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AR036137A1 - Sales novedosas de derivados anticonvulsivos - Google Patents

Sales novedosas de derivados anticonvulsivos

Info

Publication number
AR036137A1
AR036137A1 ARP020102553A ARP020102553A AR036137A1 AR 036137 A1 AR036137 A1 AR 036137A1 AR P020102553 A ARP020102553 A AR P020102553A AR P020102553 A ARP020102553 A AR P020102553A AR 036137 A1 AR036137 A1 AR 036137A1
Authority
AR
Argentina
Prior art keywords
convulsive
derivatives
new salts
salts
formula
Prior art date
Application number
ARP020102553A
Other languages
English (en)
Original Assignee
Ortho Mcneil Pharm Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=23174444&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR036137(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Ortho Mcneil Pharm Inc filed Critical Ortho Mcneil Pharm Inc
Publication of AR036137A1 publication Critical patent/AR036137A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D493/00Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/12Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains three hetero rings
    • C07D493/14Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H11/00Compounds containing saccharide radicals esterified by inorganic acids; Metal salts thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • A61P21/02Muscle relaxants, e.g. for tetanus or cramps
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Neurology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Genetics & Genomics (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Saccharide Compounds (AREA)

Abstract

Sales farmacéuticamente aceptables de un derivados anticonvulsivante de fórmula (1), en donde las sales del compuesto de fórmula (1) están formadas en el grupo sulfamato. Estas sales son útiles en el tratamiento de la epilepsia.
ARP020102553A 2001-07-09 2002-07-08 Sales novedosas de derivados anticonvulsivos AR036137A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US30396201P 2001-07-09 2001-07-09

Publications (1)

Publication Number Publication Date
AR036137A1 true AR036137A1 (es) 2004-08-11

Family

ID=23174444

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP020102553A AR036137A1 (es) 2001-07-09 2002-07-08 Sales novedosas de derivados anticonvulsivos

Country Status (26)

Country Link
US (2) US7098188B2 (es)
EP (1) EP1414824B1 (es)
JP (1) JP2005502629A (es)
KR (1) KR20040013127A (es)
CN (1) CN1288159C (es)
AR (1) AR036137A1 (es)
AT (1) ATE361304T1 (es)
AU (1) AU2002346042B2 (es)
BR (1) BR0211063A (es)
CA (1) CA2452612A1 (es)
DE (1) DE60219922T2 (es)
DK (1) DK1414824T3 (es)
ES (1) ES2284884T3 (es)
HR (1) HRP20040017A2 (es)
HU (1) HUP0401080A2 (es)
IL (2) IL159698A0 (es)
MX (1) MXPA04000232A (es)
NO (1) NO20040066L (es)
NZ (1) NZ530507A (es)
PL (1) PL367635A1 (es)
PT (1) PT1414824E (es)
RU (1) RU2320665C2 (es)
SI (1) SI21370A (es)
UA (1) UA78211C2 (es)
WO (1) WO2003006467A1 (es)
ZA (1) ZA200400970B (es)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7041650B2 (en) * 2001-07-09 2006-05-09 Ortho-Mcneil Pharmaceutical, Inc. Anticonvulsant derivative salts
UA78211C2 (en) * 2001-07-09 2007-03-15 Ortho Mcneil Pharm Inc Salts of fructopyranose derivatives as anticonvulsant
WO2003039563A1 (en) * 2001-11-06 2003-05-15 Ortho-Mcneil Pharmaceutical Inc. Treatment and prevention of paresthesia comprising co-therapy with anticonvulsant derivatives and potassium
US20100311701A1 (en) * 2002-02-15 2010-12-09 Transform Pharmaceuticals, Inc Pharmaceutical Co-Crystal Compositions
US7790905B2 (en) * 2002-02-15 2010-09-07 Mcneil-Ppc, Inc. Pharmaceutical propylene glycol solvate compositions
US20090088443A1 (en) * 2002-02-15 2009-04-02 Julius Remenar Novel crystalline forms of conazoles and methods of making and using the same
US7927613B2 (en) 2002-02-15 2011-04-19 University Of South Florida Pharmaceutical co-crystal compositions
US6559293B1 (en) * 2002-02-15 2003-05-06 Transform Pharmaceuticals, Inc. Topiramate sodium trihydrate
IL163846A0 (en) * 2002-03-01 2005-12-18 Univ South Florida Multiple-component solid phases containing at least one active pharmaceutical ingredient
US20070059356A1 (en) * 2002-05-31 2007-03-15 Almarsson Oern Pharmaceutical co-crystal compositions of drugs such as carbamazepine, celecoxib, olanzapine, itraconazole, topiramate, modafinil, 5-fluorouracil, hydrochlorothiazide, acetaminophen, aspirin, flurbiprofen, phenytoin and ibuprofen
CA2489984A1 (en) * 2002-06-21 2003-12-31 Transform Pharmaceuticals, Inc. Pharmaceutical compositions with improved dissolution
US8183290B2 (en) * 2002-12-30 2012-05-22 Mcneil-Ppc, Inc. Pharmaceutically acceptable propylene glycol solvate of naproxen
US20060088886A1 (en) * 2004-10-25 2006-04-27 Anlong Ouyang Topiramate analogs
US7638291B2 (en) 2004-10-25 2009-12-29 Seradyn, Inc. Immunoassays for topiramate
US8652527B1 (en) 2013-03-13 2014-02-18 Upsher-Smith Laboratories, Inc Extended-release topiramate capsules
US9101545B2 (en) 2013-03-15 2015-08-11 Upsher-Smith Laboratories, Inc. Extended-release topiramate capsules
US9489372B2 (en) * 2013-03-15 2016-11-08 Apple Inc. Web-based spell checker
TWI826531B (zh) 2018-09-21 2023-12-21 南韓商愛思開生物製藥股份有限公司 具有㗁二唑之化合物及包含該化合物之醫藥組合物
US20210169844A1 (en) 2019-12-10 2021-06-10 Tulex Pharmaceuticals Inc. Compositions and methods for treating epilepsy, seizures and other conditions

