AR033293A1 - Composiciones y metodos para aumentar la biodisponibilidad de agentes farmaceuticos - Google Patents
Composiciones y metodos para aumentar la biodisponibilidad de agentes farmaceuticosInfo
- Publication number
- AR033293A1 AR033293A1 ARP020101595A ARP020101595A AR033293A1 AR 033293 A1 AR033293 A1 AR 033293A1 AR P020101595 A ARP020101595 A AR P020101595A AR P020101595 A ARP020101595 A AR P020101595A AR 033293 A1 AR033293 A1 AR 033293A1
- Authority
- AR
- Argentina
- Prior art keywords
- increase
- biodisponibility
- compositions
- methods
- pharmaceutical agents
- Prior art date
Links
- 239000000203 mixture Substances 0.000 title 1
- 239000008177 pharmaceutical agent Substances 0.000 title 1
- 102100033350 ATP-dependent translocase ABCB1 Human genes 0.000 abstract 1
- KJHKTHWMRKYKJE-SUGCFTRWSA-N Kaletra Chemical compound N1([C@@H](C(C)C)C(=O)N[C@H](C[C@H](O)[C@H](CC=2C=CC=CC=2)NC(=O)COC=2C(=CC=CC=2C)C)CC=2C=CC=CC=2)CCCNC1=O KJHKTHWMRKYKJE-SUGCFTRWSA-N 0.000 abstract 1
- 108010047230 Member 1 Subfamily B ATP Binding Cassette Transporter Proteins 0.000 abstract 1
- 239000013543 active substance Substances 0.000 abstract 1
- 239000003112 inhibitor Substances 0.000 abstract 1
- 229960004525 lopinavir Drugs 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
- A61K31/7056—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing five-membered rings with nitrogen as a ring hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/426—1,3-Thiazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/513—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Molecular Biology (AREA)
- Virology (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Tropical Medicine & Parasitology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- AIDS & HIV (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
Método para aumentar la biodisponibilidad de agentes farmacéuticamente activos. Se usa lopinavir, sus equivalentes aceptables para uso farmacéutico y derivados del mismo como inhibidores de la glicoproteína P.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US36735301P | 2001-05-01 | 2001-05-01 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR033293A1 true AR033293A1 (es) | 2003-12-10 |
Family
ID=23446823
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP020101595A AR033293A1 (es) | 2001-05-01 | 2002-04-30 | Composiciones y metodos para aumentar la biodisponibilidad de agentes farmaceuticos |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US20020198160A1 (es) |
| EP (1) | EP1387684A1 (es) |
| JP (1) | JP2005511481A (es) |
| AR (1) | AR033293A1 (es) |
| CA (1) | CA2445967A1 (es) |
| MX (1) | MXPA03010054A (es) |
| PE (1) | PE20021075A1 (es) |
| TW (1) | TWI231211B (es) |
| UY (1) | UY27275A1 (es) |
| WO (1) | WO2002087585A1 (es) |
Families Citing this family (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI252847B (en) * | 2001-07-10 | 2006-04-11 | Synta Pharmaceuticals Corp | Synthesis of taxol enhancers |
| TWI332943B (en) * | 2001-07-10 | 2010-11-11 | Synta Pharmaceuticals Corp | Taxol enhancer compounds |
| TWI297335B (en) | 2001-07-10 | 2008-06-01 | Synta Pharmaceuticals Corp | Taxol enhancer compounds |
| TWI330079B (en) * | 2003-01-15 | 2010-09-11 | Synta Pharmaceuticals Corp | Treatment for cancers |
| US8025899B2 (en) | 2003-08-28 | 2011-09-27 | Abbott Laboratories | Solid pharmaceutical dosage form |
| US8377952B2 (en) * | 2003-08-28 | 2013-02-19 | Abbott Laboratories | Solid pharmaceutical dosage formulation |
| BRPI0506498A (pt) * | 2004-01-30 | 2007-02-13 | Pfizer | composições compreendendo inibidor de hiv protease e inibidor de atividade de enzima de citocromo p450 |
| US7385084B2 (en) | 2004-06-23 | 2008-06-10 | Synta Pharmaceutical Corp. | Bis(thio-hydrazide amide) salts for treatment of cancers |
| JP2008536875A (ja) * | 2005-04-15 | 2008-09-11 | シンタ ファーマシューティカルズ コーポレーション | ビス(チオヒドラジド)アミド化合物による併用癌療法 |
| WO2007021881A1 (en) | 2005-08-16 | 2007-02-22 | Synta Pharmaceuticals Corp. | Bis(thio-hydrazide amide) formulation |
| AU2007288338B2 (en) | 2006-08-21 | 2012-05-03 | Synta Pharmaceuticals Corp. | Compounds for treating proliferative disorders |
| US7939564B2 (en) * | 2006-08-31 | 2011-05-10 | Synta Pharmaceuticals Corp. | Combination with bis(thiohydrazide amides) for treating cancer |
