AR054583A1 - Pantoprazol isotopicamente sustituido - Google Patents
Pantoprazol isotopicamente sustituidoInfo
- Publication number
- AR054583A1 AR054583A1 ARP060103223A ARP060103223A AR054583A1 AR 054583 A1 AR054583 A1 AR 054583A1 AR P060103223 A ARP060103223 A AR P060103223A AR P060103223 A ARP060103223 A AR P060103223A AR 054583 A1 AR054583 A1 AR 054583A1
- Authority
- AR
- Argentina
- Prior art keywords
- replaced
- pantoprazol
- isotopically
- compounds
- solvates
- Prior art date
Links
- IQPSEEYGBUAQFF-UHFFFAOYSA-N Pantoprazole Chemical compound COC1=CC=NC(CS(=O)C=2NC3=CC=C(OC(F)F)C=C3N=2)=C1OC IQPSEEYGBUAQFF-UHFFFAOYSA-N 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 3
- 150000004677 hydrates Chemical class 0.000 abstract 2
- 125000000956 methoxy group Chemical group [H]C([H])([H])O* 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
- 239000012453 solvate Substances 0.000 abstract 2
- YZCKVEUIGOORGS-OUBTZVSYSA-N Deuterium Chemical compound [2H] YZCKVEUIGOORGS-OUBTZVSYSA-N 0.000 abstract 1
- 125000004429 atom Chemical group 0.000 abstract 1
- 229910052805 deuterium Inorganic materials 0.000 abstract 1
- 125000004786 difluoromethoxy group Chemical group [H]C(F)(F)O* 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 229940079593 drug Drugs 0.000 abstract 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
- 239000000543 intermediate Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/62—Oxygen or sulfur atoms
- C07D213/69—Two or more oxygen atoms
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Immunology (AREA)
- Pulmonology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pyridine Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP05106874 | 2005-07-26 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR054583A1 true AR054583A1 (es) | 2007-06-27 |
Family
ID=35708921
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP060103223A AR054583A1 (es) | 2005-07-26 | 2006-07-26 | Pantoprazol isotopicamente sustituido |
Country Status (8)
| Country | Link |
|---|---|
| EP (1) | EP1912947A1 (ja) |
| JP (1) | JP5289951B2 (ja) |
| CN (1) | CN101268050B (ja) |
| AR (1) | AR054583A1 (ja) |
| AU (1) | AU2006274037B2 (ja) |
| CA (1) | CA2615678C (ja) |
| TW (1) | TWI410409B (ja) |
| WO (1) | WO2007012651A1 (ja) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MX2008000901A (es) * | 2005-07-26 | 2008-03-26 | Nycomed Gmbh | Inhibidores de bomba de protones isotopicamente sustituidos. |
| EP1934201A1 (en) * | 2005-10-06 | 2008-06-25 | Auspex Pharmaceuticals Inc. | Deuterated inhibitors of gastric h+, k+-atpase with enhanced therapeutic properties |
| CA2703011A1 (en) * | 2006-10-23 | 2008-10-23 | Concert Pharmaceuticals Inc. | Oxazolidinone derivatives and methods of use |
| WO2008109175A1 (en) * | 2007-03-07 | 2008-09-12 | Concert Pharmaceuticals, Inc. | Deuterated piperazine derivatives as anti-anginal compounds |
| PL2152709T3 (pl) * | 2007-05-01 | 2012-07-31 | Concert Pharmaceuticals Inc | Związki morfinanu |
| SI3825306T1 (sl) | 2007-05-01 | 2023-10-30 | Sun Pharmaceutical Industries, Inc. | Morfinanske spojine |
| US20080312247A1 (en) * | 2007-06-13 | 2008-12-18 | Auspex Pharmaceuticals, Inc. | Substituted piperazines |