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4513008A (en) * 1982-07-30 1985-04-23 The Vinoxen Company, Inc. Virucidal compositions and therapy
US4513006A (en) * 1983-09-26 1985-04-23 Mcneil Lab., Inc. Anticonvulsant sulfamate derivatives
AU651244B2 (en) * 1991-09-19 1994-07-14 Mcneilab, Inc. Process for the preparation of chlorosulfate and sulfamate derivatives of 2,3:4,5-bis-0-(1-methylethylidene)-beta-D- fructopyranose and (1-methylcyclohexyl)methanol
US5242942A (en) * 1992-04-28 1993-09-07 Mcneilab, Inc. Anticonvulsant fructopyranose cyclic sulfites and sulfates
US5384327A (en) * 1992-12-22 1995-01-24 Mcneilab, Inc. Anticonvulsant sorbopyranose sulfamates
US5498629A (en) * 1993-12-23 1996-03-12 Ortho Pharmaceutical Corporation Anticonvulsant pseudofructopyranose sulfamates
DE4428444A1 (de) * 1994-08-11 1996-02-15 Dresden Arzneimittel Verwendung von Selegilin zur Behandlung von epileptischen Erkrankungen
US5998380A (en) * 1995-10-13 1999-12-07 New England Medical Center Hospitals, Inc. Treatment of migraine
US5952187A (en) * 1995-12-01 1999-09-14 Oxis International, Inc. Topiramate immunoassay
US6541520B1 (en) * 1998-08-05 2003-04-01 Brookhaven Science Associates Treatment of addiction and addiction-related behavior
US6323236B2 (en) * 1999-02-24 2001-11-27 University Of Cincinnati Use of sulfamate derivatives for treating impulse control disorders
UA78211C2 (en) * 2001-07-09 2007-03-15 Ortho Mcneil Pharm Inc Salts of fructopyranose derivatives as anticonvulsant
US7041650B2 (en) * 2001-07-09 2006-05-09 Ortho-Mcneil Pharmaceutical, Inc. Anticonvulsant derivative salts
US6559293B1 (en) 2002-02-15 2003-05-06 Transform Pharmaceuticals, Inc. Topiramate sodium trihydrate

Also Published As

Publication number Publication date
UA78211C2 (en) 2007-03-15
MXPA04000232A (es) 2005-03-07
ES2284884T3 (es) 2007-11-16
NO20040066L (no) 2004-03-01
EP1414824B1 (en) 2007-05-02
ZA200400970B (en) 2005-02-07
US20060105966A1 (en) 2006-05-18
ATE361304T1 (de) 2007-05-15
SI21370A (sl) 2004-06-30
IL159698A (en) 2009-09-22
CN1288159C (zh) 2006-12-06
CN1551882A (zh) 2004-12-01
AU2002346042B8 (en) 2003-01-29
DE60219922T2 (de) 2008-01-17
RU2320665C2 (ru) 2008-03-27
US20030069190A1 (en) 2003-04-10
HK1064094A1 (en) 2005-01-21
HRP20040017A2 (en) 2004-10-31
EP1414824A1 (en) 2004-05-06
CA2452612A1 (en) 2003-01-23
JP2005502629A (ja) 2005-01-27
IL159698A0 (en) 2004-06-20
AU2002346042B2 (en) 2007-10-18
BR0211063A (pt) 2004-07-20
DK1414824T3 (da) 2007-07-16
RU2004100274A (ru) 2005-06-20
NZ530507A (en) 2007-01-26
KR20040013127A (ko) 2004-02-11
DE60219922D1 (de) 2007-06-14
HUP0401080A2 (hu) 2004-09-28
PT1414824E (pt) 2007-06-27
WO2003006467A1 (en) 2003-01-23
US7098188B2 (en) 2006-08-29
PL367635A1 (en) 2005-03-07

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