AR057474A1 - Composiciones de donepezil gelificado y metodos para la fabricacion y utilizacion de las mismas - Google Patents
Composiciones de donepezil gelificado y metodos para la fabricacion y utilizacion de las mismasInfo
- Publication number
- AR057474A1 AR057474A1 ARP060103130A ARP060103130A AR057474A1 AR 057474 A1 AR057474 A1 AR 057474A1 AR P060103130 A ARP060103130 A AR P060103130A AR P060103130 A ARP060103130 A AR P060103130A AR 057474 A1 AR057474 A1 AR 057474A1
- Authority
- AR
- Argentina
- Prior art keywords
- compositions
- donepezil
- manufacture
- methods
- gelified
- Prior art date
Links
- ADEBPBSSDYVVLD-UHFFFAOYSA-N donepezil Chemical group O=C1C=2C=C(OC)C(OC)=CC=2CC1CC(CC1)CCN1CC1=CC=CC=C1 ADEBPBSSDYVVLD-UHFFFAOYSA-N 0.000 title abstract 6
- 239000000203 mixture Substances 0.000 title abstract 4
- 229960003530 donepezil Drugs 0.000 title abstract 3
- 238000004519 manufacturing process Methods 0.000 title abstract 2
- 238000000034 method Methods 0.000 title abstract 2
- 239000013543 active substance Substances 0.000 abstract 1
- 239000000839 emulsion Substances 0.000 abstract 1
- XLYOFNOQVPJJNP-UHFFFAOYSA-N water Substances O XLYOFNOQVPJJNP-UHFFFAOYSA-N 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
- A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/06—Ointments; Bases therefor; Other semi-solid forms, e.g. creams, sticks, gels
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/10—Dispersions; Emulsions
- A61K9/107—Emulsions ; Emulsion preconcentrates; Micelles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Neurosurgery (AREA)
- Nutrition Science (AREA)
- Physiology (AREA)
- Zoology (AREA)
- Engineering & Computer Science (AREA)
- Dispersion Chemistry (AREA)
- Neurology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
Abstract
Composiciones de donepezil gelificado y los métodos para fabricar y utilizar las mismas. Las composiciones incluyen un agente activo de donepezil en un vehículo oral gelificado farmacéuticamente aceptables que contienen una emulsion de agua y aceite. También se proporcionan kits de las composiciones.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US70410405P | 2005-07-28 | 2005-07-28 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR057474A1 true AR057474A1 (es) | 2007-12-05 |
Family
ID=37727633
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP060103130A AR057474A1 (es) | 2005-07-28 | 2006-07-20 | Composiciones de donepezil gelificado y metodos para la fabricacion y utilizacion de las mismas |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US20070026075A1 (es) |
| EP (1) | EP1906925A1 (es) |
| JP (1) | JP2009502917A (es) |
| AR (1) | AR057474A1 (es) |
| TW (1) | TW200726468A (es) |
| WO (1) | WO2007018801A1 (es) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0818473D0 (en) | 2008-10-08 | 2008-11-12 | Probio Nutraceuticals As | Composition |
| WO2010113325A1 (ja) * | 2009-04-03 | 2010-10-07 | 日医工ファーマ株式会社 | ペクチン含有ゼリー製剤 |
| US9125809B2 (en) * | 2009-04-03 | 2015-09-08 | Nichi-Iko Pharmaceutical Co., Ltd. | Pectin-containing jelly formulation |
| GB201006182D0 (en) * | 2010-04-14 | 2010-06-02 | Ayanda As | Composition |
| GB201006178D0 (en) * | 2010-04-14 | 2010-06-02 | Ayanda As | Composition |