| US7855204B2 (en) * | 2008-01-22 | 2010-12-21 | Concert Pharmaceuticals Inc. | Derivatives of gefitinib |
| JP5770997B2 (ja) * | 2009-12-09 | 2015-08-26 | 大塚製薬株式会社 | Cyp3a4の代謝機能測定方法 |
| CN103349655B (zh) * | 2013-07-22 | 2015-04-29 | 南通广泰生化制品有限公司 | 枸橼酸他莫昔芬肠溶胶囊 |
| EP3189007B1 (en) * | 2014-09-02 | 2019-10-02 | Bhupinder Singh | Deuterated or a non-deuterated molecule and pharmaceutical formulations |
| GB2560750A (en) * | 2017-03-24 | 2018-09-26 | Taher Darreh Shori | Biological methods |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SE7804231L (sv) * | 1978-04-14 | 1979-10-15 | Haessle Ab | Magsyrasekretionsmedel |
| ZA854287B (en) * | 1984-06-16 | 1986-02-26 | Byk Gulden Lomberg Chem Fab | Dialkoxypyridines,process for their preparation,their use and medicaments containing them |
| ATE372966T1 (de) * | 1994-03-25 | 2007-09-15 | Isotechnika Inc | Verbesserung der effektivität von arzneimitteln duren deuterierung |
| US6334997B1 (en) * | 1994-03-25 | 2002-01-01 | Isotechnika, Inc. | Method of using deuterated calcium channel blockers |
| US6884429B2 (en) * | 1997-09-05 | 2005-04-26 | Isotechnika International Inc. | Medical devices incorporating deuterated rapamycin for controlled delivery thereof |
| NO309305B1 (no) * | 1999-02-19 | 2001-01-15 | Norsk Hydro As | Anvendelse av benzaldehydderivater ved fremstilling av farmasöytiske preparater for forebygging og/eller behandling av kreft, samt visse nye benzaldehydderivater |
| DE10123129A1 (de) * | 2001-05-02 | 2002-11-14 | Berolina Drug Dev Ab Svedala | Deuterierte 3-Piperidinopropiophenone sowie diese Verbindungen enthaltende Arzneimittel |
| DE10162121A1 (de) * | 2001-12-12 | 2003-06-18 | Berolina Drug Dev Ab Svedala | Deuterierte substituierte Pyrazolyl-Benzolsulfonamide sowie diese Verbindungen enthaltende Arzneimittel |
| MX2008000901A (es) * | 2005-07-26 | 2008-03-26 | Nycomed Gmbh | Inhibidores de bomba de protones isotopicamente sustituidos. |
-
2006
- 2006-07-26 CN CN2006800344239A patent/CN101268050B/zh not_active Expired - Fee Related
- 2006-07-26 JP JP2008523355A patent/JP5289951B2/ja not_active Expired - Fee Related
- 2006-07-26 CA CA2615678A patent/CA2615678C/en not_active Expired - Fee Related
- 2006-07-26 WO PCT/EP2006/064669 patent/WO2007012651A1/en not_active Ceased
- 2006-07-26 AR ARP060103223A patent/AR054583A1/es unknown
- 2006-07-26 EP EP06777980A patent/EP1912947A1/en not_active Withdrawn
- 2006-07-26 AU AU2006274037A patent/AU2006274037B2/en not_active Ceased
- 2006-07-26 TW TW095127342A patent/TWI410409B/zh not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| WO2007012651A1 (en) | 2007-02-01 |
| CN101268050B (zh) | 2012-11-28 |
| AU2006274037B2 (en) | 2012-04-26 |
| CA2615678A1 (en) | 2007-02-01 |
| JP5289951B2 (ja) | 2013-09-11 |
| CA2615678C (en) | 2015-01-20 |
| AU2006274037A1 (en) | 2007-02-01 |
| TWI410409B (zh) | 2013-10-01 |
| JP2009502872A (ja) | 2009-01-29 |
| CN101268050A (zh) | 2008-09-17 |
| EP1912947A1 (en) | 2008-04-23 |
| TW200745039A (en) | 2007-12-16 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FB | Suspension of granting procedure |