| US7645904B2 (en) * | 2006-09-15 | 2010-01-12 | Synta Pharmaceuticals Corp. | Purification of bis(thiohydrazide amides) |
| CA2669938C (en) * | 2006-11-15 | 2016-01-05 | Abbott Laboratories | Solid pharmaceutical dosage formulations |
| PT2451445T (pt) | 2009-07-06 | 2019-07-10 | Boehringer Ingelheim Int | Processo para secagem de bibw2992, dos seus sais e de formulações farmacêuticas sólidas compreendendo este ingrediente ativo |
| NO2608792T3 (es) * | 2010-08-26 | 2018-03-10 | ||
| GB201808563D0 (en) | 2018-05-24 | 2018-07-11 | Univ Manchester | Treatments |
| GB201808564D0 (en) | 2018-05-24 | 2018-07-11 | Douglas Pharmaceuticals Ltd | Treatments |
| GB201907305D0 (en) * | 2019-05-23 | 2019-07-10 | Douglas Pharmaceuticals Ltd | Treatment of conditions |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5914332A (en) * | 1995-12-13 | 1999-06-22 | Abbott Laboratories | Retroviral protease inhibiting compounds |
-
2002
- 2002-04-29 WO PCT/US2002/013353 patent/WO2002087585A1/en not_active Ceased
- 2002-04-29 CA CA002445967A patent/CA2445967A1/en not_active Abandoned
- 2002-04-29 US US10/134,931 patent/US20020198160A1/en not_active Abandoned
- 2002-04-29 TW TW091108841A patent/TWI231211B/zh not_active IP Right Cessation
- 2002-04-29 JP JP2002584930A patent/JP2005511481A/ja active Pending
- 2002-04-29 MX MXPA03010054A patent/MXPA03010054A/es not_active Application Discontinuation
- 2002-04-29 EP EP02731543A patent/EP1387684A1/en not_active Withdrawn
- 2002-04-30 UY UY27275A patent/UY27275A1/es not_active Application Discontinuation
- 2002-04-30 AR ARP020101595A patent/AR033293A1/es not_active Application Discontinuation
- 2002-04-30 PE PE2002000367A patent/PE20021075A1/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| TWI231211B (en) | 2005-04-21 |
| CA2445967A1 (en) | 2002-11-07 |
| US20020198160A1 (en) | 2002-12-26 |
| JP2005511481A (ja) | 2005-04-28 |
| WO2002087585A1 (en) | 2002-11-07 |
| MXPA03010054A (es) | 2004-04-02 |
| PE20021075A1 (es) | 2002-12-07 |
| EP1387684A1 (en) | 2004-02-11 |
| UY27275A1 (es) | 2002-11-29 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| AR033293A1 (es) | Composiciones y metodos para aumentar la biodisponibilidad de agentes farmaceuticos | |
| ECSP22047876A (es) | Derivados de pirazolilo ?tiles como agentes anticancer?genos | |
| SV2008001369A (es) | Benzimidazoles | |
| ECSP056194A (es) | Derivados de pirazolo-quinazolina, procedimiento para su preparacion y su uso como inhibidores de quinasa | |
| UY29199A1 (es) | Derivados tiazol, composiciones que los contienen, procedimientos de preparación y aplicaciones | |
| BR112016008016A2 (pt) | inibidores de kras g12c | |
| BRPI0513841A (pt) | composto, composição farmacêutica, e uso do composto | |
| EA200870545A1 (ru) | Новые гетероциклические соединения | |
| NI200900040A (es) | Derivados de quinazolinona 5-substituidos como agentes antitumorales. | |
| DK0991407T3 (da) | Stabilisering af syresensitive benzimidazoler med amino/cyclodextrin-kombinationer | |
| ECSP055528A (es) | Composicion farmaceutica que tiene una distribución y potencia uniforme de farmaco | |
| BR112015018087A8 (pt) | composto, composição farmacêutica e uso | |
| NO20075660L (no) | Blanding for behandling av inflammatoriske sykdommer | |
| UY31430A1 (es) | Derivados de piridina y pirazina -83 | |
| UY29087A1 (es) | Derivados de adamantilo, composiciones farmaceuticas que los contienen, procesos para su preparacion y uso terapeutico | |
| ECSP083351A (es) | Composiciones farmacéuticas | |
| CY1110906T1 (el) | Φαρμακευτικη συνθεση για ρινικη χορηγηση φεντανυλης | |
| UY27381A1 (es) | 2-tio-3,5-diciano-4-fenil-6-aminopiridinas sustituidas y su uso | |
| AR031152A1 (es) | Tratamientos nuevos para el sindrome de piernas inquietas | |
| HN2003000044A (es) | Esteres hidroxamato del acido n - (4-fenil sustituido)-antranilico. | |
| ECSP055701A (es) | Nuevos derivados de pirimidinamida y el uso de los mismos | |
| PH12021550687A1 (en) | Pharmaceutical composition for oral administration comprising aminopyrimidine derivative or its salt | |
| ECSP21060917A (es) | Formulación de anticuerpos terapéuticos | |
| UY29238A1 (es) | Formulaciones de nepafenac para su administracion topica | |
| FR2873585B1 (fr) | Nouvelles formulations galeniques de principes actifs |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA | Abandonment or withdrawal |