AR049091A1 - Derivados de azepinona fusionada como reguladores del crecimiento de plantas - Google Patents
Derivados de azepinona fusionada como reguladores del crecimiento de plantasInfo
- Publication number
- AR049091A1 AR049091A1 ARP050101911A ARP050101911A AR049091A1 AR 049091 A1 AR049091 A1 AR 049091A1 AR P050101911 A ARP050101911 A AR P050101911A AR P050101911 A ARP050101911 A AR P050101911A AR 049091 A1 AR049091 A1 AR 049091A1
- Authority
- AR
- Argentina
- Prior art keywords
- alkyl
- haloalkyl
- amino
- ring
- group
- Prior art date
Links
- 125000000217 alkyl group Chemical group 0.000 abstract 11
- -1 hydroxy, amino Chemical group 0.000 abstract 10
- 125000004178 (C1-C4) alkyl group Chemical group 0.000 abstract 5
- 125000004765 (C1-C4) haloalkyl group Chemical group 0.000 abstract 5
- 229910052736 halogen Inorganic materials 0.000 abstract 5
- 150000002367 halogens Chemical class 0.000 abstract 5
- 125000001072 heteroaryl group Chemical group 0.000 abstract 5
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 abstract 5
- 125000004767 (C1-C4) haloalkoxy group Chemical group 0.000 abstract 4
- 125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 4
- 125000004453 alkoxycarbonyl group Chemical group 0.000 abstract 4
- 125000004448 alkyl carbonyl group Chemical group 0.000 abstract 4
- 125000004093 cyano group Chemical group *C#N 0.000 abstract 4
- 229910052757 nitrogen Inorganic materials 0.000 abstract 4
- 229910052760 oxygen Inorganic materials 0.000 abstract 4
- 229910052717 sulfur Inorganic materials 0.000 abstract 4
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 abstract 3
- 125000003601 C2-C6 alkynyl group Chemical group 0.000 abstract 3
- 125000003545 alkoxy group Chemical group 0.000 abstract 3
- 125000003282 alkyl amino group Chemical group 0.000 abstract 3
- 125000004432 carbon atom Chemical group C* 0.000 abstract 3
- 125000000753 cycloalkyl group Chemical group 0.000 abstract 3
- 125000005842 heteroatom Chemical group 0.000 abstract 3
- 125000006413 ring segment Chemical group 0.000 abstract 3
- 125000004397 aminosulfonyl group Chemical group NS(=O)(=O)* 0.000 abstract 2
- 125000004429 atom Chemical group 0.000 abstract 2
- 125000003917 carbamoyl group Chemical group [H]N([H])C(*)=O 0.000 abstract 2
- 125000001188 haloalkyl group Chemical group 0.000 abstract 2
- 125000005553 heteroaryloxy group Chemical group 0.000 abstract 2
- 125000005368 heteroarylthio group Chemical group 0.000 abstract 2
- 125000000623 heterocyclic group Chemical group 0.000 abstract 2
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 2
- 125000000229 (C1-C4)alkoxy group Chemical group 0.000 abstract 1
- 125000004191 (C1-C6) alkoxy group Chemical group 0.000 abstract 1
- 125000004454 (C1-C6) alkoxycarbonyl group Chemical group 0.000 abstract 1
- 125000004890 (C1-C6) alkylamino group Chemical group 0.000 abstract 1
- 125000004916 (C1-C6) alkylcarbonyl group Chemical group 0.000 abstract 1
- 125000004737 (C1-C6) haloalkoxy group Chemical group 0.000 abstract 1
- 125000000171 (C1-C6) haloalkyl group Chemical group 0.000 abstract 1
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 1
- 125000005236 alkanoylamino group Chemical group 0.000 abstract 1
- 125000004457 alkyl amino carbonyl group Chemical group 0.000 abstract 1
- 125000005153 alkyl sulfamoyl group Chemical group 0.000 abstract 1
- DXZDEAJXVCLRLE-UHFFFAOYSA-N azepin-2-one Chemical class O=C1C=CC=CC=N1 DXZDEAJXVCLRLE-UHFFFAOYSA-N 0.000 abstract 1
- 229910052799 carbon Inorganic materials 0.000 abstract 1
- 125000003178 carboxy group Chemical group [H]OC(*)=O 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- RFMQOHXWHFHOJF-UHFFFAOYSA-N cyano thiocyanate Chemical compound N#CSC#N RFMQOHXWHFHOJF-UHFFFAOYSA-N 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 230000008635 plant growth Effects 0.000 abstract 1
