AR044855A1 - Compuesto de imidazopiridina - Google Patents
Compuesto de imidazopiridinaInfo
- Publication number
- AR044855A1 AR044855A1 ARP040102166A ARP040102166A AR044855A1 AR 044855 A1 AR044855 A1 AR 044855A1 AR P040102166 A ARP040102166 A AR P040102166A AR P040102166 A ARP040102166 A AR P040102166A AR 044855 A1 AR044855 A1 AR 044855A1
- Authority
- AR
- Argentina
- Prior art keywords
- compound
- imidazopiridine
- gastric acid
- endogenously
- exogenously
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 3
- 210000004211 gastric acid Anatomy 0.000 abstract 2
- 208000017189 Gastrointestinal inflammatory disease Diseases 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 125000004857 imidazopyridinyl group Chemical class N1C(=NC2=C1C=CC=N2)* 0.000 abstract 1
- 230000002265 prevention Effects 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 230000028327 secretion Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Hospice & Palliative Care (AREA)
- Otolaryngology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
Derivados de imidazopiridinas que inhiben la secreción de ácido gástrico estimulada exógena o endógenamente. Se pueden utilizar en la prevención y tratamiento de enfermedades relacionadas con el ácido gástrico o enfermedades inflamatorias gastrointestinales. Reivindicación 1: Un compuesto de fórmula (1) o una sal farmacéuticamente aceptable de dicho compuesto.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| SE0301904A SE0301904D0 (sv) | 2003-06-26 | 2003-06-26 | Novel imidazopyridine compound II with therapeutic effect |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR044855A1 true AR044855A1 (es) | 2005-10-05 |
Family
ID=27656637
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP040102166A AR044855A1 (es) | 2003-06-26 | 2004-06-22 | Compuesto de imidazopiridina |
Country Status (28)
| Country | Link |
|---|---|
| US (1) | US7691875B2 (es) |
| EP (1) | EP1641793B1 (es) |
| JP (1) | JP4701168B2 (es) |
| KR (1) | KR20060030479A (es) |
| CN (2) | CN1809567A (es) |
| AR (1) | AR044855A1 (es) |
| AT (1) | ATE386033T1 (es) |
| AU (1) | AU2004249655B2 (es) |
| BR (1) | BRPI0411728A (es) |
| CA (1) | CA2530181A1 (es) |
| DE (1) | DE602004011773T2 (es) |
| DK (1) | DK1641793T3 (es) |
| ES (1) | ES2300796T3 (es) |
| HR (1) | HRP20080179T3 (es) |
| IL (1) | IL172530A0 (es) |
| IS (1) | IS8258A (es) |
| MX (1) | MXPA05013643A (es) |
| MY (1) | MY140718A (es) |
| NO (1) | NO20060425L (es) |
| PL (1) | PL1641793T3 (es) |
| PT (1) | PT1641793E (es) |
| RU (1) | RU2348634C2 (es) |
| SE (1) | SE0301904D0 (es) |
| TW (1) | TW200503702A (es) |
| UA (1) | UA81953C2 (es) |
| UY (1) | UY28384A1 (es) |
| WO (1) | WO2004113339A1 (es) |
| ZA (1) | ZA200510455B (es) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BRPI0719481A2 (pt) * | 2006-12-19 | 2014-02-11 | Genentech Inc | " composto, método de indução de apoptose em uma célula, de sensibilização de uma célula, para inibir a ligação de uma proteína iap a uma proteína caspase, para tratar uma doença ou condição associada com a superexpressão de uma proteína iap e para tratar câncer" |
| CN106279151A (zh) * | 2015-06-26 | 2017-01-04 | 江苏太瑞生诺生物医药科技有限公司 | 5-(2-(8-((2,6-二甲基苄基)氨基)-2,3-二甲基咪唑并[1,2-a]吡啶-6-甲酰胺基)乙氧基)-5-氧代戊酸的固体形式及其制备方法 |