| GB201006218D0 (en) | 2010-04-14 | 2010-06-02 | Ayanda As | Composition |
| US9132291B2 (en) | 2010-10-05 | 2015-09-15 | Dfb Technology, Ltd. | Water-in-oil emulsion compositions containing gellan gum for topical delivery of active ingredients to the skin or mucosa |
| GB201016900D0 (en) * | 2010-10-06 | 2010-11-17 | Probio Asa | Emulsion |
| JP2012188383A (ja) * | 2011-03-10 | 2012-10-04 | Towa Yakuhin Kk | ドネペジル塩酸塩の内用液剤 |
| US10994013B2 (en) | 2013-04-24 | 2021-05-04 | Temple University—Of the Commonwealth System of Higher Education | Solid dosage form containing arabinogalactan |
| KR102142026B1 (ko) * | 2017-05-31 | 2020-08-06 | 주식회사 대웅제약 | 방출제어가 용이한 서방성 약물 미립자의 제조방법 |
| CN114246824B (zh) * | 2022-01-24 | 2023-08-22 | 南京康川济医药科技有限公司 | 一种多奈哌齐口服凝胶及其制备方法 |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FI95572C (fi) * | 1987-06-22 | 1996-02-26 | Eisai Co Ltd | Menetelmä lääkeaineena käyttökelpoisen piperidiinijohdannaisten tai sen farmaseuttisen suolan valmistamiseksi |
| WO1997025024A1 (en) * | 1996-01-12 | 1997-07-17 | Ohta Pharmaceutical Co., Ltd. | Jellied medicinal composition for oral administration |
| TW513409B (en) * | 1996-06-07 | 2002-12-11 | Eisai Co Ltd | Polymorphs of donepezil hydrochloride |
| AU1153097A (en) * | 1996-06-07 | 1998-01-05 | Eisai Co. Ltd. | Stable polymorphs of donepezil (1-benzyl-4-{(5,6-dimethoxy-1-indanon)-2-yl}methylpiperidine ) hydrochloride and process for production |
| US6245911B1 (en) * | 1997-12-05 | 2001-06-12 | Eisai Co., Ltd. | Donepezil polycrystals and process for producing the same |
| ES2237078T3 (es) * | 1998-01-16 | 2005-07-16 | Eisai Co., Ltd. | Procedimiento para producir derivados de donepezilo. |
| US6193993B1 (en) * | 1998-03-03 | 2001-02-27 | Eisai Co., Ltd. | Suppository containing an antidementia medicament |
| US6576677B1 (en) * | 1998-08-28 | 2003-06-10 | Eisai Co., Ltd. | Medicinal compositions with relieved bitterness |
| US20060183776A9 (en) * | 2000-03-03 | 2006-08-17 | Eisai Co., Ltd. | Liquid dosage formulations of donepezil |
| IL150509A (en) * | 2002-07-01 | 2007-07-04 | Joseph Kaspi | Pharmaceutical preparations containing donafazil hydrochloride |
| US20050004104A1 (en) * | 2003-05-30 | 2005-01-06 | Cali Brian M. | Methods for the protection of memory and cognition |
| WO2005065308A2 (en) * | 2003-12-29 | 2005-07-21 | Jason Mcdevitt | Compositions and methods to treat recurrent medical conditions |
-
2006
- 2006-06-27 EP EP06774162A patent/EP1906925A1/en not_active Withdrawn
- 2006-06-27 JP JP2008523894A patent/JP2009502917A/ja active Pending
- 2006-06-27 US US11/476,410 patent/US20070026075A1/en not_active Abandoned
- 2006-06-27 WO PCT/US2006/025112 patent/WO2007018801A1/en not_active Ceased
- 2006-07-20 AR ARP060103130A patent/AR057474A1/es not_active Application Discontinuation
- 2006-07-27 TW TW095127408A patent/TW200726468A/zh unknown
Also Published As
| Publication number | Publication date |
|---|---|
| US20070026075A1 (en) | 2007-02-01 |
| JP2009502917A (ja) | 2009-01-29 |
| TW200726468A (en) | 2007-07-16 |
| EP1906925A1 (en) | 2008-04-09 |
| WO2007018801A1 (en) | 2007-02-15 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA | Abandonment or withdrawal |