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AR049210A1 - COMPOSITION WITH TENSIOACTIVE COMPOUNDS, FOR THE REDUCTION OF FAT LOCATED IN THE HUMAN BODY AND A METHOD FOR REDUCING SUCH FAT LOCALIZED - Google Patents

COMPOSITION WITH TENSIOACTIVE COMPOUNDS, FOR THE REDUCTION OF FAT LOCATED IN THE HUMAN BODY AND A METHOD FOR REDUCING SUCH FAT LOCALIZED

Info

Publication number
AR049210A1
AR049210A1 ARP050102333A ARP050102333A AR049210A1 AR 049210 A1 AR049210 A1 AR 049210A1 AR P050102333 A ARP050102333 A AR P050102333A AR P050102333 A ARP050102333 A AR P050102333A AR 049210 A1 AR049210 A1 AR 049210A1
Authority
AR
Argentina
Prior art keywords
composition
fat
reduction
human body
composition according
Prior art date
Application number
ARP050102333A
Other languages
Spanish (es)
Inventor
Marina Emiko Yagima Odo
Luiz Carlos Cuce
Original Assignee
Libbs Farmaceutica Ltda
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Libbs Farmaceutica Ltda filed Critical Libbs Farmaceutica Ltda
Publication of AR049210A1 publication Critical patent/AR049210A1/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/575Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of three or more carbon atoms, e.g. cholane, cholestane, ergosterol, sitosterol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Obesity (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Child & Adolescent Psychology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

Composicion con compuestos tensioactivos, su uso para la reduccion de la grasa localizada en el cuerpo humano y un método para reducir la grasa localizada a través del contacto de dichos tensioactivos con el tejido celular subcutáneo. Reivindicacion 1: Una composicion para la reduccion de la grasa localizada, caracterizada por el hecho de que contiene una cantidad efectiva de uno o más compuestos tensioactivos farmacéuticamente aceptables, auxiliares y excipientes, segun sea necesario. Reivindicacion 7: Una composicion, de acuerdo con la reivindicacion 3, caracterizada por el hecho de que dicho compuesto tensoactivo es uno o más de los siguientes ácidos: colico, desoxicolico, taurocolico, taurodesoxicolico, tauroursodesoxicolico, tauroquenodesoxicolico, taurolitocolico, glicocolico, glicodesoxicolico, glicolitocolico, glicoquenodesoxicolico, quénico, quenodesoxicolico, ursocolico, ursodesoxicolico, isoursodesoxicolico, lagodesoxicolico, deshidrocolico, hiocolico, hiodesoxicolico, muricolico, litocolico o ácido sulfolitocolico, así como sus sales, isomeros y derivados. Reivindicacion 13: Una composicion, de acuerdo con la reivindicacion 12, caracterizada por el hecho de que contiene 0,3% a 1% en peso de un anetésico y/o de un agente preservativo, particularmente bencil alcohol. Reivindicacion 14: Una composicion, de acuerdo con la reivindicacion 12, caracterizada por el hecho de contener 5 a 10% en peso de un co-solvente, particularmente uno o más de los glicoles o de sorbitol. Reivindicacion 15: Una composicion, de acuerdo con cualquiera de las reivindicaciones 1 a 14, caracterizada por el hecho de que contiene agentes lipolíticos adicionales, particularmente la lipasa o la papaína.Composition with surfactant compounds, their use for the reduction of localized fat in the human body and a method to reduce localized fat through the contact of said surfactants with subcutaneous cellular tissue. Claim 1: A composition for localized fat reduction, characterized in that it contains an effective amount of one or more pharmaceutically acceptable surfactant compounds, auxiliaries and excipients, as necessary. Claim 7: A composition according to claim 3, characterized in that said surfactant compound is one or more of the following acids: colic, deoxycholic, taurocolic, taurodeoxycholic, tauroursodeoxycholic, tauroquenodeoxycholic, taurolitocolic, glycololic, glycololic, glycolic, , glycokenodeoxycholic, chemical, chenodeoxycholic, ursocolic, ursodeoxycholic, isoursodeoxycholic, lake deoxycholic, dehydrocolic, hyocolic, hyodeoxycholic, muricolic, lithocolic or sulfolitocolic acid, as well as their salts, isomers and derivatives. Claim 13: A composition according to claim 12, characterized in that it contains 0.3% to 1% by weight of an anesthetic and / or a preservative agent, particularly benzyl alcohol. Claim 14: A composition, according to claim 12, characterized in that it contains 5 to 10% by weight of a co-solvent, particularly one or more of the glycols or sorbitol. Claim 15: A composition according to any one of claims 1 to 14, characterized in that it contains additional lipolytic agents, particularly lipase or papain.

