AR011008A1 - UREA-DERIVED COMPOUND 1- (3-AMINO-INDAZOL-5-IL) -3-PHENYL-METHYL-CYCLIC, PHARMACEUTICAL COMPOSITION OF HIV PROTEASE AND USEFUL PHARMACEUTICAL EQUIPMENT FOR THE TREATMENT OF SUCH INFECTION - Google Patents
UREA-DERIVED COMPOUND 1- (3-AMINO-INDAZOL-5-IL) -3-PHENYL-METHYL-CYCLIC, PHARMACEUTICAL COMPOSITION OF HIV PROTEASE AND USEFUL PHARMACEUTICAL EQUIPMENT FOR THE TREATMENT OF SUCH INFECTIONInfo
- Publication number
- AR011008A1 AR011008A1 ARP970105182A AR011008A1 AR 011008 A1 AR011008 A1 AR 011008A1 AR P970105182 A ARP970105182 A AR P970105182A AR 011008 A1 AR011008 A1 AR 011008A1
- Authority
- AR
- Argentina
- Prior art keywords
- indazol
- urea
- phenyl
- amino
- infection
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
- 108091005804 Peptidases Proteins 0.000 title 1
- 239000004365 Protease Substances 0.000 title 1
- 102100037486 Reverse transcriptase/ribonuclease H Human genes 0.000 title 1
- 208000015181 infectious disease Diseases 0.000 title 1
- -1 3-amino-indazol-5-yl Chemical group 0.000 abstract 1
- 238000009007 Diagnostic Kit Methods 0.000 abstract 1
- 108010010369 HIV Protease Proteins 0.000 abstract 1
- XSQUKJJJFZCRTK-UHFFFAOYSA-N Urea Chemical compound NC(N)=O XSQUKJJJFZCRTK-UHFFFAOYSA-N 0.000 abstract 1
- 239000004202 carbamide Substances 0.000 abstract 1
- 239000003112 inhibitor Substances 0.000 abstract 1
- 239000000651 prodrug Chemical group 0.000 abstract 1
- 229940002612 prodrug Drugs 0.000 abstract 1
- 150000003839 salts Chemical group 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Compuestos derivados de urea 1-(3-amino-indazol-5-il)-3-fenil-metil- cíclica) de las formulas (I) y (II), o una sal farmacéuticamente aceptable ouna forma de profármaco de los mismos, que son utiles como inhibidores de la proteasa del VIH,a composiciones farmacéuticas y un equipo de diagnosticoque comprende los mismos.Compounds derived from 1- (3-amino-indazol-5-yl) -3-phenyl-methylcyclic) urea of the formulas (I) and (II), or a pharmaceutically acceptable salt or a prodrug form thereof, which are useful as inhibitors of HIV protease, to pharmaceutical compositions and to a diagnostic kit comprising them.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US74710496A | 1996-11-08 | 1996-11-08 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR011008A1 true AR011008A1 (en) | 2000-08-02 |
Family
ID=25003672
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP970105182 AR011008A1 (en) | 1996-11-08 | 1997-11-06 | UREA-DERIVED COMPOUND 1- (3-AMINO-INDAZOL-5-IL) -3-PHENYL-METHYL-CYCLIC, PHARMACEUTICAL COMPOSITION OF HIV PROTEASE AND USEFUL PHARMACEUTICAL EQUIPMENT FOR THE TREATMENT OF SUCH INFECTION |
Country Status (4)
| Country | Link |
|---|---|
| AR (1) | AR011008A1 (en) |
| HR (1) | HRP970586A2 (en) |
| LT (1) | LT4676B (en) |
| ZA (1) | ZA979867B (en) |
-
1997
- 1997-11-03 ZA ZA979867A patent/ZA979867B/en unknown
- 1997-11-04 HR HRP970586 patent/HRP970586A2/en not_active Application Discontinuation
- 1997-11-06 AR ARP970105182 patent/AR011008A1/en unknown
-
1999
- 1999-05-03 LT LT99-044A patent/LT4676B/en not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| LT99044A (en) | 2000-02-25 |