- 239000005648 plant growth regulator Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 125000001424 substituent group Chemical group 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
- A01N43/46—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom rings with more than six members
Landscapes
- Life Sciences & Earth Sciences (AREA)
- Wood Science & Technology (AREA)
- Agronomy & Crop Science (AREA)
- Plant Pathology (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Dentistry (AREA)
- Pest Control & Pesticides (AREA)
- Zoology (AREA)
- General Health & Medical Sciences (AREA)
- Environmental Sciences (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Derivados de azepinona fusionada como reguladores del crecimiento de plantas, y composiciones que las contienen. Reivindicacion 1: El uso de un compuesto de formula (1) o una sal del mismo aceptable para uso en agricultura para la regulacion del crecimiento vegetal donde: X es CO2R2 o H; Y es OH; NHNR3R4, NHNHC(=Z)NR5R6 o NHNHC(=Z)CR7R8R9; o X e Y junto con los dos átomos de C a los cuales están unidos forman un anillo de formula (2) donde los átomos de C marcados 4 y 5 respectivamente corresponden a los átomos de C marcados 4 y 5 en la formula (1); Q, T, W y V son cada uno de manera independiente CR11 o un átomo de N, con la condicion de que un máximo de uno de Q, T, W y V sea un átomo de N; Z es O o S; R1 y R11 son cada uno de manera independiente H, halogeno, hidroxi, amino, nitro, formilo, carboxi, ciano, tiocianato, aminocarbonilo, alcoxi C1-6, haloalcoxi C1-6, alquil C1-6-S(O)n, haloalquil C1-6-S(O)n, alquilamino C1-6, di[alquil C1-6]amino, alquilcarbonilo C1-6, alcoxicarbonilo C1-6, alquilaminocarbonilo C1-6, di[alquil C1-6]aminocarbonilo, N-alcanoilamino C1-6, N-alcanoil C1-6-N-alquilamino C1-6, sulfamoilo, N-alquilsulfamoilo C1-6, N,N-di[alquil C1-6]sulfamoilo, cicloalquilo C3-9, alquilo C1-6, alquenilo C2-6 y alquinilo C2-6, donde cada uno de los 3 radicales mencionados en ultimo término no está sustituido con uno o más radicales seleccionados del grupo formado por halogeno, hidroxi, amino, nitro, carboxi, ciano, alcoxi C1-4, haloalcoxi C1-4, alquil C1-4-S(O)n, haloalquil C1-4-S(O)n, alquilamino C1-4, di[alquil C1-4]amino, cicloalquilo C3-9, alquilcarbonilo C1-4, alcoxicarbonilo C1-4, fenilo, fenoxi, feniltio, heterociclilo, heteroariloxi y heteroariltio, donde cada uno de los 6 ultimos radicales mencionados no está sustituido o posee uno o más sustituyentes seleccionados del grupo formado por halogeno, nitro, formilo, ciano, alquilo C1-4, alcoxi C1-4, alquil C1-4-S(O)n, haloalquil C1-4-S(O)n, haloalquilo C1-4, haloalcoxi C1-4, alquilcarbonilo C1-4 y alcoxicarbonilo C1-4; o fenilo, fenoxi, feniltio, fenilcarbonilo, heteroarilo, heteroariloxi y heteroariltio, donde cada uno de los ultimos 7 radicales mencionados no está sustituido o está sustituido con uno o más radicales seleccionados del grupo formado por halogeno, hidroxi, amino, nitro, carboxi, formilo, ciano, alquilo C1-4, haloalquilo C1-4, alcoxi C1-4, haloalcoxi C1-4, alquil C1-4-S(O)n, haloalquil C1-4-S(O)n, alquilamino C1-4, di[alquil C1-4]amino, alquilcarbonilo C1-4, alcoxicarbonilo C1-4 y en el caso de heteroarilo también oxo, donde heteroarilo en los radicales mencionados con anterioridad independientemente entre sí en cada caso es un sistema anular heteroaromático mono-, bi- o tricíclico en el cual al menos 1 anillo contiene uno o más heteroátomos seleccionados del grupo formado por N, O y S, y que contiene un total de 5 a 14 átomos anulares, donde al menos un anillo está completamente insaturado (cualquier anillo adicional está insaturado o parcialmente o completamente