| KR101777971B1 (ko) | 2016-07-05 | 2017-09-12 | 제일약품주식회사 | 이미다조[1,2-a]피리딘 유도체, 이의 제조방법 및 이의 용도 |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ZA81219B (en) | 1980-01-23 | 1982-01-27 | Schering Corp | Imidazo (1,2-a) pyridines ,process for their preparation and pharmaceutical compositions containing them |
| DE3269604D1 (en) * | 1981-06-26 | 1986-04-10 | Schering Corp | Novel imidazo(1,2-a)pyridines and pyrazines, processes for their preparation and pharmaceutical compositions containing them |
| US4725601A (en) | 1985-06-04 | 1988-02-16 | Fujisawa Pharmaceutical Co., Ltd. | Certain imidazo[1,2-a]pyridines useful in the treatment of ulcers |
| SE9700661D0 (sv) * | 1997-02-25 | 1997-02-25 | Astra Ab | New compounds |
| SE9801526D0 (sv) * | 1998-04-29 | 1998-04-29 | Astra Ab | New compounds |
| SE9802794D0 (sv) | 1998-08-21 | 1998-08-21 | Astra Ab | New compounds |
| PT1368006E (pt) | 2001-02-13 | 2006-08-31 | Astrazeneca Ab | Nova formulacao de libertacao modificada |
| SE0102808D0 (sv) | 2001-08-22 | 2001-08-22 | Astrazeneca Ab | New compounds |
-
2003
- 2003-06-26 SE SE0301904A patent/SE0301904D0/xx unknown
-
2004
- 2004-06-21 TW TW093117866A patent/TW200503702A/zh unknown
- 2004-06-22 AR ARP040102166A patent/AR044855A1/es unknown
- 2004-06-23 CA CA002530181A patent/CA2530181A1/en not_active Abandoned
- 2004-06-23 RU RU2005141059/04A patent/RU2348634C2/ru not_active IP Right Cessation
- 2004-06-23 PT PT04749051T patent/PT1641793E/pt unknown
- 2004-06-23 AU AU2004249655A patent/AU2004249655B2/en not_active Ceased
- 2004-06-23 AT AT04749051T patent/ATE386033T1/de not_active IP Right Cessation
- 2004-06-23 DE DE602004011773T patent/DE602004011773T2/de not_active Expired - Lifetime
- 2004-06-23 US US10/561,199 patent/US7691875B2/en not_active Expired - Fee Related
- 2004-06-23 HR HR20080179T patent/HRP20080179T3/xx unknown
- 2004-06-23 EP EP04749051A patent/EP1641793B1/en not_active Expired - Lifetime
- 2004-06-23 BR BRPI0411728-0A patent/BRPI0411728A/pt not_active IP Right Cessation
- 2004-06-23 CN CNA2004800175782A patent/CN1809567A/zh active Pending
- 2004-06-23 MX MXPA05013643A patent/MXPA05013643A/es active IP Right Grant
- 2004-06-23 ES ES04749051T patent/ES2300796T3/es not_active Expired - Lifetime
- 2004-06-23 DK DK04749051T patent/DK1641793T3/da active
- 2004-06-23 CN CN2010102568618A patent/CN101941968A/zh active Pending
- 2004-06-23 KR KR1020057024661A patent/KR20060030479A/ko not_active Ceased
- 2004-06-23 JP JP2006517052A patent/JP4701168B2/ja not_active Expired - Fee Related
- 2004-06-23 PL PL04749051T patent/PL1641793T3/pl unknown
- 2004-06-23 WO PCT/SE2004/001013 patent/WO2004113339A1/en not_active Ceased
- 2004-06-23 UA UAA200511721A patent/UA81953C2/uk unknown
- 2004-06-24 UY UY28384A patent/UY28384A1/es unknown
- 2004-06-24 MY MYPI20042466A patent/MY140718A/en unknown
-
2005
- 2005-12-12 IL IL172530A patent/IL172530A0/en unknown
- 2005-12-22 ZA ZA200510455A patent/ZA200510455B/en unknown
-
2006
- 2006-01-23 IS IS8258A patent/IS8258A/is unknown
- 2006-01-26 NO NO20060425A patent/NO20060425L/no not_active Application Discontinuation
Also Published As
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FB | Suspension of granting procedure |