ARP050102333A 2004-07-20 2005-06-08 COMPOSITION WITH TENSIOACTIVE COMPOUNDS, FOR THE REDUCTION OF FAT LOCATED IN THE HUMAN BODY AND A METHOD FOR REDUCING SUCH FAT LOCALIZED AR049210A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/BR2004/000123 WO2006007675A1 (en) 2004-07-20 2004-07-20 Cholic acid and/or its derivatives for the reduction of localized fat in the human body

Publications (1)

Publication Number Publication Date
AR049210A1 true AR049210A1 (en) 2006-07-05

Family

ID=35784823

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP050102333A AR049210A1 (en) 2004-07-20 2005-06-08 COMPOSITION WITH TENSIOACTIVE COMPOUNDS, FOR THE REDUCTION OF FAT LOCATED IN THE HUMAN BODY AND A METHOD FOR REDUCING SUCH FAT LOCALIZED

Country Status (3)

Country Link
AR (1) AR049210A1 (en)
BR (1) BRPI0418963A (en)
WO (1) WO2006007675A1 (en)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SI2422789T1 (en) * 2004-05-19 2018-07-31 Los Angeles Biomedical Research Institute At Harbor-Ucla Medical Center An injectable composition comprising sodium deoxycholate
US20060127468A1 (en) 2004-05-19 2006-06-15 Kolodney Michael S Methods and related compositions for reduction of fat and skin tightening
US8101593B2 (en) 2009-03-03 2012-01-24 Kythera Biopharmaceuticals, Inc. Formulations of deoxycholic acid and salts thereof
MX363465B (en) 2011-02-18 2019-03-25 Kythera Biopharmaceuticals Inc Treatment of submental fat.
US8653058B2 (en) 2011-04-05 2014-02-18 Kythera Biopharmaceuticals, Inc. Compositions comprising deoxycholic acid and salts thereof suitable for use in treating fat deposits
US9426242B2 (en) * 2013-01-29 2016-08-23 Apple Inc. Determining an invitational content item type based on predicted user attention
KR102230271B1 (en) * 2019-11-13 2021-03-19 이환석 Injectable formulation and composition for reducing of fat comprising Glycodeoxycholic acid
JP2024535386A (en) * 2022-07-05 2024-09-30 グロノバ ファーマ シーオー.,エルティディー. Injectable compositions comprising a cytolytic compound in a gel, gel-forming solution, or gel-forming suspension for fat reduction - Patents.com

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3591687A (en) * 1968-03-13 1971-07-06 George A Bray Bile acids and derivatives thereof as anorectic agents
IT1137459B (en) * 1981-04-14 1986-09-10 Erregierre Spa PRODUCTION FOR THE PREPARATION OF HIGH PURITY URSODEOXICOLIC ACID
JPS60130522A (en) * 1983-12-19 1985-07-12 Masatoshi Nakano Lipid metabolic promoter for fish
LU88373A1 (en) * 1993-07-12 1994-04-01 Michel Urso Prof Medecin Et Ch Weight loss product
US20040019027A1 (en) * 2002-04-12 2004-01-29 Barry Forman Method of treating cerebrotendinous xanthomatosis

Also Published As

Publication number Publication date
WO2006007675A1 (en) 2006-01-26
BRPI0418963A (en) 2007-12-04

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