hidrogenado); y heterociclilo es un radical heterocíclico que posee de 3 a 7 átomos anulares y de 1 a 3 heteroátomos seleccionados del grupo formado por N, O y S; R2 es alquilo C1-6, cicloalquilo C3-9, alquilo C1-6, alquenilo C2-6, alquinilo C2-6, alcoxi C1-4-alquilo C1-4; R3 es alquilo C1-6, alquenilo C2-6, alquinilo C2-6, fenil-(CH2)m o heteroarilo, donde heteroarilo es un sistema anular heteroaromático mono-, bi- o tricíclico en el cual al menos 1 anillo contiene uno o más heteroátomos seleccionados del grupo formado por N, O y S, y que contiene un total de 5 a 14 átomos anulares donde al menos un anillo está completamente insaturado, el cual no está sustituido o está sustituido con uno o más radicales seleccionados del grupo formado por halogeno, hidroxi, amino, nitro, carboxi, formilo, ciano, alquilo C1-4, haloalquilo C1-4, alcoxi C1-4, haloalcoxi C1-4, alquil C1-4-S(O)n, haloalquil C1-4-S(O)n, alquilamino C1-4, di[alquil C1- 4]amino, alquilcarbonilo C1-4, alcoxicarbonilo C1-4 y oxo; R4, R6, R8, R9 y R10 son cada uno de manera independiente H o alquilo C1-6; R5 es H o R3; R7 es segun se definio para R3 cuando m es 0; m es 0 o 1; y n es 0, 1 o 2.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP04011256 | 2004-05-12 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR049091A1 true AR049091A1 (es) | 2006-06-28 |
Family
ID=34924977
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP050101911A AR049091A1 (es) | 2004-05-12 | 2005-05-11 | Derivados de azepinona fusionada como reguladores del crecimiento de plantas |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US7767664B2 (es) |
| EP (1) | EP1748691B1 (es) |
| CN (1) | CN100551239C (es) |
| AR (1) | AR049091A1 (es) |
| AT (1) | ATE485715T1 (es) |
| AU (1) | AU2005239811B2 (es) |
| BR (1) | BRPI0511049A (es) |
| CA (1) | CA2566419A1 (es) |
| DE (1) | DE602005024385D1 (es) |
| EA (1) | EA013072B1 (es) |
| ES (1) | ES2351193T3 (es) |
| PL (1) | PL1748691T3 (es) |
| UA (1) | UA87313C2 (es) |
| WO (1) | WO2005107471A1 (es) |
Families Citing this family (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20090062124A1 (en) * | 2007-08-30 | 2009-03-05 | The United States Of America, As Represented By The Secretary Of Agriculture | Ethephon-induced enhancement of seedling development |
| EP2476680B1 (en) | 2008-01-11 | 2014-08-27 | Albany Molecular Research, Inc. | (1-Azinone)-Substituted Pyridoindoles |
| JP2012532144A (ja) | 2009-07-01 | 2012-12-13 | アルバニー モレキュラー リサーチ， インコーポレイテッド | アジノン置換アゼピノ［ｂ］インドールおよびピリド−ピロロ−アゼピンｍｃｈ−１拮抗薬、ならびにその作製方法および使用 |
| WO2011003007A1 (en) | 2009-07-01 | 2011-01-06 | Albany Molecular Research, Inc. | Azabicycloalkane-indole and azabicycloalkane-pyrrolo-pyridine mch-1 antagonists, methods of making, and use thereof |
| US8618299B2 (en) | 2009-07-01 | 2013-12-31 | Albany Molecular Research, Inc. | Azinone-substituted azapolycycle MCH-1 antagonists, methods of making, and use thereof |
| WO2011003021A1 (en) * | 2009-07-01 | 2011-01-06 | Albany Molecular Research, Inc. | Azinone-substituted azabicycloalkane-indole and azabicycloalkane-pyrrolo-pyridine mch-1 antagonists, methods of making, and use thereof |
| WO2012088038A2 (en) | 2010-12-21 | 2012-06-28 | Albany Molecular Research, Inc. | Piperazinone-substituted tetrahydro-carboline mch-1 antagonists, methods of making, and uses thereof |
| WO2012088124A2 (en) | 2010-12-21 | 2012-06-28 | Albany Molecular Research, Inc. | Tetrahydro-azacarboline mch-1 antagonists, methods of making, and uses thereof |
| CA2847569C (en) | 2011-09-08 | 2020-05-19 | Novozymes Bioag A/S | Seed treatment methods and compositions comprising lipo-chitooligosaccharides |
| RU2014113760A (ru) | 2011-09-09 | 2015-10-20 | Байер Интеллекчуал Проперти Гмбх | Ацил-гомосериновые лактоновые производные для повышения урожая растений |
