un compuesto de amonio cuaternario.
ARP070100842A 2006-03-08 2007-03-01 Medicamentos que contienen fluoroquinolonas AR059696A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE102006010643A DE102006010643A1 (de) 2006-03-08 2006-03-08 Arzneimittel enthaltend Fluorchinolone

Publications (1)

Publication Number Publication Date
AR059696A1 true AR059696A1 (es) 2008-04-23

Family

ID=38171208

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP070100842A AR059696A1 (es) 2006-03-08 2007-03-01 Medicamentos que contienen fluoroquinolonas

Country Status (31)

Country Link
US (1) US10231925B2 (es)
EP (2) EP2340809B1 (es)
JP (1) JP5584418B2 (es)
KR (2) KR20080106253A (es)
CN (2) CN101394836B (es)
AR (1) AR059696A1 (es)
AU (1) AU2007291622B2 (es)
BR (1) BRPI0708613B1 (es)
CA (1) CA2645037C (es)
CR (1) CR10270A (es)
DE (1) DE102006010643A1 (es)
DK (1) DK2340809T3 (es)
EC (1) ECSP088716A (es)
ES (1) ES2542206T3 (es)
GT (1) GT200800173A (es)
HU (1) HUE025044T2 (es)
IL (1) IL193429A0 (es)
MX (1) MX2008011344A (es)
MY (1) MY152885A (es)
NZ (1) NZ571046A (es)
PE (1) PE20071021A1 (es)
PL (1) PL2340809T3 (es)
PT (1) PT2340809E (es)
RU (1) RU2527327C2 (es)
SI (1) SI2340809T1 (es)
SV (1) SV2008003014A (es)
TW (1) TWI494105B (es)
UA (1) UA96753C2 (es)
UY (1) UY30191A1 (es)
WO (1) WO2008025380A1 (es)
ZA (1) ZA200807484B (es)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7304008B2 (en) 2001-05-15 2007-12-04 Eurokera Thermochromic material
DE102006010642A1 (de) * 2006-03-08 2007-09-27 Bayer Healthcare Aktiengesellschaft Arzneimittelformulierungen, enthaltend Fluorchinolone
WO2010069493A1 (de) * 2008-12-18 2010-06-24 Bayer Animal Health Gmbh Verbesserte wirkstoffkombination enthaltend ein antibiotikum und einen nichtsteroidalen entzündungshemmer (nsaid)
EP2332916A3 (en) 2009-11-19 2011-08-03 Krka Tovarna Zdravil, D.D., Novo Mesto A process for a preparation of marbofloxacin and intermediate thereof
CN101716141B (zh) * 2010-01-20 2011-11-30 白求恩医科大学制药厂 一种氟罗沙星注射液及其制备方法
GB2480276A (en) * 2010-05-11 2011-11-16 Michael Hilary Burke Process for the preparation of an aqueous injectable enrofloxacin antimicrobial formulation
RU2682171C2 (ru) * 2016-10-11 2019-03-15 Закрытое Акционерное Общество "Биологические Исследования И Системы" (Зао "Бис") Фармацевтическая комбинированная композиция для лечения гнойных ран на основе фторхинолонов (варианты)
CN110113942A (zh) * 2016-11-07 2019-08-09 朱比兰特生命科学有限公司 协同抗微生物组合物
ES2886088T3 (es) * 2017-02-13 2021-12-16 Bayer Animal Health Gmbh Composición líquida que contiene pradofloxacina
WO2019023842A1 (en) 2017-07-31 2019-02-07 Dow Silicones Corporation MOISTURE CURING COMPOSITIONS
WO2019027897A1 (en) 2017-07-31 2019-02-07 Dow Silicones Corporation MOISTURE CURING COMPOSITIONS
CN111620901B (zh) * 2020-06-08 2023-03-21 蚌埠医学院第二附属医院 一种含硅氧烷基的氟喹诺酮化合物、其制备方法及用途
CN119504580A (zh) * 2024-11-25 2025-02-25 华南农业大学 一种二氟沙星及其盐基化合物的晶体及其制备方法

Family Cites Families (35)

