AR012109A1 - Derivados de bencenosulfonamida, su preparacion, su aplicacion en terapeutica y composicion farmaceutica - Google Patents
Derivados de bencenosulfonamida, su preparacion, su aplicacion en terapeutica y composicion farmaceuticaInfo
- Publication number
- AR012109A1 AR012109A1 ARP980101236A ARP980101236A AR012109A1 AR 012109 A1 AR012109 A1 AR 012109A1 AR P980101236 A ARP980101236 A AR P980101236A AR P980101236 A ARP980101236 A AR P980101236A AR 012109 A1 AR012109 A1 AR 012109A1
- Authority
- AR
- Argentina
- Prior art keywords
- group
- benzenosulfonamide
- therapeutics
- derivatives
- preparation
- Prior art date
Links
- 239000003814 drug Substances 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- 125000004178 (C1-C4) alkyl group Chemical group 0.000 abstract 2
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 2
- 125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 1
- 125000006590 (C2-C6) alkenylene group Chemical group 0.000 abstract 1
- POCSEAKKTFZTJS-UHFFFAOYSA-N 2-(benzenesulfonamido)guanidine;hydrochloride Chemical compound Cl.NC(N)=NNS(=O)(=O)C1=CC=CC=C1 POCSEAKKTFZTJS-UHFFFAOYSA-N 0.000 abstract 1
- WKBOTKDWSSQWDR-UHFFFAOYSA-N Bromine atom Chemical compound [Br] WKBOTKDWSSQWDR-UHFFFAOYSA-N 0.000 abstract 1
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 abstract 1
- PXGOKWXKJXAPGV-UHFFFAOYSA-N Fluorine Chemical compound FF PXGOKWXKJXAPGV-UHFFFAOYSA-N 0.000 abstract 1
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 1
- 125000003545 alkoxy group Chemical group 0.000 abstract 1
- 125000002947 alkylene group Chemical group 0.000 abstract 1
- 125000004429 atom Chemical group 0.000 abstract 1
- GDTBXPJZTBHREO-UHFFFAOYSA-N bromine Substances BrBr GDTBXPJZTBHREO-UHFFFAOYSA-N 0.000 abstract 1
- 229910052794 bromium Inorganic materials 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 125000004093 cyano group Chemical group *C#N 0.000 abstract 1
- 230000007717 exclusion Effects 0.000 abstract 1
- -1 fluorine Chemical class 0.000 abstract 1
- 229910052731 fluorine Inorganic materials 0.000 abstract 1
- 239000011737 fluorine Substances 0.000 abstract 1
- 229910052736 halogen Inorganic materials 0.000 abstract 1
- 150000002367 halogens Chemical class 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 230000001225 therapeutic effect Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
- C07C311/30—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups
- C07C311/45—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups at least one of the singly-bound nitrogen atoms being part of any of the groups, X being a hetero atom, Y being any atom, e.g. N-acylaminosulfonamides
- C07C311/47—Y being a hetero atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D233/28—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/44—Nitrogen atoms not forming part of a nitro radical
- C07D233/50—Nitrogen atoms not forming part of a nitro radical with carbocyclic radicals directly attached to said nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/06—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D239/08—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms directly attached in position 2
- C07D239/12—Nitrogen atoms not forming part of a nitro radical
- C07D239/14—Nitrogen atoms not forming part of a nitro radical with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, attached to said nitrogen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
Compuesto de la formula (I) en la cual: A representa un átomo de hidrogeno, un halogeno tal como el fluor, el coloro o el bromo, un grupo ciano, un grupoC1-4 alquilo o un grupo alcoxi; R1 y R2 idénticos o diferentes, repesentan cada uno un átomo de hidrogeno, un grupo C1-C6 alquilo, un grupo C2-6 alquenilo o R1y R2 forman juntos una cadena C2-6 alquileno o C2-6 alquenileno y R3 representa un átomo de hidrogeno o un grupo C1-4 alquilo con la exclusion del clorhidratode 3-bencenosulfonamidoguanidina. Aplicacion en terapéutica.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR9703394A FR2761061B1 (fr) | 1997-03-20 | 1997-03-20 | Derives de benzenesulfonamide, leur preparation et leur application en therapeutique |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR012109A1 true AR012109A1 (es) | 2000-09-27 |
Family
ID=9505005
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP980101236A AR012109A1 (es) | 1997-03-20 | 1998-03-19 | Derivados de bencenosulfonamida, su preparacion, su aplicacion en terapeutica y composicion farmaceutica |
Country Status (6)
| Country | Link |
|---|---|
| EP (1) | EP0971900A1 (es) |
| AR (1) | AR012109A1 (es) |
| AU (1) | AU6924198A (es) |
| FR (1) | FR2761061B1 (es) |
| WO (1) | WO1998042679A1 (es) |
| ZA (1) | ZA982358B (es) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NZ331480A (en) * | 1997-09-04 | 2000-02-28 | F | 2-(Arylphenyl)amino-imidazoline derivatives and pharmaceutical compositions |
| US6323231B1 (en) | 2000-02-17 | 2001-11-27 | Abbott Laboratories | Use of α1A adrenoceptor agonists with α1B and α1D antagonism for the treatment of stress urinary incontinence |
| DE10106214A1 (de) * | 2001-02-10 | 2002-08-14 | Boehringer Ingelheim Pharma | Neue Alkyl-phenylimino-imidazolidin-Derivate zur Behandlung der Harninkontinenz |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2456731A1 (fr) * | 1979-05-16 | 1980-12-12 | Choay Sa | Nouveaux derives substitues d'ary |
| FR2549049B1 (fr) * | 1983-07-13 | 1986-06-20 | Chauvin Blache Lab | Nouvelles amidines, leur procede de preparation et leur application therapeutique |
| US4788195A (en) * | 1986-01-13 | 1988-11-29 | American Cyanamid Company | 4,5,6-substituted-N-(substituted-phenyl)-2-pyrimidinamines |
| FR2737494B1 (fr) * | 1995-08-04 | 1997-08-29 | Synthelabo | Derives de benzenesulfonamide, leur preparation et leur application en therapeutique |
-
1997
- 1997-03-20 FR FR9703394A patent/FR2761061B1/fr not_active Expired - Fee Related
-
1998
- 1998-03-17 EP EP98914930A patent/EP0971900A1/fr not_active Ceased
- 1998-03-17 AU AU69241/98A patent/AU6924198A/en not_active Abandoned
- 1998-03-17 WO PCT/FR1998/000530 patent/WO1998042679A1/fr not_active Ceased
- 1998-03-19 AR ARP980101236A patent/AR012109A1/es unknown
- 1998-03-19 ZA ZA982358A patent/ZA982358B/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| ZA982358B (en) | 1998-09-22 |
| WO1998042679A1 (fr) | 1998-10-01 |
| EP0971900A1 (fr) | 2000-01-19 |
| FR2761061A1 (fr) | 1998-09-25 |
| FR2761061B1 (fr) | 1999-04-23 |
| AU6924198A (en) | 1998-10-20 |
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