| CN104093680B (zh) | 2011-09-14 | 2016-08-24 | 诺维信生物农业公司 | 组合使用脂壳寡糖和/或壳寡糖与解磷微生物促植物生长 |
| EP2747567B1 (en) | 2011-09-23 | 2016-11-16 | Novozymes Bioag A/S | Chitooligosaccharides and methods for use in enhancing soybean growth |
| EP3335556A1 (en) * | 2011-09-23 | 2018-06-20 | Novozymes Bioag A/S | Use of chitooligosaccharides in a method for enhancing plant growth |
| BR112014006912A2 (pt) * | 2011-09-23 | 2017-04-11 | Novozymes Bioag As | método para intensificar o crescimento de plantas de milho |
| CN104066327A (zh) | 2011-09-23 | 2014-09-24 | 诺维信生物农业公司 | 用于增强植物生长的脂壳寡糖组合和方法 |
| WO2013139949A1 (en) | 2012-03-23 | 2013-09-26 | Bayer Intellectual Property Gmbh | Compositions comprising a strigolactame compound for enhanced plant growth and yield |
| EP2918171A1 (en) | 2014-03-14 | 2015-09-16 | University of Vienna | Novel plant growth regulators and their use in modulating organ number |
| US12004509B2 (en) | 2016-11-18 | 2024-06-11 | Indorama Ventures Oxides Australia Pty Limited | Co-formulation comprising a plant growth regulator and an oil, and methods of preparing and using said co-formulation |
| WO2022152097A1 (en) * | 2021-01-12 | 2022-07-21 | Chengdu Anticancer Bioscience, Ltd. | Fused azepine compounds and their use in the treatment of cancer |
| US20240246979A1 (en) * | 2022-12-21 | 2024-07-25 | Eli Lilly And Company | cGAS INHIBITORS |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2335115C (en) * | 1998-06-16 | 2009-01-27 | The Government Of The United States Of America, Represented By The Secretary, Department Of Health And Human Services | Fused azepinone cyclin dependent kinase inhibitors |
| FR2804959B1 (fr) * | 2000-02-15 | 2006-04-28 | Centre Nat Rech Scient | Utilisation de derives de paullones pour la fabrication de medicaments |
| DE10153348A1 (de) * | 2001-10-29 | 2003-05-08 | Gruenenthal Gmbh | Substituierte Benzo(b)azepin-2-on-Verbindungen |
-
2005
- 2005-04-30 BR BRPI0511049-1A patent/BRPI0511049A/pt not_active IP Right Cessation
- 2005-04-30 AU AU2005239811A patent/AU2005239811B2/en not_active Ceased
- 2005-04-30 AT AT05735979T patent/ATE485715T1/de not_active IP Right Cessation
- 2005-04-30 CN CNB2005800149956A patent/CN100551239C/zh not_active Expired - Fee Related
- 2005-04-30 CA CA002566419A patent/CA2566419A1/en not_active Abandoned
- 2005-04-30 EP EP05735979A patent/EP1748691B1/en not_active Expired - Lifetime
- 2005-04-30 UA UAA200613159A patent/UA87313C2/ru unknown
- 2005-04-30 DE DE602005024385T patent/DE602005024385D1/de not_active Expired - Lifetime
- 2005-04-30 EA EA200602035A patent/EA013072B1/ru not_active IP Right Cessation
- 2005-04-30 ES ES05735979T patent/ES2351193T3/es not_active Expired - Lifetime
- 2005-04-30 WO PCT/EP2005/004687 patent/WO2005107471A1/en not_active Ceased
- 2005-04-30 PL PL05735979T patent/PL1748691T3/pl unknown
- 2005-04-30 US US11/596,230 patent/US7767664B2/en not_active Expired - Fee Related
- 2005-05-11 AR ARP050101911A patent/AR049091A1/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| EA200602035A1 (ru) | 2007-04-27 |
| WO2005107471A1 (en) | 2005-11-17 |
| CN100551239C (zh) | 2009-10-21 |
| CA2566419A1 (en) | 2005-11-17 |
| ATE485715T1 (de) | 2010-11-15 |
| EP1748691A1 (en) | 2007-02-07 |
| UA87313C2 (ru) | 2009-07-10 |
| DE602005024385D1 (de) | 2010-12-09 |
| BRPI0511049A (pt) | 2007-11-27 |
| US20080269055A1 (en) | 2008-10-30 |
| CN1949976A (zh) | 2007-04-18 |
| US7767664B2 (en) | 2010-08-03 |
| AU2005239811B2 (en) | 2010-06-17 |
| ES2351193T3 (es) | 2011-02-01 |
| PL1748691T3 (pl) | 2011-04-29 |
| EP1748691B1 (en) | 2010-10-27 |
| EA013072B1 (ru) | 2010-02-26 |
| AU2005239811A1 (en) | 2005-11-17 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA | Abandonment or withdrawal |