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AR040770A1 - Benzimidazoles y benzotiazoles como inhibidores de quinasas - Google Patents

Benzimidazoles y benzotiazoles como inhibidores de quinasas

Info

Publication number
AR040770A1
AR040770A1 AR20030102781A ARP030102781A AR040770A1 AR 040770 A1 AR040770 A1 AR 040770A1 AR 20030102781 A AR20030102781 A AR 20030102781A AR P030102781 A ARP030102781 A AR P030102781A AR 040770 A1 AR040770 A1 AR 040770A1
Authority
AR
Argentina
Prior art keywords
alkyl
group
optionally substituted
halo
alkoxy
Prior art date
Application number
AR20030102781A
Other languages
English (en)
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of AR040770A1 publication Critical patent/AR040770A1/es

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/04Antineoplastic agents specific for metastasis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Reivindicación 1: Un compuesto de fórmula (1) en la que: W es como se muestra en el grupo de restos de fórmulas 2 a 11; X es N(R4) o S; R0 es (a) seleccionado entre el grupo compuesto por H, alquilo C1-6, ciano, (alquileno C1-4)-R11, 3-hidroxiprop-2-ilo, (1-fenil)-2-hidroxiet-1-ilo, (1-ciclohexil)-3-hidroxiprop-2-ilo, 4-metoxibencilo, 1,4-dioxoespiro[4,5]dec-8-ilo, tetrahidropirano, 2,2,6,6-tetrametilpiperidin-4-ilo y ciclohexan-1-on-4-ilo, (b) fenilo opcionalmente sustituido con un sustituyente seleccionado entre el grupo compuesto por nitro y amino; (c) piperidin-4-ilo opcionalmente sustituido con un sustituyente seleccionado entre el grupo compuesto por alquilo C1-4, alcoxi C1-4 carbonilo y bencilo, o (d) cicloalquilo C3-6 opcionalmente sustituido con un sustituyente seleccionado entre el grupo compuesto por alcoxi C1-4 carbonilamino, amino, hidroxi y alquileno C1-4-OH; R1 es (a) seleccionado entre el grupo compuesto por H, alquilo C1-6, alquinilo C2-4, halo, amino, azido, formilo, 1-(alcoxi C1-4carbonil)eten-2-ilo, 1-(alcoxi C1-4 carbonil)etilo, 1-(carboxi C1-4)etilo, (alquileno C1-4)benciloxi, trifluorometilo, trimetilsililetinilo, but-3-in-1-ol, cicloalquilo C3-6, tetrahidropiran-4-ilo, hidroximetilo, 2-(piperidin-1-il)metilo, N,N`,N`-[trimetil]-2-(aminoetilamino)metilo, (morfolin-4-il)metilo, dimetilaminoetilo, N-[2-(piperidin-1-il)et-1-il]aminometilo, N´,N´-dimetil-2-(aminoetilamino)metilo, piridinilo, tiazolilo, triazolilo, benzo(1,3)dioxolan-5-ilo e imidazol-2-ilo, (b) fenilo opcionalmente sustituido con uno a tres sustituyentes seleccionados independientemente entre el grupo compuesto por alquilo C1-4, halo, nitro, amino, alcoxi C1-4, trifluorometilo, trifluorometoxi, trifluorometilsulfanilo, metilsulfonilo, metilsulfonamidilo, pirrolidin-1-ilo, morfolin-4-ilo, 4-(alquil C1-4)piperazin-1-ilo, -NR6R7 y alcoxi C1-4 opcionalmente sustituido con un sustituyente seleccionado entre el grupo compuesto por piperidin-1-ilo, pirrolidin-1-ilo, morfolin-4-ilo, azepin-4-ilo y di(alquil C1-4)amino, (c) tienilo opcionalmente sustituido con un sustituyente seleccionado entre el grupo compuesto por halo, nitro, amino y alquilo C1-4, o (d) piperidin-4-ilo opcionalmente sustituido en la posición 1 del grupo compuesto por alquilo C1-4, alcoxi C1-4 carbonilo, benciloxicarbonilo y (alquileno C1-4)-R8; Como alternativa R0 y R1 pueden tomarse conjuntamente para formar una cadena de C C3-4 totalmente saturada o una cadena de C C3-4 totalmente insaturada opcionalmente sustituida con halo o alquilo C1-4; R2 es H, alquilo C1-4 o bencilo; R3 es tienilo o fenilo opcionalmente sustituido con de uno a dos sustituyentes seleccionados independientemente entre el grupo compuesto por halo, alquilo C1-4, alcoxi C1-4 y trifluorometilo; R4 es H, (alquil C1-4)sulfonilo o (cicloalquil C3-6)sulfonilo; o (alquil C1-4)2N-sulfonilo; R5 es halo, H o -NR9R10; R6 y R7 se seleccionan individualmente en cada caso entre H, carbonilo o alquilo C1-4 con la condición de que al menos uno de R6 y R7 es H; R8 es hidroxi, trifluorometilo, dimetilamino, fenilo, piridinilo o 1-metilimidazol-2-ilo; R9 es independientemente en cada caso H o alquilo C1-*4; R10 es H, alquilo C1-4 o bencilo; R11 es alcoxi C1-4, hidroxi, alcoxi C1-4carbonilo, alcoxi C1-4 carbonilamino, cicloalquilo C3-6, fenilo opcionalmente sustituido con de uno a dos sustituyentes seleccionados independientemente entre el grupo compuesto por alcoxi C1-4 y halo, morfolin-4-ilo o piridinilo; con la condición de que cuando W es como se muestra en el resto de fórmula (3) entonces (a) al menos uno de R0 y R1 es H o alquilo C1-6; o (b) R0 y R1 pueden tomarse juntos para formar una cadena de C C3-4 totalmente saturada o una cadena de C C3-4 totalmente insaturada opcionalmente sustituida con halo o alquilo C1-4; con la condición adicional de que cuando X es S, W es como se muestra en el resto de fórmula (3); o una sal farmacéuticamente aceptable o un solvato farmacéuticamente aceptable del mismo.
AR20030102781A 2002-08-09 2003-08-01 Benzimidazoles y benzotiazoles como inhibidores de quinasas AR040770A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP02380178 2002-08-09
US42193902P 2002-10-28 2002-10-28