| HRP970586A2 (en) | 1998-08-31 |
| ZA979867B (en) | 1999-05-03 |
| LT4676B (en) | 2000-07-25 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| PA8468401A1 (en) | COMPOUNDS FOR THE TREATMENT OF ISCHEMIA | |
| AR030021A1 (en) | COMPOSITE OF A REPLACED PYRIMIDINONES, PHARMACEUTICAL COMPOSITION THAT INCLUDES IT AND THE USE OF SUCH COMPOUND AND SUCH COMPOSITION IN THE MANUFACTURE OF USEFUL MEDICINES FOR THE SELECTIVE INHIBITION OF THE COAGULATION CASCADE | |
| ECSP055671A (en) | NEW ESPIROCONDENSED QUINAZOLINONES AND ITS USE AS PHOSPHODESTERESA INHIBITORS | |
| AR029216A1 (en) | NON-PEPTIDIC INHIBITING COMPOUNDS OF THE VLA-4 DEPENDENT CELL UNION IN THE TREATMENT OF INFLAMMATORY, AUTOIMMUNE AND RESPIRATORY DISEASES; PHARMACEUTICAL COMPOSITION AND TREATMENT PROCEDURE | |
| CL2004000849A1 (en) | COMPOUNDS DERIVED FROM BENZAMIDAS-2-HIDROXI-3-DIAMINOALCANS, USEFUL FOR THE TREATMENT OR PREVENTION OF ALZHEIMER, DOWN SYNDROME, HEREDITARY CEREBRAL HEMORRAGY, DEGENERATIVE DEMENCIES AND OTHERS. | |
| ATE273305T1 (en) | THROMBIN INHIBITORS | |
| ES2178037T3 (en) | CYCLOSPORINE DERIVATIVES, ITS PREPARATION AND THE PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM. | |
| ECSP045004A (en) | INHIBITORS OF THE 17BETA-HYDROXIESTEROID DEHYDROGENASE TYPE 3 FOR THE TREATMENT OF DEPENDING ANDROGEN DISEASES | |
| AR030933A1 (en) | TRIAZOL DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM | |
| ECSP034642A (en) | DERIVATIVES OF TETRALONA AS ANTITUMOR AGENTS | |
| PA8495101A1 (en) | DERIVATIVES OF 13-METHYLERITROMYCIN | |
| ES2169654B1 (en) | DEFROLING AGENT | |
| ES2188604T3 (en) | HIV PROTEASE INHIBITORS IN PHARMACEUTICAL COMBINATIONS FOR AIDS TREATMENT. | |
| ES2243579T3 (en) | DERIVATIVES OF PIRAZOLOPIRIDENO. | |
| AR029635A1 (en) | COMPOUND DERIVED FROM A REPLACED POLYCLICAL PIRIDONE, PHARMACEUTICAL COMPOSITION THAT INCLUDES IT AND THE USE OF SUCH COMPOUND AND SUCH COMPOSITION IN THE MANUFACTURE OF USEFUL DRUGS FOR THE SELECTIVE INHIBITION OF THE COAGULATION WATERFALL | |
| ES2180933T3 (en) | INHIBITOR OF SERINA-PROTEASA. | |
| UY26564A1 (en) | FACTOR XA INHIBITORS WITH ARYL - AMIDINES AND THEIR DERIVATIVES, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM | |
| CR10974A (en) | CARBOXIPEPTIDASE B PLASMATIC INHIBITORS (DIVISIONAL) | |
| ES2174921T3 (en) | HIV PROTEASE INHIBITORS. | |
| CO2023015244A2 (en) | Bicyclic heteroaromatic klk5 inhibitors | |
| ES2182035T3 (en) | DERIVATIVES OF BISARILCICLOBUTENO AS CICLOOXIGENASA INHIBITORS | |
| ES2109229T3 (en) | SUBSTITUTED SULFONAMIDES AND RELATED COMPOUNDS FOR THE TREATMENT OF ASTHMA, ARTHRITIS AND RELATED DISEASES. | |
| ES2150461T3 (en) | DERIVATIVES OF AMIDINOPHENYLALANINE, PROCESS FOR ITS PREPARATION, ITS EMPLOYMENT AND AGENTS THAT CONTAIN THEM AS ANTICOAGULANTS. | |
| AR011008A1 (en) | UREA-DERIVED COMPOUND 1- (3-AMINO-INDAZOL-5-IL) -3-PHENYL-METHYL-CYCLIC, PHARMACEUTICAL COMPOSITION OF HIV PROTEASE AND USEFUL PHARMACEUTICAL EQUIPMENT FOR THE TREATMENT OF SUCH INFECTION | |
| AR022130A1 (en) | NEW DERIVATIVES OF ARILALCANOILO, THE PROCESSES FOR THE PREPARATION, USE AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FB | Suspension of granting procedure |