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JPS5746986A (en) 1980-09-02 1982-03-17 Dai Ichi Seiyaku Co Ltd Pyrido(1,2,3-de)(1,4)benzoxazine derivative
US4670444B1 (en) 1980-09-03 1999-02-09 Bayer Ag and-naphthyridine-3-carboxylic acids and antibacte7-amino-1-cyclopropyl-4-oxo-1,4-dihydro-quinoline-rial agents containing these compounds
US4472405A (en) 1982-11-12 1984-09-18 Riker Laboratories, Inc. Antimicrobial 6,7-dihydro-5,8-dimethyl-9 fluoro-1-oxo-1H, 5H-benzo (ij) quinolizine-2-carboxylic acid and derivatives
US4730000A (en) 1984-04-09 1988-03-08 Abbott Laboratories Quinoline antibacterial compounds
US4551456A (en) * 1983-11-14 1985-11-05 Merck & Co., Inc. Ophthalmic use of norfloxacin and related antibiotics
AT392789B (de) 1985-01-23 1991-06-10 Toyama Chemical Co Ltd Verfahren zur herstellung von 1-substituierten aryl-1,4-dihydro-4-oxonaphthyridinderivaten
IN166416B (es) 1985-09-18 1990-05-05 Pfizer
DE3713672A1 (de) 1987-04-24 1988-11-17 Bayer Ag Verfahren zur herstellung von parenteral verabreichbaren chinoloncarbonsaeuren
DE3831514A1 (de) 1988-09-16 1990-03-22 Bayer Ag Ph-neutrale waessrige loesungen von chinoloncarbonsaeuren
US5225413A (en) 1988-09-16 1993-07-06 Bayer-Aktiengesellschaft pH-neutral aqueous solutions of quinolone-carboxylic acids
JP2832535B2 (ja) 1989-04-04 1998-12-09 富山化学工業株式会社 キノロンカルボン酸またはその塩の可溶化法
WO1991009616A1 (en) 1989-12-22 1991-07-11 Yale University Quinolone antibiotics encapsulated in lipid vesicles
WO1991009525A1 (en) 1989-12-29 1991-07-11 Abbott Laboratories Quinolone carboxylic acid--metal ion--acid complexes
FR2665635A1 (fr) * 1990-08-10 1992-02-14 Merck Sharp & Dohme Composition pharmaceutique fluide a base d'un complexe metallique et son procede de preparation.
WO1993005816A1 (en) 1991-09-17 1993-04-01 Alcon Laboratories, Inc. Compositions containing quinolone antibiotics and sulfonate of polystyrol
BR9612230A (pt) 1995-12-21 1999-07-13 Pfizer Formulações de quinolona injetáveis
WO1997031001A1 (de) * 1996-02-23 1997-08-28 Bayer Aktiengesellschaft Gegebenenfalls substituierte 8-cyan-1-cyclopropyl-7-(2,8-diazabicyclo-[4.3.0]-nonan-8-yl)-6-fluor-1,4-dihydro-4-oxo-3-chinolincarbonsäuren und ihre derivate
WO1998018492A1 (fr) 1996-10-25 1998-05-07 Yoshitomi Pharmaceutical Industries Ltd. Procede pour empecher la precipitation de medicaments
GB9714218D0 (en) 1997-07-04 1997-09-10 Allied Therapeutics Ltd Peritoneal dialysis fluid
DE19729879C2 (de) * 1997-07-11 1999-07-08 Mann Gerhard Chem Pharm Fab Lagerstabile ophthalmische Zusammensetzungen, umfassend Diclofenac und Ofloxacin
IL135036A0 (en) * 1997-09-15 2001-05-20 Procter & Gamble Antimicrobial quinolones, their compositions and uses
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ID21415A (id) * 1997-12-05 1999-06-10 Upjohn Co Senyawa-senyawa antibiotik magnesium quinolon
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RU2248199C1 (ru) * 2003-06-02 2005-03-20 Открытое Акционерное Общество "Акционерное Курганское общество медицинских препаратов и изделий "Синтез" (ОАО "Синтез") Глазные капли и способ их получения
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DE102004015981A1 (de) 2004-04-01 2005-10-20 Bayer Healthcare Ag Neue kirstalline Form von 8-Cyan-1-cyclopropyl-7-(1S,6S-2,8-diazabicyclo[4.3.0]nonan-8-yl)-6-fluor-1,4-dihydro-4-oxo-3-chinolincarbonsäure
MY145148A (en) * 2004-08-13 2011-12-30 Schering Plough Ltd Pharmaceutical formulation comprising an antibiotic, a triazole and a carticosteroid

Also Published As

Publication number Publication date
JP5584418B2 (ja) 2014-09-03
ZA200807484B (en) 2009-11-25
PL2340809T3 (pl) 2015-09-30
PE20071021A1 (es) 2007-11-25
NZ571046A (en) 2012-05-25
ECSP088716A (es) 2008-11-27
CN104208064A (zh) 2014-12-17
RU2527327C2 (ru) 2014-08-27
CN101394836A (zh) 2009-03-25
WO2008025380A1 (de) 2008-03-06
IL193429A0 (en) 2009-05-04
SI2340809T1 (sl) 2015-08-31
US20100009979A1 (en) 2010-01-14
MX2008011344A (es) 2008-11-12
EP2340809A3 (de) 2012-09-19
DK2340809T3 (en) 2015-07-20
ES2542206T3 (es) 2015-08-03
UY30191A1 (es) 2007-10-31
DE102006010643A1 (de) 2007-09-13
BRPI0708613B1 (pt) 2021-10-19
SV2008003014A (es) 2010-05-17
EP2340809A2 (de) 2011-07-06
KR20150046367A (ko) 2015-04-29
AU2007291622A1 (en) 2008-03-06
PT2340809E (pt) 2015-08-28
GT200800173A (es) 2009-09-14
HUE025044T2 (en) 2016-01-28
MY152885A (en) 2014-11-28
UA96753C2 (ru) 2011-12-12
EP1993510A1 (de) 2008-11-26
KR20080106253A (ko) 2008-12-04
TWI494105B (zh) 2015-08-01
TW200810756A (en) 2008-03-01
AU2007291622B2 (en) 2013-08-01
CA2645037C (en) 2016-06-28
JP2009529015A (ja) 2009-08-13
CR10270A (es) 2009-03-18
EP2340809B1 (de) 2015-04-15
CN101394836B (zh) 2017-08-29
US10231925B2 (en) 2019-03-19
BRPI0708613A2 (pt) 2011-06-07
RU2008139635A (ru) 2010-04-20
CA2645037A1 (en) 2008-03-06

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