Publications (1)

Publication Number Publication Date
AR040770A1 true AR040770A1 (es) 2005-04-20

Family

ID=31716856

Family Applications (1)

Application Number Title Priority Date Filing Date
AR20030102781A AR040770A1 (es) 2002-08-09 2003-08-01 Benzimidazoles y benzotiazoles como inhibidores de quinasas

Country Status (9)

Country Link
US (1) US7320995B2 (es)
EP (1) EP1554272B1 (es)
AR (1) AR040770A1 (es)
AT (1) ATE343572T1 (es)
AU (1) AU2003256297A1 (es)
DE (1) DE60309342T2 (es)
ES (1) ES2274302T3 (es)
TW (1) TW200404799A (es)
WO (1) WO2004014900A1 (es)

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ES2329639B1 (es) 2007-04-26 2010-09-23 Laboratorios Almirall S.A. Nuevos derivados de 4,8-difenilpoliazanaftaleno.
EP1992344A1 (en) 2007-05-18 2008-11-19 Institut Curie P38 alpha as a therapeutic target in pathologies linked to FGFR3 mutation
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WO2009005675A1 (en) 2007-06-28 2009-01-08 Abbott Laboratories Novel triazolopyridazines
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EP2113503A1 (en) 2008-04-28 2009-11-04 Laboratorios Almirall, S.A. New substituted indolin-2-one derivatives and their use as p39 mitogen-activated kinase inhibitors
EP2623101B1 (en) * 2009-04-02 2021-04-21 Merck Patent GmbH Piperidine and piperazine derivatives as autotaxin inhibitors
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Also Published As

Publication number Publication date
ATE343572T1 (de) 2006-11-15
EP1554272A1 (en) 2005-07-20
TW200404799A (en) 2004-04-01
AU2003256297A1 (en) 2004-02-25
US20050272791A1 (en) 2005-12-08
WO2004014900A1 (en) 2004-02-19
US7320995B2 (en) 2008-01-22
EP1554272B1 (en) 2006-10-25
ES2274302T3 (es) 2007-05-16
DE60309342T2 (de) 2007-05-16
DE60309342D1 (de) 2006-12-07

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